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中文名称 英文名称 CAS号 化学式 结构式图片
—— racemic 3-fluoro-4'-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-N-(2,2,2-trifluoro-1-methylethyl)biphenyl-2-sulfonamide —— C21H16F4N4O2S
racemic 3-fluoro-4'-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-N-(2,2,2-trifluoro-1-methylethyl)biphenyl-2-sulfonamide
—— (R)-5-(3-fluoro-2'-((2-methylpiperazin-1-yl)sulfonyl)-[1,1'-biphenyl]-4-yl)pyrazin-2-amine —— C21H22FN5O2S
(R)-5-(3-fluoro-2'-((2-methylpiperazin-1-yl)sulfonyl)-[1,1'-biphenyl]-4-yl)pyrazin-2-amine
—— racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine —— C22H18F4N4O2
racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine
—— racemic (endo)-4′-(5-aminopyrazin-2-yl)-N-bicyclo[2.2.1]hept-2-yl-3′-fluorobiphenyl-2-sulfonamide —— C23H23FN4O2S
racemic (endo)-4′-(5-aminopyrazin-2-yl)-N-bicyclo[2.2.1]hept-2-yl-3′-fluorobiphenyl-2-sulfonamide
—— racemic (4-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}morpholin-2-yl)methanol —— C21H21FN4O4S
racemic (4-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}morpholin-2-yl)methanol
—— racemic [2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]phenyl]-[2-(hydroxymethyl)morpholin-4-yl]methanone —— C22H21FN4O3
racemic [2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]phenyl]-[2-(hydroxymethyl)morpholin-4-yl]methanone
—— (R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-methylpiperazine-1-carboxylate —— C26H30FN5O4S
(R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-methylpiperazine-1-carboxylate
—— (R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-hydroxypropyl)-[1,1'-biphenyl]-2-sulfonamide —— C19H19FN4O3S
(R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-hydroxypropyl)-[1,1'-biphenyl]-2-sulfonamide
—— (R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-hydroxy-2-phenylethyl)-[1,1'-biphenyl]-2-sulfonamide —— C24H21FN4O3S
(R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-hydroxy-2-phenylethyl)-[1,1'-biphenyl]-2-sulfonamide
—— (R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)piperazin-2-yl)methanol —— C21H22FN5O3S
(R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)piperazin-2-yl)methanol
—— rac-tert-butyl 4-(3-isothiocyanatopyridin-4-yl)-trans-2,5-dimethylpiperazine-1-carboxylate —— C17H24N4O2S
rac-tert-butyl 4-(3-isothiocyanatopyridin-4-yl)-trans-2,5-dimethylpiperazine-1-carboxylate
—— (R)-tert-butyl 3-(4-amino-5-bromo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidine-1-carboxylate —— C16H22BrN5O2
(R)-tert-butyl 3-(4-amino-5-bromo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidine-1-carboxylate
—— (R)-2-(1-bromo-8-(2,4-dimethoxybenzylamino)imidazolo[1,5-a]pyrazin-3-yl)morpholine-4-carboxylic acid tert-butyl ester —— C24H30BrN5O5
(R)-2-(1-bromo-8-(2,4-dimethoxybenzylamino)imidazolo[1,5-a]pyrazin-3-yl)morpholine-4-carboxylic acid tert-butyl ester
—— (R)-8-chloro-1-isopropyl-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one —— C11H16ClN3O
(R)-8-chloro-1-isopropyl-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((4-fluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620678-94-5 C16H18FN3O2
(R)-8-((4-fluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-6-isopropyl-5-(2-methoxyphenyl)-2-(3-methyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)nicotinonitrile 1416138-59-4 C27H30N4O2S
(R)-6-isopropyl-5-(2-methoxyphenyl)-2-(3-methyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)nicotinonitrile
—— (R)-tert-butyl(6-(5-cyano-2-cyclopropyl-6-(3-cyclopropyl-4-(3-hydroxypropanoyl)piperazin-1-yl)pyridin-3-yl)pyridazin-4-yl)carbamate —— C28H35N7O4
(R)-tert-butyl(6-(5-cyano-2-cyclopropyl-6-(3-cyclopropyl-4-(3-hydroxypropanoyl)piperazin-1-yl)pyridin-3-yl)pyridazin-4-yl)carbamate
—— (R)-8-((3,4-difluorobenzyl)oxy)-1-isopropyl-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-43-7 C18H21F2N3O2
(R)-8-((3,4-difluorobenzyl)oxy)-1-isopropyl-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((3-fluoro-4-((2-(trifluoromethyl)pyridin-4-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620680-21-8 C22H20F4N4O3
(R)-8-((3-fluoro-4-((2-(trifluoromethyl)pyridin-4-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-N-((2R,3R)-3-Fluoro-2-(2-fluorophenyl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide —— C14H19F2NO2S
(R)-N-((2R,3R)-3-Fluoro-2-(2-fluorophenyl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-8-((3,5-difluoro-4-((2-(trifluoromethyl)pyrimidin-5-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-71-1 C21H18F5N5O3
(R)-8-((3,5-difluoro-4-((2-(trifluoromethyl)pyrimidin-5-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-(dideutero(2,4,5-trifluorophenyl)methoxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620678-97-8 C16H16F3N3O2
(R)-8-(dideutero(2,4,5-trifluorophenyl)methoxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((4-(3,4-difluorophenoxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-75-5 C22H19F4N3O3
(R)-8-((4-(3,4-difluorophenoxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-N-((S)-2-(3-chlorothiophen-2-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide 1620828-05-8 C12H18ClNO2S2
(R)-N-((S)-2-(3-chlorothiophen-2-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-((2R,3R,4R)-5,5,5-trifluoro-2-(2-fluorophenyl)-4-hydroxy-3-(2,2,2-trifluoroethoxy)pentan-2-yl)propane-2-sulfinamide 1620829-29-9 C17H22F7NO3S
(R)-2-methyl-N-((2R,3R,4R)-5,5,5-trifluoro-2-(2-fluorophenyl)-4-hydroxy-3-(2,2,2-trifluoroethoxy)pentan-2-yl)propane-2-sulfinamide
—— (R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429315-61-6 C16H18Cl2N2O4
(R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropyl-[3,3'-bipyridine]-5,5'-dicarbonitrile 1416140-53-8 C26H26N6O
(R)-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropyl-[3,3'-bipyridine]-5,5'-dicarbonitrile
—— (R)-N-(3-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)phenyl)-N-(vinylsulfonyl)ethenesulfonamide 1416140-20-9 C30H33N5O5S2
(R)-N-(3-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)phenyl)-N-(vinylsulfonyl)ethenesulfonamide
—— (R)-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropyl-2'-methyl-3,4'-bipyridine-5-carbonitrile 1416141-54-2 C26H29N5O
(R)-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropyl-2'-methyl-3,4'-bipyridine-5-carbonitrile
—— (R)-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5,6-diphenylnicotinonitrile 1416138-70-9 C27H28N4O2
(R)-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5,6-diphenylnicotinonitrile
—— (R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-4-methyl-5-(4-(trifluoromethoxy)-phenyl)nicotinonitrile 1416138-13-0 C26H29F3N4O3
(R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-4-methyl-5-(4-(trifluoromethoxy)-phenyl)nicotinonitrile
—— (R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5-(quinolin-8-yl)nicotinonitrile 1416139-54-2 C27H29N5O2
(R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5-(quinolin-8-yl)nicotinonitrile
—— (R)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-5-p-tolylnicotinonitrile 1416138-63-0 C26H28N4O2
(R)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-5-p-tolylnicotinonitrile
—— (R)-5-(3-fluorophenyl)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropylnicotinonitrile 1416138-55-0 C25H25FN4O2
(R)-5-(3-fluorophenyl)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropylnicotinonitrile
—— rac-1-(aminomethyl)[2.2]paracyclophane —— C17H19N
rac-1-(aminomethyl)[2.2]paracyclophane
—— (R)-6-isopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5-(3-(trifluoromethoxy)phenyl)nicotinonitrile 1416137-88-6 C25H29F3N4O3
(R)-6-isopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-5-(3-(trifluoromethoxy)phenyl)nicotinonitrile
—— (R)-2-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-5-(4-(trifluoromethyl)phenyl)nicotinonitrile 1416137-53-5 C26H25F3N4O2
(R)-2-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-5-(4-(trifluoromethyl)phenyl)nicotinonitrile
—— (R)-5-(3-aminophenyl)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropylnicotinonitrile 1416147-25-5 C26H29N5O
(R)-5-(3-aminophenyl)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropylnicotinonitrile
—— (R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-4-methyl-5-m-tolylnicotinonitrile 1416138-11-8 C26H32N4O2
(R)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-4-methyl-5-m-tolylnicotinonitrile
—— (R)-4-(3-fluorophenyl)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropylnicotinonitrile 1416139-14-4 C25H25FN4O2
(R)-4-(3-fluorophenyl)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropylnicotinonitrile
—— (R)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-4-o-tolylnicotinonitrile 1416139-16-6 C26H28N4O2
(R)-2-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-6-isopropyl-4-o-tolylnicotinonitrile
—— (R)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-1-(2-phenylpropyl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429314-81-7 C23H24Cl2N2O3
(R)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-1-(2-phenylpropyl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(3-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)phenyl)acrylamide 1416140-22-1 C29H31N5O2
(R)-N-(3-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)phenyl)acrylamide
—— (R)-6-cyclopropyl-2-[4-(3-methoxy-propionyl)-3-methyl-piperazin-1-yl]-5-quinolin-6-yl-nicotinonitrile 1416142-32-9 C27H29N5O2
(R)-6-cyclopropyl-2-[4-(3-methoxy-propionyl)-3-methyl-piperazin-1-yl]-5-quinolin-6-yl-nicotinonitrile
—— (R)-5-(benzo[d]thiazol-6-yl)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropylnicotinonitrile 1416140-50-5 C27H27N5OS
(R)-5-(benzo[d]thiazol-6-yl)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropylnicotinonitrile
—— (R)-5-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)isoquinoline 2-oxide 1416140-02-7 C29H29N5O2
(R)-5-(5-cyano-6-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-2-cyclopropylpyridin-3-yl)isoquinoline 2-oxide
—— (R)-2-cyclopropyl-6-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-6'-vinyl-3,3'-bipyridine-5-carbonitrile 1416141-84-8 C25H29N5O2
(R)-2-cyclopropyl-6-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-6'-vinyl-3,3'-bipyridine-5-carbonitrile
—— (R)-6-cyclopropyl-2-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-5-(2-vinylquinazolin-5-yl)nicotinonitrile 1416141-75-7 C30H32N6O2
(R)-6-cyclopropyl-2-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-5-(2-vinylquinazolin-5-yl)nicotinonitrile
—— (R)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropyl-5-(isoquinolin-5-yl)nicotinonitrile 1416139-76-8 C29H29N5O
(R)-2-(4-(cyclopropanecarbonyl)-3-cyclopropylpiperazin-1-yl)-6-cyclopropyl-5-(isoquinolin-5-yl)nicotinonitrile
—— (R)-5-(3-chloro-4-fluorophenyl)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)nicotinonitrile 1416138-05-0 C24H26ClFN4O2
(R)-5-(3-chloro-4-fluorophenyl)-6-cyclopropyl-2-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)nicotinonitrile