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—— (5S)-5-ethyl-N-methyl-N-[2-oxo-2-(2,4,6-trimethylanilino)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C23H30N2O2S
(5S)-5-ethyl-N-methyl-N-[2-oxo-2-(2,4,6-trimethylanilino)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-bromo-N-[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl]furan-2-carboxamide —— C15H14BrClN2O3
5-bromo-N-[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl]furan-2-carboxamide
—— (5-phenyl-1,3-oxazol-2-yl)methyl (5S,7S)-3-bromoadamantane-1-carboxylate —— C21H22BrNO3
(5-phenyl-1,3-oxazol-2-yl)methyl (5S,7S)-3-bromoadamantane-1-carboxylate
—— 5-chloro-N-cycloheptylthiophene-2-carboxamide —— C12H16ClNOS
5-chloro-N-cycloheptylthiophene-2-carboxamide
—— 5-bromo-N-cycloheptyl-2-fluorobenzamide —— C14H17BrFNO
5-bromo-N-cycloheptyl-2-fluorobenzamide
—— 5-bromo-N-[2-(cycloheptylamino)-2-oxoethyl]furan-2-carboxamide —— C14H19BrN2O3
5-bromo-N-[2-(cycloheptylamino)-2-oxoethyl]furan-2-carboxamide
—— (5-phenyl-1,3-oxazol-2-yl)methyl (5R,7R)-3-bromoadamantane-1-carboxylate —— C21H22BrNO3
(5-phenyl-1,3-oxazol-2-yl)methyl (5R,7R)-3-bromoadamantane-1-carboxylate
—— (5-fluoro-2-methoxyphenyl)methyl (5S,7S)-3-bromoadamantane-1-carboxylate —— C19H22BrFO3
(5-fluoro-2-methoxyphenyl)methyl (5S,7S)-3-bromoadamantane-1-carboxylate
—— (5-fluoro-2-methoxyphenyl)methyl (5R,7R)-3-bromoadamantane-1-carboxylate —— C19H22BrFO3
(5-fluoro-2-methoxyphenyl)methyl (5R,7R)-3-bromoadamantane-1-carboxylate
—— 5-bromo-N-(3-fluoro-4-methylphenyl)pyridine-3-carboxamide —— C13H10BrFN2O
5-bromo-N-(3-fluoro-4-methylphenyl)pyridine-3-carboxamide
—— 5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide —— C26H29N3O3
5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide
—— 5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide —— C26H29N3O3
5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide
—— 5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide —— C26H29N3O3
5-N-methyl-4-oxo-1-(2-phenylethyl)-3-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]pyridine-3,5-dicarboxamide
—— 5-(azepan-1-ylsulfonyl)-N-(3-fluoro-4-methylphenyl)-2-methoxybenzamide —— C21H25FN2O4S
5-(azepan-1-ylsulfonyl)-N-(3-fluoro-4-methylphenyl)-2-methoxybenzamide
—— (5-fluoro-2-methoxyphenyl)methyl (2R)-1-(thiophene-2-carbonyl)pyrrolidine-2-carboxylate —— C18H18FNO4S
(5-fluoro-2-methoxyphenyl)methyl (2R)-1-(thiophene-2-carbonyl)pyrrolidine-2-carboxylate
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-(4-fluorophenyl)-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]thiophene-2-carboxamide —— C20H17FN2O3S
5-(4-fluorophenyl)-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]thiophene-2-carboxamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-(3-acetamidopropoxy)ethoxy]ethoxy]propyl]pentanamide —— C22H40N4O6S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-(3-acetamidopropoxy)ethoxy]ethoxy]propyl]pentanamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C26H48N6O9S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide —— C21H39N3O5S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide
—— (5S,7R)-3-chloro-N-[2-(4-fluoro-3-nitroanilino)-2-oxoethyl]adamantane-1-carboxamide —— C19H21ClFN3O4
(5S,7R)-3-chloro-N-[2-(4-fluoro-3-nitroanilino)-2-oxoethyl]adamantane-1-carboxamide
—— (5Z)-5-[(7-chloro-1,3-benzodioxol-5-yl)methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H10ClNO3S2
(5Z)-5-[(7-chloro-1,3-benzodioxol-5-yl)methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-methyl-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]-1-phenylpyrazole-3-carboxamide —— C20H20N4O3
5-methyl-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]-1-phenylpyrazole-3-carboxamide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide —— C21H39N3O5S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide
—— 5-(cyclohexylsulfamoyl)-N-cyclopentyl-2-methylbenzamide —— C19H28N2O3S
5-(cyclohexylsulfamoyl)-N-cyclopentyl-2-methylbenzamide
—— 5-(diethylsulfamoyl)-N-(4-ethylphenyl)-2-fluorobenzamide —— C19H23FN2O3S
5-(diethylsulfamoyl)-N-(4-ethylphenyl)-2-fluorobenzamide
—— 5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C21H39N5O7S
5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— (5R)-2-(3,4-dimethylphenyl)-5-[(3R)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione —— C29H28N2O4
(5R)-2-(3,4-dimethylphenyl)-5-[(3R)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione
—— [5-[(4-Bromo-3,5-dimethylpyrazol-1-yl)methyl]furan-2-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C24H32BrN5O2S
[5-[(4-Bromo-3,5-dimethylpyrazol-1-yl)methyl]furan-2-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— [5-[(2-Bromophenoxy)methyl]furan-2-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C25H30BrN3O3S
[5-[(2-Bromophenoxy)methyl]furan-2-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]furan-2-carboxamide —— C20H17FN2O4
5-(4-fluorophenyl)-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]furan-2-carboxamide
—— (5R)-2-(4-chlorophenyl)-5-[(3S)-1-(4-chlorophenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione —— C25H18Cl2N2O4
(5R)-2-(4-chlorophenyl)-5-[(3S)-1-(4-chlorophenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione
—— 5-ethyl-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]-1-phenylpyrazole-4-carboxamide —— C21H22N4O3
5-ethyl-N-[4-[2-(methylamino)-2-oxoethoxy]phenyl]-1-phenylpyrazole-4-carboxamide
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-[(3S)-dithiolan-3-yl]-N-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethyl]pentanamide —— C17H33NO5S2
5-[(3S)-dithiolan-3-yl]-N-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethyl]pentanamide
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C26H50N4O9S
5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— (5S)-2-(3,4-dimethylphenyl)-5-[(3R)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione —— C29H28N2O4
(5S)-2-(3,4-dimethylphenyl)-5-[(3R)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione
—— 5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-(2-aminooxyethoxy)ethoxy]ethoxy]ethyl]pentanamide —— C18H34N4O6S
5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-(2-aminooxyethoxy)ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C21H39N5O7S
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-[3-[3-(2,5-dioxopyrrol-1-yl)propanoylamino]propoxy]ethoxy]ethoxy]propyl]pentanamide —— C27H43N5O8S
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-[3-[3-(2,5-dioxopyrrol-1-yl)propanoylamino]propoxy]ethoxy]ethoxy]propyl]pentanamide
—— (5S)-2-(3,4-dimethylphenyl)-5-[(3S)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione —— C29H28N2O4
(5S)-2-(3,4-dimethylphenyl)-5-[(3S)-1-(3,4-dimethylphenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione
—— 5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C26H48N6O9S
5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-(2-aminooxyethoxy)ethoxy]ethoxy]ethyl]pentanamide —— C18H34N4O6S
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-(2-aminooxyethoxy)ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-[3-[3-(2,5-dioxopyrrol-1-yl)propanoylamino]propoxy]ethoxy]ethoxy]propyl]pentanamide —— C27H43N5O8S
5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-[2-[3-[3-(2,5-dioxopyrrol-1-yl)propanoylamino]propoxy]ethoxy]ethoxy]propyl]pentanamide
—— (5S)-2-(4-chlorophenyl)-5-[(3R)-1-(4-chlorophenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione —— C25H18Cl2N2O4
(5S)-2-(4-chlorophenyl)-5-[(3R)-1-(4-chlorophenyl)-2,5-dioxopyrrolidin-3-yl]-7-methyl-4,5-dihydroisoindole-1,3-dione
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C21H39N5O7S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-(3-hydrazinyl-3-oxopropoxy)ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide —— C21H39N3O5S
5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[3-[2-(2-butoxyethoxy)ethoxy]propyl]pentanamide
—— 5-(dimethylsulfamoyl)-N-(4-ethylphenyl)-2-fluorobenzamide —— C17H19FN2O3S
5-(dimethylsulfamoyl)-N-(4-ethylphenyl)-2-fluorobenzamide