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—— [(6S)-6-hydroxy-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-1-yl]-(1,2-oxazol-3-yl)methanone —— C16H18N6O3
[(6S)-6-hydroxy-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-1-yl]-(1,2-oxazol-3-yl)methanone
—— (6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid —— C14H20N4O4
(6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C13H18N6O3
(6S)-1-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-[(6R)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C16H21N5O4
6-[(6R)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— (6R)-1-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C13H18N6O3
(6R)-1-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-6-methyl-N-(4-methyl-1,3-thiazol-2-yl)spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide —— C21H25N3O3S
(6R)-6-methyl-N-(4-methyl-1,3-thiazol-2-yl)spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide
—— (6S)-N-(2-benzylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide —— C19H22N2O3
(6S)-N-(2-benzylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
—— (6S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid —— C14H20N4O4
(6S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
—— (6R)-1-(1H-imidazol-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid —— C15H19N5O3
(6R)-1-(1H-imidazol-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
—— 6-methyl-1-[3-[(5S)-1-oxa-9-azaspiro[4.6]undecan-9-yl]-3-oxopropyl]pyridin-2-one —— C18H26N2O3
6-methyl-1-[3-[(5S)-1-oxa-9-azaspiro[4.6]undecan-9-yl]-3-oxopropyl]pyridin-2-one
—— 6-fluoro-N-[(2S)-1-hydroxybutan-2-yl]-4-oxo-N-(pyridin-4-ylmethyl)-1H-quinoline-3-carboxamide —— C20H20FN3O3
6-fluoro-N-[(2S)-1-hydroxybutan-2-yl]-4-oxo-N-(pyridin-4-ylmethyl)-1H-quinoline-3-carboxamide
—— 6-fluoro-N-[(2R)-1-hydroxybutan-2-yl]-4-oxo-N-(pyridin-4-ylmethyl)-1H-quinoline-3-carboxamide —— C20H20FN3O3
6-fluoro-N-[(2R)-1-hydroxybutan-2-yl]-4-oxo-N-(pyridin-4-ylmethyl)-1H-quinoline-3-carboxamide
—— (6R)-1-[2-(benzenesulfonyl)ethyl]-4-methyl-1,4-diazepan-6-ol —— C14H22N2O3S
(6R)-1-[2-(benzenesulfonyl)ethyl]-4-methyl-1,4-diazepan-6-ol
—— (6S)-1-(1H-imidazol-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid —— C15H19N5O3
(6S)-1-(1H-imidazol-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
—— (6R)-5-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H19N3O3
(6R)-5-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-5-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H19N3O3
(6S)-5-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-methyl-4-oxo-N-[2-[(3S)-3-phenylpiperidin-1-yl]ethyl]pyrido[1,2-a]pyrimidine-3-carboxamide —— C23H26N4O2
6-methyl-4-oxo-N-[2-[(3S)-3-phenylpiperidin-1-yl]ethyl]pyrido[1,2-a]pyrimidine-3-carboxamide
—— (6R)-5-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H21N5O2
(6R)-5-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-5-[[4-(pyridin-2-ylmethoxy)phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C20H20N4O3
(6S)-5-[[4-(pyridin-2-ylmethoxy)phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-5-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H21N5O2
(6S)-5-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-5-[(2,3-dichloro-6-fluorophenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C14H12Cl2FN3O2
(6S)-5-[(2,3-dichloro-6-fluorophenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6R)-5-[[4-(pyridin-2-ylmethoxy)phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C20H20N4O3
(6R)-5-[[4-(pyridin-2-ylmethoxy)phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-(4-Cyclohexylthiosemicarbazono)methyl-2,3-dimethoxy-benzoic acid —— C17H23N3O4S
6-(4-Cyclohexylthiosemicarbazono)methyl-2,3-dimethoxy-benzoic acid
—— (6R)-5-[(2,3-dichloro-6-fluorophenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C14H12Cl2FN3O2
(6R)-5-[(2,3-dichloro-6-fluorophenyl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[3-[(1S)-1-pyrrolidin-1-ylethyl]phenyl]pyrimidin-4-amine —— C16H20N4
6-[3-[(1S)-1-pyrrolidin-1-ylethyl]phenyl]pyrimidin-4-amine
—— 6-[3-[(1R)-1-pyrrolidin-1-ylethyl]phenyl]pyrimidin-4-amine —— C16H20N4
6-[3-[(1R)-1-pyrrolidin-1-ylethyl]phenyl]pyrimidin-4-amine
—— 6-[(5S)-3-(2-hydroxyethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carboxamide —— C18H28N4O3
6-[(5S)-3-(2-hydroxyethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carboxamide
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2,6,8-trimethylquinolin-4-yl)methanone —— C18H22N2O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2,6,8-trimethylquinolin-4-yl)methanone
—— 6-[(5R)-3-(2-hydroxyethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carboxamide —— C18H28N4O3
6-[(5R)-3-(2-hydroxyethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carboxamide
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2,6,8-trimethylquinolin-4-yl)methanone —— C18H22N2O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2,6,8-trimethylquinolin-4-yl)methanone
—— [(6R)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-morpholin-4-ylmethanone —— C16H22N6O3
[(6R)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-morpholin-4-ylmethanone
—— 6-fluoro-N-[2-[(3R)-3-(hydroxymethyl)piperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide —— C18H22FN3O3
6-fluoro-N-[2-[(3R)-3-(hydroxymethyl)piperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide
—— [(6S)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-morpholin-4-ylmethanone —— C16H22N6O3
[(6S)-6-hydroxy-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl]-morpholin-4-ylmethanone
—— 6-fluoro-N-[2-[(3S)-3-(hydroxymethyl)piperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide —— C18H22FN3O3
6-fluoro-N-[2-[(3S)-3-(hydroxymethyl)piperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide
—— 6-(3-bromophenoxy)-N-cyclopropyl-N-[(3S)-2,5-dioxopyrrolidin-3-yl]pyridine-3-carboxamide —— C19H16BrN3O4
6-(3-bromophenoxy)-N-cyclopropyl-N-[(3S)-2,5-dioxopyrrolidin-3-yl]pyridine-3-carboxamide
—— (6S)-1-[(1-benzylimidazol-2-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C17H22N4O2
(6S)-1-[(1-benzylimidazol-2-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-1-[(1-benzylimidazol-2-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C17H22N4O2
(6R)-1-[(1-benzylimidazol-2-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-(4-fluorophenyl)-N-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]thieno[3,2-d]pyrimidin-4-amine —— C19H17FN6S
6-(4-fluorophenyl)-N-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]thieno[3,2-d]pyrimidin-4-amine
—— 6-chloro-N-[(E)-1-(7-methoxy-1-benzofuran-2-yl)ethylideneamino]pyridazin-3-amine —— C15H13ClN4O2
6-chloro-N-[(E)-1-(7-methoxy-1-benzofuran-2-yl)ethylideneamino]pyridazin-3-amine
—— (6Z)-6-[(4-hydroxy-3-nitrophenyl)methylidene]-2-phenyl-4,5-dihydro-1,3-benzothiazol-7-one —— C20H14N2O4S
(6Z)-6-[(4-hydroxy-3-nitrophenyl)methylidene]-2-phenyl-4,5-dihydro-1,3-benzothiazol-7-one
—— 6-[2-[(2E)-2-[(4-methoxyphenyl)methylidene]hydrazinyl]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one —— C19H16N4O3S
6-[2-[(2E)-2-[(4-methoxyphenyl)methylidene]hydrazinyl]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one
—— (6R)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-6-ol —— C13H19N5O2S
(6R)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-6-ol
—— [(6R)-4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C16H24N2O4
[(6R)-4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— [(6S)-4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C16H24N2O4
[(6S)-4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— 6-methyl-2-[(2E)-2-(3,4,5-trimethoxybenzylidene)hydrazinyl]pyrimidin-4(3H)-one —— C15H18N4O4
6-methyl-2-[(2E)-2-(3,4,5-trimethoxybenzylidene)hydrazinyl]pyrimidin-4(3H)-one
—— 6-bromo-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide —— C14H10BrF2N5O
6-bromo-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
—— 6-bromo-N-[(1S)-1-(3,4-difluorophenyl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide —— C14H10BrF2N5O
6-bromo-N-[(1S)-1-(3,4-difluorophenyl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
—— 6-methyl-3-[(2E)-2-(1-pyridin-4-ylethylidene)hydrazinyl]-4H-1,2,4-triazin-5-one —— C11H12N6O
6-methyl-3-[(2E)-2-(1-pyridin-4-ylethylidene)hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-methyl-3-[(2E)-2-(1-pyridin-3-ylethylidene)hydrazinyl]-4H-1,2,4-triazin-5-one —— C11H12N6O
6-methyl-3-[(2E)-2-(1-pyridin-3-ylethylidene)hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-chloro-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide —— C16H16ClNO5
6-chloro-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide