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—— (6S)-6-[3-[(4-bromophenyl)carbamoylamino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C28H26BrN5O2S
(6S)-6-[3-[(4-bromophenyl)carbamoylamino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-[2-[[5-(2-methylprop-2-enylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C16H15N3O3S3
6-[2-[[5-(2-methylprop-2-enylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— (6S)-6-[4-[(4-chlorobenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C29H27ClN4O3S
(6S)-6-[4-[(4-chlorobenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6R)-6-[4-[(4-chlorobenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C29H27ClN4O3S
(6R)-6-[4-[(4-chlorobenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-[(1S,2R,9S,10S,11S,12S,16S)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O5S2
6-[(1S,2R,9S,10S,11S,12S,16S)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6,7-Dimethyl-4-[[5-(2-methylprop-2-enylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C18H18N2O2S3
6,7-Dimethyl-4-[[5-(2-methylprop-2-enylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 6-[(1R,2S,9R,10S,11R,12R,16S)-9-(4-methoxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O6S2
6-[(1R,2S,9R,10S,11R,12R,16S)-9-(4-methoxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16S)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C23H24N2O5S3
6-[(1S,2R,9S,10S,11S,12S,16S)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O5S2
6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16R)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C23H24N2O5S3
6-[(1S,2R,9S,10S,11S,12S,16R)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25FN2O5S2
6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O5S2
6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1R,2S,9R,10S,11R,12R,16S)-9-(4-hydroxy-3-methoxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O7S2
6-[(1R,2S,9R,10S,11R,12R,16S)-9-(4-hydroxy-3-methoxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25FN2O5S2
6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25ClN2O5S2
6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25ClN2O5S2
6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25FN2O5S2
6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-fluorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H25ClN2O5S2
6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-chlorophenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C26H28N2O5S2
6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-methylphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16R)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C23H24N2O5S3
6-[(1S,2R,9S,10S,11S,12R,16R)-6,13,15-trioxo-9-thiophen-2-yl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-methyl-1,2-oxazole-5-carboxylate —— C14H12N2O7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-methyl-1,2-oxazole-5-carboxylate
—— [6-[(3-methylphenyl)methyl]thieno[2,3-b]pyrrol-5-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C25H30N2OS
[6-[(3-methylphenyl)methyl]thieno[2,3-b]pyrrol-5-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 6-[(Z)-2-phenylethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C22H22N6S
6-[(Z)-2-phenylethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6S)-6-[3-[(4-butylbenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C33H36N4O3S
(6S)-6-[3-[(4-butylbenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6R)-6-[3-[(4-butylbenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C33H36N4O3S
(6R)-6-[3-[(4-butylbenzoyl)amino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-[(Z)-2-(2-methoxyphenyl)ethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C23H24N6OS
6-[(Z)-2-(2-methoxyphenyl)ethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C23H24N6OS
6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-[(4-phenylpiperazin-1-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6S)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2S)-2-(2-fluorophenoxy)butanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H29FN2O5S2
(6S)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2S)-2-(2-fluorophenoxy)butanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-6-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2R)-2-(4-fluorophenoxy)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H33FN2O5S2
(6S)-6-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2R)-2-(4-fluorophenoxy)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Chloro-4-[(4-ethoxyanilino)methyl]-7-methylchromen-2-one —— C19H18ClNO3
6-Chloro-4-[(4-ethoxyanilino)methyl]-7-methylchromen-2-one
—— (6S)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2R)-2-(2-fluorophenoxy)butanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H29FN2O5S2
(6S)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[[(2R)-2-(2-fluorophenoxy)butanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate —— C22H22N2O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]propanoate —— C23H23N3O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]propanoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2R)-2-(4-fluorophenoxy)propanoate —— C19H17FN2O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2R)-2-(4-fluorophenoxy)propanoate
—— 6-Methyl-2-[(4-pentyl-1,2,4-triazol-3-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C17H21N5OS
6-Methyl-2-[(4-pentyl-1,2,4-triazol-3-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 6-Methyl-2-[(10-methyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C20H18N4OS2
6-Methyl-2-[(10-methyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate —— C20H21N3O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(1,3-benzothiazol-2-yl)butanoate —— C21H19N3O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(1,3-benzothiazol-2-yl)butanoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-ethoxybenzoyl)amino]acetate —— C21H21N3O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-ethoxybenzoyl)amino]acetate
—— 6,7-dimethoxy-2-(4-methyl-3-nitrophenyl)sulfonyl-3,4-dihydro-1H-isoquinoline —— C18H20N2O6S
6,7-dimethoxy-2-(4-methyl-3-nitrophenyl)sulfonyl-3,4-dihydro-1H-isoquinoline
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(1,3-benzodioxole-5-carbonylamino)acetate —— C20H17N3O6
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(1,3-benzodioxole-5-carbonylamino)acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-chlorobenzoyl)amino]acetate —— C19H16ClN3O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-chlorobenzoyl)amino]acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate —— C19H16FN3O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate
—— 6-[[Methyl(naphthalen-2-yl)amino]methyl]-1,3,5-triazine-2,4-diamine —— C15H16N6
6-[[Methyl(naphthalen-2-yl)amino]methyl]-1,3,5-triazine-2,4-diamine
—— 6-methyl-N-naphthalen-2-yl-1-(2-nitrophenyl)-4-oxopyridazine-3-carboxamide —— C22H16N4O4
6-methyl-N-naphthalen-2-yl-1-(2-nitrophenyl)-4-oxopyridazine-3-carboxamide
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-(4-chlorophenyl)sulfanylpropanoate —— C19H17ClN2O3S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-(4-chlorophenyl)sulfanylpropanoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C18H19N3O4S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 6-chloro-2-[(2S)-2-hydroxy-3-morpholin-4-ium-4-ylpropyl]sulfanyl-3-prop-2-enylquinazolin-4-one —— C18H23ClN3O3S+
6-chloro-2-[(2S)-2-hydroxy-3-morpholin-4-ium-4-ylpropyl]sulfanyl-3-prop-2-enylquinazolin-4-one
—— 6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-pyridin-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C17H13N5OS
6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-pyridin-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-Ethyl-3-(3-methoxyphenyl)-5-methyl-2-(2-methylsulfanylethylsulfanyl)thieno[2,3-d]pyrimidin-4-one —— C19H22N2O2S3
6-Ethyl-3-(3-methoxyphenyl)-5-methyl-2-(2-methylsulfanylethylsulfanyl)thieno[2,3-d]pyrimidin-4-one