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—— 6-acetamido-N-[3-[(2R,4R,6S)-4-[[[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C35H45N3O7
6-acetamido-N-[3-[(2R,4R,6S)-4-[[[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-[(3R,3aR,6aS)-4,6-dioxo-2-phenyl-5-(4-propoxyphenyl)-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]-2,3-dimethoxybenzoic acid —— C29H28N2O8
6-[(3R,3aR,6aS)-4,6-dioxo-2-phenyl-5-(4-propoxyphenyl)-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]-2,3-dimethoxybenzoic acid
—— 6-(dimethylamino)-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C23H33N3O
6-(dimethylamino)-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1R)-1-naphthalen-2-ylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C46H53N3O5
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1R)-1-naphthalen-2-ylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-butoxy-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C25H36N2O2
6-butoxy-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-acetamido-N-[3-[(2R,4R,6S)-4-[(dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C40H47N3O5
6-acetamido-N-[3-[(2R,4R,6S)-4-[(dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4R,6S)-4-(1,3-benzothiazol-2-ylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H39N3O5S2
6-acetamido-N-[[4-[(2R,4R,6S)-4-(1,3-benzothiazol-2-ylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-chloro-2,8-dimethyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C22H29ClN2O
6-chloro-2,8-dimethyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-butyl-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C25H36N2O
6-butyl-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-(diethylamino)-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C25H37N3O
6-(diethylamino)-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-imino-2-oxo-N-[(1S)-1-phenylethyl]-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C26H29N5O3
6-imino-2-oxo-N-[(1S)-1-phenylethyl]-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C36H47N3O6
6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H40Cl2N4O5
6-acetamido-N-[[3-[3-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-imino-2-oxo-N-[(1R)-1-phenylethyl]-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C26H29N5O3
6-imino-2-oxo-N-[(1R)-1-phenylethyl]-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-acetamido-N-[[3-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H51N3O7
6-acetamido-N-[[3-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H57N3O5
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-amino-5-[(S)-[5-(4-chlorophenyl)furan-2-yl]-(4-phenylpiperazin-1-yl)methyl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C29H32ClN5O3
6-amino-5-[(S)-[5-(4-chlorophenyl)furan-2-yl]-(4-phenylpiperazin-1-yl)methyl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— (6S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C23H18N4O2
(6S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— (6R)-3-(3,4-dimethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C25H22N4O2
(6R)-3-(3,4-dimethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— (6S)-3-(4-fluorophenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C23H17FN4O2
(6S)-3-(4-fluorophenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-fluoro-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C21H27FN2O
6-fluoro-2-methyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— 6-amino-5-[(R)-[5-(4-chlorophenyl)furan-2-yl]-(4-phenylpiperazin-1-yl)methyl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C29H32ClN5O3
6-amino-5-[(R)-[5-(4-chlorophenyl)furan-2-yl]-(4-phenylpiperazin-1-yl)methyl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— (6R)-3-(4-ethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C25H22N4O2
(6R)-3-(4-ethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H56N4O5
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6R)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C23H18N4O2
(6R)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— (6R)-3-(4-fluorophenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C23H17FN4O2
(6R)-3-(4-fluorophenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— (6S)-3-(3,4-dimethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C25H22N4O2
(6S)-3-(3,4-dimethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-acetamido-N-[[4-[(2R,4R,6S)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C35H45N3O5
6-acetamido-N-[[4-[(2R,4R,6S)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— (6S)-3-(4-ethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C25H22N4O2
(6S)-3-(4-ethylphenyl)-6-(4-methoxyphenyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-acetamido-N-[[2-[4-[(2R,4R,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H53N3O5
6-acetamido-N-[[2-[4-[(2R,4R,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H43N3O6S
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-[4-(4-bromophenyl)-2-[(3R)-3,5-diphenyl-3,4-dihydropyrazol-2-yl]-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one —— C31H23BrN4O
6-[4-(4-bromophenyl)-2-[(3R)-3,5-diphenyl-3,4-dihydropyrazol-2-yl]-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one
—— 6-acetamido-N-[[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H40N4O5
6-acetamido-N-[[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C29H38N6O5S
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-[4-(4-bromophenyl)-2-[(3S)-3,5-diphenyl-3,4-dihydropyrazol-2-yl]-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one —— C31H23BrN4O
6-[4-(4-bromophenyl)-2-[(3S)-3,5-diphenyl-3,4-dihydropyrazol-2-yl]-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H49N3O6
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H43N3O5S
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]hexanamide —— C28H35N5O5S
6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C46H55N5O6
6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[(dioctylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C49H73N3O5
6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[(dioctylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H44N6O5S
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6S,9R,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione —— C14H14O3
(6S,9R,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione
—— 6-acetamido-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C33H38N6O6S
6-acetamido-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H53N3O6
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6R,9S,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione —— C14H14O3
(6R,9S,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H53N3O6
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6R)-2-[[(1S,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H24N2O2S
(6R)-2-[[(1S,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S,9S,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione —— C14H14O3
(6S,9S,12S,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione
—— 6-acetamido-N-[3-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C29H34Cl2N4O5
6-acetamido-N-[3-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— (6S,9R,12R,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione —— C14H14O3
(6S,9R,12R,15R)-3-oxahexacyclo[7.6.0.01,5.05,12.06,10.011,15]pentadecane-2,4-dione