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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(2-{[2-(morpholin-4-yl)-2-oxoethyl]sulfanyl}-1,3-benzothiazol-6-yl)acetamide 5777-02-6 C24H24N6O3S3
2-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(2-{[2-(morpholin-4-yl)-2-oxoethyl]sulfanyl}-1,3-benzothiazol-6-yl)acetamide
—— 6-N-benzyl-2-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxopyran-2,6-dicarboxamide 1095513-90-8 C31H27N7O6
6-N-benzyl-2-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxopyran-2,6-dicarboxamide
—— diethyl 3-(3-chloro-4-fluoroanilino)-1H-pyrazole-4,5-dicarboxylate 142115-61-5 C15H15ClFN3O4
diethyl 3-(3-chloro-4-fluoroanilino)-1H-pyrazole-4,5-dicarboxylate
—— 2-methoxy-5-p-nitrophenyloxazole 80224-86-8 C10H8N2O4
2-methoxy-5-p-nitrophenyloxazole
—— N-[2-(2-bromophenyl)-1,3-benzoxazol-5-yl]-2-chlorobenzamide 5638-59-5 C20H12BrClN2O2
N-[2-(2-bromophenyl)-1,3-benzoxazol-5-yl]-2-chlorobenzamide
—— 2-(4-Methylphenyl)sulfonyl-3-[1-phenyl-3-(4-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enenitrile 6616-22-4 C30H28N4O4S2
2-(4-Methylphenyl)sulfonyl-3-[1-phenyl-3-(4-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enenitrile
—— 11-(4-tert-butylphenyl)-N-(3,4-dichlorophenyl)-10-methyl-8-phenyl-8,11-dihydropyrazolo[3',4':4,5]pyrimido[1,2-a]quinoxalin-6-amine 5720-22-9 C35H30Cl2N6
11-(4-tert-butylphenyl)-N-(3,4-dichlorophenyl)-10-methyl-8-phenyl-8,11-dihydropyrazolo[3',4':4,5]pyrimido[1,2-a]quinoxalin-6-amine
—— 2-[[4-(4-chlorophenyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,4-dimethylphenyl)acetamide 5305-25-9 C25H23ClN4OS
2-[[4-(4-chlorophenyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,4-dimethylphenyl)acetamide
—— 7-[(5-Methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one 5621-62-5 C16H13N5OS2
7-[(5-Methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 4-(2-methanesulfonyloxy-ethyl)-2-phenoxymethyl-oxazole-5-carboxylic acid ethyl ester 1454302-78-3 C16H19NO7S
4-(2-methanesulfonyloxy-ethyl)-2-phenoxymethyl-oxazole-5-carboxylic acid ethyl ester
—— 5-p-cyanophenyl-2-methoxyoxazole 80224-87-9 C11H8N2O2
5-p-cyanophenyl-2-methoxyoxazole
—— (R)-N-(2,2-dimethoxyethyl)-N-(3,3-dimethylbutan-2-yl)-3-(3-(1-ethyl-1H-pyrazol-4-yl)phenethoxy)propanamide 1201641-27-1 C26H41N3O4
(R)-N-(2,2-dimethoxyethyl)-N-(3,3-dimethylbutan-2-yl)-3-(3-(1-ethyl-1H-pyrazol-4-yl)phenethoxy)propanamide
—— (R)-2-phenoxymethyl-4-[2-(1 ,2,2-trimethyl-propylamino)-ethyl]-oxazole-5-carboxylic acid ethyl ester 1454302-79-4 C21H30N2O4
(R)-2-phenoxymethyl-4-[2-(1 ,2,2-trimethyl-propylamino)-ethyl]-oxazole-5-carboxylic acid ethyl ester
—— 4-[(4-Chlorophenyl)sulfanyl]-3-methyl-1-phenyl-1H-pyrazol-5-yl 2-(4-chlorophenoxy)-2-methylpropanoate 6235-01-4 C26H22Cl2N2O3S
4-[(4-Chlorophenyl)sulfanyl]-3-methyl-1-phenyl-1H-pyrazol-5-yl 2-(4-chlorophenoxy)-2-methylpropanoate
—— N-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(3-methoxyphenyl)imidazol-2-yl]sulfanyl-acetamide 6242-94-0 C19H15ClF3N3O2S
N-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(3-methoxyphenyl)imidazol-2-yl]sulfanyl-acetamide
—— 7-[4-(Benzyloxy)-2-hydroxyphenyl]-10-bromo-2-phenyl-5,7,12,12a-tetrahydro-1H-benzo[g][1,2,4]triazolo[1,2-a]cinnoline-1,3,8,11(2H)-tetrone 6057-95-0 C33H24BrN3O6
7-[4-(Benzyloxy)-2-hydroxyphenyl]-10-bromo-2-phenyl-5,7,12,12a-tetrahydro-1H-benzo[g][1,2,4]triazolo[1,2-a]cinnoline-1,3,8,11(2H)-tetrone
—— [2-(4-Fluorophenyl)-5-propylpyrazol-3-yl] 4-butoxybenzoate 5878-92-2 C23H25FN2O3
[2-(4-Fluorophenyl)-5-propylpyrazol-3-yl] 4-butoxybenzoate
—— 2,3-dihydro-3-ethyl-2,4-dioxo-4H-<1,3,4>thiadiazolo<3,2-a><1,3,5>triazine-7-sulfonamide 109907-77-9 C6H7N5O4S2
2,3-dihydro-3-ethyl-2,4-dioxo-4H-<1,3,4>thiadiazolo<3,2-a><1,3,5>triazine-7-sulfonamide
—— 5-(N'-ethylureido)-1,3,4-thiadiazole-2-sulfonamide 109907-73-5 C5H9N5O3S2
5-(N'-ethylureido)-1,3,4-thiadiazole-2-sulfonamide
—— 3-methyl-5-(o-nitrophenyl)-1,2,4-oxadiazole 76629-46-4 C9H7N3O3
3-methyl-5-(o-nitrophenyl)-1,2,4-oxadiazole
—— 4-Phenyl-2-sulfamoyl-thiazol 90417-48-4 C9H8N2O2S2
4-Phenyl-2-sulfamoyl-thiazol
—— N-[5-tert-butyl-2-(4-chlorophenyl)pyrazol-3-yl]-2-[butyl-[(3-methylphenyl)carbamoyl]amino]acetamide 5880-14-8 C27H34ClN5O2
N-[5-tert-butyl-2-(4-chlorophenyl)pyrazol-3-yl]-2-[butyl-[(3-methylphenyl)carbamoyl]amino]acetamide
—— N-butan-2-yl-2-(2,4-dimethylphenyl)-5-(3,4-dimethylphenyl)pyrazole-3-carboxamide 5985-08-0 C24H29N3O
N-butan-2-yl-2-(2,4-dimethylphenyl)-5-(3,4-dimethylphenyl)pyrazole-3-carboxamide
—— (R)-tert-butyl3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidine-1-carboxylate 1221743-93-6 C28H29F3N8O3
(R)-tert-butyl3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidine-1-carboxylate
—— 1-[4-(3-Phenylprop-2-en-1-yl)piperazin-1-yl]-2-[(1,4,5-triphenyl-1H-imidazol-2-yl)sulfanyl]ethan-1-one 5924-26-5 C36H34N4OS
1-[4-(3-Phenylprop-2-en-1-yl)piperazin-1-yl]-2-[(1,4,5-triphenyl-1H-imidazol-2-yl)sulfanyl]ethan-1-one
—— 1-(5-Cyclobutyl-2-phenylpyrazol-3-yl)-3-[3-(trifluoromethyl)phenyl]urea 1448705-38-1 C21H19F3N4O
1-(5-Cyclobutyl-2-phenylpyrazol-3-yl)-3-[3-(trifluoromethyl)phenyl]urea
—— 1-(4-(4-amino-1-((R)-tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-d]pyrirmdin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1221743-79-8 C23H20F3N7O2
1-(4-(4-amino-1-((R)-tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-d]pyrirmdin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— 1-(2-Phenyl-5-propan-2-ylpyrazol-3-yl)-3-[3-(trifluoromethyl)phenyl]urea 1448705-19-8 C20H19F3N4O
1-(2-Phenyl-5-propan-2-ylpyrazol-3-yl)-3-[3-(trifluoromethyl)phenyl]urea
—— 1-(4-(4-amino-1-((R)-pyrrolidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1221743-89-0 C23H21F3N8O
1-(4-(4-amino-1-((R)-pyrrolidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— 1,4,5-Trimethyl-3-[3-(trifluoromethyl)phenyl]imidazol-2-one 127931-88-8 C13H13F3N2O
1,4,5-Trimethyl-3-[3-(trifluoromethyl)phenyl]imidazol-2-one
—— 1-[5-(Cyclopropylmethyl)-2-phenylpyrazol-3-yl]-3-[3-(trifluoromethyl)phenyl]urea 1448705-33-6 C21H19F3N4O
1-[5-(Cyclopropylmethyl)-2-phenylpyrazol-3-yl]-3-[3-(trifluoromethyl)phenyl]urea
—— 2,3-Dihydro-6-p-chlorophenylimidazo<2,1-b>thiazol-5-ylmethyl m-Trifluoromethylphenylcarbamate 123772-55-4 C20H15ClF3N3O2S
2,3-Dihydro-6-p-chlorophenylimidazo<2,1-b>thiazol-5-ylmethyl m-Trifluoromethylphenylcarbamate
—— 1-(2-(4-(6-(3-hydroxyphenyl)imidazo[2,1-b]thiazol-5-yl)pyrimidin-2-ylamino)ethyl)-3-(3-(trifluoromethyl)phenyl)urea 1350454-78-2 C25H20F3N7O2S
1-(2-(4-(6-(3-hydroxyphenyl)imidazo[2,1-b]thiazol-5-yl)pyrimidin-2-ylamino)ethyl)-3-(3-(trifluoromethyl)phenyl)urea
—— (S)-3-(4-amino-3-(4-aminophenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-N-(3-(trifluoromethyl)phenyl)pyrrolidine-1-carboxamide 1221743-84-5 C23H21F3N8O
(S)-3-(4-amino-3-(4-aminophenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-N-(3-(trifluoromethyl)phenyl)pyrrolidine-1-carboxamide
—— 1-(2-(4-(6-(3-methoxyphenyl)imidazo[2,1-b]thiazol-5-yl)pyrimidin-2-ylamino)ethyl)-3-(3-(trifluoromethyl)phenyl)urea 1350454-75-9 C26H22F3N7O2S
1-(2-(4-(6-(3-methoxyphenyl)imidazo[2,1-b]thiazol-5-yl)pyrimidin-2-ylamino)ethyl)-3-(3-(trifluoromethyl)phenyl)urea
—— (S)-1-(4-(1-(2-(2-hydroxypropylamino)pyrimidin-4-yl)-1H-imidazol-2-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1220701-46-1 C24H22F3N7O2
(S)-1-(4-(1-(2-(2-hydroxypropylamino)pyrimidin-4-yl)-1H-imidazol-2-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— 3-[(4-(2-(2-phenyl-4-oxazolyl)ethoxy)phenyl)methyl]1,2,4-thiadiazolin-5-one 179170-53-7 C20H17N3O3S
3-[(4-(2-(2-phenyl-4-oxazolyl)ethoxy)phenyl)methyl]1,2,4-thiadiazolin-5-one
—— (S)-1-(3-(1-(2-(2-hydroxypropylamino)pyrimidin-4-yl)-1H-imidazol-2-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1220701-41-6 C24H22F3N7O2
(S)-1-(3-(1-(2-(2-hydroxypropylamino)pyrimidin-4-yl)-1H-imidazol-2-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— 1-{3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]propyl}-3-(3-trifluoromethylphenyl)urea 1287760-93-3 C27H25F3N4O3S
1-{3-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-yl]propyl}-3-(3-trifluoromethylphenyl)urea
—— 3-[1-(4-Methylsulfonylphenyl)-5-phenylpyrazol-3-yl]propan-1-amine 1287761-12-9 C19H21N3O2S
3-[1-(4-Methylsulfonylphenyl)-5-phenylpyrazol-3-yl]propan-1-amine
—— 1-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-ylmethyl]-3-(3-trifluoromethylphenyl)urea 1287760-89-7 C25H21F3N4O3S
1-[1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazol-3-ylmethyl]-3-(3-trifluoromethylphenyl)urea
—— 1-(4-(4-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1221743-62-9 C20H16F3N7O
1-(4-(4-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— 4-(2-(2-phenyl-4-oxazolyl)ethoxy)benzeneethanimidamide hydrochloride 179170-54-8 C19H19N3O2*ClH
4-(2-(2-phenyl-4-oxazolyl)ethoxy)benzeneethanimidamide hydrochloride
—— AD57 1093380-42-7 C22H20F3N7O
AD57
—— 4-(5-phenyl-3-{3-[3-(3-trifluoromethylphenyl)ureido]propyl}pyrazol-1-yl)benzenesulfonamide 1287760-94-4 C26H24F3N5O3S
4-(5-phenyl-3-{3-[3-(3-trifluoromethylphenyl)ureido]propyl}pyrazol-1-yl)benzenesulfonamide
—— 1-[5-chloro-2-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-3-(3-trifluoromethyl-phenyl)-urea 697278-53-8 C16H10ClF3N4O3
1-[5-chloro-2-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-3-(3-trifluoromethyl-phenyl)-urea
—— (S)-3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-N-(3-(trifluoromethyl)phenyl)pyrrolidine-1-carboxamide 1221743-85-6 C31H25F6N9O2
(S)-3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-N-(3-(trifluoromethyl)phenyl)pyrrolidine-1-carboxamide
—— (S)-tert-butyl3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidine-1-carboxylate 1221743-92-5 C28H29F3N8O3
(S)-tert-butyl3-(4-amino-3-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidine-1-carboxylate
—— 1-[4-[4-Amino-1-[3-[tert-butyl(dimethyl)silyl]oxypropyl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]-3-[3-(trifluoromethyl)phenyl]urea 1293140-49-4 C28H34F3N7O2Si
1-[4-[4-Amino-1-[3-[tert-butyl(dimethyl)silyl]oxypropyl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]-3-[3-(trifluoromethyl)phenyl]urea
—— 1-(4-(4-amino-1-((S)-tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-d]pyrirmdin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1221743-71-0 C23H20F3N7O2
1-(4-(4-amino-1-((S)-tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-d]pyrirmdin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea