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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl (6R)-6-[3-chloro-4-(difluoromethoxy)-5-methoxyphenyl]-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C18H19ClF2N2O5
methyl (6R)-6-[3-chloro-4-(difluoromethoxy)-5-methoxyphenyl]-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-cyclopropyl-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C20H24F2N2O5
ethyl (6S)-3-cyclopropyl-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 2-methoxyethyl (6R)-6-(5-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C16H19BrN2O4S
2-methoxyethyl (6R)-6-(5-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 2-[[2-[(1R)-1-ethoxyethyl]-1,3-thiazol-4-yl]methyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C17H22N4O2S
2-[[2-[(1R)-1-ethoxyethyl]-1,3-thiazol-4-yl]methyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— 2-[[2-[(1S)-1-ethoxyethyl]-1,3-thiazol-4-yl]methyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C17H22N4O2S
2-[[2-[(1S)-1-ethoxyethyl]-1,3-thiazol-4-yl]methyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— methyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(2,4-dimethylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H23N3O4
methyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(2,4-dimethylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 3-amino-N-[(1R,3S)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide —— C14H20N4O2
3-amino-N-[(1R,3S)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide
—— 3-amino-N-[(1R,3R)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide —— C14H20N4O2
3-amino-N-[(1R,3R)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide
—— 3-amino-N-[(1R)-1-(5-ethylfuran-2-yl)-2-methoxyethyl]pyrazine-2-carboxamide —— C14H18N4O3
3-amino-N-[(1R)-1-(5-ethylfuran-2-yl)-2-methoxyethyl]pyrazine-2-carboxamide
—— 3-amino-N-[(1S,3R)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide —— C14H20N4O2
3-amino-N-[(1S,3R)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide
—— 3-amino-N-[(1S,3S)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide —— C14H20N4O2
3-amino-N-[(1S,3S)-3-ethoxyspiro[3.3]heptan-1-yl]pyrazine-2-carboxamide
—— [2-[(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-propylamino]-2-oxoethyl] (E)-but-2-enoate —— C20H24N4O5
[2-[(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-propylamino]-2-oxoethyl] (E)-but-2-enoate
—— [2-[(6-amino-1-butyl-2,4-dioxopyrimidin-5-yl)-cyclopentylamino]-2-oxoethyl] (E)-but-2-enoate —— C19H28N4O5
[2-[(6-amino-1-butyl-2,4-dioxopyrimidin-5-yl)-cyclopentylamino]-2-oxoethyl] (E)-but-2-enoate
—— [2-[(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-ethylamino]-2-oxoethyl] 2-thiophen-3-ylacetate —— C18H24N4O5S
[2-[(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-ethylamino]-2-oxoethyl] 2-thiophen-3-ylacetate
—— ethyl (4S)-6-[[5-(butylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H25N5O3S2
ethyl (4S)-6-[[5-(butylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[5-(butylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H25N5O3S2
ethyl (4R)-6-[[5-(butylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[4-benzyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H25N5O4S
ethyl (4S)-6-[[4-benzyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[4-benzyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H25N5O4S
ethyl (4R)-6-[[4-benzyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 3-[[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]amino]pyrazine-2-carbonitrile —— C12H14N6O
3-[[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]amino]pyrazine-2-carbonitrile
—— N-[[(1R,2R)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O
N-[[(1R,2R)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide
—— N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide —— C20H25N3O2
N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide
—— N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-pyrimidin-5-ylbenzamide —— C19H21N5O
N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-pyrimidin-5-ylbenzamide
—— (2R)-1-[(5-bromopyrimidin-2-yl)amino]-2-(1-methylpyrazol-4-yl)propan-2-ol —— C11H14BrN5O
(2R)-1-[(5-bromopyrimidin-2-yl)amino]-2-(1-methylpyrazol-4-yl)propan-2-ol
—— N-[[(1S,2R)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O
N-[[(1S,2R)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide
—— N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-pyrimidin-5-ylbenzamide —— C19H21N5O
N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-pyrimidin-5-ylbenzamide
—— N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide —— C20H25N3O2
N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide
—— N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide —— C20H25N3O2
N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide
—— N-[[(1R,2S)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O
N-[[(1R,2S)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide
—— N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide —— C20H25N3O2
N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-2-pyrimidin-5-ylbenzamide
—— 3-[[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]amino]pyrazine-2-carbonitrile —— C12H14N6O
3-[[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]amino]pyrazine-2-carbonitrile
—— (2S)-1-[(5-bromopyrimidin-2-yl)amino]-2-(1-methylpyrazol-4-yl)propan-2-ol —— C11H14BrN5O
(2S)-1-[(5-bromopyrimidin-2-yl)amino]-2-(1-methylpyrazol-4-yl)propan-2-ol
—— N-[[(1S,2S)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O
N-[[(1S,2S)-2-phenylcyclopropyl]methyl]-2-pyrimidin-5-ylbenzamide
—— 6-[(2R)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]pyrido[2,3-d]pyridazin-5-one —— C15H15N3O3S
6-[(2R)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]pyrido[2,3-d]pyridazin-5-one —— C15H15N3O3S
6-[(2S)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]pyrido[2,3-d]pyridazin-5-one
—— N-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide —— C18H24N4O2
N-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
—— 3-[3-[[(3R)-oxolan-3-yl]methoxy]propylamino]pyrazine-2-carbonitrile —— C13H18N4O2
3-[3-[[(3R)-oxolan-3-yl]methoxy]propylamino]pyrazine-2-carbonitrile
—— N-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-N-methyl-2-(3-methyl-6-oxopyridazin-1-yl)acetamide —— C18H27N3O3
N-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-N-methyl-2-(3-methyl-6-oxopyridazin-1-yl)acetamide
—— (2S)-1-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-2-thiophen-2-ylpropan-2-ol —— C16H19N5OS
(2S)-1-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-2-thiophen-2-ylpropan-2-ol
—— N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide —— C18H24N4O2
N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
—— 3-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyrazine-2-carbonitrile —— C10H14N4OS
3-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyrazine-2-carbonitrile
—— 3-[[(2S)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyrazine-2-carbonitrile —— C10H14N4OS
3-[[(2S)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]pyrazine-2-carbonitrile
—— N-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide —— C18H24N4O2
N-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
—— N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methyl-2-(3-methyl-6-oxopyridazin-1-yl)acetamide —— C18H27N3O3
N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methyl-2-(3-methyl-6-oxopyridazin-1-yl)acetamide
—— 3-[[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]amino]pyrazine-2-carbonitrile —— C16H20N6S
3-[[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]amino]pyrazine-2-carbonitrile
—— (3R)-4-methylsulfanyl-3-[(2-phenylpyrimidin-4-yl)amino]butan-1-ol —— C15H19N3OS
(3R)-4-methylsulfanyl-3-[(2-phenylpyrimidin-4-yl)amino]butan-1-ol
—— 6-chloro-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyrazin-2-amine —— C12H18ClN3O2
6-chloro-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]pyrazin-2-amine
—— 3-amino-N-[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide —— C16H22N6OS
3-amino-N-[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide
—— (2S)-1-[(6-chloropyrazin-2-yl)amino]-2-thiophen-3-ylpropan-2-ol —— C11H12ClN3OS
(2S)-1-[(6-chloropyrazin-2-yl)amino]-2-thiophen-3-ylpropan-2-ol
—— (4S)-4-[(5-bromopyrimidin-2-yl)amino]-4-phenylbutan-1-ol —— C14H16BrN3O
(4S)-4-[(5-bromopyrimidin-2-yl)amino]-4-phenylbutan-1-ol
—— 3-[[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]amino]pyrazine-2-carbonitrile —— C16H20N6S
3-[[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]amino]pyrazine-2-carbonitrile