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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[2-[(2R)-2,4-dimethylpiperazin-1-yl]-2-oxoethyl]-4-methyl-2-pyridin-3-yl-1H-pyrimidin-6-one —— C18H23N5O2
5-[2-[(2R)-2,4-dimethylpiperazin-1-yl]-2-oxoethyl]-4-methyl-2-pyridin-3-yl-1H-pyrimidin-6-one
—— 2-tert-butyl-N-[(2S)-2-hydroxy-3-phenylpropyl]-4-methyl-6-oxo-1H-pyrimidine-5-carboxamide —— C19H25N3O3
2-tert-butyl-N-[(2S)-2-hydroxy-3-phenylpropyl]-4-methyl-6-oxo-1H-pyrimidine-5-carboxamide
—— (4aR,7aR)-4-benzyl-6-(6-methoxypyrazin-2-yl)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine —— C18H22N4O2
(4aR,7aR)-4-benzyl-6-(6-methoxypyrazin-2-yl)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine
—— (4aS,7aR)-4-benzyl-6-(6-methoxypyrazin-2-yl)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine —— C18H22N4O2
(4aS,7aR)-4-benzyl-6-(6-methoxypyrazin-2-yl)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine
—— 6-chloro-2-[(3R)-5-(2-methoxyphenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C28H21ClN4OS
6-chloro-2-[(3R)-5-(2-methoxyphenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 6-chloro-2-[(3S)-5-(2-methoxyphenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C28H21ClN4OS
6-chloro-2-[(3S)-5-(2-methoxyphenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 4-(4-chlorophenyl)-2-[(3R)-3-(4-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]quinazoline —— C30H22ClFN4O
4-(4-chlorophenyl)-2-[(3R)-3-(4-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]quinazoline
—— 2-[(3R)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C31H26N4O2
2-[(3R)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 4-(4-chlorophenyl)-2-[(3S)-3-(4-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]quinazoline —— C30H22ClFN4O
4-(4-chlorophenyl)-2-[(3S)-3-(4-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]quinazoline
—— 2-[(3R)-5-(3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C30H24N4O
2-[(3R)-5-(3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 2-[(3S)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C31H26N4O2
2-[(3S)-3,5-bis(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 2-[(3S)-5-(3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C30H24N4O
2-[(3S)-5-(3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— 6-methoxy-5-[[[(2R,3R)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine —— C17H25N5OS
6-methoxy-5-[[[(2R,3R)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine
—— 6-methoxy-5-[[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine —— C17H25N5OS
6-methoxy-5-[[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine
—— (2R)-N-methyl-2-phenoxy-N-(6-phenylpyridazin-3-yl)propanamide —— C20H19N3O2
(2R)-N-methyl-2-phenoxy-N-(6-phenylpyridazin-3-yl)propanamide
—— (2S)-N-methyl-2-phenoxy-N-(6-phenylpyridazin-3-yl)propanamide —— C20H19N3O2
(2S)-N-methyl-2-phenoxy-N-(6-phenylpyridazin-3-yl)propanamide
—— (1R,6S)-N-methyl-N-(6-phenylpyridazin-3-yl)bicyclo[4.1.0]heptane-7-carboxamide —— C19H21N3O
(1R,6S)-N-methyl-N-(6-phenylpyridazin-3-yl)bicyclo[4.1.0]heptane-7-carboxamide
—— (3S,4S)-N,N-dimethyl-4-methylsulfanyl-1-(10-pyridin-3-yl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl)pyrrolidin-3-amine —— C21H25N5S2
(3S,4S)-N,N-dimethyl-4-methylsulfanyl-1-(10-pyridin-3-yl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl)pyrrolidin-3-amine
—— (3R,4S)-N,N-dimethyl-4-methylsulfanyl-1-(10-pyridin-3-yl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl)pyrrolidin-3-amine —— C21H25N5S2
(3R,4S)-N,N-dimethyl-4-methylsulfanyl-1-(10-pyridin-3-yl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl)pyrrolidin-3-amine
—— N-[[(2S)-4-[(1-ethylimidazol-2-yl)methyl]morpholin-2-yl]methyl]pyridazin-3-amine —— C15H22N6O
N-[[(2S)-4-[(1-ethylimidazol-2-yl)methyl]morpholin-2-yl]methyl]pyridazin-3-amine
—— N-[[(2R)-4-[(1-ethylimidazol-2-yl)methyl]morpholin-2-yl]methyl]pyridazin-3-amine —— C15H22N6O
N-[[(2R)-4-[(1-ethylimidazol-2-yl)methyl]morpholin-2-yl]methyl]pyridazin-3-amine
—— 4-ethyl-2-[[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl-methylamino]methyl]-1H-pyrimidin-6-one —— C15H22N4O2S
4-ethyl-2-[[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl-methylamino]methyl]-1H-pyrimidin-6-one
—— 4-ethyl-2-[[methyl-[(1R,2S)-2-methylsulfanylcyclopentyl]amino]methyl]-1H-pyrimidin-6-one —— C14H23N3OS
4-ethyl-2-[[methyl-[(1R,2S)-2-methylsulfanylcyclopentyl]amino]methyl]-1H-pyrimidin-6-one
—— (3S)-1-cyclopropyl-3-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one —— C18H21N5O
(3S)-1-cyclopropyl-3-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one
—— 6-chloro-4-N-[(R)-(4-ethylphenyl)-thiophen-2-ylmethyl]pyrimidine-2,4-diamine —— C17H17ClN4S
6-chloro-4-N-[(R)-(4-ethylphenyl)-thiophen-2-ylmethyl]pyrimidine-2,4-diamine
—— 2-methyl-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C14H16N6O2S
2-methyl-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-methyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C14H16N6O2S
2-methyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 6-chloro-4-N-[(S)-(4-ethylphenyl)-thiophen-2-ylmethyl]pyrimidine-2,4-diamine —— C17H17ClN4S
6-chloro-4-N-[(S)-(4-ethylphenyl)-thiophen-2-ylmethyl]pyrimidine-2,4-diamine
—— 4-ethyl-2-[[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl-methylamino]methyl]-1H-pyrimidin-6-one —— C15H22N4O2S
4-ethyl-2-[[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl-methylamino]methyl]-1H-pyrimidin-6-one
—— 6-ethyl-2-[6-[methyl-[[(2R)-oxan-2-yl]methyl]amino]pyridin-3-yl]-1H-pyrimidin-4-one —— C18H24N4O2
6-ethyl-2-[6-[methyl-[[(2R)-oxan-2-yl]methyl]amino]pyridin-3-yl]-1H-pyrimidin-4-one
—— 4-ethyl-2-[6-[[(2R)-1-ethylpiperidin-2-yl]methylamino]pyridin-3-yl]-1H-pyrimidin-6-one —— C19H27N5O
4-ethyl-2-[6-[[(2R)-1-ethylpiperidin-2-yl]methylamino]pyridin-3-yl]-1H-pyrimidin-6-one
—— 4-ethyl-2-[[(2R)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methyl]-1H-pyrimidin-6-one —— C17H26N6O
4-ethyl-2-[[(2R)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methyl]-1H-pyrimidin-6-one
—— 3,4-diethyl-6-oxo-N-[(1R)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]-1H-pyridazine-5-carboxamide —— C17H24N4O2S
3,4-diethyl-6-oxo-N-[(1R)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]-1H-pyridazine-5-carboxamide
—— 5-[(1S)-2,2-dimethyl-1-oxo-1,4-thiazinane-4-carbonyl]-3,4-diethyl-1H-pyridazin-6-one —— C15H23N3O3S
5-[(1S)-2,2-dimethyl-1-oxo-1,4-thiazinane-4-carbonyl]-3,4-diethyl-1H-pyridazin-6-one
—— 4-ethyl-2-[[[(2R)-1-ethylsulfanylpropan-2-yl]-methylamino]methyl]-1H-pyrimidin-6-one —— C13H23N3OS
4-ethyl-2-[[[(2R)-1-ethylsulfanylpropan-2-yl]-methylamino]methyl]-1H-pyrimidin-6-one
—— 4-ethyl-2-[[[(2S)-1-ethylsulfanylpropan-2-yl]-methylamino]methyl]-1H-pyrimidin-6-one —— C13H23N3OS
4-ethyl-2-[[[(2S)-1-ethylsulfanylpropan-2-yl]-methylamino]methyl]-1H-pyrimidin-6-one
—— 1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S)-1-(5-methyl-1,3-thiazol-2-yl)ethyl]urea —— C16H23N5O2S
1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S)-1-(5-methyl-1,3-thiazol-2-yl)ethyl]urea
—— 1-[(4-ethyl-6-oxo-1H-pyrimidin-2-yl)methyl]-1,2,4-triazole-3-carbonitrile —— C10H10N6O
1-[(4-ethyl-6-oxo-1H-pyrimidin-2-yl)methyl]-1,2,4-triazole-3-carbonitrile
—— 4-ethyl-2-[[methyl-[(1S,2S)-2-methylsulfanylcyclopentyl]amino]methyl]-1H-pyrimidin-6-one —— C14H23N3OS
4-ethyl-2-[[methyl-[(1S,2S)-2-methylsulfanylcyclopentyl]amino]methyl]-1H-pyrimidin-6-one
—— 2-[(1R)-cyclohex-2-en-1-yl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C15H19N3O
2-[(1R)-cyclohex-2-en-1-yl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— 1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S,2S)-2-phenylcyclopropyl]urea —— C19H24N4O2
1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S,2S)-2-phenylcyclopropyl]urea
—— 4-ethyl-2-[[(2S)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methyl]-1H-pyrimidin-6-one —— C17H26N6O
4-ethyl-2-[[(2S)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methyl]-1H-pyrimidin-6-one
—— 2-[(1S)-cyclohex-2-en-1-yl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C15H19N3O
2-[(1S)-cyclohex-2-en-1-yl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— (2R)-1-[4-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]piperidin-1-yl]butan-2-ol —— C20H29N5O
(2R)-1-[4-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]piperidin-1-yl]butan-2-ol
—— 5-[(1R)-2,2-dimethyl-1-oxo-1,4-thiazinane-4-carbonyl]-3,4-diethyl-1H-pyridazin-6-one —— C15H23N3O3S
5-[(1R)-2,2-dimethyl-1-oxo-1,4-thiazinane-4-carbonyl]-3,4-diethyl-1H-pyridazin-6-one
—— 1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1R,2R)-2-phenylcyclopropyl]urea —— C19H24N4O2
1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1R,2R)-2-phenylcyclopropyl]urea
—— 1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1R,2S)-2-phenylcyclopropyl]urea —— C19H24N4O2
1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1R,2S)-2-phenylcyclopropyl]urea
—— 1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S,2R)-2-phenylcyclopropyl]urea —— C19H24N4O2
1-[(3,4-diethyl-6-oxo-1H-pyridazin-5-yl)methyl]-3-[(1S,2R)-2-phenylcyclopropyl]urea
—— (3R)-1-cyclopropyl-3-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one —— C18H21N5O
(3R)-1-cyclopropyl-3-[(6-ethyl-2-pyridin-2-ylpyrimidin-4-yl)amino]pyrrolidin-2-one
—— 4-ethyl-2-[6-[[(2S)-1-ethylpiperidin-2-yl]methylamino]pyridin-3-yl]-1H-pyrimidin-6-one —— C19H27N5O
4-ethyl-2-[6-[[(2S)-1-ethylpiperidin-2-yl]methylamino]pyridin-3-yl]-1H-pyrimidin-6-one