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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (1S,6R)-3-(7-phenylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C25H29N5O3
tert-butyl (1S,6R)-3-(7-phenylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— 2-[(3R)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-6-methyl-4-phenylquinazoline —— C32H28N4O2
2-[(3R)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-6-methyl-4-phenylquinazoline
—— 2-[(3R)-5-(3-methoxyphenyl)-3-(3-nitrophenyl)-3,4-dihydropyrazol-2-yl]-6-methyl-4-phenylquinazoline —— C31H25N5O3
2-[(3R)-5-(3-methoxyphenyl)-3-(3-nitrophenyl)-3,4-dihydropyrazol-2-yl]-6-methyl-4-phenylquinazoline
—— 4-bromo-2-methyl-5-[[(1S)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridazin-3-one —— C12H14BrN3OS
4-bromo-2-methyl-5-[[(1S)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridazin-3-one
—— 4-bromo-2-methyl-5-[[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridazin-3-one —— C12H14BrN3OS
4-bromo-2-methyl-5-[[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridazin-3-one
—— imidazo[1,2-a]pyrazin-8-yl-[(3R)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methanone —— C16H16N4O2S
imidazo[1,2-a]pyrazin-8-yl-[(3R)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methanone
—— 2,5,6-trimethyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]-3-oxopyridazine-4-carboxamide —— C15H19N3O2S
2,5,6-trimethyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]-3-oxopyridazine-4-carboxamide
—— imidazo[1,2-a]pyrazin-8-yl-[(3S)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methanone —— C16H16N4O2S
imidazo[1,2-a]pyrazin-8-yl-[(3S)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methanone
—— 2,5,6-trimethyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]-3-oxopyridazine-4-carboxamide —— C15H19N3O2S
2,5,6-trimethyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]-3-oxopyridazine-4-carboxamide
—— N-[(1S,2S)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine —— C15H22FN3O
N-[(1S,2S)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine
—— N-[(1R,2S)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine —— C15H22FN3O
N-[(1R,2S)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine
—— N-[(1R,2R)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine —— C15H22FN3O
N-[(1R,2R)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine
—— 6-chloro-4-N-[(1S,2S)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine —— C15H23ClN4O
6-chloro-4-N-[(1S,2S)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine
—— N-[(1S,2R)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine —— C15H22FN3O
N-[(1S,2R)-2-cyclopentyloxycyclohexyl]-5-fluoropyrimidin-2-amine
—— 6-chloro-4-N-[(1R,2R)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine —— C15H23ClN4O
6-chloro-4-N-[(1R,2R)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine
—— (2S)-1-methoxy-3-[4-[(4-methoxypyrimidin-2-yl)amino]piperidin-1-yl]propan-2-ol —— C14H24N4O3
(2S)-1-methoxy-3-[4-[(4-methoxypyrimidin-2-yl)amino]piperidin-1-yl]propan-2-ol
—— 6-chloro-4-N-[(1S,2R)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine —— C15H23ClN4O
6-chloro-4-N-[(1S,2R)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine
—— 6-chloro-4-N-[(1R,2S)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine —— C15H23ClN4O
6-chloro-4-N-[(1R,2S)-2-cyclopentyloxycyclohexyl]pyrimidine-2,4-diamine
—— methyl (6S)-6-(3-chloro-4-hydroxyphenyl)-3-(3-fluoro-4-methylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C20H18ClFN2O4
methyl (6S)-6-(3-chloro-4-hydroxyphenyl)-3-(3-fluoro-4-methylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— N-[(2R)-1-hydroxy-4,4-dimethylpentan-2-yl]-2-phenylpyrimidine-5-carboxamide —— C18H23N3O2
N-[(2R)-1-hydroxy-4,4-dimethylpentan-2-yl]-2-phenylpyrimidine-5-carboxamide
—— N-[(2S)-1-hydroxy-4,4-dimethylpentan-2-yl]-2-phenylpyrimidine-5-carboxamide —— C18H23N3O2
N-[(2S)-1-hydroxy-4,4-dimethylpentan-2-yl]-2-phenylpyrimidine-5-carboxamide
—— methyl (6R)-6-(3-chloro-4-hydroxyphenyl)-3-(3-fluoro-4-methylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C20H18ClFN2O4
methyl (6R)-6-(3-chloro-4-hydroxyphenyl)-3-(3-fluoro-4-methylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (2R)-2-phenyl-N-(1-pyrimidin-2-ylpyrazol-4-yl)propane-1-sulfonamide —— C16H17N5O2S
(2R)-2-phenyl-N-(1-pyrimidin-2-ylpyrazol-4-yl)propane-1-sulfonamide
—— (2S)-2-phenyl-N-(1-pyrimidin-2-ylpyrazol-4-yl)propane-1-sulfonamide —— C16H17N5O2S
(2S)-2-phenyl-N-(1-pyrimidin-2-ylpyrazol-4-yl)propane-1-sulfonamide
—— [(3R)-3-(3-chlorophenoxy)pyrrolidin-1-yl]-pyrazin-2-ylmethanone —— C15H14ClN3O2
[(3R)-3-(3-chlorophenoxy)pyrrolidin-1-yl]-pyrazin-2-ylmethanone
—— [(3S)-3-(3-chlorophenoxy)pyrrolidin-1-yl]-pyrazin-2-ylmethanone —— C15H14ClN3O2
[(3S)-3-(3-chlorophenoxy)pyrrolidin-1-yl]-pyrazin-2-ylmethanone
—— (2S,5R)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide —— C17H20N4O3
(2S,5R)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide
—— 2,6-dimethyl-N-[(E)-1-[(1R,2R)-2-phenylcyclopropyl]ethylideneamino]pyrimidin-4-amine —— C17H20N4
2,6-dimethyl-N-[(E)-1-[(1R,2R)-2-phenylcyclopropyl]ethylideneamino]pyrimidin-4-amine
—— N-benzyl-6-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-2-ylpyrimidin-4-amine —— C22H24N4O
N-benzyl-6-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-2-ylpyrimidin-4-amine
—— (3S)-1-cyclopropyl-3-[(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3S)-1-cyclopropyl-3-[(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one
—— (3S)-3-benzyl-4-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)morpholine —— C21H22N4O
(3S)-3-benzyl-4-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)morpholine
—— 4-methyl-6-[(3S)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]-2-pyridin-2-ylpyrimidine —— C20H25N7
4-methyl-6-[(3S)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]-2-pyridin-2-ylpyrimidine
—— 5-fluoro-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]pyrimidin-2-amine —— C13H19FN4O
5-fluoro-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]pyrimidin-2-amine
—— (4aS,8aS)-6-methyl-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-2,3,4,4a,5,7,8,8a-octahydro-1,6-naphthyridine —— C19H25N5
(4aS,8aS)-6-methyl-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-2,3,4,4a,5,7,8,8a-octahydro-1,6-naphthyridine
—— (2S,5S)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide —— C17H20N4O3
(2S,5S)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide
—— (3R)-1-[2-(4-chlorophenyl)-6-methylpyrimidine-4-carbonyl]-N-pyridin-2-ylpiperidine-3-carboxamide —— C23H22ClN5O2
(3R)-1-[2-(4-chlorophenyl)-6-methylpyrimidine-4-carbonyl]-N-pyridin-2-ylpiperidine-3-carboxamide
—— 5-fluoro-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]pyrimidin-2-amine —— C13H19FN4O
5-fluoro-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]pyrimidin-2-amine
—— 2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]-N-[(1R)-3-hydroxy-1-phenylpropyl]-N-methylacetamide —— C23H29N5O2
2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]-N-[(1R)-3-hydroxy-1-phenylpropyl]-N-methylacetamide
—— 2-cyclopropyl-6-methyl-N-[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]pyrimidin-4-amine —— C14H19N3O
2-cyclopropyl-6-methyl-N-[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]pyrimidin-4-amine
—— N-[(3R)-1-[6-(3-fluorophenyl)-4-methylpyridazin-3-yl]piperidin-3-yl]acetamide —— C18H21FN4O
N-[(3R)-1-[6-(3-fluorophenyl)-4-methylpyridazin-3-yl]piperidin-3-yl]acetamide
—— N-benzyl-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-ylpyrimidin-4-amine —— C22H24N4O
N-benzyl-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-ylpyrimidin-4-amine
—— (2R,5R)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide —— C17H20N4O3
(2R,5R)-5-[[(4-phenylmethoxypyrimidin-2-yl)amino]methyl]oxolane-2-carboxamide
—— (3S)-1-[2-(4-chlorophenyl)-6-methylpyrimidine-4-carbonyl]-N-pyridin-2-ylpiperidine-3-carboxamide —— C23H22ClN5O2
(3S)-1-[2-(4-chlorophenyl)-6-methylpyrimidine-4-carbonyl]-N-pyridin-2-ylpiperidine-3-carboxamide
—— (2S)-2-cyano-2-(4,6-dimethylpyrimidin-2-yl)-N-propan-2-ylacetamide —— C12H16N4O
(2S)-2-cyano-2-(4,6-dimethylpyrimidin-2-yl)-N-propan-2-ylacetamide
—— N-[(3S)-1-[6-(3-fluorophenyl)-4-methylpyridazin-3-yl]piperidin-3-yl]acetamide —— C18H21FN4O
N-[(3S)-1-[6-(3-fluorophenyl)-4-methylpyridazin-3-yl]piperidin-3-yl]acetamide
—— (3R)-1-cyclopropyl-3-[(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3R)-1-cyclopropyl-3-[(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one
—— (4aR,8aS)-6-methyl-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-2,3,4,4a,5,7,8,8a-octahydro-1,6-naphthyridine —— C19H25N5
(4aR,8aS)-6-methyl-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-2,3,4,4a,5,7,8,8a-octahydro-1,6-naphthyridine
—— N-[(2S)-2-(4-methoxyphenyl)-2-morpholin-4-ylethyl]-6-methylpyrimidine-4-carboxamide —— C19H24N4O3
N-[(2S)-2-(4-methoxyphenyl)-2-morpholin-4-ylethyl]-6-methylpyrimidine-4-carboxamide
—— N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]-4-phenylmethoxypyrimidin-2-amine —— C17H19N5O
N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]-4-phenylmethoxypyrimidin-2-amine
—— 2,6-dimethyl-N-[(E)-1-[(1S,2R)-2-phenylcyclopropyl]ethylideneamino]pyrimidin-4-amine —— C17H20N4
2,6-dimethyl-N-[(E)-1-[(1S,2R)-2-phenylcyclopropyl]ethylideneamino]pyrimidin-4-amine