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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(2-hydroxyethyl)-N-methyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H22N4O2
6-(2-hydroxyethyl)-N-methyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-1-(5-chloropyridin-2-yl)-4-[2-(dimethylamino)ethyl]-1,4-diazepan-6-ol —— C14H23ClN4O
(6R)-1-(5-chloropyridin-2-yl)-4-[2-(dimethylamino)ethyl]-1,4-diazepan-6-ol
—— 6-methyl-N-[(3R)-1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H19N5O2S
6-methyl-N-[(3R)-1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[(4-hydroxyphenyl)methyl]-1-[(Z)-3-phenylprop-2-enyl]-3-pyridin-4-yl-7,8-dihydro-5H-1,6-naphthyridin-2-one —— C29H27N3O2
6-[(4-hydroxyphenyl)methyl]-1-[(Z)-3-phenylprop-2-enyl]-3-pyridin-4-yl-7,8-dihydro-5H-1,6-naphthyridin-2-one
—— (6S)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H23N3O3
(6S)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-methyl-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H19N5O2S
6-methyl-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one —— C23H34N4O3
(6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
—— (6R)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H23N3O3
(6R)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-4-[(Z)-3-(4-methoxyphenyl)prop-2-enyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one —— C27H35N3O4
(6S)-4-[(Z)-3-(4-methoxyphenyl)prop-2-enyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
—— [(6R)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-(6-methylpyridin-2-yl)methanone —— C17H23N3O2
[(6R)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-(6-methylpyridin-2-yl)methanone
—— [(6S)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-(6-methylpyridin-2-yl)methanone —— C17H23N3O2
[(6S)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-(6-methylpyridin-2-yl)methanone
—— (6S)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-(oxan-4-ylmethyl)-6-phenylmethoxy-1,4-diazepan-2-one —— C28H36N2O5
(6S)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-(oxan-4-ylmethyl)-6-phenylmethoxy-1,4-diazepan-2-one
—— (6R)-1-[2-(methylamino)acetyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid —— C14H25N3O4
(6R)-1-[2-(methylamino)acetyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
—— 6-(1H-indol-3-ylmethyl)-3-[(Z)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-7,8-dihydro-5H-1,6-naphthyridin-2-one —— C31H28N4O
6-(1H-indol-3-ylmethyl)-3-[(Z)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-7,8-dihydro-5H-1,6-naphthyridin-2-one
—— 6-bromo-3-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one —— C20H19BrN2O3
6-bromo-3-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one
—— 6-chloro-3-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one —— C20H19ClN2O3
6-chloro-3-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one
—— 6-chloro-3-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one —— C20H19ClN2O3
6-chloro-3-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one
—— 6-bromo-3-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one —— C20H19BrN2O3
6-bromo-3-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]quinazolin-4-one
—— 6-nitro-N-[(1R)-1-phenylethyl]quinolin-2-amine —— C17H15N3O2
6-nitro-N-[(1R)-1-phenylethyl]quinolin-2-amine
—— 6-cyclopropyl-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H25N3O4
6-cyclopropyl-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-4-carboxamide —— C23H28N4O3
6-cyclopropyl-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H25N3O4
6-cyclopropyl-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C23H26FN3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-4-carboxamide —— C23H28N4O3
6-cyclopropyl-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-4-carboxamide
—— (6R)-1-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-1,4-diazepane-6-carboxylic acid —— C15H22N4O3
(6R)-1-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-1,4-diazepane-6-carboxylic acid
—— 6-cyclopropyl-N-[(2R)-1-hydroxypropan-2-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C16H21N3O3
6-cyclopropyl-N-[(2R)-1-hydroxypropan-2-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H22FN3O3
6-cyclopropyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C23H26FN3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(2S)-1-hydroxypropan-2-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C16H21N3O3
6-cyclopropyl-N-[(2S)-1-hydroxypropan-2-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C24H20FN3O3
6-cyclopropyl-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(S)-phenyl(pyridin-4-yl)methyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C25H24N4O2
6-cyclopropyl-N-[(S)-phenyl(pyridin-4-yl)methyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H22F2N4O3
6-cyclopropyl-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H27N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-1-hydroxypropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C18H25N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-1-hydroxypropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-2-hydroxypropyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C18H25N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-2-hydroxypropyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(2R)-2-hydroxypropyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C16H21N3O3
6-cyclopropyl-N-[(2R)-2-hydroxypropyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-2-hydroxypropyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C18H25N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2R)-2-hydroxypropyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H27N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6S)-1-[2-(cyclopropylamino)acetyl]-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H24N4O4
(6S)-1-[2-(cyclopropylamino)acetyl]-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-1-hydroxypropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C18H25N3O3
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(2S)-1-hydroxypropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6R)-1-[2-(cyclopropylamino)acetyl]-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H24N4O4
(6R)-1-[2-(cyclopropylamino)acetyl]-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-cyclopropyl-N-[(2S)-2-hydroxypropyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C16H21N3O3
6-cyclopropyl-N-[(2S)-2-hydroxypropyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C24H20FN3O3
6-cyclopropyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H22F2N4O3
6-cyclopropyl-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[(R)-phenyl(pyridin-4-yl)methyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C25H24N4O2
6-cyclopropyl-N-[(R)-phenyl(pyridin-4-yl)methyl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6S)-5-[(7-methoxy-1,3-benzodioxol-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C16H17N3O5
(6S)-5-[(7-methoxy-1,3-benzodioxol-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-5-[4-(4-tert-butylphenyl)-4-oxobutyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C21H27N3O3
(6S)-5-[4-(4-tert-butylphenyl)-4-oxobutyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— [(6R)-4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C15H20N8O2
[(6R)-4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— (6R)-5-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H17FN4O2
(6R)-5-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-(dimethylamino)-N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methylpyridine-3-carboxamide —— C17H22N4O2
6-(dimethylamino)-N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methylpyridine-3-carboxamide