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—— 5-amino-3-(4-carboxy-phenyl)-4-oxo-3,4-dihydro-thieno[3,4-d]pyridazine-1-carboxylic acid ethyl ester —— C16H13N3O5S
5-amino-3-(4-carboxy-phenyl)-4-oxo-3,4-dihydro-thieno[3,4-d]pyridazine-1-carboxylic acid ethyl ester
—— 5-(((2S)-6-amino-2-((2,2-dimethylpropanoyl)amino)hexanoyl)amino)-3'-hydroxy(1,1'-biphenyl)-2-carboxylic acid 250789-61-8 C24H31N3O5
5-(((2S)-6-amino-2-((2,2-dimethylpropanoyl)amino)hexanoyl)amino)-3'-hydroxy(1,1'-biphenyl)-2-carboxylic acid
—— 5-{3-[3-tert-Butyl-2-(2,2-difluoro-ethoxy)-5-ethyl-phenyl]-thiophen-2-yl}-3-methyl-penta-2,4-dienoic acid —— C24H28F2O3S
5-{3-[3-tert-Butyl-2-(2,2-difluoro-ethoxy)-5-ethyl-phenyl]-thiophen-2-yl}-3-methyl-penta-2,4-dienoic acid
—— (5Z)-5-[[3-methoxy-2-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C26H29NO3S
(5Z)-5-[[3-methoxy-2-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-5-ethenyl-2,2,2-triphenyl-1,2lambda5-oxaphospholane —— C23H23OP
(5S)-5-ethenyl-2,2,2-triphenyl-1,2lambda5-oxaphospholane
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethylsulfanyl)butan-2-yl]pyridine-3-carboxamide —— C13H12F8N2OS
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethylsulfanyl)butan-2-yl]pyridine-3-carboxamide
—— 5-Chloro-2-[2-[3-(4-fluorophenoxy)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethoxy]benzamide —— C22H22ClFN2O4
5-Chloro-2-[2-[3-(4-fluorophenoxy)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethoxy]benzamide
—— (5S,10bS)-2-(4-methylphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C31H36N2O2
(5S,10bS)-2-(4-methylphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,6S)-6-[(1R)-1-hydroxyethyl]-7-oxo-3-[4-(pyridin-4-ylsulfanylmethyl)phenyl]-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid —— C21H20N2O4S
(5R,6S)-6-[(1R)-1-hydroxyethyl]-7-oxo-3-[4-(pyridin-4-ylsulfanylmethyl)phenyl]-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethylsulfanyl)butan-2-yl]pyridine-3-carboxamide —— C13H12F8N2OS
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethylsulfanyl)butan-2-yl]pyridine-3-carboxamide
—— (5R,10bS)-5-(4-bromophenyl)-7,9-dichloro-2-(3,4-dimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H19BrCl2N2O3
(5R,10bS)-5-(4-bromophenyl)-7,9-dichloro-2-(3,4-dimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethylsulfanyl)propan-2-yl]pyridine-3-carboxamide —— C12H10F8N2OS
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethylsulfanyl)propan-2-yl]pyridine-3-carboxamide
—— 5-[2-[4-(5-Fluorobenzotriazol-1-yl)piperidin-1-yl]ethyl]-4-(4-fluorophenyl)-2-methyl-1,3-thiazole —— C23H23F2N5S
5-[2-[4-(5-Fluorobenzotriazol-1-yl)piperidin-1-yl]ethyl]-4-(4-fluorophenyl)-2-methyl-1,3-thiazole
—— (5R,10bS)-2-(4-methoxyphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C31H36N2O3
(5R,10bS)-2-(4-methoxyphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-Phenyl-2-(6,7,8,9-tetrahydrodibenzofuran-3-ylsulfonylamino)pentanoic acid —— C23H25NO5S
5-Phenyl-2-(6,7,8,9-tetrahydrodibenzofuran-3-ylsulfonylamino)pentanoic acid
—— 5-Cyclopropyl-2-(2-dimethylamino-ethyl)-7-(2,6-dimethyl-pyridin-4-yl)-6,8-difluoro-2,5-dihydro-pyrazolo[4,3-c]quinolin-3-one —— C24H25F2N5O
5-Cyclopropyl-2-(2-dimethylamino-ethyl)-7-(2,6-dimethyl-pyridin-4-yl)-6,8-difluoro-2,5-dihydro-pyrazolo[4,3-c]quinolin-3-one
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethoxy)propan-2-yl]pyridine-3-carboxamide —— C12H10F8N2O2
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethoxy)propan-2-yl]pyridine-3-carboxamide
—— (5S)-5-[[4-(azidomethyl)triazol-1-yl]methyl]-3-[3-fluoro-4-(1-oxo-3,6-dihydro-2H-thiopyran-4-yl)phenyl]-1,3-oxazolidin-2-one —— C18H18FN7O3S
(5S)-5-[[4-(azidomethyl)triazol-1-yl]methyl]-3-[3-fluoro-4-(1-oxo-3,6-dihydro-2H-thiopyran-4-yl)phenyl]-1,3-oxazolidin-2-one
—— (5R,10bS)-2-(4-methylphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C31H36N2O2
(5R,10bS)-2-(4-methylphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-(4-methoxyphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C31H36N2O3
(5S,10bS)-2-(4-methoxyphenyl)-5-(4-octoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5Z)-5-[[6-methoxy-5-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)pyridin-3-yl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C25H29N3O2S
(5Z)-5-[[6-methoxy-5-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)pyridin-3-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide —— C13H12F8N2O2
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2R)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethoxy)propan-2-yl]pyridine-3-carboxamide —— C12H10F8N2O2
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethoxy)propan-2-yl]pyridine-3-carboxamide
—— 5-[(7R)-4,6a-dimethyl-7-(6-methylheptan-2-yl)-2-oxo-4a,5,6,7,8,9,9a,9b-octahydro-1H-cyclopenta[f]isochromen-4-yl]pentanoic acid —— C27H46O4
5-[(7R)-4,6a-dimethyl-7-(6-methylheptan-2-yl)-2-oxo-4a,5,6,7,8,9,9a,9b-octahydro-1H-cyclopenta[f]isochromen-4-yl]pentanoic acid
—— 5-[(3-bromophenyl)methylsulfanyl]-7-(1-hydroxypropan-2-ylamino)-3H-[1,3]thiazolo[4,5-d]pyrimidin-2-one —— C15H15BrN4O2S2
5-[(3-bromophenyl)methylsulfanyl]-7-(1-hydroxypropan-2-ylamino)-3H-[1,3]thiazolo[4,5-d]pyrimidin-2-one
—— 5-[[4-[3-(5-Methyl-2-phenyl-4,5-dihydro-1,3-oxazol-4-yl)propanoyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C23H22N2O4S
5-[[4-[3-(5-Methyl-2-phenyl-4,5-dihydro-1,3-oxazol-4-yl)propanoyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— 5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide —— C13H12F8N2O2
5-(1,1,2,2,2-pentafluoroethyl)-N-[(2S)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide
—— 5-[2-[4-(5-Fluorobenzotriazol-1-yl)piperidin-1-yl]ethyl]-4-(4-fluorophenyl)-1,3-thiazole —— C22H21F2N5S
5-[2-[4-(5-Fluorobenzotriazol-1-yl)piperidin-1-yl]ethyl]-4-(4-fluorophenyl)-1,3-thiazole
—— 5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione nitrate 403731-62-4 C18H19N3O3S*HNO3
5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione nitrate
—— 5-[[3-Tert-butyl-4-hydroxy-5-(phenylsulfanylmethyl)phenyl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H23NO2S3
5-[[3-Tert-butyl-4-hydroxy-5-(phenylsulfanylmethyl)phenyl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[4-[(E)-3-(4-fluorophenyl)-2-methylprop-2-enyl]piperazin-1-yl]methyl]-4,8-dioxa-3,11-diazatricyclo[7.4.0.02,6]trideca-1(9),2,10,12-tetraene —— C24H27FN4O2
5-[[4-[(E)-3-(4-fluorophenyl)-2-methylprop-2-enyl]piperazin-1-yl]methyl]-4,8-dioxa-3,11-diazatricyclo[7.4.0.02,6]trideca-1(9),2,10,12-tetraene
—— (5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H20BrClF3N5O5
(5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[3-(1,4,5,6-Tetrahydropyrimidin-2-ylamino)propoxy]tetracyclo[8.6.1.03,8.013,17]heptadeca-1(17),3(8),4,6,13,15-hexaene-11-carboxylic acid —— C25H29N3O3
5-[3-(1,4,5,6-Tetrahydropyrimidin-2-ylamino)propoxy]tetracyclo[8.6.1.03,8.013,17]heptadeca-1(17),3(8),4,6,13,15-hexaene-11-carboxylic acid
—— (5R,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H20BrClF3N5O5
(5R,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(3,4-dichlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C28H16Cl3F3N4O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3S)-5-(3,4-dichlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5R,7R)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H23BrF3N5O5
(5R,7R)-5-(4-bromophenyl)-N-[3-(4-ethoxyphenoxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H17Br2ClF3N5O4
(5S,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-5-(2,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C29H21ClF3N5O4S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-5-(2,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H17Br2ClF3N5O4
(5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H20BrClF3N5O5
(5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C32H32F3N5O4
(5S,7S)-N-[(Z)-[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylideneamino]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H18Br2F3N5O4
(5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H18Br2F3N5O4
(5S,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H17Br2ClF3N5O4
(5R,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3R)-5-(3,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C30H22ClF3N4O4S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3R)-5-(3,4-dimethoxyphenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-(2-hydroxyphenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C33H21ClF3N5O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-(2-hydroxyphenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H18Br2F3N5O4
(5S,7S)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H17Br2ClF3N5O4
(5R,7R)-N-[3-(4-bromophenoxy)-5-nitrophenyl]-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3R)-5-(3,4-dichlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone —— C28H16Cl3F3N4O2S
[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]-[(3R)-5-(3,4-dichlorophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]methanone
—— (5R,7S)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C29H23BrF3N5O4
(5R,7S)-5-(4-bromophenyl)-N-[3-(2,3-dihydro-1H-inden-5-yloxy)-5-nitrophenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide