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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-fluoro-3-[(2S)-2-(1H-imidazol-5-ylmethyl)-3-oxopiperazine-1-carbonyl]-1H-quinolin-4-one —— C18H16FN5O3
6-fluoro-3-[(2S)-2-(1H-imidazol-5-ylmethyl)-3-oxopiperazine-1-carbonyl]-1H-quinolin-4-one
—— [(6S)-4-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1,2,5-oxadiazol-3-yl)methanone —— C15H19N7O3
[(6S)-4-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1,2,5-oxadiazol-3-yl)methanone
—— [(6R)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-2-yl)methanone —— C14H18N6O2
[(6R)-4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-2-yl)methanone
—— [(6R)-4-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1,2,5-oxadiazol-3-yl)methanone —— C15H19N7O3
[(6R)-4-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1,2,5-oxadiazol-3-yl)methanone
—— (6R)-6-methyl-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide —— C25H29N5O3
(6R)-6-methyl-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide
—— (6S)-6-methyl-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide —— C25H29N5O3
(6S)-6-methyl-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide
—— (6S)-6-methyl-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide —— C25H29N5O3
(6S)-6-methyl-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide
—— 6-chloro-4-[(Z)-3-phenylprop-2-enyl]-1,4-benzoxazin-3-one —— C17H14ClNO2
6-chloro-4-[(Z)-3-phenylprop-2-enyl]-1,4-benzoxazin-3-one
—— 6-[(Z)-3-phenylprop-2-enoxy]-1,3-benzoxathiol-2-one —— C16H12O3S
6-[(Z)-3-phenylprop-2-enoxy]-1,3-benzoxathiol-2-one
—— (6R)-6-methyl-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide —— C25H29N5O3
(6R)-6-methyl-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]spiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-carboxamide
—— 6-ethoxy-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C11H16N2O3
6-ethoxy-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C11H16N2O3
6-ethoxy-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(4-bromophenoxy)-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(4-bromophenoxy)-N-[(2R)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(4-bromophenoxy)-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]pyridine-3-carboxamide —— C20H25N3O2
6-ethoxy-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(4-bromophenoxy)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]pyridine-3-carboxamide —— C20H25N3O2
6-ethoxy-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide —— C11H16N2O3
6-ethoxy-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]pyridine-3-carboxamide —— C20H16BrN5O2
6-(4-bromophenoxy)-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]pyridine-3-carboxamide
—— 6-(4-bromophenoxy)-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]pyridine-3-carboxamide —— C20H16BrN5O2
6-(4-bromophenoxy)-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(2S)-5-methylhexan-2-yl]pyridine-3-carboxamide —— C15H24N2O2
6-ethoxy-N-[(2S)-5-methylhexan-2-yl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide —— C11H16N2O3
6-ethoxy-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(2R)-5-methylhexan-2-yl]pyridine-3-carboxamide —— C15H24N2O2
6-ethoxy-N-[(2R)-5-methylhexan-2-yl]pyridine-3-carboxamide
—— 6-phenoxy-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide —— C19H18N2O2S
6-phenoxy-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide
—— 6-(3-bromophenoxy)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(3-bromophenoxy)-N-[(2S)-1-hydroxypropan-2-yl]pyridine-3-carboxamide
—— 6-(3-bromophenoxy)-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(3-bromophenoxy)-N-[(2R)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-(3-bromophenoxy)-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide —— C15H15BrN2O3
6-(3-bromophenoxy)-N-[(2S)-2-hydroxypropyl]pyridine-3-carboxamide
—— 6-phenoxy-N-[(R)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide —— C24H19N3O2
6-phenoxy-N-[(R)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide
—— 6-phenoxy-N-[(S)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide —— C24H19N3O2
6-phenoxy-N-[(S)-phenyl(pyridin-4-yl)methyl]pyridine-3-carboxamide
—— 6-methyl-4-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-3-sulfanylidene-2H-1,2,4-triazin-5-one —— C15H17N5O2S
6-methyl-4-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-3-sulfanylidene-2H-1,2,4-triazin-5-one
—— (6R)-1-pyrazin-2-yl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-6-ol —— C15H17N7O
(6R)-1-pyrazin-2-yl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,4-diazepan-6-ol
—— [(6S)-6-hydroxy-4-pyridin-4-yl-1,4-diazepan-1-yl]-(4-methylpiperazin-1-yl)methanone —— C16H25N5O2
[(6S)-6-hydroxy-4-pyridin-4-yl-1,4-diazepan-1-yl]-(4-methylpiperazin-1-yl)methanone
—— [(6S)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-[3-(tetrazol-1-yl)-1H-pyrazol-5-yl]methanone —— C15H20N8O2
[(6S)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-[3-(tetrazol-1-yl)-1H-pyrazol-5-yl]methanone
—— 6-[[methyl-[2-[(2S)-oxan-2-yl]ethyl]amino]methyl]naphthalen-2-ol —— C19H25NO2
6-[[methyl-[2-[(2S)-oxan-2-yl]ethyl]amino]methyl]naphthalen-2-ol
—— [(6R)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-[3-(tetrazol-1-yl)-1H-pyrazol-5-yl]methanone —— C15H20N8O2
[(6R)-6-hydroxy-4-pent-2-ynyl-1,4-diazepan-1-yl]-[3-(tetrazol-1-yl)-1H-pyrazol-5-yl]methanone
—— 6-[[methyl-[2-[(2R)-oxan-2-yl]ethyl]amino]methyl]naphthalen-2-ol —— C19H25NO2
6-[[methyl-[2-[(2R)-oxan-2-yl]ethyl]amino]methyl]naphthalen-2-ol
—— [(6R)-6-hydroxy-4-pyridin-4-yl-1,4-diazepan-1-yl]-(4-methylpiperazin-1-yl)methanone —— C16H25N5O2
[(6R)-6-hydroxy-4-pyridin-4-yl-1,4-diazepan-1-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-methyl-5-phenyl-2-[(Z)-2-phenylethenyl]-1H-pyrimidin-4-one —— C19H16N2O
6-methyl-5-phenyl-2-[(Z)-2-phenylethenyl]-1H-pyrimidin-4-one
—— [(6S)-4-[2-(diethylamino)ethyl]-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrazol-5-yl)methanone —— C15H27N5O2
[(6S)-4-[2-(diethylamino)ethyl]-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrazol-5-yl)methanone
—— (6S)-1-cyclopropylsulfonyl-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid —— C14H24N2O5S
(6S)-1-cyclopropylsulfonyl-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid —— C16H19FN2O3
(6S)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid
—— [(6S)-6-hydroxy-4-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone —— C17H25N5O3
[(6S)-6-hydroxy-4-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone
—— (6R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid —— C16H19FN2O3
(6R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(cyclobutylmethyl)-4-(furan-2-carbonyl)-1,4-diazepane-6-carboxylic acid —— C16H22N2O4
(6S)-1-(cyclobutylmethyl)-4-(furan-2-carbonyl)-1,4-diazepane-6-carboxylic acid
—— (6R)-1-(cyclobutylmethyl)-4-(furan-2-carbonyl)-1,4-diazepane-6-carboxylic acid —— C16H22N2O4
(6R)-1-(cyclobutylmethyl)-4-(furan-2-carbonyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-1,4-diazepan-6-ol —— C16H24N2O2
(6S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-1,4-diazepan-6-ol
—— (6R)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-1,4-diazepan-6-ol —— C16H24N2O2
(6R)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-1,4-diazepan-6-ol
—— [(6R)-6-hydroxy-4-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone —— C17H25N5O3
[(6R)-6-hydroxy-4-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone
—— (6R)-1-[3-(1,3-dihydroisoindol-2-yl)propanoyl]-1,4-diazepane-6-carboxylic acid —— C17H23N3O3
(6R)-1-[3-(1,3-dihydroisoindol-2-yl)propanoyl]-1,4-diazepane-6-carboxylic acid