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—— (5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(E)-3-chloroprop-2-enyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one —— C18H14Cl2N2O2S2
(5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(E)-3-chloroprop-2-enyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one
—— (5R)-N-(8-methylquinolin-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C19H22N4O3
(5R)-N-(8-methylquinolin-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— 5-(benzenesulfonyl)-N-[3-[4-[3-[[5-(benzenesulfonyl)thiophen-2-yl]sulfonylamino]propylamino]butylamino]propyl]thiophene-2-sulfonamide —— C30H38N4O8S6
5-(benzenesulfonyl)-N-[3-[4-[3-[[5-(benzenesulfonyl)thiophen-2-yl]sulfonylamino]propylamino]butylamino]propyl]thiophene-2-sulfonamide
—— [(5S)-9-[(3-ethyl-1H-pyrazol-5-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C21H32N4O2
[(5S)-9-[(3-ethyl-1H-pyrazol-5-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [5'-[6-(butanoyloxymethyl)-3,4,5-trihydroxyoxan-2-yl]oxy-3',4,6-trihydroxy-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-4'-yl] (2E,4E,12E)-7-hydroxy-2,8,14-trimethylhexadeca-2,4,12-trienoate —— C42H62O16
[5'-[6-(butanoyloxymethyl)-3,4,5-trihydroxyoxan-2-yl]oxy-3',4,6-trihydroxy-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-4'-yl] (2E,4E,12E)-7-hydroxy-2,8,14-trimethylhexadeca-2,4,12-trienoate
—— (5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-5-(thiophen-2-ylmethylidene)imidazol-4-one —— C24H19ClN4O2S2
(5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-5-(thiophen-2-ylmethylidene)imidazol-4-one
—— (5Z)-3-(3-methoxyphenyl)-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]sulfanyl-5-[(4-propan-2-ylphenyl)methylidene]imidazol-4-one —— C28H33N3O3S
(5Z)-3-(3-methoxyphenyl)-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]sulfanyl-5-[(4-propan-2-ylphenyl)methylidene]imidazol-4-one
—— 5-methyl-3-[(2S)-1-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]piperidin-2-yl]-1,2-oxazole —— C20H24N4O
5-methyl-3-[(2S)-1-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]piperidin-2-yl]-1,2-oxazole
—— (5Z)-3-(5-chloro-2-methoxyphenyl)-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-5-[(3-methylthiophen-2-yl)methylidene]imidazol-4-one —— C24H26ClN3O4S2
(5Z)-3-(5-chloro-2-methoxyphenyl)-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-5-[(3-methylthiophen-2-yl)methylidene]imidazol-4-one
—— 5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole;4-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide —— C39H40F3N5O4S2
5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole;4-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide
—— (5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(2S)-3-oxobutan-2-yl]sulfanylimidazol-4-one —— C22H21ClN2O4S
(5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(2S)-3-oxobutan-2-yl]sulfanylimidazol-4-one
—— (5Z)-3-(3-chloro-4-methoxyphenyl)-2-[2-(1H-indol-3-yl)-2-oxoethyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one —— C25H18ClN3O3S2
(5Z)-3-(3-chloro-4-methoxyphenyl)-2-[2-(1H-indol-3-yl)-2-oxoethyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one
—— 5-[[4-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione;(1R,2S,3R)-1-[5-[(2S,3R)-2,3,4-trihydroxybutyl]pyrazin-2-yl]butane-1,2,3,4-tetrol —— C36H47N3O12S
5-[[4-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione;(1R,2S,3R)-1-[5-[(2S,3R)-2,3,4-trihydroxybutyl]pyrazin-2-yl]butane-1,2,3,4-tetrol
—— 5-methyl-3-[(2R)-1-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]piperidin-2-yl]-1,2-oxazole —— C20H24N4O
5-methyl-3-[(2R)-1-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]piperidin-2-yl]-1,2-oxazole
—— 5-[5-[[4-[5-[[4-[5-[Acetyl(hydroxy)amino]pentylamino]-4-oxobutanoyl]-hydroxyamino]pentylamino]-4-oxobutanoyl]-hydroxyamino]pentylamino]-5-oxo-3-phenylpentanoic acid —— C36H58N6O11
5-[5-[[4-[5-[[4-[5-[Acetyl(hydroxy)amino]pentylamino]-4-oxobutanoyl]-hydroxyamino]pentylamino]-4-oxobutanoyl]-hydroxyamino]pentylamino]-5-oxo-3-phenylpentanoic acid
—— 5-(dimethylsulfamoyl)-N-[(1S)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide —— C20H26N4O3S
5-(dimethylsulfamoyl)-N-[(1S)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide
—— (5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]imidazol-4-one —— C27H23ClN4O3S
(5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]imidazol-4-one
—— (5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(2S)-3-oxobutan-2-yl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one —— C19H17ClN2O3S2
(5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(2S)-3-oxobutan-2-yl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one
—— [5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl (Z)-3-[4-(cyanomethoxy)-3-methoxyphenyl]prop-2-enoate —— C24H23N3O8
[5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl (Z)-3-[4-(cyanomethoxy)-3-methoxyphenyl]prop-2-enoate
—— (5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(2R)-3-oxobutan-2-yl]sulfanylimidazol-4-one —— C22H21ClN2O4S
(5E)-3-(4-chloro-3-methoxyphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[(2R)-3-oxobutan-2-yl]sulfanylimidazol-4-one
—— (5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-3-(4-methylphenyl)imidazol-4-one —— C27H22N4O3S
(5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-3-(4-methylphenyl)imidazol-4-one
—— (5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(Z)-3-chloroprop-2-enyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one —— C18H14Cl2N2O2S2
(5Z)-3-(3-chloro-4-methoxyphenyl)-2-[(Z)-3-chloroprop-2-enyl]sulfanyl-5-(thiophen-2-ylmethylidene)imidazol-4-one
—— (5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-(4-methylphenyl)-2-[(3R)-2-oxooxolan-3-yl]sulfanylimidazol-4-one —— C22H18N2O5S
(5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-(4-methylphenyl)-2-[(3R)-2-oxooxolan-3-yl]sulfanylimidazol-4-one
—— (5R)-3-methyl-9-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H24N4O2
(5R)-3-methyl-9-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-(dimethylsulfamoyl)-N-[(1R)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide —— C20H26N4O3S
5-(dimethylsulfamoyl)-N-[(1R)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide
—— 5-[(3,5-dibutyl-1,2,4-triazol-1-yl)methyl]-2-[2-(2H-tetrazol-5-yl)phenyl]pyridine;(7R,8R,10R,13S,14S,17R)-10,13-dimethyl-7-sulfanylspiro[2,6,7,8,9,11,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthrene-17,5'-oxolane]-2',3-dione —— C45H58N8O3S
5-[(3,5-dibutyl-1,2,4-triazol-1-yl)methyl]-2-[2-(2H-tetrazol-5-yl)phenyl]pyridine;(7R,8R,10R,13S,14S,17R)-10,13-dimethyl-7-sulfanylspiro[2,6,7,8,9,11,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthrene-17,5'-oxolane]-2',3-dione
—— (5S)-3-methyl-9-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H24N4O2
(5S)-3-methyl-9-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]carbamoyl]thiophene-2-carboxylic acid —— C18H21N3O3S
5-[[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]carbamoyl]thiophene-2-carboxylic acid
—— 5-[2-[[4-[4-[(4aS,8aR)-4-(3,4-dimethoxyphenyl)-1-oxo-4a,5,8,8a-tetrahydrophthalazin-2-yl]piperidin-1-yl]-4-oxobutyl]amino]-1-hydroxyethyl]-2-amino-3-chlorobenzonitrile;(E)-but-2-enedioic acid —— C38H45ClN6O9
5-[2-[[4-[4-[(4aS,8aR)-4-(3,4-dimethoxyphenyl)-1-oxo-4a,5,8,8a-tetrahydrophthalazin-2-yl]piperidin-1-yl]-4-oxobutyl]amino]-1-hydroxyethyl]-2-amino-3-chlorobenzonitrile;(E)-but-2-enedioic acid
—— 5-(diethylsulfamoyl)-N-[(1R)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide —— C22H30N4O3S
5-(diethylsulfamoyl)-N-[(1R)-1-pyridin-4-ylethyl]-2-pyrrolidin-1-ylbenzamide
—— [5-(4-bromophenyl)-1,3,4-oxadiazol-2-yl]methyl (Z)-3-(4-methylphenyl)prop-2-enoate —— C19H15BrN2O3
[5-(4-bromophenyl)-1,3,4-oxadiazol-2-yl]methyl (Z)-3-(4-methylphenyl)prop-2-enoate
—— 5-[[4-[2-(5-Ethylpyridin-2-yl)ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione;6-[1-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)cyclopropyl]pyridine-3-carboxylic acid —— C43H49N3O5S
5-[[4-[2-(5-Ethylpyridin-2-yl)ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione;6-[1-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)cyclopropyl]pyridine-3-carboxylic acid
—— 5-(5-methylfuran-2-yl)-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-1H-pyrazole-3-carboxamide —— C21H24N4O2
5-(5-methylfuran-2-yl)-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-1H-pyrazole-3-carboxamide
—— [(5S)-9-(cyclopropylmethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(furan-2-yl)methanone —— C19H28N2O3
[(5S)-9-(cyclopropylmethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(furan-2-yl)methanone
—— (5S,5aR,8aR,9R)-5-[[7,8-dihydroxy-2-[(E)-1-phenylprop-1-en-2-yl]-4,4a,6,7,8,8a-hexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy]-9-(4-hydroxy-3,5-dimethoxyphenyl)-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[6,5-f][1,3]benzodioxol-8-one —— C37H38O13
(5S,5aR,8aR,9R)-5-[[7,8-dihydroxy-2-[(E)-1-phenylprop-1-en-2-yl]-4,4a,6,7,8,8a-hexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy]-9-(4-hydroxy-3,5-dimethoxyphenyl)-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[6,5-f][1,3]benzodioxol-8-one
—— 5,6-dimethyl-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridine-3-carboxamide —— C15H23N3O
5,6-dimethyl-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridine-3-carboxamide
—— 5-(4-{2-[4-((R)-3,10-Dibromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-piperidin-1-yl]-2-oxo-ethyl}-piperidin-1-yl)-5-oxo-pentanoic acid amide —— C31H37Br2ClN4O3
5-(4-{2-[4-((R)-3,10-Dibromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-piperidin-1-yl]-2-oxo-ethyl}-piperidin-1-yl)-5-oxo-pentanoic acid amide
—— [(5R)-9-(cyclopropylmethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(furan-2-yl)methanone —— C19H28N2O3
[(5R)-9-(cyclopropylmethyl)-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(furan-2-yl)methanone
—— 5,6-dimethyl-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyridine-3-carboxamide —— C15H23N3O
5,6-dimethyl-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyridine-3-carboxamide
—— (5-methyl-2-methylidenehexyl) (E)-2-hydroxy-6-[(4E,6E,14E,16E,19E)-11-hydroxy-24-(hydroxymethyl)-12,24-dimethyl-3-oxo-2,22,26-trioxatricyclo[19.3.1.19,13]hexacosa-4,6,14,16,19-pentaen-23-yl]hex-4-enoate —— C40H58O9
(5-methyl-2-methylidenehexyl) (E)-2-hydroxy-6-[(4E,6E,14E,16E,19E)-11-hydroxy-24-(hydroxymethyl)-12,24-dimethyl-3-oxo-2,22,26-trioxatricyclo[19.3.1.19,13]hexacosa-4,6,14,16,19-pentaen-23-yl]hex-4-enoate
—— 5-methyl-N-[[4-[(3R)-3-methylpiperidin-1-yl]phenyl]methyl]-1,3-oxazole-4-carboxamide —— C18H23N3O2
5-methyl-N-[[4-[(3R)-3-methylpiperidin-1-yl]phenyl]methyl]-1,3-oxazole-4-carboxamide
—— 5-[5-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)piperazin-1-yl]sulfonyl-2-ethoxypyridin-3-yl]-3-propyl-2-(pyridin-2-ylmethyl)-6H-pyrazolo[4,3-d]pyrimidin-7-one —— C34H38N8O6S
5-[5-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)piperazin-1-yl]sulfonyl-2-ethoxypyridin-3-yl]-3-propyl-2-(pyridin-2-ylmethyl)-6H-pyrazolo[4,3-d]pyrimidin-7-one
—— 5-methoxy-2-[(3S)-3-(methylsulfanylmethyl)piperidine-1-carbonyl]-1H-pyridin-4-one —— C14H20N2O3S
5-methoxy-2-[(3S)-3-(methylsulfanylmethyl)piperidine-1-carbonyl]-1H-pyridin-4-one
—— [5-[(1R)-1-piperidin-1-ylethyl]furan-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone —— C21H28N4O2
[5-[(1R)-1-piperidin-1-ylethyl]furan-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone
—— 5-O-[2-[[2-[3-(5-cyano-2-methyl-6-oxo-1H-pyridin-3-yl)phenoxy]acetyl]amino]ethyl] 3-O-methyl 4-(2,3-dichlorophenyl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate —— C33H30Cl2N4O7
5-O-[2-[[2-[3-(5-cyano-2-methyl-6-oxo-1H-pyridin-3-yl)phenoxy]acetyl]amino]ethyl] 3-O-methyl 4-(2,3-dichlorophenyl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate
—— 5-(pyrrolidin-1-ylmethyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-3-ylethyl]furan-2-carboxamide —— C17H18F3N3O2
5-(pyrrolidin-1-ylmethyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-3-ylethyl]furan-2-carboxamide
—— [5-[(1S)-1-piperidin-1-ylethyl]furan-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone —— C21H28N4O2
[5-[(1S)-1-piperidin-1-ylethyl]furan-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone
—— (5E)-3-[(3-chlorophenyl)methyl]-5-[[4-(morpholine-4-carbonyl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C22H19ClN2O4S
(5E)-3-[(3-chlorophenyl)methyl]-5-[[4-(morpholine-4-carbonyl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— [(5R)-5-(hydroxymethyl)-9-(3-methoxypropyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(1H-pyrrol-3-yl)methanone —— C19H31N3O3
[(5R)-5-(hydroxymethyl)-9-(3-methoxypropyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(1H-pyrrol-3-yl)methanone
—— 5-methyl-N-[(3-methylphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-oxazole-4-carboxamide —— C18H22N2O3
5-methyl-N-[(3-methylphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-oxazole-4-carboxamide