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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-N'-(4-cyanophenyl)-3-(1-(4-cyanophenyl)ethoxy)benzimidamide hydrochloride 1616242-08-0 C23H18N4O*ClH
(R)-N'-(4-cyanophenyl)-3-(1-(4-cyanophenyl)ethoxy)benzimidamide hydrochloride
—— (R)-3-(N-(4-(1-aminoethyl)phenyl)-N-methylsulfamoyl)-N-(4-cyanophenyl)-benzamide 1616338-14-7 C23H22N4O3S
(R)-3-(N-(4-(1-aminoethyl)phenyl)-N-methylsulfamoyl)-N-(4-cyanophenyl)-benzamide
—— (R)-N-(4-acetylphenyl)-3-(1-(4-acetylphenyl)ethoxy)benzamide 1616243-07-2 C25H23NO4
(R)-N-(4-acetylphenyl)-3-(1-(4-acetylphenyl)ethoxy)benzamide
—— (R)-3,4-Dimethyl-cyclohexanone —— C8H14O
(R)-3,4-Dimethyl-cyclohexanone
—— (R)-6-((1-cyclobutylethyl)amino)-7-((4-methylenecyclohexyl)methyl)-7H-purine-2-carbonitrile 1621912-16-0 C20H26N6
(R)-6-((1-cyclobutylethyl)amino)-7-((4-methylenecyclohexyl)methyl)-7H-purine-2-carbonitrile
—— (R)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)piperidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-53-8 C22H25F3N6O3S
(R)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)piperidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-4-(2-acrylamidophenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide 1622001-76-6 C26H27N7O5
(R)-4-(2-acrylamidophenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide
—— rel-(3aR,5R)-5-(5-methyl pyrazin-2-yl)-3,3a,4,5-tetrahydro-7H-pyrano[3,4-c][1,2]oxazole —— C11H13N3O2
rel-(3aR,5R)-5-(5-methyl pyrazin-2-yl)-3,3a,4,5-tetrahydro-7H-pyrano[3,4-c][1,2]oxazole
—— (R)-1-ethyl-4-hydroxy-5-oxo-N-(4-phenyl-2,3 dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429345-48-1 C22H22N2O3
(R)-1-ethyl-4-hydroxy-5-oxo-N-(4-phenyl-2,3 dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-1-ethyl-4-hydroxy-5-oxo-N-(6-(trifluoromethyl)-2,3-dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-81-9 C17H17F3N2O3
(R)-1-ethyl-4-hydroxy-5-oxo-N-(6-(trifluoromethyl)-2,3-dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(3'-fluorobiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-35-3 C20H19FN2O3
(R)-N-(1-(3'-fluorobiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-4-hydroxy-1-methyl-5-oxo-N-(1-(3'-(trimethylsilyl)biphenyl-3-yl)ethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-50-2 C23H28N2O3Si
(R)-4-hydroxy-1-methyl-5-oxo-N-(1-(3'-(trimethylsilyl)biphenyl-3-yl)ethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(3-(2,4-dimethylthiazol-5-yl)phenyl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-59-1 C19H21N3O3S
(R)-N-(1-(3-(2,4-dimethylthiazol-5-yl)phenyl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(2’,6’-dimethylbiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-48-8 C22H24N2O3
(R)-N-(1-(2’,6’-dimethylbiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-1-ethyl-4-hydroxy-5-oxo-N-(6-phenyl-2,3-dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429345-50-5 C22H22N2O3
(R)-1-ethyl-4-hydroxy-5-oxo-N-(6-phenyl-2,3-dihydro-1H-inden-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-4-(2-acrylamidophenoxy)-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide 1622001-73-3 C26H28N6O5
(R)-4-(2-acrylamidophenoxy)-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide
—— (R)-4-hydroxy-1-methyl-5-oxo-N-(1-(2’-(trifluoromethoxy)biphenyl-3-yl)ethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-41-1 C21H19F3N2O4
(R)-4-hydroxy-1-methyl-5-oxo-N-(1-(2’-(trifluoromethoxy)biphenyl-3-yl)ethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(4’-fluoro-2’-hydroxybiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-53-5 C20H19FN2O4
(R)-N-(1-(4’-fluoro-2’-hydroxybiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(4'-(acetamidomethyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-47-7 C23H25N3O4
(R)-N-(1-(4'-(acetamidomethyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(4’-(N-cyclopropylsulfamoyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-56-8 C23H25N3O5S
(R)-N-(1-(4’-(N-cyclopropylsulfamoyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-4-hydroxy-1-methyl-N-(1-(3-(1-methyl-1H-imidazol-5-yl)phenyl)ethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-60-4 C18H20N4O3
(R)-4-hydroxy-1-methyl-N-(1-(3-(1-methyl-1H-imidazol-5-yl)phenyl)ethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-tert-butyl (1-((2-bromophenyl)sulfonyl)pyrrolidin-3-yl)carbamate —— C15H21BrN2O4S
(R)-tert-butyl (1-((2-bromophenyl)sulfonyl)pyrrolidin-3-yl)carbamate
—— (R)-5-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5'-ethoxy-1",2",3",6"-tetrahydro-[3,3':6',4"-terpyridin]-6-amine —— C25H25Cl2FN4O2
(R)-5-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5'-ethoxy-1",2",3",6"-tetrahydro-[3,3':6',4"-terpyridin]-6-amine
—— (R)-4-(1-(1-2,5,8,11-tetraoxatetradecanepiperidin-3-yl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419216-94-6 C33H39F3N8O6
(R)-4-(1-(1-2,5,8,11-tetraoxatetradecanepiperidin-3-yl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— racemic tert-butyl (1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}piperidin-3-yl)carbamate —— C26H30FN5O4S
racemic tert-butyl (1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}piperidin-3-yl)carbamate
—— (R)-4-(4-amino-7-(piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419216-88-8 C23H21F3N8O
(R)-4-(4-amino-7-(piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(4-amino-7-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419216-91-3 C28H27F3N8O3
(R)-4-(4-amino-7-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(4-amino-7-(1-(2-fluoro-2-methylpropanoyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419216-87-7 C27H26F4N8O2
(R)-4-(4-amino-7-(1-(2-fluoro-2-methylpropanoyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(3-(1-2,5,8,11,14,17,20,23-octaoxahexacosanepiperidin-3-yl)-8-aminoimidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419214-46-2 C42H56F3N7O10
(R)-4-(3-(1-2,5,8,11,14,17,20,23-octaoxahexacosanepiperidin-3-yl)-8-aminoimidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(4-amino-7-(1-(3-ethoxypropanoyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419216-89-9 C28H29F3N8O3
(R)-4-(4-amino-7-(1-(3-ethoxypropanoyl)piperidin-3-yl)imidazo[1,5-f][1,2,4]triazin-5-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-(4-chlorophenyl)-[5-(2-chloropyridin-4-yl)-2-(1H-imidazol-2-yl)thiophen-3-yl]methanol —— C19H13Cl2N3OS
(R)-(4-chlorophenyl)-[5-(2-chloropyridin-4-yl)-2-(1H-imidazol-2-yl)thiophen-3-yl]methanol
—— (R)-2-((R)-4-(1-(1-(difluoromethyl)-6-oxo-1,6-dihydropyridin-3-yl)-4-fluoro-1H-pyrazol-3-yl)-3-oxomorpholin-2-yl)-2-methyl-2-hydroxyacetic acid 1621526-10-0 C16H15F3N4O6
(R)-2-((R)-4-(1-(1-(difluoromethyl)-6-oxo-1,6-dihydropyridin-3-yl)-4-fluoro-1H-pyrazol-3-yl)-3-oxomorpholin-2-yl)-2-methyl-2-hydroxyacetic acid
—— (R)-8-benzyl-6-((1-cyclobutylethyl)amino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylic acid —— C27H26F3N5O2
(R)-8-benzyl-6-((1-cyclobutylethyl)amino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylic acid
—— (R)-2-((R)-4-(1-(1-(difluoromethyl)-6-oxo-1,6-dihydropyridin-3-yl)-1H-pyrazol-3-yl)-3-oxomorpholin-2-yl)-2-hydroxypropanoic acid 1621525-83-4 C16H16F2N4O6
(R)-2-((R)-4-(1-(1-(difluoromethyl)-6-oxo-1,6-dihydropyridin-3-yl)-1H-pyrazol-3-yl)-3-oxomorpholin-2-yl)-2-hydroxypropanoic acid
—— (R)-6-((1-cyclobutylethyl)amino)-8-(4-cyclopropyl-2-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile —— C30H29F3N6
(R)-6-((1-cyclobutylethyl)amino)-8-(4-cyclopropyl-2-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile
—— (R)-methyl 6-((1-cyclobutylethyl)amino)-8-(methylamino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate —— C22H25F3N6O2
(R)-methyl 6-((1-cyclobutylethyl)amino)-8-(methylamino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate
—— (R)-6-((1-cyclobutylethyl)amino)-8-(phenoxymethyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile —— C27H25F3N6O
(R)-6-((1-cyclobutylethyl)amino)-8-(phenoxymethyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile
—— (r)-7-(4-Chlorobenzyl)-6-((1-cyclopropylethyl) amino)-8-(2-(3-methoxypropoxy)-5-methylphenyl)-7h-purine-2-carboxylic acid —— C29H32ClN5O4
(r)-7-(4-Chlorobenzyl)-6-((1-cyclopropylethyl) amino)-8-(2-(3-methoxypropoxy)-5-methylphenyl)-7h-purine-2-carboxylic acid
—— (R)-methyl 6-((1-cyclobutyl-4-((methylsulfonyl)oxy)butyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate —— C31H34F3N5O5S
(R)-methyl 6-((1-cyclobutyl-4-((methylsulfonyl)oxy)butyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate
—— (R)-methyl 6-((1-cyclobutylethyl)amino)-8-(3-methoxyphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate 1621222-52-3 C28H28F3N5O3
(R)-methyl 6-((1-cyclobutylethyl)amino)-8-(3-methoxyphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate
—— (R)-methyl 4-cyclobutyl-4-((8-(4-isopropylpyridin-2-yl)-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-yl)amino)butanoate —— C30H33F3N6O2
(R)-methyl 4-cyclobutyl-4-((8-(4-isopropylpyridin-2-yl)-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-yl)amino)butanoate
—— (r)-8-(2-(3-(Bis(2-methoxyethyl)amino) propoxy)-5-methyl-phenyl)-7-(4-chlorobenzyl)-6-((1-cyclopropylethyl)amino)-7h-purine-2-carboxylic acid —— C34H43ClN6O5
(r)-8-(2-(3-(Bis(2-methoxyethyl)amino) propoxy)-5-methyl-phenyl)-7-(4-chlorobenzyl)-6-((1-cyclopropylethyl)amino)-7h-purine-2-carboxylic acid
—— (RS)-7-ethyl-4-hydroxy-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxylic acid —— C13H14N2O3S
(RS)-7-ethyl-4-hydroxy-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carboxylic acid
—— (R)-methyl 6-((1-cyclobutyl-4-(dimethylamino)butyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate —— C32H37F3N6O2
(R)-methyl 6-((1-cyclobutyl-4-(dimethylamino)butyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate
—— (R)-N-(4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)-2-chloro-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-amine —— C34H43ClF3N5OSi
(R)-N-(4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)-2-chloro-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-amine
—— (r)-7-(4-Chlorobenzyl)-6-((1-cyclopropylethyl) amino)-8-(2-(2-methoxyethoxy)-5-methylphenyl)-7h-purine-2-carboxylic acid —— C28H30ClN5O4
(r)-7-(4-Chlorobenzyl)-6-((1-cyclopropylethyl) amino)-8-(2-(2-methoxyethoxy)-5-methylphenyl)-7h-purine-2-carboxylic acid
—— (R)-methyl 6-((4-amino-1-cyclobutyl-4-oxobutyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate —— C30H31F3N6O3
(R)-methyl 6-((4-amino-1-cyclobutyl-4-oxobutyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carboxylate
—— (R)-4-((2-chloro-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-yl)amino)-4-cyclobutylbutanoic acid —— C21H21ClF3N5O2
(R)-4-((2-chloro-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-yl)amino)-4-cyclobutylbutanoic acid
—— (R)-[(4S)-4-[amino-(3-aminopiperazin-2-yl)methyl]cyclohexa-1,5-dien-1-yl]-[[4-(trifluoromethyl)-1,2-dihydropyridin-2-yl]amino]methanol —— C18H27F3N6O
(R)-[(4S)-4-[amino-(3-aminopiperazin-2-yl)methyl]cyclohexa-1,5-dien-1-yl]-[[4-(trifluoromethyl)-1,2-dihydropyridin-2-yl]amino]methanol
—— (R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-oxopiperidin-3-yl)biphenyl-2-sulfonamide —— C21H20FN5O3S
(R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(2-oxopiperidin-3-yl)biphenyl-2-sulfonamide