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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-2-(3-fluoropyrrolidin-1-yl)[1,2,4]triazolo[1,5-a]pyridin-7-amine —— C10H12FN5
(R)-2-(3-fluoropyrrolidin-1-yl)[1,2,4]triazolo[1,5-a]pyridin-7-amine
—— (R)-N-(2-(3-fluoropyrrolidin-1-yl)[1,2,4]triazolo[1,5-a]pyridin-7-yl)-1-methyl-4-(4-(trifluoromethyl)thiazol-2-yl)-1H-pyrazol-5-carboxamide —— C19H16F4N8OS
(R)-N-(2-(3-fluoropyrrolidin-1-yl)[1,2,4]triazolo[1,5-a]pyridin-7-yl)-1-methyl-4-(4-(trifluoromethyl)thiazol-2-yl)-1H-pyrazol-5-carboxamide
—— (R)-N-[(2S,4Z)-2-(2,3-difluorophenyl)-4-(dimethylhydrazinylidene)-1,5,5,5-tetrafluoropentan-2-yl]-2-methylpropane-2-sulfinamide —— C17H23F6N3OS
(R)-N-[(2S,4Z)-2-(2,3-difluorophenyl)-4-(dimethylhydrazinylidene)-1,5,5,5-tetrafluoropentan-2-yl]-2-methylpropane-2-sulfinamide
—— (R,E)-N-(1-(5-bromo-2-fluorophenyl)-2-fluoroethylidene)-2-methylpropane-2-sulfinamide —— C12H14BrF2NOS
(R,E)-N-(1-(5-bromo-2-fluorophenyl)-2-fluoroethylidene)-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-2-(5-bromo-2-fluoropyridin-3-yl)-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide —— C13H20BrFN2O2S
(R)-N-[(2S)-2-(5-bromo-2-fluoropyridin-3-yl)-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-[(2R,3S)-1,3,4-tributoxybutan-2-yl]oxymethanol —— C23H40N4O5
(R)-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-[(2R,3S)-1,3,4-tributoxybutan-2-yl]oxymethanol
—— (R)-3-{2-[4-(4-CHLORo-PHENYL)-PIperazin-1-YL]-5-OXO-6,7-DIHYDRO-5H-5λ4-THIENO[3,2-d]PYRIMIDIN-4-YLAMINO}-PYRROLIDIN-1-carboxylic acid-tert-BUTYLESTER —— C25H33ClN6O3S
(R)-3-{2-[4-(4-CHLORo-PHENYL)-PIperazin-1-YL]-5-OXO-6,7-DIHYDRO-5H-5λ4-THIENO[3,2-d]PYRIMIDIN-4-YLAMINO}-PYRROLIDIN-1-carboxylic acid-tert-BUTYLESTER
—— (R)-2-phenyl-5-azidopentane —— C11H15N3
(R)-2-phenyl-5-azidopentane
—— (R)-3-(2-chloro-4-(5-(1,2-dihydroxyethyl)-1,3,4-oxadiazol-2-yl)phenyl)-N-(3-chloro-4-(trifluoromethyl)phenyl)propiolamide 1412944-69-4 C20H12Cl2F3N3O4
(R)-3-(2-chloro-4-(5-(1,2-dihydroxyethyl)-1,3,4-oxadiazol-2-yl)phenyl)-N-(3-chloro-4-(trifluoromethyl)phenyl)propiolamide
—— (R)-2-(6-chloro-5-methylpyridin-3-yl)-5-(2,2-dimethyl-1,3-dioxolan-4-yl)-1,3,4-oxadiazole —— C13H14ClN3O3
(R)-2-(6-chloro-5-methylpyridin-3-yl)-5-(2,2-dimethyl-1,3-dioxolan-4-yl)-1,3,4-oxadiazole
—— (R)-2-(4-(4-cyanophenyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-1,2,5,6,7,8-hexahydroquinazolin-3(4H)-yl)-N,N-dimethylacetamide 1625670-24-7 C26H23F3N4O3
(R)-2-(4-(4-cyanophenyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-1,2,5,6,7,8-hexahydroquinazolin-3(4H)-yl)-N,N-dimethylacetamide
—— (R)-N-[(2S,4R)-2-(5-bromo-2-fluorophenyl)-1,5,5,5-tetrafluoro-4-hydroxypentan-2-yl]-2-methylpropane-2-sulfinamide —— C15H19BrF5NO2S
(R)-N-[(2S,4R)-2-(5-bromo-2-fluorophenyl)-1,5,5,5-tetrafluoro-4-hydroxypentan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-((4S)-2-(2,3-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide —— C15H20F5NO2S
(R)-N-((4S)-2-(2,3-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-(2-(3-bromophenyl)-1,5,5,5-tetrafluoro-4-oxopentan-2-yl)-2-methylpropane-2-sulfinamide —— C15H18BrF4NO2S
(R)-N-(2-(3-bromophenyl)-1,5,5,5-tetrafluoro-4-oxopentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-[2-(3-chloro-2-fluorophenyl)-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide —— C14H21ClFNO2S
(R)-N-[2-(3-chloro-2-fluorophenyl)-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-((S)-2-(3-bromophenyl)-1,5,5,5-tetrafluoro-4-oxopentan-2-yl)-2-methylpropane-2-sulfinamide —— C15H18BrF4NO2S
(R)-N-((S)-2-(3-bromophenyl)-1,5,5,5-tetrafluoro-4-oxopentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-1-(2,5-bis(trifluoromethyl)phenyl)ethyl methanesulfonate —— C11H10F6O3S
(R)-1-(2,5-bis(trifluoromethyl)phenyl)ethyl methanesulfonate
—— (R)-N-(2-(3-chloro-2-fluorophenyl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide —— C14H21ClFNO2S
(R)-N-(2-(3-chloro-2-fluorophenyl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-(2-(2,3-difluorophenyl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide —— C14H21F2NO2S
(R)-N-(2-(2,3-difluorophenyl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-ethyl 2-((2S,3R,6S)-2,3-bis(4-chlorophenyl)-5-oxo-6-(4-((trifluoromethyl)sulfonyl)benzyl)morpholino)pentanoate —— C31H30Cl2F3NO6S
(R)-ethyl 2-((2S,3R,6S)-2,3-bis(4-chlorophenyl)-5-oxo-6-(4-((trifluoromethyl)sulfonyl)benzyl)morpholino)pentanoate
—— (R)-N-[(2R,3S)-2-(5-bromo-2-fluorophenyl)-1,1,3-trifluoro-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide —— C14H18BrF4NO2S
(R)-N-[(2R,3S)-2-(5-bromo-2-fluorophenyl)-1,1,3-trifluoro-4-hydroxybutan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-[(2R)-5-[(4-methylphenyl)methyl]-3,4-dihydro-2H-pyrrol-2-yl]-phenylmethanol —— C19H21NO
(R)-[(2R)-5-[(4-methylphenyl)methyl]-3,4-dihydro-2H-pyrrol-2-yl]-phenylmethanol
—— (R)-4-amino-6-(5-(5-methyl-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4,5-dihydro-1H-pyrazol-1-yl)pyrimidine-5-carbonitrile —— C23H18N8O
(R)-4-amino-6-(5-(5-methyl-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4,5-dihydro-1H-pyrazol-1-yl)pyrimidine-5-carbonitrile
—— (R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]piperidine-3-carboxylic acid —— C28H31Cl2N3O3
(R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]piperidine-3-carboxylic acid
—— (R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-3-hydroxy-1-isobutyl-2-oxo-1,2-dihydroquinoline-4-carboxamide 1429186-13-9 C24H26Cl2N2O4
(R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-3-hydroxy-1-isobutyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— (R)-1-bromo-3-(4-methoxy-3-methylphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-17-8 C16H19BrN2O2
(R)-1-bromo-3-(4-methoxy-3-methylphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
——  (R)-N-(1-(3-(4-ethylpiperazin-1-yl)phenyl)ethyl)-3-hydroxy-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide 1429187-47-2 C25H30N4O3
 (R)-N-(1-(3-(4-ethylpiperazin-1-yl)phenyl)ethyl)-3-hydroxy-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— (R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]piperidine-3-carboxylic acid ethyl ester —— C30H35Cl2N3O3
(R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]piperidine-3-carboxylic acid ethyl ester
—— (R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]pyrrolidine-3-carboxylic acid methyl ester —— C28H31Cl2N3O3
(R)-1-[1-chloro-6-(3-chloro-1-isopropyl-1H-indazol-5-ylmethoxy)-3,4-dihydronaphthalen-2-ylmethyl]pyrrolidine-3-carboxylic acid methyl ester
——  (R)-3-hydroxy-1-methyl-2-oxo-N-(1-(3-(4-phenylpiperidin-1-yl)phenyl)ethyl)-1,2-dihydroquinoline-4-carboxamide 1429187-45-0 C30H31N3O3
 (R)-3-hydroxy-1-methyl-2-oxo-N-(1-(3-(4-phenylpiperidin-1-yl)phenyl)ethyl)-1,2-dihydroquinoline-4-carboxamide
—— (R)-1-bromo-3-(4-ethyl-3-methoxyphenyl)-6-methyl-5,6,8,9,-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-06-5 C17H21BrN2O2
(R)-1-bromo-3-(4-ethyl-3-methoxyphenyl)-6-methyl-5,6,8,9,-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-(4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)pyridin-2-yl)methanol 1623764-29-3 C21H22ClN3O3
(R)-(4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)pyridin-2-yl)methanol
——  (R)-3-hydroxy-N-(1-(3-(4-hydroxy-4-phenylpiperidin-1-yl)phenyl)-ethyl)-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide 1429187-44-9 C30H31N3O4
 (R)-3-hydroxy-N-(1-(3-(4-hydroxy-4-phenylpiperidin-1-yl)phenyl)-ethyl)-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— (R)-1-bromo-3-(3-chloro-4-(difluoromethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-23-6 C15H14BrClF2N2O2
(R)-1-bromo-3-(3-chloro-4-(difluoromethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-(5-(6-methyl-1-(2-methylpyridin-4-yl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-3-yl)-2-(trifluoromethoxy)phenyl)methanol 1623766-14-2 C22H22F3N3O3
(R)-(5-(6-methyl-1-(2-methylpyridin-4-yl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-3-yl)-2-(trifluoromethoxy)phenyl)methanol
——  (R)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydroquinoline-4-carboxamide 1429187-17-6 C21H20N2O3
 (R)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydroquinoline-4-carboxamide
—— (R)-4-(2,4-dimethoxybenzyl)-2-ethyl-1,4-oxazepan-5-one 1623766-51-7 C16H23NO4
(R)-4-(2,4-dimethoxybenzyl)-2-ethyl-1,4-oxazepan-5-one
—— (R)-methyl 3-(4-ethyl-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine-1-carboxylate —— C19H24N2O4
(R)-methyl 3-(4-ethyl-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine-1-carboxylate
—— (R)-2-ethyl-5-methoxy-2,3,6,7-tetrahydro-1,4-oxazepine 1623766-53-9 C8H15NO2
(R)-2-ethyl-5-methoxy-2,3,6,7-tetrahydro-1,4-oxazepine
—— rel-5-{[(3S,4S)-4-amino-1,1-dioxidotetrahydro-2H-thiopyran-3-yl]amino}-3-[(4-methoxy-6-methylpyridin-2-yl)amino]pyridine-2-carbonitrile —— C18H22N6O3S
rel-5-{[(3S,4S)-4-amino-1,1-dioxidotetrahydro-2H-thiopyran-3-yl]amino}-3-[(4-methoxy-6-methylpyridin-2-yl)amino]pyridine-2-carbonitrile
—— (R)-4-(2,4-dimethoxybenzyl)-2-ethyl-3,4-dihydro-1,4-oxazepin-5(2H)-one 1623766-50-6 C16H21NO4
(R)-4-(2,4-dimethoxybenzyl)-2-ethyl-3,4-dihydro-1,4-oxazepin-5(2H)-one
—— (R)-methyl 3-(4-bromo-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine-1-carboxylate —— C17H19BrN2O4
(R)-methyl 3-(4-bromo-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine-1-carboxylate
—— (R)-1-bromo-6-methyl-3-(3-methyl-4-(trifluoromethoxy)phenyl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-02-1 C16H16BrF3N2O2
(R)-1-bromo-6-methyl-3-(3-methyl-4-(trifluoromethoxy)phenyl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-N-[(1S)-1-(2,5-difluoro-4-propan-2-ylphenyl)ethyl]-2-methylpropane-2-sulfinamide —— C15H23F2NOS
(R)-N-[(1S)-1-(2,5-difluoro-4-propan-2-ylphenyl)ethyl]-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-[(1S)-1-[4-(1-methylpyrazol-4-yl)phenyl]ethyl]propane-2-sulfinamide —— C16H23N3OS
(R)-2-methyl-N-[(1S)-1-[4-(1-methylpyrazol-4-yl)phenyl]ethyl]propane-2-sulfinamide
—— (R)-2-methyl-N-[(1S)-1-[6-(1-methylcyclopropyl)pyridin-3-yl]ethyl]propane-2-sulfinamide —— C15H24N2OS
(R)-2-methyl-N-[(1S)-1-[6-(1-methylcyclopropyl)pyridin-3-yl]ethyl]propane-2-sulfinamide
—— (R)-N-(4-acetylphenyl)-5-(1-(4-acetylphenyl)ethoxy)nicotinamide 1616243-41-4 C24H22N2O4
(R)-N-(4-acetylphenyl)-5-(1-(4-acetylphenyl)ethoxy)nicotinamide
—— (R)-6-(3-fluoro-5-(trifluoromethyl)phenyl)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-4-carboxamide 1429216-37-4 C24H20F4N2O3
(R)-6-(3-fluoro-5-(trifluoromethyl)phenyl)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-4-carboxamide
—— (R)-N-((S)-1-(5-chloro-6-(1,1-difluoroethyl)pyridin-3-yl)ethyl)-2-methylpropane-2-sulfinamide —— C13H19ClF2N2OS
(R)-N-((S)-1-(5-chloro-6-(1,1-difluoroethyl)pyridin-3-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-3-(1-(4-acetylphenyl)ethoxy)-N-(4-cyanophenyl)benzamide 1616242-91-1 C24H20N2O3
(R)-3-(1-(4-acetylphenyl)ethoxy)-N-(4-cyanophenyl)benzamide