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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-1'-acetyl-5-cyano-N-(5-fluorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C18H16FN5O2S
(R)-1'-acetyl-5-cyano-N-(5-fluorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide
—— (R)-2-methyl-N-[(1S)-1-(2-pyridin-3-yl-2,3-dihydro-1,3-thiazol-5-yl)ethyl]propane-2-sulfinamide —— C14H21N3OS2
(R)-2-methyl-N-[(1S)-1-(2-pyridin-3-yl-2,3-dihydro-1,3-thiazol-5-yl)ethyl]propane-2-sulfinamide
—— (R)-3-(tert-butoxy)-N-(5-chloro-3-cyclobutyl-3H-imidazo[4,5-b]pyridin-2-yl)butanamide —— C18H25ClN4O2
(R)-3-(tert-butoxy)-N-(5-chloro-3-cyclobutyl-3H-imidazo[4,5-b]pyridin-2-yl)butanamide
—— (R)-2-chloro-1-(3-hydroxy-pyrrolidin-1-yl)-ethanone —— C6H10ClNO2
(R)-2-chloro-1-(3-hydroxy-pyrrolidin-1-yl)-ethanone
—— (R)-1-(5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl)ethanamine —— C5H6F3N3O
(R)-1-(5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl)ethanamine
—— (R)-(1-ethylpyrazol-4-yl)-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]methanol —— C22H29N7O2
(R)-(1-ethylpyrazol-4-yl)-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]methanol
—— (R)-2-(2-cyanopropan-2-yl)-N-(4-methyl-3-(4-(3-methylmorpholino)-1H-imidazo[4,5-c]pyridin-6-yl)phenyl)isonicotinamide —— C28H29N7O2
(R)-2-(2-cyanopropan-2-yl)-N-(4-methyl-3-(4-(3-methylmorpholino)-1H-imidazo[4,5-c]pyridin-6-yl)phenyl)isonicotinamide
—— (R/S)-(2-(2H-1,2,3-triazol-2-yl)phenyl)-2-((5-(trifluoromethyl)pyridin-2-yl)oxy)-7-azabicyclo[2.2.1]heptan-7-yl)methanone —— C21H18F3N5O2
(R/S)-(2-(2H-1,2,3-triazol-2-yl)phenyl)-2-((5-(trifluoromethyl)pyridin-2-yl)oxy)-7-azabicyclo[2.2.1]heptan-7-yl)methanone
—— (rac-2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-4-((6-methylpyridin2-yl)amino)-N-(pyrrolidin-3-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide —— C25H33N5O2
(rac-2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-4-((6-methylpyridin2-yl)amino)-N-(pyrrolidin-3-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
—— rac-benzyl ((2S,3R,4R)-1-acetyl-2-cyclopropyl-6-methoxy-3-methyl-1,2,3,4-tetrahydro-1,5-naphthyridin-4-yl)carbamate —— C23H27N3O4
rac-benzyl ((2S,3R,4R)-1-acetyl-2-cyclopropyl-6-methoxy-3-methyl-1,2,3,4-tetrahydro-1,5-naphthyridin-4-yl)carbamate
—— rac-1-((2S,3R,4R)-4-amino-2-cyclopropyl-3-methyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone —— C14H19N3O
rac-1-((2S,3R,4R)-4-amino-2-cyclopropyl-3-methyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone
—— rac-6-(((2S,3R,4R)-1-acetyl-2,3-dimethyl-6-(1,2,3,4-tetrahydropyridin-4-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)nicotinonitrile —— C24H27N5O
rac-6-(((2S,3R,4R)-1-acetyl-2,3-dimethyl-6-(1,2,3,4-tetrahydropyridin-4-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)nicotinonitrile
—— rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-((6-methylpyridin-2-yl)amino)-1,2,3,4-tetrahydroquinolin-6-yl)-5,6-dihydropyridine-1(2H)-carboxylate —— C31H40N4O3
rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-((6-methylpyridin-2-yl)amino)-1,2,3,4-tetrahydroquinolin-6-yl)-5,6-dihydropyridine-1(2H)-carboxylate
—— rac-1-((2S,3R,4R)-4-Amino-2,3-dimethyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone —— C12H17N3O
rac-1-((2S,3R,4R)-4-Amino-2,3-dimethyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-1-acetyl-2,3-dimethyl-4-((6-yl)amino)-N-(tetrahydro-2H-pyran-4-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide —— C25H32N4O3
rac-(2S,3R,4R)-1-acetyl-2,3-dimethyl-4-((6-yl)amino)-N-(tetrahydro-2H-pyran-4-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
—— rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2-cyclopropyl-4-((6-methoxypyridin-2-yl)amino)-3-methyl-1,2,3,4-tetrahydroquinolin-6-yl)-5,6-dihydropyridine-1(2H)-carboxylate —— C31H40N4O4
rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2-cyclopropyl-4-((6-methoxypyridin-2-yl)amino)-3-methyl-1,2,3,4-tetrahydroquinolin-6-yl)-5,6-dihydropyridine-1(2H)-carboxylate
—— rac-1-((2S,3R,4R)-4-Amino-2-cyclopropyl-6-methoxy-3-methyl-3,4-dihydro-1,5-naphthyridin-1(2H)-yl)ethanone —— C15H21N3O2
rac-1-((2S,3R,4R)-4-Amino-2-cyclopropyl-6-methoxy-3-methyl-3,4-dihydro-1,5-naphthyridin-1(2H)-yl)ethanone
—— (R)-7-(4-chlorobenzyl)-1-(2-hydroxypropyl)-3-methyl-8-(3-(trifluoromethoxy)phenoxy)-1H-purine-2,6(3H,7H)-dione —— C23H20ClF3N4O5
(R)-7-(4-chlorobenzyl)-1-(2-hydroxypropyl)-3-methyl-8-(3-(trifluoromethoxy)phenoxy)-1H-purine-2,6(3H,7H)-dione
—— (R)-2-amino-2,5-dimethylhex-4-enoic acid tert-butyl ester —— C12H23NO2
(R)-2-amino-2,5-dimethylhex-4-enoic acid tert-butyl ester
—— rac-(2S,3R,4R)-1-Acetyl-4-(((benzyloxy)carbonyl)amino)-2,3-dimethyl-1,2,3,4-tetra hydro-1,7-naphthyridin-8-yl trifluoromethanesulfonate —— C21H22F3N3O6S
rac-(2S,3R,4R)-1-Acetyl-4-(((benzyloxy)carbonyl)amino)-2,3-dimethyl-1,2,3,4-tetra hydro-1,7-naphthyridin-8-yl trifluoromethanesulfonate
—— rac-(2S,3S,4R)-methyl 2-cyclopropyl-4-(phenylamino)-1,2,3,4-tetrahydroquinoline-3-carboxylate —— C20H22N2O2
rac-(2S,3S,4R)-methyl 2-cyclopropyl-4-(phenylamino)-1,2,3,4-tetrahydroquinoline-3-carboxylate
—— rac-1-((2S,3R,4R)-2-cyclopropyl-3-methyl-4-(phenylamino)-6-(piperazin-1-yl)-3,4-dihydro-1,5-naphthyridin-1(2H)-yl)ethanone —— C24H31N5O
rac-1-((2S,3R,4R)-2-cyclopropyl-3-methyl-4-(phenylamino)-6-(piperazin-1-yl)-3,4-dihydro-1,5-naphthyridin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-1-acetyl-4-amino-2-ethyl-N,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxamide —— C16H23N3O2
rac-(2S,3R,4R)-1-acetyl-4-amino-2-ethyl-N,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxamide
—— (R)-1-[4-[4-[2,5-dimethyl-4-(1-phenylethoxycarbonylamino)pyrazol-3-yl]phenyl]-phenyl]cyclopropane carboxylic acid methyl ester —— C31H31N3O4
(R)-1-[4-[4-[2,5-dimethyl-4-(1-phenylethoxycarbonylamino)pyrazol-3-yl]phenyl]-phenyl]cyclopropane carboxylic acid methyl ester
—— (R)-1-(4-{5-[4-Methyl-5-(1-phenyl-ethoxycarbonylamino)-pyrazol-1-yl]-pyridin-2-yl}-phenyl)-cyclopropanecarboxylic acid methyl ester —— C29H28N4O4
(R)-1-(4-{5-[4-Methyl-5-(1-phenyl-ethoxycarbonylamino)-pyrazol-1-yl]-pyridin-2-yl}-phenyl)-cyclopropanecarboxylic acid methyl ester
—— rac-4-(((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-6-(piperazin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)benzonitrile —— C25H31N5O
rac-4-(((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-6-(piperazin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)benzonitrile
—— rac-1-((2S,3R,4R)-2-cyclopropyl-3-methyl-4-((6-methylpyridin-2-yl)amino)-6-(1,2,3,6-tetrahydropyridin-4-yl)-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C26H32N4O
rac-1-((2S,3R,4R)-2-cyclopropyl-3-methyl-4-((6-methylpyridin-2-yl)amino)-6-(1,2,3,6-tetrahydropyridin-4-yl)-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— (RS)-3-Cyclopropyl-2-{4-[3-methyl-4-((R)-1-phenyl-ethoxycarbonylamino)-isoxazol-5-yl]-benzyloxy}-propionic acid methyl ester —— C27H30N2O6
(RS)-3-Cyclopropyl-2-{4-[3-methyl-4-((R)-1-phenyl-ethoxycarbonylamino)-isoxazol-5-yl]-benzyloxy}-propionic acid methyl ester
—— rac-tert-butyl 4-((6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(Phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl)piperazine-1-carboxylate —— C29H39N5O3
rac-tert-butyl 4-((6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(Phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl)piperazine-1-carboxylate
—— (R)-tert-butyl 3-(3-bromophenoxy)-2-hydroxypropyl(methyl)carbamate —— C15H22BrNO4
(R)-tert-butyl 3-(3-bromophenoxy)-2-hydroxypropyl(methyl)carbamate
—— racemic cis-3-fluoro-4-[4-(4-fluoro-3-methyl-phenyl)-1H-imidazol-2-yl]-piperidine-1-carboxylic acid benzyl ester —— C23H23F2N3O2
racemic cis-3-fluoro-4-[4-(4-fluoro-3-methyl-phenyl)-1H-imidazol-2-yl]-piperidine-1-carboxylic acid benzyl ester
—— racemic cis-3-fluoro-4-[4-(4-fluoro-3-methyl-phenyl)-1H-imidazol-2-yl]-piperidine-1-carboxylic acid tert-butyl ester —— C20H25F2N3O2
racemic cis-3-fluoro-4-[4-(4-fluoro-3-methyl-phenyl)-1H-imidazol-2-yl]-piperidine-1-carboxylic acid tert-butyl ester
—— (R)-1-(3-(4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(5H-pyrrolo[3,4-d]pyrimidin-6(7H)-yl)pyrimidin-2-yl)-4-(trifluoromethyl)phenoxy)-3-(methylamino)propan-2-ol —— C27H28F3N7O3
(R)-1-(3-(4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(5H-pyrrolo[3,4-d]pyrimidin-6(7H)-yl)pyrimidin-2-yl)-4-(trifluoromethyl)phenoxy)-3-(methylamino)propan-2-ol
—— (R)-3-Methyl-2-((methylamino)methyl)butanoic acid —— C7H15NO2
(R)-3-Methyl-2-((methylamino)methyl)butanoic acid
—— racemic cis-3-fluoro-4-{4-(4-fluoro-3-methyl-phenyl)-1-[2-(tetrahydro-pyran-2-yloxy)-ethyl]-1H-imidazol-2-yl}-piperidine-1-carboxylic acid tert-butyl ester —— C27H37F2N3O4
racemic cis-3-fluoro-4-{4-(4-fluoro-3-methyl-phenyl)-1-[2-(tetrahydro-pyran-2-yloxy)-ethyl]-1H-imidazol-2-yl}-piperidine-1-carboxylic acid tert-butyl ester
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2’-(tert-butyl)-[3,4’-bipyridin]-6-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C29H38N6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2’-(tert-butyl)-[3,4’-bipyridin]-6-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-cyclopropyl-4-methyl-3-(2-(((R)-1-(4-((3,3,4-trimethylpiperazin-1-yl)methyl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C27H38N6O2
(R)-4-cyclopropyl-4-methyl-3-(2-(((R)-1-(4-((3,3,4-trimethylpiperazin-1-yl)methyl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-tert-butyl 4-(4-(5-fluoro-2-methoxyphenyl)-1-tosyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-methyl-5,6-dihydropyridine-1(2H)-carboxylate —— C32H34FN3O5S
(R)-tert-butyl 4-(4-(5-fluoro-2-methoxyphenyl)-1-tosyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-methyl-5,6-dihydropyridine-1(2H)-carboxylate
—— (R)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)-8-methylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone —— C30H36FN7O2S
(R)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)-8-methylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone
—— (R)-tert-butyl 4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-(hydroxymethyl)-5,6-dihydropyridine-1(2H)-carboxylate —— C25H28FN3O4
(R)-tert-butyl 4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-(hydroxymethyl)-5,6-dihydropyridine-1(2H)-carboxylate
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H26F4N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H25F5N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H27F3N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(trifluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(4-(difluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H27ClF2N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(4-(difluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(difluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H28F2N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(difluoromethoxy)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2,5-difluoropyrimidin-4-yl)-4-((S)-1-hydroxyethyl)oxazolidin-2-one —— C9H9F2N3O3
(R)-3-(2,5-difluoropyrimidin-4-yl)-4-((S)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl)piperidin-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C29H41F3N6O3
(R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl)piperidin-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-isobutoxyphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H36N4O4
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-isobutoxyphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((R)-1-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H18ClF3N6O5
(R)-3-(2-(((R)-1-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(6-chloro-2-(((S)-1-(5-phenylthiophen-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C21H21ClN4O3S
(R)-3-(6-chloro-2-(((S)-1-(5-phenylthiophen-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one