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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(3S)-3-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C17H24N6O2
5-[(3S)-3-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 6-cyclopropyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine —— C15H24N4O2S
6-cyclopropyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine
—— 2-(dimethylamino)-N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N,4-dimethylpyrimidine-5-carboxamide —— C17H23N5O2
2-(dimethylamino)-N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N,4-dimethylpyrimidine-5-carboxamide
—— (E)-N-[[(2R)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C16H21N3O2S
(E)-N-[[(2R)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— (E)-N-[[(2S)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3S)-thiolan-3-yl]prop-2-enamide —— C16H21N3O2S
(E)-N-[[(2S)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3S)-thiolan-3-yl]prop-2-enamide
—— [(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2-morpholin-4-ylpyrimidin-5-yl)methanone —— C18H24N6O2
[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2-morpholin-4-ylpyrimidin-5-yl)methanone
—— N-methyl-N-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C22H23N5O
N-methyl-N-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— [(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2-morpholin-4-ylpyrimidin-5-yl)methanone —— C18H24N6O2
[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2-morpholin-4-ylpyrimidin-5-yl)methanone
—— (E)-N-[[(2S)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C16H21N3O2S
(E)-N-[[(2S)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— 2-methyl-5-methylsulfonyl-N-[(1S)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine —— C17H20N6O2S
2-methyl-5-methylsulfonyl-N-[(1S)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
—— (5S)-5-[[6-(methoxymethyl)pyrimidin-4-yl]amino]-1-methylpiperidin-2-one —— C12H18N4O2
(5S)-5-[[6-(methoxymethyl)pyrimidin-4-yl]amino]-1-methylpiperidin-2-one
—— (E)-N-[[(2R)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3S)-thiolan-3-yl]prop-2-enamide —— C16H21N3O2S
(E)-N-[[(2R)-oxolan-2-yl]methyl]-3-pyrazin-2-yl-N-[(3S)-thiolan-3-yl]prop-2-enamide
—— 2-methoxyethyl (4S)-6-methyl-2-oxo-4-(2,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N2O7
2-methoxyethyl (4S)-6-methyl-2-oxo-4-(2,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)-3-[(3R)-1-methylpiperidin-3-yl]propanamide —— C17H26N4O
N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)-3-[(3R)-1-methylpiperidin-3-yl]propanamide
—— 5-(Ethyliminomethyl)-1,3-dimethyl-1,3-diazinane-2,4,6-trione —— C9H13N3O3
5-(Ethyliminomethyl)-1,3-dimethyl-1,3-diazinane-2,4,6-trione
—— (5R)-5-[[6-(methoxymethyl)pyrimidin-4-yl]amino]-1-methylpiperidin-2-one —— C12H18N4O2
(5R)-5-[[6-(methoxymethyl)pyrimidin-4-yl]amino]-1-methylpiperidin-2-one
—— 3,6-dimethyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine —— C20H22N6O
3,6-dimethyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
—— 2-ethyl-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidine-5-carboxamide —— C18H23N3O4
2-ethyl-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidine-5-carboxamide
—— 5-[1-[(1S)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]triazol-4-yl]pyrimidine —— C17H16N8
5-[1-[(1S)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]triazol-4-yl]pyrimidine
—— N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)-3-[(3S)-1-methylpiperidin-3-yl]propanamide —— C17H26N4O
N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)-3-[(3S)-1-methylpiperidin-3-yl]propanamide
—— 3,6-dimethyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine —— C20H22N6O
3,6-dimethyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
—— 2-anilino-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-5-carboxamide —— C14H14N8O
2-anilino-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-5-carboxamide
—— 5-ethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-2-amine —— C17H23N5O
5-ethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-2-amine
—— 2-ethyl-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidine-5-carboxamide —— C18H23N3O4
2-ethyl-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidine-5-carboxamide
—— 5-[1-[(1R)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]triazol-4-yl]pyrimidine —— C17H16N8
5-[1-[(1R)-1-phenyl-3-(1,2,4-triazol-1-yl)propyl]triazol-4-yl]pyrimidine
—— 5-ethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-2-amine —— C17H23N5O
5-ethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-2-amine
—— N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C17H18N6O2
N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C18H19N5OS
N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— 2-[2-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]-N,N-dimethylethanamine —— C17H26N6O
2-[2-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]-N,N-dimethylethanamine
—— 5-ethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine —— C17H23N5O
5-ethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine
—— N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C18H19N5OS
N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— 5-ethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine —— C17H23N5O
5-ethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine
—— 5-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C21H19N5
5-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— [4-[(1S)-1-(dimethylamino)ethyl]piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone —— C20H27N5O
[4-[(1S)-1-(dimethylamino)ethyl]piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone
—— 2-[2-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]-N,N-dimethylethanamine —— C17H26N6O
2-[2-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]-N,N-dimethylethanamine
—— [4-[(1R)-1-(dimethylamino)ethyl]piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone —— C20H27N5O
[4-[(1R)-1-(dimethylamino)ethyl]piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone
—— pyridin-3-yl-[(3S)-1-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperidin-3-yl]methanone —— C21H19N5O2
pyridin-3-yl-[(3S)-1-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperidin-3-yl]methanone
—— (3R)-5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C23H23N5O2
(3R)-5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— (2-cyclopropyl-4-methylpyrimidin-5-yl)-[(3R)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone —— C20H27N5O
(2-cyclopropyl-4-methylpyrimidin-5-yl)-[(3R)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone
—— 3-[2-amino-4-methyl-6-[[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]pyrimidin-5-yl]propanoic acid —— C13H19N7O2
3-[2-amino-4-methyl-6-[[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]pyrimidin-5-yl]propanoic acid
—— 2-methoxyethyl (4S)-4-(2,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H16Cl2N2O4
2-methoxyethyl (4S)-4-(2,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (3S)-5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C23H23N5O2
(3S)-5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— N-[[(3R)-1-(2-methylphenyl)pyrrolidin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C22H23N5O
N-[[(3R)-1-(2-methylphenyl)pyrrolidin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— N-[[(3S)-1-(2-methylphenyl)pyrrolidin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C22H23N5O
N-[[(3S)-1-(2-methylphenyl)pyrrolidin-3-yl]methyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— 3-[2-amino-4-methyl-6-[[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]pyrimidin-5-yl]propanoic acid —— C13H19N7O2
3-[2-amino-4-methyl-6-[[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]pyrimidin-5-yl]propanoic acid
—— pyridin-3-yl-[(3R)-1-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperidin-3-yl]methanone —— C21H19N5O2
pyridin-3-yl-[(3R)-1-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperidin-3-yl]methanone
—— (2-cyclopropyl-4-methylpyrimidin-5-yl)-[(3S)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone —— C20H27N5O
(2-cyclopropyl-4-methylpyrimidin-5-yl)-[(3S)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone
—— (6S)-6-[(5-ethylpyrimidin-2-yl)amino]-2-methylheptan-2-ol —— C14H25N3O
(6S)-6-[(5-ethylpyrimidin-2-yl)amino]-2-methylheptan-2-ol
—— (6R)-6-[(5-ethylpyrimidin-2-yl)amino]-2-methylheptan-2-ol —— C14H25N3O
(6R)-6-[(5-ethylpyrimidin-2-yl)amino]-2-methylheptan-2-ol
—— (3R)-3-methyl-1-[(3-methylphenyl)methyl]-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one —— C23H23N5O2
(3R)-3-methyl-1-[(3-methylphenyl)methyl]-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one