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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-3-benzyl-N-(3-ethoxyphenyl)-4-oxo-2-[4-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide —— C27H24F3N3O3S
(6R)-3-benzyl-N-(3-ethoxyphenyl)-4-oxo-2-[4-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide
—— (6S)-3-butyl-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-N-(4-ethoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C24H25ClF3N3O3S
(6S)-3-butyl-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-N-(4-ethoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-3-benzyl-N-(3-chloro-4-methylphenyl)-4-oxo-2-[4-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide —— C26H21ClF3N3O2S
(6S)-3-benzyl-N-(3-chloro-4-methylphenyl)-4-oxo-2-[4-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide
—— 6-ethyl-7-hydroxy-2-methyl-3-(1H-pyrazol-3-yl)-4H-chromen-4-one —— C15H14N2O3
6-ethyl-7-hydroxy-2-methyl-3-(1H-pyrazol-3-yl)-4H-chromen-4-one
—— (6S)-N-(3-chlorophenyl)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C27H25ClFN3O4S
(6S)-N-(3-chlorophenyl)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(3-chlorophenyl)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C27H25ClFN3O4S
(6R)-N-(3-chlorophenyl)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H28N2O4
(6S,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C32H29N3O5
(6S,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C32H29N3O5
(6S,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C28H28FN3O5S
(6R)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C32H29N3O5
(6R,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-N-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6Z)-2-(3,4-dimethoxybenzyl)-5-imino-6-(1H-indol-3-ylmethylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H19N5O3S
(6Z)-2-(3,4-dimethoxybenzyl)-5-imino-6-(1H-indol-3-ylmethylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(2,4-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H19Cl2N5OS
(6E)-6-{[1-(2,4-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C29H30FN3O5S
(6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6Z)-2-(benzylsulfanyl)-5-imino-6-(4-methoxybenzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H16N4O2S2
(6Z)-2-(benzylsulfanyl)-5-imino-6-(4-methoxybenzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-2-(4-chlorophenyl)imino-N-(3-ethoxyphenyl)-3-[2-(4-fluorophenyl)ethyl]-4-oxo-1,3-thiazinane-6-carboxamide —— C27H25ClFN3O3S
(6S)-2-(4-chlorophenyl)imino-N-(3-ethoxyphenyl)-3-[2-(4-fluorophenyl)ethyl]-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H28N2O4
(6R,9R)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6Z)-2-ethyl-5-imino-6-{3-methoxy-4-[2-(3-methylphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O4S
(6Z)-2-ethyl-5-imino-6-{3-methoxy-4-[2-(3-methylphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C28H28FN3O5S
(6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2-fluorophenyl)imino-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H28N2O4
(6R,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H22Cl2N2O3
(6S,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-3-[2-(3,4-dimethoxyphenyl)ethyl]-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C29H30FN3O5S
(6R)-3-[2-(3,4-dimethoxyphenyl)ethyl]-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-ethyl-2-[(3S)-1-(imidazole-1-carbonyl)piperidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2
6-ethyl-2-[(3S)-1-(imidazole-1-carbonyl)piperidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-chloro-3-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one —— C22H19ClN4O2
6-chloro-3-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one
—— (6Z)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H20FN5OS
(6Z)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-(imidazole-1-carbonyl)piperidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2
6-ethyl-2-[(3R)-1-(imidazole-1-carbonyl)piperidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6R,9R)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H22Cl2N2O3
(6R,9R)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[[4-(1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2,4-dichlorocyclohexa-2,4-dien-1-one —— C21H14Cl2N2O2
(6E)-6-[[4-(1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2,4-dichlorocyclohexa-2,4-dien-1-one
—— (6R,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H22Cl2N2O3
(6R,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6Z)-6-{4-[(2-chlorobenzyl)oxy]-3-methoxybenzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H18Cl2N4O3S
(6Z)-6-{4-[(2-chlorobenzyl)oxy]-3-methoxybenzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O3
6-ethyl-5-methyl-2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6S,9R)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H22Cl2N2O3
(6S,9R)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-methyl-3-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one —— C23H22N4O2
6-methyl-3-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one
—— 6-[(E)-2-(4-bromo-3-nitrophenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione —— C12H7BrN4O6
6-[(E)-2-(4-bromo-3-nitrophenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione
—— (6S,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H28N2O4
(6S,9S)-9-(furan-2-yl)-6-(2-methoxyphenyl)-5-(naphthalene-1-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-chloro-3-[[(1S,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one —— C22H19ClN4O2
6-chloro-3-[[(1S,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H28N4O5
6-ethyl-5-methyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6Z)-2-ethyl-6-{4-[2-(3-ethyl-5-methylphenoxy)ethoxy]-3-methoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N4O4S
(6Z)-2-ethyl-6-{4-[2-(3-ethyl-5-methylphenoxy)ethoxy]-3-methoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[2-[4-(1,1,1,3,3,3-hexafluoropropan-2-yloxy)-6-(4-nitroanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C19H12F6N8O6
(6E)-6-[[2-[4-(1,1,1,3,3,3-hexafluoropropan-2-yloxy)-6-(4-nitroanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6R)-3-[(3,4-dimethoxyphenyl)methyl]-N-(3-ethoxyphenyl)-2-(4-methoxyphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C29H31N3O6S
(6R)-3-[(3,4-dimethoxyphenyl)methyl]-N-(3-ethoxyphenyl)-2-(4-methoxyphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-ethyl-5-methyl-2-[(2S)-1-[(1S,2S,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O3
6-ethyl-5-methyl-2-[(2S)-1-[(1S,2S,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[(1S,2S,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O3
6-ethyl-5-methyl-2-[(2R)-1-[(1S,2S,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[(1S,2R,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O3
6-ethyl-5-methyl-2-[(2S)-1-[(1S,2R,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[(1S,2R,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O3
6-ethyl-5-methyl-2-[(2R)-1-[(1S,2R,4R)-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H28N4O5
6-ethyl-5-methyl-2-[(2R)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6E)-4,5-dibromo-2-ethoxy-6-[[[2-(4-methoxyphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C23H18Br2N2O4
(6E)-4,5-dibromo-2-ethoxy-6-[[[2-(4-methoxyphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-benzyl-6-{[1-(3,4-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5OS
(6Z)-2-benzyl-6-{[1-(3,4-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2,4-dibromo-6-[[2-(4-morpholin-4-ylsulfonyl-2-nitrophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C17H16Br2N4O6S
(6E)-2,4-dibromo-6-[[2-(4-morpholin-4-ylsulfonyl-2-nitrophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(E)-2-(2,4-diethoxyphenyl)ethenyl]-5-nitropyrimidine-2,4-diol —— C16H17N3O6
6-[(E)-2-(2,4-diethoxyphenyl)ethenyl]-5-nitropyrimidine-2,4-diol
—— (6E)-6-[amino(nitroso)methylidene]-N,N-diphenyl-4-pyrrolidin-1-yl-1H-1,3,5-triazin-2-amine —— C20H21N7O
(6E)-6-[amino(nitroso)methylidene]-N,N-diphenyl-4-pyrrolidin-1-yl-1H-1,3,5-triazin-2-amine