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—— (5S,7S)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C29H23BrF3N5O4
(5S,7S)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H23BrF3N5O5
(5R,7S)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C33H21ClF3N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— 5-[2-[(3S)-3-(2-methoxyphenyl)pyrrolidin-1-yl]ethyl]-8-thia-3,5,13-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene-4,6-dione —— C22H22N4O3S
5-[2-[(3S)-3-(2-methoxyphenyl)pyrrolidin-1-yl]ethyl]-8-thia-3,5,13-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene-4,6-dione
—— (5E)-4-bromo-3-(1-bromohexyl)-5-(bromomethylidene)furan-2-one —— C11H13Br3O2
(5E)-4-bromo-3-(1-bromohexyl)-5-(bromomethylidene)furan-2-one
—— (5E)-5-[[2-[(3,4-dichlorophenyl)methylsulfanyl]pyrimidin-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C15H9Cl2N3OS3
(5E)-5-[[2-[(3,4-dichlorophenyl)methylsulfanyl]pyrimidin-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-Cyclohexyloxy-3-(1-methyl-2-pyrrolidinylmethyl)-1-benzoylindole —— C27H32N2O2
5-Cyclohexyloxy-3-(1-methyl-2-pyrrolidinylmethyl)-1-benzoylindole
—— (5E)-5-[[3-amino-4-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C25H28N2O2S
(5E)-5-[[3-amino-4-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5S,7R)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C29H23BrF3N5O4
(5S,7R)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H23BrF3N5O5
(5S,7R)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-5-(2,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C29H21ClF3N5O4S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-5-(2,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5,6-Dimethyl-3-pyridin-2-yl-4,7,9-triazatricyclo[7.4.0.02,7]trideca-3,5,10,12-tetraen-8-ylidene)-dimethylazanium;perchlorate —— C19H22ClN5O4
(5,6-Dimethyl-3-pyridin-2-yl-4,7,9-triazatricyclo[7.4.0.02,7]trideca-3,5,10,12-tetraen-8-ylidene)-dimethylazanium;perchlorate
—— 5-chloro-4-N-(cyclopropylmethyl)-6-N-(5,7-dimethyl-2,1,3-benzothiadiazol-4-yl)-2-methyl-4-N-propylpyrimidine-4,6-diamine —— C20H25ClN6S
5-chloro-4-N-(cyclopropylmethyl)-6-N-(5,7-dimethyl-2,1,3-benzothiadiazol-4-yl)-2-methyl-4-N-propylpyrimidine-4,6-diamine
—— 5-chloro-3-[1-(2-phenylethyl)piperidin-4-yl]-2-phenyl-1H-indole —— C27H27ClN2
5-chloro-3-[1-(2-phenylethyl)piperidin-4-yl]-2-phenyl-1H-indole
—— 5-(methylsulfamoyl)-N-(4-morpholin-4-ylphenyl)-2,3-dihydroindole-1-carboxamide —— C20H24N4O4S
5-(methylsulfamoyl)-N-(4-morpholin-4-ylphenyl)-2,3-dihydroindole-1-carboxamide
—— 5-{1-[3-(2-Phenyl-1,3-dioxolan-2-yl)phenyl]ethyl}-N-tetrahydro-2(1H)-pyrimidinylidene-1,3,4-oxadiazol-2-amine 321873-90-9 C23H25N5O3
5-{1-[3-(2-Phenyl-1,3-dioxolan-2-yl)phenyl]ethyl}-N-tetrahydro-2(1H)-pyrimidinylidene-1,3,4-oxadiazol-2-amine
—— (5-Bromo-2-methylindol-1-yl)sulfonyl-(4-chlorophenyl)methanone —— C16H11BrClNO3S
(5-Bromo-2-methylindol-1-yl)sulfonyl-(4-chlorophenyl)methanone
—— 5,7-Dimethoxy-2-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]chromen-4-one —— C23H25BO6
5,7-Dimethoxy-2-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]chromen-4-one
—— (5Z)-5-[[3-methyl-2-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C26H29NO2S
(5Z)-5-[[3-methyl-2-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (+/-)-5-[[(2,3-difluorophenyl)methyl]thio]-7-[[2-hydroxy-1-(methoxymethyl)ethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one —— C16H16F2N4O3S2
(+/-)-5-[[(2,3-difluorophenyl)methyl]thio]-7-[[2-hydroxy-1-(methoxymethyl)ethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one
—— [5-fluoro-2-methylidene-1-(3-morpholin-4-ylpropyl)-3H-indol-3-yl]-(4-methoxyphenyl)methanone —— C24H27FN2O3
[5-fluoro-2-methylidene-1-(3-morpholin-4-ylpropyl)-3H-indol-3-yl]-(4-methoxyphenyl)methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C27H16ClF4N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]methanone —— C31H19ClF3N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]methanone
—— 5-(3,5-Dioxo-1,2,4-triazin-2-yl)-1-(4-methylsulfonylphenyl)-2,3-dihydroindene-1-carbonitrile —— C20H16N4O4S
5-(3,5-Dioxo-1,2,4-triazin-2-yl)-1-(4-methylsulfonylphenyl)-2,3-dihydroindene-1-carbonitrile
—— (5S,7S)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H23BrF3N5O5
(5S,7S)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(5-Acetyl-2-butoxy-3-pyridinyl)-3-ethyl-2-(2-methoxyethyl)-2,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one —— C21H27N5O4
5-(5-Acetyl-2-butoxy-3-pyridinyl)-3-ethyl-2-(2-methoxyethyl)-2,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one
—— 5-Bromo-2-(1-(4-cyanobenzyl)-5-imidazolylmethyl)-1,2,3,4-tetrahydroisoquinoline —— C21H19BrN4
5-Bromo-2-(1-(4-cyanobenzyl)-5-imidazolylmethyl)-1,2,3,4-tetrahydroisoquinoline
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(2,5-dimethylphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C30H22ClF3N4O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(2,5-dimethylphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5R,7R)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C29H23BrF3N5O4
(5R,7R)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C32H32F3N5O4
(5S,7R)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H19BrF3N5O4
(5R,7S)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5-Amino-1-benzofuran-2-yl)-[8-(chloromethyl)-4-hydroxy-2-methyl-7,8-dihydrothieno[2,3-e]indol-6-yl]methanone —— C21H17ClN2O3S
(5-Amino-1-benzofuran-2-yl)-[8-(chloromethyl)-4-hydroxy-2-methyl-7,8-dihydrothieno[2,3-e]indol-6-yl]methanone
—— 5-[8-(4-phenylphenyl)-7H-[1,2,4]triazolo[5,1-f]purin-5-yl]pentanoic acid —— C23H20N6O2
5-[8-(4-phenylphenyl)-7H-[1,2,4]triazolo[5,1-f]purin-5-yl]pentanoic acid
—— 5-(Tributylstannyl)-3-pyridinemethanoic acid —— C18H31NO2Sn
5-(Tributylstannyl)-3-pyridinemethanoic acid
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C28H19ClF3N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(3,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C30H22ClF3N4O4S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(3,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C28H19ClF3N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C28H19ClF3N5O3S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-(2-hydroxyphenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5R,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C32H32F3N5O4
(5R,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C27H16ClF4N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-5-(4-fluorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5S,7R)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H19BrF3N5O4
(5S,7R)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H19BrF3N5O4
(5S,7S)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H19BrF3N5O4
(5R,7R)-5-(4-bromophenyl)-N-(3-nitro-5-phenoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-Amino-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-methylthiopyrazole-3-thiocarboxamide —— C12H9Cl2F3N4S2
5-Amino-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-methylthiopyrazole-3-thiocarboxamide
—— (5Z)-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H28FN5O3S2
(5Z)-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[[2-(4-bromophenoxy)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H18BrN3O4S2
(5Z)-5-[[2-(4-bromophenoxy)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-Fluoro-3-[[3-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]-4-oxopentanoic acid —— C19H25FN2O6
5-Fluoro-3-[[3-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]-4-oxopentanoic acid
—— (5Z)-5-[[3-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H23Cl2N3O4S3
(5Z)-5-[[3-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-chloro-3-[(2Z,4E)-5-(2,6-dimethyl-3-oxocyclohexyl)-3-methylpenta-2,4-dienyl]-2-hydroxy-4-methoxy-6-methylbenzaldehyde —— C23H29ClO4
5-chloro-3-[(2Z,4E)-5-(2,6-dimethyl-3-oxocyclohexyl)-3-methylpenta-2,4-dienyl]-2-hydroxy-4-methoxy-6-methylbenzaldehyde
—— [5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-(6-phenyl-thieno[3,2-d]pyrimidin-4-yl)-amine 225382-80-9 C21H14ClN5S
[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-(6-phenyl-thieno[3,2-d]pyrimidin-4-yl)-amine