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中文名称 英文名称 CAS号 化学式 结构式图片
—— rac-N-(2-amino-2-methylpentyl)-8-[(2-fluoro-3-methylbenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C24H31FN4O2
rac-N-(2-amino-2-methylpentyl)-8-[(2-fluoro-3-methylbenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-Difluorobenzyl)oxy]-N-(6-methoxy-1,2,3,4-tetrahydroquinolin-4-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C27H26F2N4O3
rac-8-[(2,6-Difluorobenzyl)oxy]-N-(6-methoxy-1,2,3,4-tetrahydroquinolin-4-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— (R)-3-methyl-2-[5-oxo-2-(4-pyridin-4-yl-piperazin-1-yl)-6,7-dihydro-5H-5λ<sup>4</sup>-thieno[3,2-d]pyrimidin-4-ylamino]-butan-1-ol trifluoroacetate —— (x)C2HF3O2*C20H28N6O2S
(R)-3-methyl-2-[5-oxo-2-(4-pyridin-4-yl-piperazin-1-yl)-6,7-dihydro-5H-5λ<sup>4</sup>-thieno[3,2-d]pyrimidin-4-ylamino]-butan-1-ol trifluoroacetate
—— (R)-N-[(1R)-2-methoxy-1-(4-methoxyphenyl)ethyl]-2-methylpropane-2-sulfinamide —— C14H23NO3S
(R)-N-[(1R)-2-methoxy-1-(4-methoxyphenyl)ethyl]-2-methylpropane-2-sulfinamide
—— (R)-2-((5-bromopyridin-3-yl)amino)-2-phenylacetamide —— C13H12BrN3O
(R)-2-((5-bromopyridin-3-yl)amino)-2-phenylacetamide
—— (R)-6-[(R)-1-(1,3-dimethylazetidin-3-yl)ethyl]-7-[2-(1-hydroxy-1-methylethyl)phenyl]-4-methyl-2,10-dihydro-9-oxa-1,2,4a-triazaphenanthren-3-one 1613718-04-9 C27H34N4O3
(R)-6-[(R)-1-(1,3-dimethylazetidin-3-yl)ethyl]-7-[2-(1-hydroxy-1-methylethyl)phenyl]-4-methyl-2,10-dihydro-9-oxa-1,2,4a-triazaphenanthren-3-one
—— (R)-N-(1-(4-fluorophenyl)ethyl)-4-(2,2,3,3-tetradeuterio-1,2,3,4-tetrahydropyrido[3,2-b]pyrazine-7-sulfonamido)cyclohexanecarboxamide —— C22H28FN5O3S
(R)-N-(1-(4-fluorophenyl)ethyl)-4-(2,2,3,3-tetradeuterio-1,2,3,4-tetrahydropyrido[3,2-b]pyrazine-7-sulfonamido)cyclohexanecarboxamide
—— (R)-N-(1-(4-fluorophenyl)ethyl)-4-(1,2,3,4-tetrahydropyrido[3,2-b]pyrazine-7-sulfonamido)bicyclo[2.2.2]octane-1-carboxamide 1357274-54-4 C24H30FN5O3S
(R)-N-(1-(4-fluorophenyl)ethyl)-4-(1,2,3,4-tetrahydropyrido[3,2-b]pyrazine-7-sulfonamido)bicyclo[2.2.2]octane-1-carboxamide
—— (R)-Quinuclidin-3-yl ((S)-(3-(2-((3-formylphenyl)amino)-2-oxoethoxy)phenyl)-(phenyl)methyl)carbamate —— C30H31N3O5
(R)-Quinuclidin-3-yl ((S)-(3-(2-((3-formylphenyl)amino)-2-oxoethoxy)phenyl)-(phenyl)methyl)carbamate
—— rac-cyclopentyl(4-(5-fluoro-2-methyl-3-nitrobenzyl)-2-methylpiperazin-1-yl)methanone —— C19H26FN3O3
rac-cyclopentyl(4-(5-fluoro-2-methyl-3-nitrobenzyl)-2-methylpiperazin-1-yl)methanone
—— (R)-2-amino-6-fluoro-N-(5-fluoro-4-(4-(3-methylpiperazine-1-carbonyl)piperidin-1-yl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1613196-95-4 C23H27F2N9O2
(R)-2-amino-6-fluoro-N-(5-fluoro-4-(4-(3-methylpiperazine-1-carbonyl)piperidin-1-yl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (R)-quinuclidin-3-yl ((S)-(3-((1-(4-(2-(((R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)ethyl)benzoyl)piperidin-4-yl)methoxy)phenyl)(phenyl)methyl)carbamate 1613464-23-5 C47H53N5O7
(R)-quinuclidin-3-yl ((S)-(3-((1-(4-(2-(((R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)ethyl)benzoyl)piperidin-4-yl)methoxy)phenyl)(phenyl)methyl)carbamate
—— (R)-quinuclidin-3-yl ((S)-(3-((5-(benzyl(3-(((R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)propyl)carbamoyl)furan-2-yl)methoxy)phenyl)(phenyl)methyl)carbamate 1613464-56-4 C48H51N5O8
(R)-quinuclidin-3-yl ((S)-(3-((5-(benzyl(3-(((R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)propyl)carbamoyl)furan-2-yl)methoxy)phenyl)(phenyl)methyl)carbamate
—— [(R)-[[6-(3-chloro-4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-phenylmethyl]phosphonic acid —— C20H17ClN3O3PS
[(R)-[[6-(3-chloro-4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-phenylmethyl]phosphonic acid
—— (R)-1-{1-((R)-sec-Butyl)-6-[2-(1-ethanesulfonyl-1H-pyrazol-4-yl)pyrimidin-4-ylamino]-1H-imidazo[4,5-c]pyridin-2-yl}ethanol —— C21H26N8O3S
(R)-1-{1-((R)-sec-Butyl)-6-[2-(1-ethanesulfonyl-1H-pyrazol-4-yl)pyrimidin-4-ylamino]-1H-imidazo[4,5-c]pyridin-2-yl}ethanol
—— (R)-1-[6-Chloro-1-((R)-2,2,2-trifluoro-1-methylethyl)-1H-imidazo[4,5-c]pyridin-2-yl]ethanol —— C11H11ClF3N3O
(R)-1-[6-Chloro-1-((R)-2,2,2-trifluoro-1-methylethyl)-1H-imidazo[4,5-c]pyridin-2-yl]ethanol
—— (R)-ethyl 3-((2-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-ylamino)methyl)piperidine-1-carboxylate —— C20H23ClN6O2
(R)-ethyl 3-((2-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-ylamino)methyl)piperidine-1-carboxylate
—— (R,E)-1-(3-(4-amino-6-chloro-5-(4-chlorophenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)pyrrolidin-1-yl)-4-(dimethylamino)but-2-en-1-one 1610697-23-8 C22H24Cl2N6O
(R,E)-1-(3-(4-amino-6-chloro-5-(4-chlorophenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)pyrrolidin-1-yl)-4-(dimethylamino)but-2-en-1-one
—— (RS)-1-([3-(tert-butyl-dimethyl-silanyloxy)-propyl]-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-amino)-9-fluoro-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one —— C34H43FN4O5SSi
(RS)-1-([3-(tert-butyl-dimethyl-silanyloxy)-propyl]-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-amino)-9-fluoro-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one
—— (R)-2-(3-(3-(4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-1-yl)propylamino)-2-(tert-butoxycarbonylamino)-3-oxopropylthio)ethyl palmitate 1610431-55-4 C42H68N6O6S
(R)-2-(3-(3-(4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-1-yl)propylamino)-2-(tert-butoxycarbonylamino)-3-oxopropylthio)ethyl palmitate
—— (RS)-1-([2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-amino)-9-fluoro-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one —— C33H41FN4O5SSi
(RS)-1-([2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-amino)-9-fluoro-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one
—— (R)-3-(Ethyl(tetrahydro-2H-pyran-4-yl)amino)-5-((1-(2-hydroxypropyl)piperidin-4-yl)ethynyl)-N-((4-isopropyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methylbenzamide —— C35H50N4O4
(R)-3-(Ethyl(tetrahydro-2H-pyran-4-yl)amino)-5-((1-(2-hydroxypropyl)piperidin-4-yl)ethynyl)-N-((4-isopropyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methylbenzamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,2,3,4-tetrahydroisoquiolin-1-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide 1609340-90-0 C26H24F2N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,2,3,4-tetrahydroisoquiolin-1-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
—— rac-benzyl 1-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3-azabicyclo[4.1.0]heptane-3-carboxylate 1609345-59-6 C30H28F2N4O4
rac-benzyl 1-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3-azabicyclo[4.1.0]heptane-3-carboxylate
—— (R)-1-cyclopropyl-3-(dibenzylamino)-2-fluoropropan-1-one 1609546-52-2 C20H22FNO
(R)-1-cyclopropyl-3-(dibenzylamino)-2-fluoropropan-1-one
—— rac-tert-butyl {2-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]-2-phenylethyl}carbamate 1609344-77-5 C29H30F2N4O4
rac-tert-butyl {2-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]-2-phenylethyl}carbamate
—— rac-benzyl [3-(3,4-difluorophenoxy)-2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)propyl]carbamate 1609345-37-0 C25H20F2N2O5
rac-benzyl [3-(3,4-difluorophenoxy)-2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)propyl]carbamate
—— (R)-N-(4-(4-(2-methoxyethyl)-3-methylpiperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377259-58-9 C24H27N7OS
(R)-N-(4-(4-(2-methoxyethyl)-3-methylpiperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— rac-6-(5-fluoropyrimidin-2-yl)-7a-(2-pyridyl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-amine 1607432-79-0 C15H15FN6S
rac-6-(5-fluoropyrimidin-2-yl)-7a-(2-pyridyl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-amine
—— (R)-N-(4-(4-(2-methoxyethyl)-2-methylpiperazin-1-yl)pyridin-2-yl)-5-(5-methyl-1H-pyrazol-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377260-46-2 C23H28N8OS
(R)-N-(4-(4-(2-methoxyethyl)-2-methylpiperazin-1-yl)pyridin-2-yl)-5-(5-methyl-1H-pyrazol-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— rac-7a-(5-fluoro-2-pyridyl)-6-(5-fluoropyrimidin-2-yl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-amine 1607432-80-3 C15H14F2N6S
rac-7a-(5-fluoro-2-pyridyl)-6-(5-fluoropyrimidin-2-yl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-amine
—— rac-N-[7a-(5-fluoro-2-pyridyl)-6-(5-fluoropyrimidin-2-yl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-yl]benzamide 1607432-40-5 C22H18F2N6OS
rac-N-[7a-(5-fluoro-2-pyridyl)-6-(5-fluoropyrimidin-2-yl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-2-yl]benzamide
—— (R)-4-benzyl-3-[2-(4-benzyloxy-3-chlorophenyl)cyclopropanecarbonyl]oxazolidin-2-one —— C27H24ClNO4
(R)-4-benzyl-3-[2-(4-benzyloxy-3-chlorophenyl)cyclopropanecarbonyl]oxazolidin-2-one
—— rac-4,4,4-Trifluorobutane-1,2-diamine dihydrochloride 1609345-92-7 C4H11Cl2F3N2
rac-4,4,4-Trifluorobutane-1,2-diamine dihydrochloride
—— rac-N-(2-amino-2-methylbutyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609342-13-3 C21H23ClF2N4O2
rac-N-(2-amino-2-methylbutyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,2,3,4-tetrahydroquinolin-4-yl)imidazo[1,2-a]-pyridine-3-carboxamide 1609340-61-5 C25H22F2N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,2,3,4-tetrahydroquinolin-4-yl)imidazo[1,2-a]-pyridine-3-carboxamide
—— (R)-methyl 2-((R)-1-(tert-butyldimethylsilyloxy)-10-(1-phenyl-1H-tetrazol-5-ylsulfonyl)decyl)-26-(pivaloyloxy)hexacosanoate —— C55H100N4O7SSi
(R)-methyl 2-((R)-1-(tert-butyldimethylsilyloxy)-10-(1-phenyl-1H-tetrazol-5-ylsulfonyl)decyl)-26-(pivaloyloxy)hexacosanoate
—— (R)-5-(2-(4-fluorophenyl)-6-(4-(4-fluorophenyl)-2-methylpiperazine-1-carbonyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid —— C32H31F2N3O4
(R)-5-(2-(4-fluorophenyl)-6-(4-(4-fluorophenyl)-2-methylpiperazine-1-carbonyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
—— (R)-1-(7-fluoro-3-oxoindan-5-yl)-3-[6-(2,2,2-trifluoroethoxy)pyridin-3-yloxy]pyrrolidin-2-one 1593699-17-2 C20H16F4N2O4
(R)-1-(7-fluoro-3-oxoindan-5-yl)-3-[6-(2,2,2-trifluoroethoxy)pyridin-3-yloxy]pyrrolidin-2-one
—— (R)-3-(6-sec-butoxypyridin-3-yloxy)-1-(7-fluoro-3-oxoindan-5-yl)pyrrolidin-2-one 1593697-88-1 C22H23FN2O4
(R)-3-(6-sec-butoxypyridin-3-yloxy)-1-(7-fluoro-3-oxoindan-5-yl)pyrrolidin-2-one
—— rac-(4aR,8aR)-6-[3-(6-fluoro-1H-benzimidazol-2-yl)-5-(3-fluoro-5-methoxyphenyl)-4-pyridinyl]octahydro-1H-pyrido[3,4-b][1,4]oxazine —— C26H25F2N5O2
rac-(4aR,8aR)-6-[3-(6-fluoro-1H-benzimidazol-2-yl)-5-(3-fluoro-5-methoxyphenyl)-4-pyridinyl]octahydro-1H-pyrido[3,4-b][1,4]oxazine
—— (R)-[2-[[2-amino-7-[4-fluoro-2-(6-methoxypyridin-2-yl)phenyl]-4-methyl-7,8-dihydropyrido[4,3-d]pyrimidin-5-yl]amino]oxyacetyl]-(2-methoxyethyl)-methyl-phenylazanium —— C32H35FN7O4+
(R)-[2-[[2-amino-7-[4-fluoro-2-(6-methoxypyridin-2-yl)phenyl]-4-methyl-7,8-dihydropyrido[4,3-d]pyrimidin-5-yl]amino]oxyacetyl]-(2-methoxyethyl)-methyl-phenylazanium
—— (R)-(-)-dimethyl (3-methyl-2-oxo-6-phenylhexyl)phosphonate 1544280-13-8 C15H23O4P
(R)-(-)-dimethyl (3-methyl-2-oxo-6-phenylhexyl)phosphonate
—— (R)-1-(4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)benzoyl)piperidin-2-carboxamide —— C28H37FN4O3
(R)-1-(4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)benzoyl)piperidin-2-carboxamide
—— (R)-(4-(4-((6-(2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-7-yl)imidazo[1,2-a]pyrazin-8-yl)amino)-2-methoxyphenyl)morpholin-2-yl)methanol —— C25H27N7O4
(R)-(4-(4-((6-(2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-7-yl)imidazo[1,2-a]pyrazin-8-yl)amino)-2-methoxyphenyl)morpholin-2-yl)methanol
—— (RS)-N-(2-hydroxyethyl)-4-[(6-isopropoxy-1H-indazol-5-yl)amino]-N-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxamide —— C24H28N6O3S
(RS)-N-(2-hydroxyethyl)-4-[(6-isopropoxy-1H-indazol-5-yl)amino]-N-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxamide
—— ((R)-4-chloro-2-(4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-4-yl)-phenoxy)-acetic acid ethyl ester hydrochloride —— C16H17ClN2O3S*(x)ClH
((R)-4-chloro-2-(4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-4-yl)-phenoxy)-acetic acid ethyl ester hydrochloride
—— (R)-(3-hydroxypyrrolidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)methanone —— C29H35F3N2O3
(R)-(3-hydroxypyrrolidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)methanone
—— (RS)-N-benzyl-4-chloro-N-[2-(dimethylamino)ethyl]-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxamide —— C22H25ClN4OS
(RS)-N-benzyl-4-chloro-N-[2-(dimethylamino)ethyl]-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxamide
—— (R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-2,3'-difluorobiphenyl-4-yl)(2-(hydroxymethyl)pyrrolidin-1-yl)methanone —— C30H39F3N2O3
(R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-2,3'-difluorobiphenyl-4-yl)(2-(hydroxymethyl)pyrrolidin-1-yl)methanone