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—— (R)-tert-butyl 3-(2-((1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-2,2-dimethylbut-3-en-1-yl)carbamoyl)phenoxy)azetidine-1-carboxylate —— C37H40F2N4O4
(R)-tert-butyl 3-(2-((1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-2,2-dimethylbut-3-en-1-yl)carbamoyl)phenoxy)azetidine-1-carboxylate
—— (R)-4-(5-bromo-2-ethoxypyridin-3-yl)-3-methylmorpholine —— C12H17BrN2O2
(R)-4-(5-bromo-2-ethoxypyridin-3-yl)-3-methylmorpholine
—— (R)-1-((6-(5-amino-2-methylphenyl)-2-morpholinopyrimidin-4-yl)amino)propan-2-ol —— C18H25N5O2
(R)-1-((6-(5-amino-2-methylphenyl)-2-morpholinopyrimidin-4-yl)amino)propan-2-ol
—— (R)-N-(6'-((1-methoxypropan-2-yl)oxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide —— C27H29F3N4O4
(R)-N-(6'-((1-methoxypropan-2-yl)oxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide
—— (R)-6-chloro-2-methyl-4-(3-methylmorpholino)pyridazin-3(2H)-one —— C10H14ClN3O2
(R)-6-chloro-2-methyl-4-(3-methylmorpholino)pyridazin-3(2H)-one
—— (R)-3-(6-chloro-2-(((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-methoxyethyl)oxazolidin-2-one —— C19H19ClF4N4O3
(R)-3-(6-chloro-2-(((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-methoxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3,5-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C21H25F3N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3,5-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-chloro-2-(((S)-1-(5-(2-(trifluoromethyl)pyridin-4-yl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C25H27ClF3N7O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-chloro-2-(((S)-1-(5-(2-(trifluoromethyl)pyridin-4-yl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(1,1-difluoroethyl)-2-fluorophenyl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C24H31F3N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(1,1-difluoroethyl)-2-fluorophenyl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(4-fluoro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20F4N6O3
(R)-3-(2-((1-(5-(4-fluoro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-2-methyl-N-((S)-1-(5-phenylthiophen-2-yl)ethyl)propane-2-sulfinamide —— C16H21NOS2
(R)-2-methyl-N-((S)-1-(5-phenylthiophen-2-yl)ethyl)propane-2-sulfinamide
—— (R)-N-((S)-1-(5-(4-fluorophenyl)isoxazol-3-yl)ethyl)-2-methylpropane-2-sulfinamide —— C15H19FN2O2S
(R)-N-((S)-1-(5-(4-fluorophenyl)isoxazol-3-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-imidazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C25H31ClN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-imidazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-N-((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)-2-methylpropane-2-sulfinamide —— C15H19ClN2OS2
(R)-N-((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C24H29ClN6O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-2-methyl-N-((S)-1-(5-phenylisoxazol-3-yl)ethyl)propane-2-sulfinamide —— C15H20N2O2S
(R)-2-methyl-N-((S)-1-(5-phenylisoxazol-3-yl)ethyl)propane-2-sulfinamide
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(4-(1-ethoxycyclopropyl)-2-fluorophenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C26H35FN4O4
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(4-(1-ethoxycyclopropyl)-2-fluorophenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C22H26F4N4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-{2-[1-(5-pyridin-3-yl-[1,3,4]-oxadiazol-2-yl)ethylamino]pyrimidin-4-yl}oxazolidin-2-one —— C18H19N7O4
(R)-4-((R)-1-hydroxyethyl)-3-{2-[1-(5-pyridin-3-yl-[1,3,4]-oxadiazol-2-yl)ethylamino]pyrimidin-4-yl}oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C24H29FN6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H33ClN6O5
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H28Cl2N6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R,E)-2-methyl-N-((2-(6-(trifluoromethyl)pyridin-3-yl)thiazol-5-yl)methylene)propane-2-sulfinamide —— C14H14F3N3OS2
(R,E)-2-methyl-N-((2-(6-(trifluoromethyl)pyridin-3-yl)thiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-di-tert-butyl 2-((3-(5-(methoxycarbonyl)-thiophen-2-yl)prop-2-yn-1-yl)amino)pentanedioate —— C22H31NO6S
(R)-di-tert-butyl 2-((3-(5-(methoxycarbonyl)-thiophen-2-yl)prop-2-yn-1-yl)amino)pentanedioate
—— (R)-1-(3-(5-(methoxycarbonyl)thiophen-2-yl)prop-2-yn-1-yl)-5-oxopyrrolidine-2-carboxylic acid —— C14H13NO5S
(R)-1-(3-(5-(methoxycarbonyl)thiophen-2-yl)prop-2-yn-1-yl)-5-oxopyrrolidine-2-carboxylic acid
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(o-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C20H22N6O4
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(o-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-isopropylphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C24H32F2N4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-isopropylphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-{1-[3-(3,4-difluorophenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H18F2N6O4
(R)-3-(2-{1-[3-(3,4-difluorophenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-chlorophenyl)-1,3,4-thiadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H26Cl2N6O3S
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-chlorophenyl)-1,3,4-thiadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C24H27ClFN5O3S
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(3-(4-chlorophenyl)isoxazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H27Cl2N5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(3-(4-chlorophenyl)isoxazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-imidazol-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-(fluoromethyl)oxazolidin-2-one —— C19H17ClF2N6O2
(R)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-imidazol-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-(fluoromethyl)oxazolidin-2-one
—— (R)-3-(2-((1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19ClN6O4
(R)-3-(2-((1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H33ClN6O5
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-3-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C25H31ClN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-3-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethanamine —— C10H17N3O2
(R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethanamine
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-phenylisoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H28ClN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-phenylisoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H27Cl2N7O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-(R)-(1-hydroxyethyl)oxazolidin-2-one —— C20H18ClF3N6O5
(R)-3-(2-((1-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-(R)-(1-hydroxyethyl)oxazolidin-2-one
—— (R)-methyl 5-(3-(2-(hydroxymethyl)-5-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate —— C14H15NO4S
(R)-methyl 5-(3-(2-(hydroxymethyl)-5-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2-(4-(difluoromethyl)phenyl)thiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C25H29F2N5O3S
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2-(4-(difluoromethyl)phenyl)thiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1-methylcyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H32F2N4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1-methylcyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R,E)-2-methyl-N-((5-(pyridin-2-yl)thiophen-2-yl)methylene)propane-2-sulfinamide —— C14H16N2OS2
(R,E)-2-methyl-N-((5-(pyridin-2-yl)thiophen-2-yl)methylene)propane-2-sulfinamide
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C24H28ClFN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C24H30ClN7O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-5-chloro-N1'-methyl-N1-(5-methylthiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C18H20ClN5O2S
(R)-5-chloro-N1'-methyl-N1-(5-methylthiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-5-cyano-N1-(5-methoxythiazol-2-yl)-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C19H20N6O3S
(R)-5-cyano-N1-(5-methoxythiazol-2-yl)-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-t-butyl 5-bromospiro[indoline-3,3'-pyrrolidine]-1'-carboxylate —— C16H21BrN2O2
(R)-t-butyl 5-bromospiro[indoline-3,3'-pyrrolidine]-1'-carboxylate
—— (R)-N1-(5-Fluorothiazol-2-yl)-N1'-methyl-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C18H17F4N5O2S
(R)-N1-(5-Fluorothiazol-2-yl)-N1'-methyl-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-5-chloro-N-(5-chlorothiazol-2-yl)-1'-formyl spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C16H14Cl2N4O2S
(R)-5-chloro-N-(5-chlorothiazol-2-yl)-1'-formyl spiro[indoline-3,3'-pyrrolidine]-1-carboxamide