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—— 5-methyl-3-[(2S)-1-[(5-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-1,2,4-triazole —— C12H18N6
5-methyl-3-[(2S)-1-[(5-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-1,2,4-triazole
—— (5S)-5-[[(2S)-3-(1-benzothiophen-3-yl)-2-[[(2S)-2-methyl-1-[(2S)-2-[[(2S)-2-(phenanthrene-4-carbonylamino)-3-[4-(sulfomethyl)phenyl]propanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-6-(tert-butylamino)-6-oxohexanoic acid —— C57H66N6O11S2
(5S)-5-[[(2S)-3-(1-benzothiophen-3-yl)-2-[[(2S)-2-methyl-1-[(2S)-2-[[(2S)-2-(phenanthrene-4-carbonylamino)-3-[4-(sulfomethyl)phenyl]propanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-6-(tert-butylamino)-6-oxohexanoic acid
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(7-methylimidazo[1,2-a]pyridin-2-yl)methanone —— C18H23N3O3
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(7-methylimidazo[1,2-a]pyridin-2-yl)methanone
—— 5-[(3S)-3-phenylpiperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile —— C16H16N4O
5-[(3S)-3-phenylpiperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile
—— 5-methoxy-N-[(3-methylphenyl)methyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyridine-2-carboxamide —— C20H24N2O4
5-methoxy-N-[(3-methylphenyl)methyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyridine-2-carboxamide
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(7-methylimidazo[1,2-a]pyridin-2-yl)methanone —— C18H23N3O3
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(7-methylimidazo[1,2-a]pyridin-2-yl)methanone
—— [(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-pyrazolo[1,5-a]pyrimidin-2-ylmethanone —— C17H22N4O3
[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-pyrazolo[1,5-a]pyrimidin-2-ylmethanone
—— (5S)-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C20H25N3O4
(5S)-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— 5-methoxy-N-[(3-methylphenyl)methyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyridine-2-carboxamide —— C20H24N2O4
5-methoxy-N-[(3-methylphenyl)methyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyridine-2-carboxamide
—— [(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-pyrazolo[1,5-a]pyrimidin-2-ylmethanone —— C17H22N4O3
[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-pyrazolo[1,5-a]pyrimidin-2-ylmethanone
—— (5R)-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C20H25N3O4
(5R)-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— [(5R)-9-[(2-aminopyrimidin-5-yl)methyl]-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(1H-pyrrol-3-yl)methanone —— C20H28N6O2
[(5R)-9-[(2-aminopyrimidin-5-yl)methyl]-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(1H-pyrrol-3-yl)methanone
—— 5-[[4-[(3-Carboxy-1-cyclopropyl-6,8-difluoro-4-oxo-7-piperazin-1-ylquinolin-5-yl)amino]cyclohexyl]amino]-1-cyclopropyl-6,8-difluoro-4-oxo-7-piperazin-1-ylquinoline-3-carboxylic acid —— C40H44F4N8O6
5-[[4-[(3-Carboxy-1-cyclopropyl-6,8-difluoro-4-oxo-7-piperazin-1-ylquinolin-5-yl)amino]cyclohexyl]amino]-1-cyclopropyl-6,8-difluoro-4-oxo-7-piperazin-1-ylquinoline-3-carboxylic acid
—— 5-[5-[(3S)-oxolan-3-yl]-2-pyridin-3-yl-1,2,4-triazol-3-yl]pyridine-2-carbonitrile —— C17H14N6O
5-[5-[(3S)-oxolan-3-yl]-2-pyridin-3-yl-1,2,4-triazol-3-yl]pyridine-2-carbonitrile
—— 5-bromo-2-[6-[[(2R,4R)-1-[(2S)-5-(diaminomethylideneamino)-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8-yl)sulfonylamino]pentanoyl]-4-methylpiperidine-2-carbonyl]amino]hexanoyloxy]benzoic acid —— C36H50BrN7O8S
5-bromo-2-[6-[[(2R,4R)-1-[(2S)-5-(diaminomethylideneamino)-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8-yl)sulfonylamino]pentanoyl]-4-methylpiperidine-2-carbonyl]amino]hexanoyloxy]benzoic acid
—— 5,10,15-Tris(2,3,4,5,6-pentafluorophenyl)-22-(pyridin-2-ylmethyl)-21,24-dihydrocorrin —— C43H16F15N5
5,10,15-Tris(2,3,4,5,6-pentafluorophenyl)-22-(pyridin-2-ylmethyl)-21,24-dihydrocorrin
—— 5-[[(2R)-2-(2-aminoethyl)morpholin-4-yl]methyl]-N-ethylpyrimidin-2-amine —— C13H23N5O
5-[[(2R)-2-(2-aminoethyl)morpholin-4-yl]methyl]-N-ethylpyrimidin-2-amine
—— 5-(5-ethyl-3H-1,3,4-oxadiazol-2-ylidene)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrole-3-sulfonamide —— C18H20N4O3S
5-(5-ethyl-3H-1,3,4-oxadiazol-2-ylidene)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrole-3-sulfonamide
—— 5-[[(2S)-2-(2-aminoethyl)morpholin-4-yl]methyl]-N-ethylpyrimidin-2-amine —— C13H23N5O
5-[[(2S)-2-(2-aminoethyl)morpholin-4-yl]methyl]-N-ethylpyrimidin-2-amine
—— 5-[2-[2-[2-[2-[Bis(carboxymethyl)amino]ethyl-(carboxymethyl)amino]ethyl-(carboxymethyl)amino]acetyl]hydrazinyl]-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-oxopentanoic acid —— C34H45N13O13
5-[2-[2-[2-[2-[Bis(carboxymethyl)amino]ethyl-(carboxymethyl)amino]ethyl-(carboxymethyl)amino]acetyl]hydrazinyl]-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-oxopentanoic acid
—— (5'S,10E,12S,14E,16E,21R,24S)-21,24-dihydroxy-12-[(4S,5S,6S)-5-[(2S,4S,5S,6S)-5-hydroxy-4-methoxy-6-methyloxan-2-yl]oxy-4-methoxy-6-methyloxan-2-yl]oxy-5',11,13,22-tetramethylspiro[3,7,19-trioxatetracyclo[15.6.1.14,8.020,24]pentacosa-10,14,16,22-tetraene-6,2'-oxane]-2-one —— C44H66O14
(5'S,10E,12S,14E,16E,21R,24S)-21,24-dihydroxy-12-[(4S,5S,6S)-5-[(2S,4S,5S,6S)-5-hydroxy-4-methoxy-6-methyloxan-2-yl]oxy-4-methoxy-6-methyloxan-2-yl]oxy-5',11,13,22-tetramethylspiro[3,7,19-trioxatetracyclo[15.6.1.14,8.020,24]pentacosa-10,14,16,22-tetraene-6,2'-oxane]-2-one
—— 5-[(3R)-3-phenylpiperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile —— C16H16N4O
5-[(3R)-3-phenylpiperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile
—— 5-[5-[(3R)-oxolan-3-yl]-2-pyridin-3-yl-1,2,4-triazol-3-yl]pyridine-2-carbonitrile —— C17H14N6O
5-[5-[(3R)-oxolan-3-yl]-2-pyridin-3-yl-1,2,4-triazol-3-yl]pyridine-2-carbonitrile
—— 5-[[2-[[(2S,3S,5R)-2-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-2-oxoethyl]carbamothioylamino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid —— C33H32N5O19P3S
5-[[2-[[(2S,3S,5R)-2-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-2-oxoethyl]carbamothioylamino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid
—— [(5S)-9-(1H-imidazol-2-ylmethyl)-3-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C22H32N4O
[(5S)-9-(1H-imidazol-2-ylmethyl)-3-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-[[4-[[(3R)-3-ethyl-4-methylpiperazin-1-yl]methyl]phenoxy]methyl]furan-2-carboxylic acid —— C20H26N2O4
5-[[4-[[(3R)-3-ethyl-4-methylpiperazin-1-yl]methyl]phenoxy]methyl]furan-2-carboxylic acid
—— 5-[(1R)-1-piperidin-1-ylethyl]-N-(2H-tetrazol-5-ylmethyl)furan-2-carboxamide —— C14H20N6O2
5-[(1R)-1-piperidin-1-ylethyl]-N-(2H-tetrazol-5-ylmethyl)furan-2-carboxamide
—— [(5R)-9-(1H-imidazol-2-ylmethyl)-3-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C22H32N4O
[(5R)-9-(1H-imidazol-2-ylmethyl)-3-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-[(6S)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile —— C14H17N7O2
5-[(6S)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile
—— 5-chloro-N-[6-[[4-[[6-[(5-chloronaphthalen-1-yl)sulfonylamino]hexylamino]methyl]phenyl]methylamino]hexyl]naphthalene-1-sulfonamide —— C40H48Cl2N4O4S2
5-chloro-N-[6-[[4-[[6-[(5-chloronaphthalen-1-yl)sulfonylamino]hexylamino]methyl]phenyl]methylamino]hexyl]naphthalene-1-sulfonamide
—— 5-[[4-[[(3S)-3-ethyl-4-methylpiperazin-1-yl]methyl]phenoxy]methyl]furan-2-carboxylic acid —— C20H26N2O4
5-[[4-[[(3S)-3-ethyl-4-methylpiperazin-1-yl]methyl]phenoxy]methyl]furan-2-carboxylic acid
—— 5-[(6R)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile —— C14H17N7O2
5-[(6R)-6-hydroxy-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile
—— 5-[(2R)-1,4-dioxan-2-yl]-1-[(3-methylphenyl)methyl]-3-(oxan-4-yl)-1,2,4-triazole —— C19H25N3O3
5-[(2R)-1,4-dioxan-2-yl]-1-[(3-methylphenyl)methyl]-3-(oxan-4-yl)-1,2,4-triazole
—— 5-[[4-[[methyl-[[(2R)-1-methylpiperidin-2-yl]methyl]amino]methyl]phenoxy]methyl]furan-2-carboxylic acid —— C21H28N2O4
5-[[4-[[methyl-[[(2R)-1-methylpiperidin-2-yl]methyl]amino]methyl]phenoxy]methyl]furan-2-carboxylic acid
—— 5-[(2S)-1,4-dioxan-2-yl]-1-[(3-methylphenyl)methyl]-3-(oxan-4-yl)-1,2,4-triazole —— C19H25N3O3
5-[(2S)-1,4-dioxan-2-yl]-1-[(3-methylphenyl)methyl]-3-(oxan-4-yl)-1,2,4-triazole
—— 5-methyl-3-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,2,4-oxadiazole —— C13H21N3O2
5-methyl-3-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,2,4-oxadiazole
—— 5-[[4-[[methyl-[[(2S)-1-methylpiperidin-2-yl]methyl]amino]methyl]phenoxy]methyl]furan-2-carboxylic acid —— C21H28N2O4
5-[[4-[[methyl-[[(2S)-1-methylpiperidin-2-yl]methyl]amino]methyl]phenoxy]methyl]furan-2-carboxylic acid
—— [(5S)-9-[(2,3-dimethylimidazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C21H32N4O2
[(5S)-9-[(2,3-dimethylimidazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [(5R)-9-[(2,3-dimethylimidazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C21H32N4O2
[(5R)-9-[(2,3-dimethylimidazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-Bromo-N-{(S)-1-[(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-4-guanidino-butylcarbamoyl]-2-cyclohexyl-ethyl}-nicotinamide —— C30H41BrN8O4
5-Bromo-N-{(S)-1-[(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-4-guanidino-butylcarbamoyl]-2-cyclohexyl-ethyl}-nicotinamide
—— [(5S)-3-[(8-methylquinolin-5-yl)methyl]-9-propan-2-yl-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C24H35N3O
[(5S)-3-[(8-methylquinolin-5-yl)methyl]-9-propan-2-yl-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— (5S,5aR,8aR,9R)-5-[[(4aR,6R,7R,8R,8aS)-2-cyclohex-3-en-1-yl-7-(dimethylamino)-8-hydroxy-4,4a,6,7,8,8a-hexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy]-9-(4-hydroxy-3,5-dimethoxyphenyl)-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[6,5-f][1,3]benzodioxol-8-one —— C36H43NO12
(5S,5aR,8aR,9R)-5-[[(4aR,6R,7R,8R,8aS)-2-cyclohex-3-en-1-yl-7-(dimethylamino)-8-hydroxy-4,4a,6,7,8,8a-hexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy]-9-(4-hydroxy-3,5-dimethoxyphenyl)-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[6,5-f][1,3]benzodioxol-8-one
—— 5-methoxy-2-[(2S)-2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyridin-4-one —— C18H20N2O3
5-methoxy-2-[(2S)-2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyridin-4-one
—— 5-[(2R)-oxolan-2-yl]-N-[[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl]thiophene-2-carboxamide —— C17H17N3O3S2
5-[(2R)-oxolan-2-yl]-N-[[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl]thiophene-2-carboxamide
—— 5-(oxan-4-yl)-3-[5-[(2S)-pyrrolidin-2-yl]thiophen-2-yl]-1H-1,2,4-triazole —— C15H20N4OS
5-(oxan-4-yl)-3-[5-[(2S)-pyrrolidin-2-yl]thiophen-2-yl]-1H-1,2,4-triazole
—— [(5R)-3-[(8-methylquinolin-5-yl)methyl]-9-propan-2-yl-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C24H35N3O
[(5R)-3-[(8-methylquinolin-5-yl)methyl]-9-propan-2-yl-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— (5R)-5-[4-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one —— C17H26N4O2S
(5R)-5-[4-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
—— (5R)-5-[4-[[4-(4-aza-1-azoniabicyclo[2.2.2]octan-1-ylmethyl)phenyl]methoxy]phenyl]-3,3-dibutyl-N,N-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6,4-benzothiazepin-7-amine;chloride —— C39H55ClN4O3S
(5R)-5-[4-[[4-(4-aza-1-azoniabicyclo[2.2.2]octan-1-ylmethyl)phenyl]methoxy]phenyl]-3,3-dibutyl-N,N-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6,4-benzothiazepin-7-amine;chloride
—— [(5R)-3-[(4-chlorophenyl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C22H33ClN2O2
[(5R)-3-[(4-chlorophenyl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-[(2S)-oxolan-2-yl]-N-[1-(thian-4-yl)piperidin-4-yl]thiophene-2-carboxamide —— C19H28N2O2S2
5-[(2S)-oxolan-2-yl]-N-[1-(thian-4-yl)piperidin-4-yl]thiophene-2-carboxamide