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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-6-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methylheptan-2-ol —— C14H25N3O
(6R)-6-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methylheptan-2-ol
—— 2-[(4-tert-butylphenoxy)methyl]-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C22H26N4O4
2-[(4-tert-butylphenoxy)methyl]-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 2-(1-adamantyl)-5-[(3S)-3-hydroxypiperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H27N3O3
2-(1-adamantyl)-5-[(3S)-3-hydroxypiperidine-1-carbonyl]-1H-pyrimidin-6-one
—— 2-[(4-tert-butylphenoxy)methyl]-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C22H26N4O4
2-[(4-tert-butylphenoxy)methyl]-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 2-(1-adamantyl)-5-[(3R)-3-hydroxypiperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H27N3O3
2-(1-adamantyl)-5-[(3R)-3-hydroxypiperidine-1-carbonyl]-1H-pyrimidin-6-one
—— (6S)-6-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methylheptan-2-ol —— C14H25N3O
(6S)-6-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methylheptan-2-ol
—— [2-(ethylamino)pyrimidin-5-yl]-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]methanone —— C15H24N4O2
[2-(ethylamino)pyrimidin-5-yl]-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]methanone
—— 6-[[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C17H28N4O4
6-[[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— [2-(ethylamino)pyrimidin-5-yl]-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]methanone —— C15H24N4O2
[2-(ethylamino)pyrimidin-5-yl]-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]methanone
—— 6-[[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C17H28N4O4
6-[[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— [(3R)-1-[3-[(2,5,6-trimethylpyrimidin-4-yl)amino]propyl]piperidin-3-yl]methanol —— C16H28N4O
[(3R)-1-[3-[(2,5,6-trimethylpyrimidin-4-yl)amino]propyl]piperidin-3-yl]methanol
—— [(3S)-1-[3-[(2,5,6-trimethylpyrimidin-4-yl)amino]propyl]piperidin-3-yl]methanol —— C16H28N4O
[(3S)-1-[3-[(2,5,6-trimethylpyrimidin-4-yl)amino]propyl]piperidin-3-yl]methanol
—— N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide —— C17H23N5O3S
N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide
—— (6S)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N5O2
(6S)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 2-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C17H22N4O4
2-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— (6R)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N5O2
(6R)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 2-methyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C17H22N4O4
2-methyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 4-(1H-pyrazol-4-yl)-N-[(5R)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide —— C20H22N6O
4-(1H-pyrazol-4-yl)-N-[(5R)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide
—— (4R)-6-ethyl-5-nitro-4-(2-propoxyphenyl)-3,4-dihydro-1H-pyrimidin-2-one —— C15H19N3O4
(4R)-6-ethyl-5-nitro-4-(2-propoxyphenyl)-3,4-dihydro-1H-pyrimidin-2-one
—— [(2S)-1-[3-[(5,6-dimethylpyrimidin-4-yl)amino]propyl]piperidin-2-yl]methanol —— C15H26N4O
[(2S)-1-[3-[(5,6-dimethylpyrimidin-4-yl)amino]propyl]piperidin-2-yl]methanol
—— N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidine-5-carboxamide —— C16H19N7O2S
N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidine-5-carboxamide
—— 4-(1H-pyrazol-4-yl)-N-[(5S)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide —— C20H22N6O
4-(1H-pyrazol-4-yl)-N-[(5S)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide
—— N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidine-5-carboxamide —— C16H19N7O2S
N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidine-5-carboxamide
—— N-[(1S)-1-(2-chlorophenyl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C18H15ClN4O2
N-[(1S)-1-(2-chlorophenyl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— N-[(1R)-1-(2-chlorophenyl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C18H15ClN4O2
N-[(1R)-1-(2-chlorophenyl)ethyl]-6-oxo-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide —— C17H23N5O3S
N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-1H-pyrimidine-5-carboxamide
—— 2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide —— C14H16N4O3S
2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide
—— 2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide —— C14H16N4O3S
2-(2-methyl-1,3-thiazol-4-yl)-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide
—— [(2R)-1-[3-[(5,6-dimethylpyrimidin-4-yl)amino]propyl]piperidin-2-yl]methanol —— C15H26N4O
[(2R)-1-[3-[(5,6-dimethylpyrimidin-4-yl)amino]propyl]piperidin-2-yl]methanol
—— 6-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H21N5O2S
6-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (3S)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]-3,4-dihydro-2H-chromene-3-carboxamide —— C22H21N3O3
(3S)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]-3,4-dihydro-2H-chromene-3-carboxamide
—— 2-[(2,6-dichlorophenyl)methyl]-6-oxo-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrimidine-5-carboxamide —— C17H16Cl2N6O2
2-[(2,6-dichlorophenyl)methyl]-6-oxo-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrimidine-5-carboxamide
—— 6-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H21N5O2S
6-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2,6-dichlorophenyl)methyl]-6-oxo-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrimidine-5-carboxamide —— C17H16Cl2N6O2
2-[(2,6-dichlorophenyl)methyl]-6-oxo-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrimidine-5-carboxamide
—— (3R)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]-3,4-dihydro-2H-chromene-3-carboxamide —— C22H21N3O3
(3R)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]-3,4-dihydro-2H-chromene-3-carboxamide
—— N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-6-oxo-2-pyridin-3-yl-1H-pyrimidine-5-carboxamide —— C17H18N6O3
N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-6-oxo-2-pyridin-3-yl-1H-pyrimidine-5-carboxamide
—— N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-6-oxo-2-pyridin-3-yl-1H-pyrimidine-5-carboxamide —— C17H18N6O3
N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-6-oxo-2-pyridin-3-yl-1H-pyrimidine-5-carboxamide
—— 2-(ethylamino)-N-[(4-methoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidine-5-carboxamide —— C20H26N4O3
2-(ethylamino)-N-[(4-methoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidine-5-carboxamide
—— 2-(ethylamino)-N-[(4-methoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidine-5-carboxamide —— C20H26N4O3
2-(ethylamino)-N-[(4-methoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidine-5-carboxamide
—— N-Tert-butyl-2-({7-oxo-5-phenyl-7H,8H-[1,2,4]triazolo[4,3-A]pyrimidin-3-YL}sulfanyl)acetamide —— C17H19N5O2S
N-Tert-butyl-2-({7-oxo-5-phenyl-7H,8H-[1,2,4]triazolo[4,3-A]pyrimidin-3-YL}sulfanyl)acetamide
—— (2S)-1-N-(6-cyclopropylpyrimidin-4-yl)-2-N-ethyl-2-N-methylbutane-1,2-diamine —— C14H24N4
(2S)-1-N-(6-cyclopropylpyrimidin-4-yl)-2-N-ethyl-2-N-methylbutane-1,2-diamine
—— 2-(4-methylphenyl)-5-[(2S)-2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H20N4O2S
2-(4-methylphenyl)-5-[(2S)-2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— 2-(4-methylphenyl)-5-[(2R)-2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H20N4O2S
2-(4-methylphenyl)-5-[(2R)-2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— (2-methylpyrimidin-5-yl)-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N6O
(2-methylpyrimidin-5-yl)-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— 6-oxo-2-thiophen-2-yl-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide —— C19H20N4O2S2
6-oxo-2-thiophen-2-yl-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide
—— (2-methylpyrimidin-5-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N6O
(2-methylpyrimidin-5-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (3S)-1-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid —— C17H23N3O5
(3S)-1-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
—— 2-(4-methylphenyl)-5-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyrimidin-6-one —— C19H18N4O2S
2-(4-methylphenyl)-5-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyrimidin-6-one
—— (3R)-1-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid —— C17H23N3O5
(3R)-1-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
—— 5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C12H12N6O
5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole