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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-1-(2-amino-4-methylpyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid —— C15H22N4O4
(3R)-1-(2-amino-4-methylpyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
—— 3-phenylpropyl (6S)-3,4-dimethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C20H22N2O3S
3-phenylpropyl (6S)-3,4-dimethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— N-[(5R)-2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-pyridin-2-ylpyrimidine-5-carboxamide —— C20H21N7O
N-[(5R)-2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-pyridin-2-ylpyrimidine-5-carboxamide
—— 2-cyclopropyl-5-[(2R)-2-(3-fluorophenyl)azepane-1-carbonyl]-1H-pyrimidin-6-one —— C20H22FN3O2
2-cyclopropyl-5-[(2R)-2-(3-fluorophenyl)azepane-1-carbonyl]-1H-pyrimidin-6-one
—— 2-cyclopropyl-5-[(2S)-2-(3-fluorophenyl)azepane-1-carbonyl]-1H-pyrimidin-6-one —— C20H22FN3O2
2-cyclopropyl-5-[(2S)-2-(3-fluorophenyl)azepane-1-carbonyl]-1H-pyrimidin-6-one
—— N-[(2R)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyrimidin-2-amine —— C15H19N5O
N-[(2R)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyrimidin-2-amine
—— 3-[(3R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl]-N,N-dimethylpropanamide —— C18H29N5O2
3-[(3R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl]-N,N-dimethylpropanamide
—— 2,5,6-trimethyl-N-[4-[(2R)-oxolan-2-yl]butyl]pyrimidin-4-amine —— C15H25N3O
2,5,6-trimethyl-N-[4-[(2R)-oxolan-2-yl]butyl]pyrimidin-4-amine
—— 2,5,6-trimethyl-N-[4-[(2S)-oxolan-2-yl]butyl]pyrimidin-4-amine —— C15H25N3O
2,5,6-trimethyl-N-[4-[(2S)-oxolan-2-yl]butyl]pyrimidin-4-amine
—— N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine —— C12H16N4O
N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine
—— (3R)-3-(cyclopropylmethyl)-1-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]piperidine-3-carboxylic acid —— C20H24N4O2
(3R)-3-(cyclopropylmethyl)-1-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]piperidine-3-carboxylic acid
—— 3-[(3S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl]-N,N-dimethylpropanamide —— C18H29N5O2
3-[(3S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl]-N,N-dimethylpropanamide
—— [(3R)-1-[2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl]piperidin-3-yl]methanol —— C15H27N5O
[(3R)-1-[2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl]piperidin-3-yl]methanol
—— N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine —— C12H16N4O
N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine
—— (3R)-3-[4-(2-cyclohexylpyrimidin-5-yl)triazol-1-yl]-1-methylpyrrolidin-2-one —— C17H22N6O
(3R)-3-[4-(2-cyclohexylpyrimidin-5-yl)triazol-1-yl]-1-methylpyrrolidin-2-one
—— (3S)-3-[4-(2-cyclohexylpyrimidin-5-yl)triazol-1-yl]-1-methylpyrrolidin-2-one —— C17H22N6O
(3S)-3-[4-(2-cyclohexylpyrimidin-5-yl)triazol-1-yl]-1-methylpyrrolidin-2-one
—— dimethyl (6R)-8-methyl-4-oxo-6-thiophen-2-yl-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate —— C16H14N2O5S2
dimethyl (6R)-8-methyl-4-oxo-6-thiophen-2-yl-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate
—— 6-ethoxy-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]pyrazin-2-amine —— C12H19N3O2
6-ethoxy-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]pyrazin-2-amine
—— N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine —— C12H16N4O
N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine
—— (3S)-3-(cyclopropylmethyl)-1-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]piperidine-3-carboxylic acid —— C20H24N4O2
(3S)-3-(cyclopropylmethyl)-1-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]piperidine-3-carboxylic acid
—— [(3S)-1-[2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl]piperidin-3-yl]methanol —— C15H27N5O
[(3S)-1-[2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl]piperidin-3-yl]methanol
—— 6-ethoxy-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]pyrazin-2-amine —— C12H19N3O2
6-ethoxy-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]pyrazin-2-amine
—— N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine —— C12H16N4O
N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]imidazo[1,2-b]pyridazin-6-amine
—— (2S)-N-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-pyrazol-1-ylbutanamide —— C15H21N5O2
(2S)-N-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-pyrazol-1-ylbutanamide
—— N-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-6-oxo-2-thiophen-2-yl-1H-pyrimidine-5-carboxamide —— C13H11N3O4S2
N-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-6-oxo-2-thiophen-2-yl-1H-pyrimidine-5-carboxamide
—— 6-ethoxy-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]pyrazin-2-amine —— C12H19N3O2
6-ethoxy-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]pyrazin-2-amine
—— 6-ethoxy-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyrazin-2-amine —— C12H19N3O2
6-ethoxy-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyrazin-2-amine
—— (2R)-N-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-pyrazol-1-ylbutanamide —— C15H21N5O2
(2R)-N-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-pyrazol-1-ylbutanamide
—— N-[(5S)-2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-pyridin-2-ylpyrimidine-5-carboxamide —— C20H21N7O
N-[(5S)-2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-pyridin-2-ylpyrimidine-5-carboxamide
—— N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C19H19N5O3
N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— N-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-2-(ethylamino)pyrimidine-5-carboxamide —— C12H18N4O3S
N-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-2-(ethylamino)pyrimidine-5-carboxamide
—— N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-6-oxo-2-thiophen-2-yl-1H-pyrimidine-5-carboxamide —— C13H11N3O4S2
N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-6-oxo-2-thiophen-2-yl-1H-pyrimidine-5-carboxamide
—— N-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-2-(ethylamino)pyrimidine-5-carboxamide —— C12H18N4O3S
N-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-2-(ethylamino)pyrimidine-5-carboxamide
—— N-[[(2R)-1,4-dioxan-2-yl]methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide —— C15H18N4O4S
N-[[(2R)-1,4-dioxan-2-yl]methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide
—— N-[[(2S)-1,4-dioxan-2-yl]methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide —— C15H18N4O4S
N-[[(2S)-1,4-dioxan-2-yl]methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide
—— N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C16H15N5O3
N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C19H19N5O3
N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— (2S)-2-N,2-N-dimethyl-1-N-(2,5,6-trimethylpyrimidin-4-yl)pentane-1,2-diamine —— C14H26N4
(2S)-2-N,2-N-dimethyl-1-N-(2,5,6-trimethylpyrimidin-4-yl)pentane-1,2-diamine
—— 2-methoxyethyl (6R)-3-benzyl-6-(2-chlorophenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23ClN2O4
2-methoxyethyl (6R)-3-benzyl-6-(2-chlorophenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 6-oxo-2-pyridin-2-yl-N-[(2S)-1-thiophen-3-ylpropan-2-yl]-1H-pyrimidine-5-carboxamide —— C17H16N4O2S
6-oxo-2-pyridin-2-yl-N-[(2S)-1-thiophen-3-ylpropan-2-yl]-1H-pyrimidine-5-carboxamide
—— (2R)-2-N,2-N-dimethyl-1-N-(2,5,6-trimethylpyrimidin-4-yl)pentane-1,2-diamine —— C14H26N4
(2R)-2-N,2-N-dimethyl-1-N-(2,5,6-trimethylpyrimidin-4-yl)pentane-1,2-diamine
—— 6-oxo-2-pyridin-2-yl-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1H-pyrimidine-5-carboxamide —— C17H16N4O2S
6-oxo-2-pyridin-2-yl-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1H-pyrimidine-5-carboxamide
—— N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C15H15N5O3S
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 5-[(2S)-2-(aminomethyl)piperidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one —— C18H20Cl2N4O2
5-[(2S)-2-(aminomethyl)piperidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one
—— N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide —— C18H19N5OS
N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
—— 6-[[(3R)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C14H23N3O3
6-[[(3R)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— [(3S)-3-(hydroxymethyl)-3-(3-methylbut-2-enyl)piperidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C17H26N4O2
[(3S)-3-(hydroxymethyl)-3-(3-methylbut-2-enyl)piperidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— 5,6-dimethyl-4-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidine-2,4-diamine —— C14H25N5O2S
5,6-dimethyl-4-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidine-2,4-diamine
—— N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C15H15N5O3S
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 5-[(2R)-2-butyl-4-methyl-3-oxopiperazine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C19H23N5O3
5-[(2R)-2-butyl-4-methyl-3-oxopiperazine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one