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—— (6S)-1-(2-cyclobutylacetyl)-4-(furan-2-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C17H24N2O4
(6S)-1-(2-cyclobutylacetyl)-4-(furan-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— 6-[[(2S)-2-pyridin-3-ylmorpholin-4-yl]methyl]pyridine-2-carboxylic acid —— C16H17N3O3
6-[[(2S)-2-pyridin-3-ylmorpholin-4-yl]methyl]pyridine-2-carboxylic acid
—— 6-chloro-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-indole-2-carboxamide —— C17H15ClN2O2
6-chloro-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-indole-2-carboxamide
—— (6R)-1-[[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl]-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-6-ol —— C16H24N6O3
(6R)-1-[[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl]-4-(2H-triazol-4-ylmethyl)-1,4-diazepan-6-ol
—— 6-[[(2R)-2-pyridin-3-ylmorpholin-4-yl]methyl]pyridine-2-carboxylic acid —— C16H17N3O3
6-[[(2R)-2-pyridin-3-ylmorpholin-4-yl]methyl]pyridine-2-carboxylic acid
—— 6-methyl-1-[3-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-3-oxopropyl]pyridin-2-one —— C18H27N3O2
6-methyl-1-[3-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-3-oxopropyl]pyridin-2-one
—— (6S)-1-[[3-(furan-2-yl)phenyl]methyl]-1,4-diazepane-6-carboxylic acid —— C17H20N2O3
(6S)-1-[[3-(furan-2-yl)phenyl]methyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-5-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H20N6O2
(6R)-5-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— [(6S)-6-hydroxy-4-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]-[2-(methylamino)pyridin-3-yl]methanone —— C16H23N7O2
[(6S)-6-hydroxy-4-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]-[2-(methylamino)pyridin-3-yl]methanone
—— [(6S)-6-hydroxy-4-(3-methoxypropyl)-1,4-diazepan-1-yl]-(1,2,3,4-tetrahydroquinolin-8-yl)methanone —— C19H29N3O3
[(6S)-6-hydroxy-4-(3-methoxypropyl)-1,4-diazepan-1-yl]-(1,2,3,4-tetrahydroquinolin-8-yl)methanone
—— [(6R)-6-hydroxy-4-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]-[2-(methylamino)pyridin-3-yl]methanone —— C16H23N7O2
[(6R)-6-hydroxy-4-[(4-methyl-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]-[2-(methylamino)pyridin-3-yl]methanone
—— 6-methyl-1-[3-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-3-oxopropyl]pyridin-2-one —— C18H27N3O2
6-methyl-1-[3-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-3-oxopropyl]pyridin-2-one
—— (6R)-1-[[3-(furan-2-yl)phenyl]methyl]-1,4-diazepane-6-carboxylic acid —— C17H20N2O3
(6R)-1-[[3-(furan-2-yl)phenyl]methyl]-1,4-diazepane-6-carboxylic acid
—— 6-[2-[2-(4-bromophenyl)-2-oxoethyl]-5-[(Z)-2-(4-methoxyphenyl)ethenyl]-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C25H20BrN3O3
6-[2-[2-(4-bromophenyl)-2-oxoethyl]-5-[(Z)-2-(4-methoxyphenyl)ethenyl]-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(Z)-2-(2-methoxyphenyl)ethenyl]-3-(2-methylfuran-3-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C17H14N4O2S
6-[(Z)-2-(2-methoxyphenyl)ethenyl]-3-(2-methylfuran-3-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-(dimethylamino)-N-[(2S,6R)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide —— C16H25N3O
6-(dimethylamino)-N-[(2S,6R)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(S)-(4-fluorophenyl)-phenylmethyl]pyridine-3-carboxamide —— C21H20FN3O
6-(dimethylamino)-N-[(S)-(4-fluorophenyl)-phenylmethyl]pyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide —— C15H19N3O2
6-(dimethylamino)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(2R,6R)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide —— C16H25N3O
6-(dimethylamino)-N-[(2R,6R)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(R)-(4-fluorophenyl)-phenylmethyl]pyridine-3-carboxamide —— C21H20FN3O
6-(dimethylamino)-N-[(R)-(4-fluorophenyl)-phenylmethyl]pyridine-3-carboxamide
—— 6-ethyl-3-[(E)-pyridin-3-ylmethylideneamino]thieno[2,3-d]pyrimidin-4-one —— C14H12N4OS
6-ethyl-3-[(E)-pyridin-3-ylmethylideneamino]thieno[2,3-d]pyrimidin-4-one
—— 6-(dimethylamino)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide —— C15H19N3O2
6-(dimethylamino)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(2S,6S)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide —— C16H25N3O
6-(dimethylamino)-N-[(2S,6S)-2,6-dimethylcyclohexyl]pyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(R)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide —— C20H20N4O
6-(dimethylamino)-N-[(R)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide
—— 6-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H14FN3O3S
6-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H14FN3O3S
6-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[(6R)-6-hydroxy-4-(1H-indol-2-ylmethyl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile —— C20H21N5O
6-[(6R)-6-hydroxy-4-(1H-indol-2-ylmethyl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile
—— [(6R)-2-oxa-8-azaspiro[5.5]undecan-8-yl]-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methanone —— C19H20F3N3O3
[(6R)-2-oxa-8-azaspiro[5.5]undecan-8-yl]-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methanone
—— [(6S)-2-oxa-8-azaspiro[5.5]undecan-8-yl]-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methanone —— C19H20F3N3O3
[(6S)-2-oxa-8-azaspiro[5.5]undecan-8-yl]-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methanone
—— (6S)-1-[2-(benzimidazol-1-yl)ethyl]-4-(cyclopropylmethyl)-1,4-diazepane-6-carboxylic acid —— C19H26N4O2
(6S)-1-[2-(benzimidazol-1-yl)ethyl]-4-(cyclopropylmethyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(3,3,3-trifluoropropyl)-1,4-diazepan-6-ol —— C17H23F3N2O
(6S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(3,3,3-trifluoropropyl)-1,4-diazepan-6-ol
—— 6-[2-[(3R)-3-(5-ethylfuran-2-yl)morpholin-4-yl]ethoxy]-3,4-dihydro-1H-quinolin-2-one —— C21H26N2O4
6-[2-[(3R)-3-(5-ethylfuran-2-yl)morpholin-4-yl]ethoxy]-3,4-dihydro-1H-quinolin-2-one
—— 6-cyclopropyl-3-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H28N4O4
6-cyclopropyl-3-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C21H31N5O3
6-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide
—— 6-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C21H31N5O3
6-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide
—— 6-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C21H31N5O3
6-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H28N4O4
6-cyclopropyl-3-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H28N4O4
6-cyclopropyl-3-methyl-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-3-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H28N4O4
6-cyclopropyl-3-methyl-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6-chloropyridin-3-yl)methyl (2S)-2-(3-fluorophenoxy)propanoate —— C15H13ClFNO3
(6-chloropyridin-3-yl)methyl (2S)-2-(3-fluorophenoxy)propanoate
—— (6-chloropyridin-3-yl)methyl (2R)-2-(3-fluorophenoxy)propanoate —— C15H13ClFNO3
(6-chloropyridin-3-yl)methyl (2R)-2-(3-fluorophenoxy)propanoate
—— 6-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-N-(pyridin-3-ylmethyl)-1H-pyridine-3-carboxamide —— C18H21N3O3
6-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-N-(pyridin-3-ylmethyl)-1H-pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C15H23N3O2
6-(azepan-1-yl)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C15H23N3O2
6-(azepan-1-yl)-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]pyridine-3-carboxamide —— C21H24F2N4O2
6-(azepan-1-yl)-N-[(1S)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]pyridine-3-carboxamide —— C21H24F2N4O2
6-(azepan-1-yl)-N-[(1R)-1-(3,4-difluorophenyl)-2-(methylamino)-2-oxoethyl]pyridine-3-carboxamide
—— 6-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-N-(pyridin-3-ylmethyl)-1H-pyridine-3-carboxamide —— C18H21N3O3
6-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-N-(pyridin-3-ylmethyl)-1H-pyridine-3-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2R)-1-hydroxypropan-2-yl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C19H24N4O3
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-1-hydroxypropan-2-yl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide
—— 6-methyl-3-[(2E)-2-[(2,4,6-trimethylphenyl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C14H17N5O
6-methyl-3-[(2E)-2-[(2,4,6-trimethylphenyl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-hydroxypropan-2-yl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C19H24N4O3
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-hydroxypropan-2-yl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide