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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-[3-(2-methylpyrimidin-4-yl)phenyl]-2-(5-methyl-1H-1,2,4-triazol-3-yl)pyrrolidine-1-carboxamide —— C19H21N7O
(2R)-N-[3-(2-methylpyrimidin-4-yl)phenyl]-2-(5-methyl-1H-1,2,4-triazol-3-yl)pyrrolidine-1-carboxamide
—— 3-(6-methylpyridazin-3-yl)-5-[(1S)-1-propoxyethyl]-1,2,4-oxadiazole —— C12H16N4O2
3-(6-methylpyridazin-3-yl)-5-[(1S)-1-propoxyethyl]-1,2,4-oxadiazole
—— [(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C19H28N6O
[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— N-ethyl-N-[[(3S)-1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl]methyl]pyrazine-2-carboxamide —— C22H30N4O2
N-ethyl-N-[[(3S)-1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl]methyl]pyrazine-2-carboxamide
—— [(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C19H28N6O
[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— 1-[(R)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-3-[3-(2-methylpyrimidin-4-yl)phenyl]urea —— C20H22N6O
1-[(R)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-3-[3-(2-methylpyrimidin-4-yl)phenyl]urea
—— N-(3-morpholin-4-ylpropyl)-2-pyridin-3-ylquinazolin-4-amine —— C20H23N5O
N-(3-morpholin-4-ylpropyl)-2-pyridin-3-ylquinazolin-4-amine
—— N-ethyl-N-[[(3R)-1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl]methyl]pyrazine-2-carboxamide —— C22H30N4O2
N-ethyl-N-[[(3R)-1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl]methyl]pyrazine-2-carboxamide
—— 2-[2-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]acetamide —— C15H20N6O2
2-[2-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]acetamide
—— 1-[(S)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-3-[3-(2-methylpyrimidin-4-yl)phenyl]urea —— C20H22N6O
1-[(S)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-3-[3-(2-methylpyrimidin-4-yl)phenyl]urea
—— 2-[2-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]acetamide —— C15H20N6O2
2-[2-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]imidazol-1-yl]acetamide
—— N-[[(3S)-1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl]methyl]-N-methyl-2-(methylamino)pyrimidine-5-carboxamide —— C21H28FN5O
N-[[(3S)-1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl]methyl]-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
—— N-[(3,4-difluorophenyl)methyl]-3-[(3S)-1-(6-oxo-1H-pyrimidine-5-carbonyl)piperidin-3-yl]propanamide —— C20H22F2N4O3
N-[(3,4-difluorophenyl)methyl]-3-[(3S)-1-(6-oxo-1H-pyrimidine-5-carbonyl)piperidin-3-yl]propanamide
—— N-[[(3R)-1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl]methyl]-N-methyl-2-(methylamino)pyrimidine-5-carboxamide —— C21H28FN5O
N-[[(3R)-1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl]methyl]-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
—— [(3S)-3-methyl-3-phenylpiperidin-1-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone —— C22H22N4O
[(3S)-3-methyl-3-phenylpiperidin-1-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone
—— N-[(3,4-difluorophenyl)methyl]-3-[(3R)-1-(6-oxo-1H-pyrimidine-5-carbonyl)piperidin-3-yl]propanamide —— C20H22F2N4O3
N-[(3,4-difluorophenyl)methyl]-3-[(3R)-1-(6-oxo-1H-pyrimidine-5-carbonyl)piperidin-3-yl]propanamide
—— [(3R)-3-methyl-3-phenylpiperidin-1-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone —— C22H22N4O
[(3R)-3-methyl-3-phenylpiperidin-1-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone
—— N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxopyrimidine-4-carboxamide —— C15H20N4O3S
N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxopyrimidine-4-carboxamide
—— N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxopyrimidine-4-carboxamide —— C15H20N4O3S
N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxopyrimidine-4-carboxamide
—— 1-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-3-[2-[(1S)-1-phenylethyl]pyrazol-3-yl]urea —— C20H24N6O2
1-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-3-[2-[(1S)-1-phenylethyl]pyrazol-3-yl]urea
—— 1,3-dimethyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C13H16N6S
1,3-dimethyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— ethyl (4R)-4-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C11H16N6O3S
ethyl (4R)-4-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-3-[2-[(1R)-1-phenylethyl]pyrazol-3-yl]urea —— C20H24N6O2
1-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-3-[2-[(1R)-1-phenylethyl]pyrazol-3-yl]urea
—— 1,3-dimethyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C13H16N6S
1,3-dimethyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide —— C22H34N4O3
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide
—— N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide —— C22H34N4O3
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrimidine-5-carboxamide
—— 1,3-dimethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]-2,6-dioxopyrimidine-4-carboxamide —— C16H20N4O3
1,3-dimethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]-2,6-dioxopyrimidine-4-carboxamide
—— 1-[2-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-3-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]urea —— C18H24N6O2
1-[2-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-3-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]urea
—— 1-[2-[[(1S)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-3-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]urea —— C18H24N6O2
1-[2-[[(1S)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-3-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]urea
—— 6-[(3S)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H24N4O5
6-[(3S)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(3R)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H24N4O5
6-[(3R)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 1,3-dimethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]-2,6-dioxopyrimidine-4-carboxamide —— C16H20N4O3
1,3-dimethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]-2,6-dioxopyrimidine-4-carboxamide
—— ethyl (4R)-4-(4-butylphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N2O3
ethyl (4R)-4-(4-butylphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carboxylate —— C18H12ClN3O4S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carboxylate
—— [(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C19H28N6O
[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— [(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C19H28N6O
[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— methyl N-[(1R)-1-(3-pyridazin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]carbamate —— C10H11N5O3
methyl N-[(1R)-1-(3-pyridazin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]carbamate
—— methyl N-[(1S)-1-(3-pyridazin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]carbamate —— C10H11N5O3
methyl N-[(1S)-1-(3-pyridazin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]carbamate
—— 6-[(2S)-2-(3-fluorophenyl)azepane-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H22FN3O3
6-[(2S)-2-(3-fluorophenyl)azepane-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(2R)-2-(3-fluorophenyl)azepane-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H22FN3O3
6-[(2R)-2-(3-fluorophenyl)azepane-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— (4S)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide —— C23H23N3O2
(4S)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
—— (4R)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide —— C23H23N3O2
(4R)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
—— [2-[[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-(2-methoxyethyl)amino]-2-oxoethyl] (1S,2S)-2-methylcyclopropane-1-carboxylate —— C18H28N4O6
[2-[[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-(2-methoxyethyl)amino]-2-oxoethyl] (1S,2S)-2-methylcyclopropane-1-carboxylate
—— methyl (4R)-4-(4-chlorophenyl)-6-propyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H17ClN2O2S
methyl (4R)-4-(4-chlorophenyl)-6-propyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [2-[[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-(2-methoxyethyl)amino]-2-oxoethyl] (1R,2R)-2-methylcyclopropane-1-carboxylate —— C18H28N4O6
[2-[[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-(2-methoxyethyl)amino]-2-oxoethyl] (1R,2R)-2-methylcyclopropane-1-carboxylate
—— N-[(R)-(2,5-dimethylphenyl)-pyridin-3-ylmethyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide —— C21H22N4O3
N-[(R)-(2,5-dimethylphenyl)-pyridin-3-ylmethyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide
—— 4-[(2S)-2-methylpiperidin-1-yl]-2-pyridin-3-ylquinazoline —— C19H20N4
4-[(2S)-2-methylpiperidin-1-yl]-2-pyridin-3-ylquinazoline
—— N-[(S)-(2,5-dimethylphenyl)-pyridin-3-ylmethyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide —— C21H22N4O3
N-[(S)-(2,5-dimethylphenyl)-pyridin-3-ylmethyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide
—— ethyl (4R)-4-ethyl-2-oxo-6-(pyridine-2-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H19N3O5
ethyl (4R)-4-ethyl-2-oxo-6-(pyridine-2-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(3-methoxyphenyl)methyl]-3-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]propanamide —— C22H28N4O3
N-[(3-methoxyphenyl)methyl]-3-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]propanamide