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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R,9S)-5-propanoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O8
(6R,9S)-5-propanoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-N-(3,4-dichlorophenyl)-6-(3-fluorophenyl)-9-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C33H26Cl2FN3O3
(6S,9S)-N-(3,4-dichlorophenyl)-6-(3-fluorophenyl)-9-(4-methoxyphenyl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R,9S)-5-benzyl-9-(4-tert-butylphenyl)-6-(2,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C36H34Cl2N2O
(6R,9S)-5-benzyl-9-(4-tert-butylphenyl)-6-(2,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H39ClN2O2
(6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-6-(3,5-ditert-butyl-4-hydroxyphenyl)-9-(4-fluorophenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C36H41FN2O3
(6R,9R)-6-(3,5-ditert-butyl-4-hydroxyphenyl)-9-(4-fluorophenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-chloro-N-[2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]quinolin-2-amine —— C22H25ClN4O
6-chloro-N-[2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]quinolin-2-amine
—— (6R)-6-tert-butyl-2-[[2-(2-chloro-5-methylphenoxy)acetyl]amino]-N-(2-ethoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C30H35ClN2O4S
(6R)-6-tert-butyl-2-[[2-(2-chloro-5-methylphenoxy)acetyl]amino]-N-(2-ethoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-5-benzoyl-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C37H35ClN2O4
(6S)-5-benzoyl-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-N-(3,4-dichlorophenyl)-6-(2-fluorophenyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C32H24Cl2FN3O2
(6S,9S)-N-(3,4-dichlorophenyl)-6-(2-fluorophenyl)-7-oxo-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S)-5-acetyl-6-[3-(1-adamantyl)-1-phenylpyrazol-4-yl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H40N4O2
(6S)-5-acetyl-6-[3-(1-adamantyl)-1-phenylpyrazol-4-yl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H30ClN3O2
(6R,9S)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(2-Aminocyclohexyl)amino]-2-(3-bromoanilino)pyridine-3-carboxamide —— C18H22BrN5O
6-[(2-Aminocyclohexyl)amino]-2-(3-bromoanilino)pyridine-3-carboxamide
—— (6R,9S)-5-benzoyl-6-(4-chlorophenyl)-9-(3,4-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H29ClN2O4
(6R,9S)-5-benzoyl-6-(4-chlorophenyl)-9-(3,4-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-acetyl-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C32H33ClN2O4
(6S)-5-acetyl-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-Chloro-4-[2-(2-chlorophenyl)ethynyl]-4-(trifluoromethyl)-1,3-dihydroquinazoline-2-thione —— C17H9Cl2F3N2S
6-Chloro-4-[2-(2-chlorophenyl)ethynyl]-4-(trifluoromethyl)-1,3-dihydroquinazoline-2-thione
—— (6R)-9,9-dimethyl-5-(2-phenylacetyl)-6-(4-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H34N2O3
(6R)-9,9-dimethyl-5-(2-phenylacetyl)-6-(4-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6Z)-4-bromo-3-fluoro-6-[(3-hydroxy-1-oxidopyridin-1-ium-2-yl)-[(2-methylpropan-2-yl)oxyamino]methylidene]cyclohexa-2,4-dien-1-one —— C16H16BrFN2O4
(6Z)-4-bromo-3-fluoro-6-[(3-hydroxy-1-oxidopyridin-1-ium-2-yl)-[(2-methylpropan-2-yl)oxyamino]methylidene]cyclohexa-2,4-dien-1-one
—— (6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-(thiophene-2-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H31ClN2O2S
(6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-(thiophene-2-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,7R)-7-[[(2S)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H23ClN6O4S3
(6R,7R)-7-[[(2S)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,9R)-9-(3,4-dimethoxyphenyl)-6-(4-fluorophenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H35FN2O4
(6R,9R)-9-(3,4-dimethoxyphenyl)-6-(4-fluorophenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,7R)-7-[[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H23ClN6O4S3
(6R,7R)-7-[[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,9S)-6-(3-bromophenyl)-5-hexanoyl-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H33BrN2O2
(6S,9S)-6-(3-bromophenyl)-5-hexanoyl-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,7R)-7-[[(2S)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H23ClN6O4S3
(6R,7R)-7-[[(2S)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-[(3S,4R)-3-hydroxy-2,2-dimethyl-6-(trifluoromethoxy)-3,4-dihydrochromen-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C19H17F3N2O4
6-[(3S,4R)-3-hydroxy-2,2-dimethyl-6-(trifluoromethoxy)-3,4-dihydrochromen-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— 6-[5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-bicyclo[3.1.0]hex-2-en-2-yl]-nicotinic acid —— C27H31NO2
6-[5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-bicyclo[3.1.0]hex-2-en-2-yl]-nicotinic acid
—— (6S,7S)-7-[(4-bromo-1,5-dimethylpyrazole-3-carbonyl)amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17BrN6O4S3
(6S,7S)-7-[(4-bromo-1,5-dimethylpyrazole-3-carbonyl)amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,9S)-6-[2-[(2S)-butan-2-yl]oxyphenyl]-9-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O5
(6R,9S)-6-[2-[(2S)-butan-2-yl]oxyphenyl]-9-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-9-(4-fluorophenyl)-6-(4-pentoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H30F4N2O3
(6S,9S)-9-(4-fluorophenyl)-6-(4-pentoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-9-(4-fluorophenyl)-6-(4-pentoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H30F4N2O3
(6S,9R)-9-(4-fluorophenyl)-6-(4-pentoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C31H28ClF3N2O2
(6R,9S)-9-(4-tert-butylphenyl)-6-(2-chlorophenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C36H34N2O3
(6S,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-5-benzoyl-6-(3-bromophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27BrN2O2
(6R,9S)-5-benzoyl-6-(3-bromophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-6-(4-acetylphenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H38N2O5
(6S,9R)-6-(4-acetylphenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-tert-butyl-2-[[2-(2-chloro-5-methylphenoxy)acetyl]amino]-N-(2-ethoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C30H35ClN2O4S
(6S)-6-tert-butyl-2-[[2-(2-chloro-5-methylphenoxy)acetyl]amino]-N-(2-ethoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R,9S)-6-(4-acetylphenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H38N2O5
(6R,9S)-6-(4-acetylphenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-5-benzoyl-6-(4-chlorophenyl)-9-(3,4-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H29ClN2O4
(6S,9R)-5-benzoyl-6-(4-chlorophenyl)-9-(3,4-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,7S)-7-[[(2S)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H23ClN6O4S3
(6R,7S)-7-[[(2S)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,9R)-5-benzoyl-6-(3-bromophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27BrN2O2
(6S,9R)-5-benzoyl-6-(3-bromophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-cyclobutyl-3-(2,6-difluorophenyl)-5-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,3-triazolo[4,5-b]pyridine 252750-07-5 C19H17F2N7O
6-cyclobutyl-3-(2,6-difluorophenyl)-5-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,3-triazolo[4,5-b]pyridine
—— (6R,9S)-5-hexanoyl-6-(4-methoxyphenyl)-9-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H33F3N2O3
(6R,9S)-5-hexanoyl-6-(4-methoxyphenyl)-9-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H30ClN3O2
(6R,9R)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— [6-Benzyl-7-ethyl-3-methyl-8-oxamoylpyrrolo[1,2-a]pyrazin-1-yl]oxyacetic acid 245756-89-2 C21H21N3O5
[6-Benzyl-7-ethyl-3-methyl-8-oxamoylpyrrolo[1,2-a]pyrazin-1-yl]oxyacetic acid
—— (6S,9S)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H30ClN3O2
(6S,9S)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H30ClN3O2
(6S,9R)-5-(4-chlorobenzoyl)-6-[4-(dimethylamino)phenyl]-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,7S)-7-[[(2R)-2-(4-bromopyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17BrN6O4S3
(6S,7S)-7-[[(2R)-2-(4-bromopyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-[(1S,2R,6S,7R,8R,9S)-8,9-dibromo-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(4-ethoxyphenyl)hexanamide —— C23H28Br2N2O4
6-[(1S,2R,6S,7R,8R,9S)-8,9-dibromo-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(4-ethoxyphenyl)hexanamide
—— (6R)-5-(2-fluorobenzoyl)-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C35H31FN2O3
(6R)-5-(2-fluorobenzoyl)-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-6-[2-[(2R)-butan-2-yl]oxyphenyl]-9-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O5
(6R,9S)-6-[2-[(2R)-butan-2-yl]oxyphenyl]-9-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-(N-carbamoyl-2,6-difluoroanilino)-2-(4-fluoro-2-methylphenyl)pyridine-3-carboxamide —— C20H15F3N4O2
6-(N-carbamoyl-2,6-difluoroanilino)-2-(4-fluoro-2-methylphenyl)pyridine-3-carboxamide
—— (6R,7R)-7-[[(2R)-2-(4-bromopyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17BrN6O4S3
(6R,7R)-7-[[(2R)-2-(4-bromopyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid