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—— (6E)-5-imino-2-(methylsulfanyl)-6-[(6-phenylimidazo[2,1-b][1,3]thiazol-5-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C18H12N6OS3
(6E)-5-imino-2-(methylsulfanyl)-6-[(6-phenylimidazo[2,1-b][1,3]thiazol-5-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-2-benzoyl-6-(4-fluoro-3-phenoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C34H29FN2O3
(6S)-2-benzoyl-6-(4-fluoro-3-phenoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6Z)-6-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H34N4O4S
(6Z)-6-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H34N4O4S
(6Z)-6-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H34N4O4S
(6Z)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-ethoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-ethyl-7-hydroxy-2-methyl-3-(1-methylbenzimidazol-2-yl)-8-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]chromen-4-one —— C31H37N3O3
6-ethyl-7-hydroxy-2-methyl-3-(1-methylbenzimidazol-2-yl)-8-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]chromen-4-one
—— (6Z)-6-[[5-bromo-2-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O3S
(6Z)-6-[[5-bromo-2-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(5E)-5-[(4-methoxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-[5-[(4-methylphenyl)methyl]-1,3-thiazol-2-yl]hexanamide —— C28H29N3O3S3
6-[(5E)-5-[(4-methoxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-[5-[(4-methylphenyl)methyl]-1,3-thiazol-2-yl]hexanamide
—— 6-[3-[(5E)-5-[(E)-2-methyl-3-phenylprop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoylamino]hexanoic acid —— C22H26N2O4S2
6-[3-[(5E)-5-[(E)-2-methyl-3-phenylprop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoylamino]hexanoic acid
—— 6-ethyl-7-hydroxy-3-(1-methylbenzimidazol-2-yl)-2-propan-2-yl-8-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]chromen-4-one —— C33H41N3O3
6-ethyl-7-hydroxy-3-(1-methylbenzimidazol-2-yl)-2-propan-2-yl-8-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]chromen-4-one
—— 6-[ethyl-[(Z)-2-methylpropylideneamino]amino]-3-methyl-1H-pyrimidine-2,4-dione —— C11H18N4O2
6-[ethyl-[(Z)-2-methylpropylideneamino]amino]-3-methyl-1H-pyrimidine-2,4-dione
—— 6-amino-5-[2-[(4Z)-1-[4-(difluoromethoxy)phenyl]-4-(furan-2-ylmethylidene)-5-oxoimidazol-2-yl]sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione —— C23H19F2N5O6S
6-amino-5-[2-[(4Z)-1-[4-(difluoromethoxy)phenyl]-4-(furan-2-ylmethylidene)-5-oxoimidazol-2-yl]sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6E)-6-({1-[2-(2,6-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H27N5O2S
(6E)-6-({1-[2-(2,6-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-chlorophenyl)-N-[1-(4-chlorophenyl)ethylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine —— C19H14Cl2F3N4+
6-(4-chlorophenyl)-N-[1-(4-chlorophenyl)ethylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine
—— 6-[[(1S,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]hexanoic acid —— C14H21NO3
6-[[(1S,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]hexanoic acid
—— (6E)-2-butyl-5-imino-6-[[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H25N5O2S
(6E)-2-butyl-5-imino-6-[[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-bromo-4-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinazoline —— C18H22BrN3
6-bromo-4-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinazoline
—— (6R)-6-nitro-2-phenyl-6H-indole-3,5-dione —— C14H8N2O4
(6R)-6-nitro-2-phenyl-6H-indole-3,5-dione
—— 6-bromo-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinazoline —— C18H22BrN3
6-bromo-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinazoline
—— 6-imino-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C29H27N5O2
6-imino-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6E)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H24FN5OS
(6E)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[1-(4-ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C22H22N4OS
(6Z)-6-[[1-(4-ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-8-methyl-6-(2-methylhexylidene)-1,2,3,5,7,8a-hexahydroindolizine-7,8-diol —— C16H29NO2
(6Z)-8-methyl-6-(2-methylhexylidene)-1,2,3,5,7,8a-hexahydroindolizine-7,8-diol
—— (6Z)-6-[[3-bromo-4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O4S
(6Z)-6-[[3-bromo-4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[1-(4-ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N6O2S
(6Z)-6-[[1-(4-ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-6-nitro-2-phenyl-6H-indole-3,5-dione —— C14H8N2O4
(6S)-6-nitro-2-phenyl-6H-indole-3,5-dione
—— (6E)-3-(4-chlorophenyl)-6-[[4-(diethylamino)phenyl]methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C21H19ClN4OS
(6E)-3-(4-chlorophenyl)-6-[[4-(diethylamino)phenyl]methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-imino-11-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C29H27N5O2
6-imino-11-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-(2-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6Z)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-chloro-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29ClN4O4S
(6Z)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-chloro-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-imino-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H25N5O2
6-imino-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-imino-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-7-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C22H25N5O4
6-imino-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-7-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6Z)-6-[[3-bromo-4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H31BrN4O4S
(6Z)-6-[[3-bromo-4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[5-bromo-2-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H27BrN4O3S
(6Z)-6-[[5-bromo-2-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H28FN5OS
(6E)-6-{[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H31BrN4O4S
(6Z)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-butyl-5-imino-6-[[4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O3S
(6E)-2-butyl-5-imino-6-[[4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O4S
(6Z)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-imino-11-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H25N5O2
6-imino-11-methyl-2-oxo-N-[(1R)-1-phenylethyl]-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6E)-6-[(4-chloroanilino)methylidene]-4-[(3E)-3-[(4-chloroanilino)methylidene]-4-oxocyclohexa-1,5-dien-1-yl]sulfonylcyclohexa-2,4-dien-1-one —— C26H18Cl2N2O4S
(6E)-6-[(4-chloroanilino)methylidene]-4-[(3E)-3-[(4-chloroanilino)methylidene]-4-oxocyclohexa-1,5-dien-1-yl]sulfonylcyclohexa-2,4-dien-1-one
—— (6E)-6-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H30N4O3S
(6E)-6-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-5-[(2E)-2-(1-phenylpropylidene)hydrazinyl]-1,2,4-triazin-3(2H)-one —— C13H15N5O
6-methyl-5-[(2E)-2-(1-phenylpropylidene)hydrazinyl]-1,2,4-triazin-3(2H)-one
—— 6-imino-7-(2-methoxyethyl)-13-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C21H25N5O4
6-imino-7-(2-methoxyethyl)-13-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6E)-6-[[4-[2-(4-cyclohexylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H30N4O3S
(6E)-6-[[4-[2-(4-cyclohexylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(4-chlorobenzyl)-1H-indol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H24ClN5OS
(6E)-6-{[1-(4-chlorobenzyl)-1H-indol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-imino-7-(2-methoxyethyl)-11-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C21H25N5O4
6-imino-7-(2-methoxyethyl)-11-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-imino-7-(3-methoxypropyl)-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C25H27N5O3
6-imino-7-(3-methoxypropyl)-11-methyl-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-imino-7-(3-methoxypropyl)-13-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C22H27N5O4
6-imino-7-(3-methoxypropyl)-13-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-amino-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]hexanamide —— C15H28N2O
6-amino-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]hexanamide
—— (6E)-6-[(4-ethoxyphenyl)methylidene]-3-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C22H21N3O5S
(6E)-6-[(4-ethoxyphenyl)methylidene]-3-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-amino-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]hexanamide —— C15H28N2O
6-amino-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]hexanamide