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—— (6R)-N-[(4-bromophenyl)methyl]-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C19H16BrClN4O2
(6R)-N-[(4-bromophenyl)methyl]-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6S)-N-[(4-bromophenyl)methyl]-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C19H16BrClN4O2
(6S)-N-[(4-bromophenyl)methyl]-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— 6-{(2E)-2-[1-(4-chlorophenyl)ethylidene]hydrazinyl}-5-nitropyrimidin-4-amine —— C12H11ClN6O2
6-{(2E)-2-[1-(4-chlorophenyl)ethylidene]hydrazinyl}-5-nitropyrimidin-4-amine
—— (6S)-6-(4-bromophenyl)-N-(2-phenylethyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C20H19BrN4O2
(6S)-6-(4-bromophenyl)-N-(2-phenylethyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6R)-6-(4-bromophenyl)-N-(2-phenylethyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C20H19BrN4O2
(6R)-6-(4-bromophenyl)-N-(2-phenylethyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6R)-6-(4-bromophenyl)-N-[(2,4-difluorophenyl)methyl]-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C19H15BrF2N4O2
(6R)-6-(4-bromophenyl)-N-[(2,4-difluorophenyl)methyl]-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— [(6S)-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazin-3-yl]-[4-(1-phenylcyclopropanecarbonyl)piperazin-1-yl]methanone —— C26H26ClN5O3
[(6S)-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazin-3-yl]-[4-(1-phenylcyclopropanecarbonyl)piperazin-1-yl]methanone
—— (6R)-N-(2,3-dihydro-1H-inden-5-yl)-6-(4-fluorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C21H19FN4O2
(6R)-N-(2,3-dihydro-1H-inden-5-yl)-6-(4-fluorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4R)-3-[(E)-3-phenylprop-2-enoyl]-1,3-thiazolidine-4-carboxylate —— C22H20BrNO5S
(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4R)-3-[(E)-3-phenylprop-2-enoyl]-1,3-thiazolidine-4-carboxylate
—— 6-ethoxy-N-[(1R)-1-(4-methoxyphenyl)propyl]imidazo[1,2-b]pyridazine-2-carboxamide —— C19H22N4O3
6-ethoxy-N-[(1R)-1-(4-methoxyphenyl)propyl]imidazo[1,2-b]pyridazine-2-carboxamide
—— (6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4R)-3-(benzenesulfonyl)-1,3-thiazolidine-4-carboxylate —— C19H18BrNO6S2
(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4R)-3-(benzenesulfonyl)-1,3-thiazolidine-4-carboxylate
—— 6-bromo-7-[[(R)-[(2R)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C15H19BrO4S
6-bromo-7-[[(R)-[(2R)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (6S)-6-(4-bromophenyl)-N-[(2,4-difluorophenyl)methyl]-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C19H15BrF2N4O2
(6S)-6-(4-bromophenyl)-N-[(2,4-difluorophenyl)methyl]-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6S)-N-(2,3-dihydro-1H-inden-5-yl)-6-(4-fluorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C21H19FN4O2
(6S)-N-(2,3-dihydro-1H-inden-5-yl)-6-(4-fluorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— (6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4S)-3-[(E)-3-phenylprop-2-enoyl]-1,3-thiazolidine-4-carboxylate —— C22H20BrNO5S
(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)methyl (4S)-3-[(E)-3-phenylprop-2-enoyl]-1,3-thiazolidine-4-carboxylate
—— 6-ethoxy-N-[(1S)-1-(4-methoxyphenyl)propyl]imidazo[1,2-b]pyridazine-2-carboxamide —— C19H22N4O3
6-ethoxy-N-[(1S)-1-(4-methoxyphenyl)propyl]imidazo[1,2-b]pyridazine-2-carboxamide
—— 6-[(2E)-2-(3,4-dimethoxybenzylidene)hydrazinyl]-N,N'-diethyl-1,3,5-triazine-2,4-diamine —— C16H23N7O2
6-[(2E)-2-(3,4-dimethoxybenzylidene)hydrazinyl]-N,N'-diethyl-1,3,5-triazine-2,4-diamine
—— 6-bromo-7-[[(S)-[(2R)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C15H19BrO4S
6-bromo-7-[[(S)-[(2R)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (6R)-6-(4-fluorophenyl)-2-[3-(4-phenylmethoxyphenyl)-1,2,4-oxadiazol-5-yl]-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine —— C27H21FN4O3
(6R)-6-(4-fluorophenyl)-2-[3-(4-phenylmethoxyphenyl)-1,2,4-oxadiazol-5-yl]-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine
—— (6R)-6-(4-bromophenyl)-N-(3-phenylpropyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide —— C21H21BrN4O2
(6R)-6-(4-bromophenyl)-N-(3-phenylpropyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carboxamide
—— [(6R)-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazin-3-yl]-[4-(1-phenylcyclopropanecarbonyl)piperazin-1-yl]methanone —— C26H26ClN5O3
[(6R)-6-(4-chlorophenyl)-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazin-3-yl]-[4-(1-phenylcyclopropanecarbonyl)piperazin-1-yl]methanone
—— 6-bromo-7-[[(S)-[(2S)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C15H19BrO4S
6-bromo-7-[[(S)-[(2S)-oxan-2-yl]methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (6S)-6-(4-fluorophenyl)-2-[3-(4-phenylmethoxyphenyl)-1,2,4-oxadiazol-5-yl]-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine —— C27H21FN4O3
(6S)-6-(4-fluorophenyl)-2-[3-(4-phenylmethoxyphenyl)-1,2,4-oxadiazol-5-yl]-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine
—— 6-phenyl-N-[(E)-(2-piperidin-1-yl-4-thiophen-2-yl-1,3-thiazol-5-yl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C25H22N6S3
6-phenyl-N-[(E)-(2-piperidin-1-yl-4-thiophen-2-yl-1,3-thiazol-5-yl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 6-(3,5-dimethylpyrazol-1-yl)-4-N-(4-methylphenyl)-2-N-[(E)-1-(4-nitrophenyl)ethylideneamino]-1,3,5-triazine-2,4-diamine —— C23H23N9O2
6-(3,5-dimethylpyrazol-1-yl)-4-N-(4-methylphenyl)-2-N-[(E)-1-(4-nitrophenyl)ethylideneamino]-1,3,5-triazine-2,4-diamine
—— 6-bromo-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-1H-indole-2-carboxamide —— C18H14BrF2N3O2
6-bromo-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-1H-indole-2-carboxamide
—— 6-bromo-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-1H-indole-2-carboxamide —— C18H14BrF2N3O2
6-bromo-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-1H-indole-2-carboxamide
—— [(6R)-6-hydroxy-1,4-diazepan-1-yl]-(1-phenylcyclopentyl)methanone —— C17H24N2O2
[(6R)-6-hydroxy-1,4-diazepan-1-yl]-(1-phenylcyclopentyl)methanone
—— [(6S)-6-hydroxy-1,4-diazepan-1-yl]-(1-phenylcyclopentyl)methanone —— C17H24N2O2
[(6S)-6-hydroxy-1,4-diazepan-1-yl]-(1-phenylcyclopentyl)methanone
—— (6S)-5-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H20ClN3O4
(6S)-5-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[(6S)-6-hydroxy-4-(5-methyl-2H-triazole-4-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C14H18N8O3
6-[(6S)-6-hydroxy-4-(5-methyl-2H-triazole-4-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— 6-[(Z)-2-[3-(difluoromethoxy)-4-methoxyphenyl]ethenyl]pyridine-3-carbonitrile —— C16H12F2N2O2
6-[(Z)-2-[3-(difluoromethoxy)-4-methoxyphenyl]ethenyl]pyridine-3-carbonitrile
—— (6S)-1-[(2-aminopyridin-3-yl)methyl]-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol —— C16H23N7O
(6S)-1-[(2-aminopyridin-3-yl)methyl]-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
—— 6-[(Z)-2-[5-(4-fluorophenyl)furan-2-yl]ethenyl]pyridine-3-carbonitrile —— C18H11FN2O
6-[(Z)-2-[5-(4-fluorophenyl)furan-2-yl]ethenyl]pyridine-3-carbonitrile
—— 6-{(E)-[2-(3-carboxyphenyl)hydraziniumylidene]methyl}-2,3-dimethoxybenzoate —— C17H16N2O6
6-{(E)-[2-(3-carboxyphenyl)hydraziniumylidene]methyl}-2,3-dimethoxybenzoate
—— 6-[(Z)-2-[4-(1,3-thiazol-4-ylmethoxy)phenyl]ethenyl]pyridine-3-carbonitrile —— C18H13N3OS
6-[(Z)-2-[4-(1,3-thiazol-4-ylmethoxy)phenyl]ethenyl]pyridine-3-carbonitrile
—— 6-[(2E)-2-[4-(1,3-benzodioxol-5-yl)butan-2-ylidene]hydrazinyl]-2H-1,2,4-triazine-3,5-dione —— C14H15N5O4
6-[(2E)-2-[4-(1,3-benzodioxol-5-yl)butan-2-ylidene]hydrazinyl]-2H-1,2,4-triazine-3,5-dione
—— 6-[(6R)-6-hydroxy-4-(5-methyl-2H-triazole-4-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C14H18N8O3
6-[(6R)-6-hydroxy-4-(5-methyl-2H-triazole-4-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— (6R)-5-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H20ClN3O4
(6R)-5-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[2-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)imino-3-[(E)-2-ethylbutylideneamino]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one —— C28H30N6O3S
6-[2-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)imino-3-[(E)-2-ethylbutylideneamino]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one
—— 6-methylsulfonyl-N-[[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]methyl]pyridin-3-amine —— C15H19N3O2S2
6-methylsulfonyl-N-[[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]methyl]pyridin-3-amine
—— 6-methylsulfonyl-N-[[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]methyl]pyridin-3-amine —— C15H19N3O2S2
6-methylsulfonyl-N-[[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]methyl]pyridin-3-amine
—— 6-[(2E)-2-[[5-(4-chlorophenyl)furan-2-yl]methylidene]hydrazinyl]-2H-1,2,4-triazine-3,5-dione —— C14H10ClN5O3
6-[(2E)-2-[[5-(4-chlorophenyl)furan-2-yl]methylidene]hydrazinyl]-2H-1,2,4-triazine-3,5-dione
—— (6R)-1-(furan-3-carbonyl)-4-[(5-methylthiophen-2-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C17H20N2O4S
(6R)-1-(furan-3-carbonyl)-4-[(5-methylthiophen-2-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-N-[[(2S)-oxolan-2-yl]methyl]-6-N-(thiophen-2-ylmethyl)-7H-purine-2,6-diamine —— C15H18N6OS
6-N-[[(2S)-oxolan-2-yl]methyl]-6-N-(thiophen-2-ylmethyl)-7H-purine-2,6-diamine
—— 6-[(5R)-4-benzyl-5-methyl-1,4-diazepan-1-yl]-7H-purin-2-amine —— C18H23N7
6-[(5R)-4-benzyl-5-methyl-1,4-diazepan-1-yl]-7H-purin-2-amine
—— 6-[(2R)-2-methyl-2-phenylmorpholin-4-yl]-7H-purin-2-amine —— C16H18N6O
6-[(2R)-2-methyl-2-phenylmorpholin-4-yl]-7H-purin-2-amine
—— 6-[(3S)-3-pyridin-3-yloxypyrrolidin-1-yl]-7H-purin-2-amine —— C14H15N7O
6-[(3S)-3-pyridin-3-yloxypyrrolidin-1-yl]-7H-purin-2-amine
—— 6-[(3R)-3-benzylpyrrolidin-1-yl]-7H-purin-2-amine —— C16H18N6
6-[(3R)-3-benzylpyrrolidin-1-yl]-7H-purin-2-amine
—— 6-[(2S,4S)-4-(4-methoxyphenyl)-2-methylpyrrolidin-1-yl]-7H-purin-2-amine —— C17H20N6O
6-[(2S,4S)-4-(4-methoxyphenyl)-2-methylpyrrolidin-1-yl]-7H-purin-2-amine