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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(2,4-dichlorophenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H19Cl2N3O2S2
2-[(2,4-dichlorophenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-(6-oxo-3-phenylpyridazin-1-yl)acetamide —— C19H20N4O2S
N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-(6-oxo-3-phenylpyridazin-1-yl)acetamide
—— 2-[(3-bromophenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H22BrN3O3S
2-[(3-bromophenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-(6-oxo-3-phenylpyridazin-1-yl)acetamide —— C19H20N4O2S
N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-(6-oxo-3-phenylpyridazin-1-yl)acetamide
—— N-[(1R)-2-ethyl-1-thiophen-2-ylbutyl]-2-(3-methyl-2,4-dioxopyrimidin-1-yl)acetamide —— C17H23N3O3S
N-[(1R)-2-ethyl-1-thiophen-2-ylbutyl]-2-(3-methyl-2,4-dioxopyrimidin-1-yl)acetamide
—— N-[(1S)-2-ethyl-1-thiophen-2-ylbutyl]-2-(3-methyl-2,4-dioxopyrimidin-1-yl)acetamide —— C17H23N3O3S
N-[(1S)-2-ethyl-1-thiophen-2-ylbutyl]-2-(3-methyl-2,4-dioxopyrimidin-1-yl)acetamide
—— 2-[(2,3-dichlorophenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H19Cl2N3O2S2
2-[(2,3-dichlorophenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[[4-(dimethylamino)phenyl]methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H26N4O2S2
2-[[4-(dimethylamino)phenyl]methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[(4-methoxyphenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H25N3O4S
2-[(4-methoxyphenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[(5-bromo-2-hydroxyphenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H20BrN3O3S2
2-[(5-bromo-2-hydroxyphenyl)methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[(4-chlorophenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H22ClN3O3S
2-[(4-chlorophenyl)methylidene]-7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[[4-(diethylamino)phenyl]methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H30N4O2S2
2-[[4-(diethylamino)phenyl]methylidene]-7-methyl-N-(2-methylphenyl)-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 7-methyl-N-(2-methylphenyl)-2-[(4-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H20N4O4S2
7-methyl-N-(2-methylphenyl)-2-[(4-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— N-cyclohexyl-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide —— C23H30N6O
N-cyclohexyl-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide
—— 4-(azepan-1-yl)-6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C26H31N5O2S
4-(azepan-1-yl)-6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (3-methoxyphenyl)-(4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)methanone —— C25H27N5O2
(3-methoxyphenyl)-(4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)methanone
—— 3-[(2-pyridin-2-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)sulfonyl]benzonitrile —— C23H22N6O2S
3-[(2-pyridin-2-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)sulfonyl]benzonitrile
—— 6-[2-(benzenesulfonyl)ethyl]-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C24H27N5O2S
6-[2-(benzenesulfonyl)ethyl]-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-piperidin-1-yl-6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H25N5
4-piperidin-1-yl-6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— ethyl 1-[6-(3-methoxyphenyl)sulfonyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C27H31N5O5S
ethyl 1-[6-(3-methoxyphenyl)sulfonyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— 4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine —— C24H27N5O3S
4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine
—— 6-[2-(benzenesulfonyl)ethyl]-4-(4-methylpiperazin-1-yl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C25H30N6O2S
6-[2-(benzenesulfonyl)ethyl]-4-(4-methylpiperazin-1-yl)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-piperidin-1-yl-6-prop-2-enyl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H25N5
4-piperidin-1-yl-6-prop-2-enyl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine —— C24H27N5O3S
4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine
—— ethyl 1-(6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C23H29N5O2
ethyl 1-(6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— Ethyl 1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C20H25N5O2
Ethyl 1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— 6-prop-2-enyl-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23N5
6-prop-2-enyl-2-pyridin-3-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 2-Pyridin-2-yl-4-pyrrolidin-1-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine —— C16H19N5
2-Pyridin-2-yl-4-pyrrolidin-1-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— [4-(azepan-1-yl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(3-methoxyphenyl)methanone —— C26H29N5O2
[4-(azepan-1-yl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(3-methoxyphenyl)methanone
—— ethyl 1-[6-(ethylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C23H30N6O3
ethyl 1-[6-(ethylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— 6-prop-2-enyl-2-pyridin-2-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23N5
6-prop-2-enyl-2-pyridin-2-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— ethyl 1-[6-[(3-cyanophenyl)carbamoyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H29N7O3
ethyl 1-[6-[(3-cyanophenyl)carbamoyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— Ethane ethyl 1-{6-[2-(benzenesulfonyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl}piperidine-4-carboxylate —— C28H33N5O4S
Ethane ethyl 1-{6-[2-(benzenesulfonyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl}piperidine-4-carboxylate
—— ethyl 1-[2-pyridin-2-yl-6-(thiophene-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C25H27N5O3S
ethyl 1-[2-pyridin-2-yl-6-(thiophene-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— 4-(azepan-1-yl)-2-pyridin-3-yl-6-(pyridin-3-ylmethyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C24H28N6
4-(azepan-1-yl)-2-pyridin-3-yl-6-(pyridin-3-ylmethyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine —— C24H27N5O3S
4-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]morpholine
—— 6-[2-(benzenesulfonyl)ethyl]-4-piperidin-1-yl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C25H29N5O2S
6-[2-(benzenesulfonyl)ethyl]-4-piperidin-1-yl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C24H27N5O2S
6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-4-pyrrolidin-1-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)morpholine —— C19H23N5O
4-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)morpholine
—— ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O4S
ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— 6-[2-(benzenesulfonyl)ethyl]-4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C25H29N5O2S
6-[2-(benzenesulfonyl)ethyl]-4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— ethyl 1-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C23H29N5O2
ethyl 1-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— ethyl 1-[6-[(3-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O3
ethyl 1-[6-[(3-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O4S
ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— 6-[2-(benzenesulfonyl)ethyl]-4-(4-methylpiperazin-1-yl)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C25H30N6O2S
6-[2-(benzenesulfonyl)ethyl]-4-(4-methylpiperazin-1-yl)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 4-(4-methylpiperazin-1-yl)-6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N6
4-(4-methylpiperazin-1-yl)-6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— ethyl 1-[6-(benzenesulfonylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C27H30N6O5S
ethyl 1-[6-(benzenesulfonylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— N-cyclohexyl-4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide —— C24H32N6O
N-cyclohexyl-4-piperidin-1-yl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide
—— ethyl 1-(2-pyridin-2-yl-6-thiophen-2-ylsulfonyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C24H27N5O4S2
ethyl 1-(2-pyridin-2-yl-6-thiophen-2-ylsulfonyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— 4-(4-methylpiperazin-1-yl)-6-prop-2-enyl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N6
4-(4-methylpiperazin-1-yl)-6-prop-2-enyl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine