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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(cyclopropylmethoxy)-N-[[(3R)-1-(2-phenylethyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C23H29N3O2
6-(cyclopropylmethoxy)-N-[[(3R)-1-(2-phenylethyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— 6-(3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-(4-methoxyphenyl)pentyl]pyridine-3-carboxamide —— C23H28N4O2
6-(3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-(4-methoxyphenyl)pentyl]pyridine-3-carboxamide
—— 6-(furan-2-yl)-N-[(1S)-1-(4-methoxyphenyl)pentyl]-2-oxo-1H-pyridine-3-carboxamide —— C22H24N2O4
6-(furan-2-yl)-N-[(1S)-1-(4-methoxyphenyl)pentyl]-2-oxo-1H-pyridine-3-carboxamide
—— 6-(3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(4-methoxyphenyl)pentyl]pyridine-3-carboxamide —— C23H28N4O2
6-(3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(4-methoxyphenyl)pentyl]pyridine-3-carboxamide
—— 6-chloro-4-[2-[2-[[3-[[1-[(2R,5S)-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-4-yl]amino]propylamino]methyl]cyclopropyl]ethynyl]-4-(trifluoromethyl)-1H-3,1-benzoxazin-2-one —— C27H29ClF3N5O5
6-chloro-4-[2-[2-[[3-[[1-[(2R,5S)-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-4-yl]amino]propylamino]methyl]cyclopropyl]ethynyl]-4-(trifluoromethyl)-1H-3,1-benzoxazin-2-one
—— 6-(furan-2-yl)-N-[(1R)-1-(4-methoxyphenyl)pentyl]-2-oxo-1H-pyridine-3-carboxamide —— C22H24N2O4
6-(furan-2-yl)-N-[(1R)-1-(4-methoxyphenyl)pentyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R,7R)-3-[[3-amino-4-(2-aminoethyl)-2-methylpyrazol-1-ium-1-yl]methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(2-carboxypropan-2-yloxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C22H29N10O7S2+
(6R,7R)-3-[[3-amino-4-(2-aminoethyl)-2-methylpyrazol-1-ium-1-yl]methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(2-carboxypropan-2-yloxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— [(6E,8E,10E,16Z)-15-hydroxy-5-methoxy-14,16-dimethyl-3,22,24-trioxo-2-azabicyclo[18.3.1]tetracosa-1(23),6,8,10,16,20-hexaen-13-yl] 2-(cyclopropanecarbonylamino)propanoate —— C33H42N2O8
[(6E,8E,10E,16Z)-15-hydroxy-5-methoxy-14,16-dimethyl-3,22,24-trioxo-2-azabicyclo[18.3.1]tetracosa-1(23),6,8,10,16,20-hexaen-13-yl] 2-(cyclopropanecarbonylamino)propanoate
—— (6R)-1-(1H-indol-5-ylmethyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol —— C19H27N3O2
(6R)-1-(1H-indol-5-ylmethyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
—— 6-(4-methoxy-benzyl)-7-(((5-methoxy-1H-indole-2-carbonyl)amino)-methyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid —— C29H28N4O8S
6-(4-methoxy-benzyl)-7-(((5-methoxy-1H-indole-2-carbonyl)amino)-methyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid
—— [(6S)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-imidazo[1,2-a]pyridin-3-ylmethanone —— C16H19N7O2
[(6S)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-imidazo[1,2-a]pyridin-3-ylmethanone
—— [(6R)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C15H23N5O3
[(6R)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— 6-[2-ethoxy-5-(4-ethylpiperazin-1-yl)sulfonylpyridin-3-yl]-1-propyl-3-(pyrazin-2-ylmethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C26H33N9O4S
6-[2-ethoxy-5-(4-ethylpiperazin-1-yl)sulfonylpyridin-3-yl]-1-propyl-3-(pyrazin-2-ylmethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[4-(4-Imino-1-methyl-2-phenyl-4a,8a-dihydroquinolin-6-yl)-6-methylsulfanyl-1,3,5-triazin-2-yl]-1-methyl-2-phenylquinolin-4-imine —— C36H31N7S
6-[4-(4-Imino-1-methyl-2-phenyl-4a,8a-dihydroquinolin-6-yl)-6-methylsulfanyl-1,3,5-triazin-2-yl]-1-methyl-2-phenylquinolin-4-imine
—— [(6R)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-imidazo[1,2-a]pyridin-3-ylmethanone —— C16H19N7O2
[(6R)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-imidazo[1,2-a]pyridin-3-ylmethanone
—— [(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(2-thiophen-2-ylpyrimidin-5-yl)methanone —— C16H20N4O3S
[(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(2-thiophen-2-ylpyrimidin-5-yl)methanone
—— (6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-3-[(E)-[2-oxo-1-[(3R)-pyrrolidin-3-yl]pyrrolidin-3-ylidene]methyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H22ClN7O6S2
(6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-3-[(E)-[2-oxo-1-[(3R)-pyrrolidin-3-yl]pyrrolidin-3-ylidene]methyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R)-1-(1H-indol-2-ylmethyl)-4-pyridin-4-yl-1,4-diazepan-6-ol —— C19H22N4O
(6R)-1-(1H-indol-2-ylmethyl)-4-pyridin-4-yl-1,4-diazepan-6-ol
—— (6R,7R)-3-[[4-(2-aminoethylsulfanylmethyl)-1,3-thiazol-5-yl]sulfanyl]-7-[[(2Z)-2-(6-amino-1H-pyridin-2-ylidene)-2-nitrosoacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H21N7O5S4
(6R,7R)-3-[[4-(2-aminoethylsulfanylmethyl)-1,3-thiazol-5-yl]sulfanyl]-7-[[(2Z)-2-(6-amino-1H-pyridin-2-ylidene)-2-nitrosoacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,7R)-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-3-[(E)-3-imidazo[5,1-b][1,3]thiazol-6-ium-6-ylprop-1-enyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H18FN8O5S3+
(6R,7R)-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-3-[(E)-3-imidazo[5,1-b][1,3]thiazol-6-ium-6-ylprop-1-enyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-(dimethylamino)-N-[2-(3-methyl-7-oxo-5-thia-10-azatetracyclo[7.4.0.01,12.02,6]trideca-2(6),3,8-triene-10-carbonyl)-1H-indol-5-yl]-1H-indole-2-carboxamide —— C32H27N5O3S
6-(dimethylamino)-N-[2-(3-methyl-7-oxo-5-thia-10-azatetracyclo[7.4.0.01,12.02,6]trideca-2(6),3,8-triene-10-carbonyl)-1H-indol-5-yl]-1H-indole-2-carboxamide
—— 6,11-dihydro-11-[1-[2-[4-(2-quinolinylmethoxy)phenyl]ethyl]-4-piperidinylidene]-5H-imidazo[2,1-b][3]benzazepine-3-methanol —— C36H36N4O2
6,11-dihydro-11-[1-[2-[4-(2-quinolinylmethoxy)phenyl]ethyl]-4-piperidinylidene]-5H-imidazo[2,1-b][3]benzazepine-3-methanol
—— (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-[(4-carbamoyl-6,7-dihydro-5H-cyclopenta[b]pyridin-1-ium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C23H24N7O6S2+
(6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-[(4-carbamoyl-6,7-dihydro-5H-cyclopenta[b]pyridin-1-ium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6,20-dihydroxy-13-(2-hydroxyethyl)-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione —— C28H25N3O10
6,20-dihydroxy-13-(2-hydroxyethyl)-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione
—— (6R,7R)-3-[(E)-2-[1-(2-amino-2-oxoethyl)pyridin-1-ium-4-yl]sulfanylethenyl]-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C21H19N7O6S3
(6R,7R)-3-[(E)-2-[1-(2-amino-2-oxoethyl)pyridin-1-ium-4-yl]sulfanylethenyl]-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— 6-{3-[benzothiazol-2-yl-(2,4-bis-trifluoromethyl-benzyl)-amino]-propoxy}-pyridine-2-carboxylic acid —— C25H19F6N3O3S
6-{3-[benzothiazol-2-yl-(2,4-bis-trifluoromethyl-benzyl)-amino]-propoxy}-pyridine-2-carboxylic acid
—— (6R,7R)-3-[(7-aminopyrazolo[1,5-a]pyrimidin-4-ium-4-yl)methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C19H17FN10O5S2
(6R,7R)-3-[(7-aminopyrazolo[1,5-a]pyrimidin-4-ium-4-yl)methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— 6,7-dichloro-3-(1-phenylimidazol-2-yl)-N-(4-pyrrolidin-1-ylbutyl)quinoxalin-2-amine;dihydrochloride —— C25H28Cl4N6
6,7-dichloro-3-(1-phenylimidazol-2-yl)-N-(4-pyrrolidin-1-ylbutyl)quinoxalin-2-amine;dihydrochloride
—— (6R,7R)-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-3-[(E)-(3-ethyl-2-methyliminoimidazolidin-1-yl)iminomethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H23FN10O5S2
(6R,7R)-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-3-[(E)-(3-ethyl-2-methyliminoimidazolidin-1-yl)iminomethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S)-1-(3-carbamoylpyridin-2-yl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C15H19N7O3
(6S)-1-(3-carbamoylpyridin-2-yl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— [(6S)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C15H23N5O3
[(6S)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— (6S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H22N2O4
(6S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6R,7R)-3-[(7-aminopyrazolo[1,5-a]pyrimidin-4-ium-4-yl)methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H18FN10O5S2+
(6R,7R)-3-[(7-aminopyrazolo[1,5-a]pyrimidin-4-ium-4-yl)methyl]-7-[[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(fluoromethoxyimino)acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-[Amino-(4-chlorophenyl)-(3-methylimidazol-4-yl)methyl]-4-(3-bromophenyl)-1-methylquinolin-2-one —— C27H22BrClN4O
6-[Amino-(4-chlorophenyl)-(3-methylimidazol-4-yl)methyl]-4-(3-bromophenyl)-1-methylquinolin-2-one
—— 6-[(8aS)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-5-methoxy-N-[5-(2-methylpyridin-3-yl)naphthalen-1-yl]-2,3-dihydroindole-1-carboxamide —— C33H35N5O2
6-[(8aS)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-5-methoxy-N-[5-(2-methylpyridin-3-yl)naphthalen-1-yl]-2,3-dihydroindole-1-carboxamide
—— 6-[5-(5,7-Dihydroxy-4-oxochromen-3-yl)-2-hydroxyphenyl]-5,7-dihydroxy-3-(4-hydroxyphenyl)chromen-4-one —— C30H18O10
6-[5-(5,7-Dihydroxy-4-oxochromen-3-yl)-2-hydroxyphenyl]-5,7-dihydroxy-3-(4-hydroxyphenyl)chromen-4-one
—— 6-(2-aminoethyl)-3,19,21-trihydroxy-15-methoxy-20-methyl-6,7-diazahexacyclo[12.12.0.02,11.04,9.016,25.018,23]hexacosa-1,3,8,10,14,16(25),18,20,22-nonaene-5,17,24,26-tetrone —— C28H23N3O8
6-(2-aminoethyl)-3,19,21-trihydroxy-15-methoxy-20-methyl-6,7-diazahexacyclo[12.12.0.02,11.04,9.016,25.018,23]hexacosa-1,3,8,10,14,16(25),18,20,22-nonaene-5,17,24,26-tetrone
—— (6E,8E,10E,12E,14E,16E,18E,20E,22E)-3-hydroxy-23-(4-hydroxy-2,6,6-trimethylcyclohexen-1-yl)-9,12,17,21-tetramethyltricosa-6,8,10,12,14,16,18,20,22-nonaen-5-one —— C36H50O3
(6E,8E,10E,12E,14E,16E,18E,20E,22E)-3-hydroxy-23-(4-hydroxy-2,6,6-trimethylcyclohexen-1-yl)-9,12,17,21-tetramethyltricosa-6,8,10,12,14,16,18,20,22-nonaen-5-one
—— (6R)-1-(4-aminopyrimidin-2-yl)-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1,4-diazepan-6-ol —— C13H18N6O2S
(6R)-1-(4-aminopyrimidin-2-yl)-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1,4-diazepan-6-ol
—— 6-fluoro-N-{7-[(6-fluoro-1,2,3,4-tetrahydroacridin-9-yl)amino]heptyl}-1,2,3,4-tetrahydroacridin-9-amine —— C33H38F2N4
6-fluoro-N-{7-[(6-fluoro-1,2,3,4-tetrahydroacridin-9-yl)amino]heptyl}-1,2,3,4-tetrahydroacridin-9-amine
—— (6R)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H22N2O4
(6R)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-[[4-(4-fluorophenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione —— C22H18FN5O2S
6-[[4-(4-fluorophenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-[[4-(3-methoxyphenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione —— C23H21N5O3S
6-[[4-(3-methoxyphenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione
—— [(6R)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-(2H-triazol-4-yl)methanone —— C14H16N8O2
[(6R)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-(2H-triazol-4-yl)methanone
—— [(6S)-6-hydroxy-1,4-diazepan-1-yl]-(2-methyl-5-phenylpyrazol-3-yl)methanone —— C16H20N4O2
[(6S)-6-hydroxy-1,4-diazepan-1-yl]-(2-methyl-5-phenylpyrazol-3-yl)methanone
—— 6,7-Dimethoxy-2-[4-[(3-phenylmethoxyphenyl)methyl]piperazin-1-yl]quinazolin-4-amine —— C28H31N5O3
6,7-Dimethoxy-2-[4-[(3-phenylmethoxyphenyl)methyl]piperazin-1-yl]quinazolin-4-amine
—— 6,7-Dimethoxy-2-[4-[(3-phenylmethoxyphenyl)methyl]piperazin-1-yl]quinazolin-4-amine;hydrochloride —— C28H32ClN5O3
6,7-Dimethoxy-2-[4-[(3-phenylmethoxyphenyl)methyl]piperazin-1-yl]quinazolin-4-amine;hydrochloride
—— [(6R)-6-hydroxy-1,4-diazepan-1-yl]-(2-methyl-5-phenylpyrazol-3-yl)methanone —— C16H20N4O2
[(6R)-6-hydroxy-1,4-diazepan-1-yl]-(2-methyl-5-phenylpyrazol-3-yl)methanone
—— [(6R)-6-hydroxy-4-(2-morpholin-4-ylethyl)-1,4-diazepan-1-yl]-(1H-imidazol-5-yl)methanone —— C15H25N5O3
[(6R)-6-hydroxy-4-(2-morpholin-4-ylethyl)-1,4-diazepan-1-yl]-(1H-imidazol-5-yl)methanone
—— 6-butyl-11-methyl-5-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-2,5,7,10-tetrazatetracyclo[9.2.2.02,10.04,8]pentadeca-4(8),6-dien-3-one —— C30H34N8O
6-butyl-11-methyl-5-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]-2,5,7,10-tetrazatetracyclo[9.2.2.02,10.04,8]pentadeca-4(8),6-dien-3-one