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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1R)-1-[6-(2-amino-4-nitrophenyl)-3-chloropyridazin-4-yl]but-3-enyl]carbamate —— C15H13ClN5O4-
N-[(1R)-1-[6-(2-amino-4-nitrophenyl)-3-chloropyridazin-4-yl]but-3-enyl]carbamate
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2R)-2-hydroxypropyl]benzenesulfonamide —— C19H19FN4O3S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2R)-2-hydroxypropyl]benzenesulfonamide
—— 5-[4-[2-(6-Aminopyrazin-2-yl)sulfanylphenyl]-2-fluorophenyl]pyrimidin-2-amine;formic acid —— C21H17FN6O2S
5-[4-[2-(6-Aminopyrazin-2-yl)sulfanylphenyl]-2-fluorophenyl]pyrimidin-2-amine;formic acid
—— 2-({3-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]pyridin-2-yl}oxy)ethanol —— C17H15FN4O2
2-({3-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]pyridin-2-yl}oxy)ethanol
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-4-(trifluoromethyl)biphenyl-2-ol —— C17H11F4N3O
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-4-(trifluoromethyl)biphenyl-2-ol
—— 5-(3-fluoro-2'-{[(3R)-3-methylmorpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine —— C22H21FN4O2
5-(3-fluoro-2'-{[(3R)-3-methylmorpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine
—— 5-[2-Fluoro-3-(1-methylbenzimidazol-2-yl)sulfonyl-4-phenylphenyl]pyrimidin-2-amine —— C24H18FN5O2S
5-[2-Fluoro-3-(1-methylbenzimidazol-2-yl)sulfonyl-4-phenylphenyl]pyrimidin-2-amine
—— 6-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]oxy}pyridine-2-carbonitrile —— C22H14FN5O
6-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]oxy}pyridine-2-carbonitrile
—— 5-{3-fluoro-2'-[(5-methoxypyrimidin-2-yl)oxy]biphenyl-4-yl}pyrimidin-2-amine —— C21H16FN5O2
5-{3-fluoro-2'-[(5-methoxypyrimidin-2-yl)oxy]biphenyl-4-yl}pyrimidin-2-amine
—— 5-(4-Bromo-2-fluorophenyl)-6-cyanopyrazin-2-amine —— C11H6BrFN4
5-(4-Bromo-2-fluorophenyl)-6-cyanopyrazin-2-amine
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(3R)-2-oxopiperidin-3-yl]biphenyl-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C21H20FN5O3S
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(3R)-2-oxopiperidin-3-yl]biphenyl-2-sulfonamide trifluoroacetic acid salt
—— [[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-[(3S)-2-oxopiperidin-3-yl]amino] 2,2,2-trifluoroacetate —— C23H19F4N5O5S
[[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-[(3S)-2-oxopiperidin-3-yl]amino] 2,2,2-trifluoroacetate
—— 1-{[4'-(2-Aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-N-methylazetidine-3-carboxamide —— C21H20FN5O3S
1-{[4'-(2-Aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-N-methylazetidine-3-carboxamide
—— 5-{4-[2-(cyclopropylsulfonyl)pyridin-3-yl]-2-fluorophenyl}pyrimidin-2-amine —— C18H15FN4O2S
5-{4-[2-(cyclopropylsulfonyl)pyridin-3-yl]-2-fluorophenyl}pyrimidin-2-amine
—— 4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-methylpiperazine-1-carboxylic acid —— C22H22FN5O4S
4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-methylpiperazine-1-carboxylic acid
—— 5-[2-fluoro-3-[3-(trifluoromethyl)phenyl]phenyl]-N-methylpyrimidin-2-amine —— C18H13F4N3
5-[2-fluoro-3-[3-(trifluoromethyl)phenyl]phenyl]-N-methylpyrimidin-2-amine
—— 5-[4-(2-Cyclopropylsulfonylpyridin-3-yl)-2-fluorophenyl]pyrimidin-2-amine;formic acid —— C19H17FN4O4S
5-[4-(2-Cyclopropylsulfonylpyridin-3-yl)-2-fluorophenyl]pyrimidin-2-amine;formic acid
—— 2-[4-(2-amino-4-methylpyrimidin-5-yl)-3-fluorophenyl]-N-tert-butylbenzenesulfonamide;2,2,2-trifluoroacetic acid —— C23H24F4N4O4S
2-[4-(2-amino-4-methylpyrimidin-5-yl)-3-fluorophenyl]-N-tert-butylbenzenesulfonamide;2,2,2-trifluoroacetic acid
—— 5-[3-fluoro-2'-(pyrimidin-4-ylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine —— C20H14FN5O2S
5-[3-fluoro-2'-(pyrimidin-4-ylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine
—— 5-[3-fluoro-2'-(methylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine trifluoroacetic acid salt —— (x)C2HF3O2*C17H14FN3O2S
5-[3-fluoro-2'-(methylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine trifluoroacetic acid salt
—— racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine —— C22H18F4N4O2
racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrimidin-2-amine
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(2-hydroxy-2-methylpropyl)biphenyl-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C20H21FN4O3S
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(2-hydroxy-2-methylpropyl)biphenyl-2-sulfonamide trifluoroacetic acid salt
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]benzenesulfonamide —— C21H23FN4O3S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]benzenesulfonamide
—— [[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-[(3R)-2-oxopiperidin-3-yl]amino] 2,2,2-trifluoroacetate —— C23H19F4N5O5S
[[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-[(3R)-2-oxopiperidin-3-yl]amino] 2,2,2-trifluoroacetate
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-(2-hydroxy-2-methylpropyl)benzenesulfonamide —— C20H21FN4O3S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-(2-hydroxy-2-methylpropyl)benzenesulfonamide
—— racemic [2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]phenyl]-[2-(hydroxymethyl)morpholin-4-yl]methanone —— C22H21FN4O3
racemic [2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]phenyl]-[2-(hydroxymethyl)morpholin-4-yl]methanone
—— 5-(4-{2-[(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)oxy]pyridin-3-yl}-2-fluorophenyl)pyrimidin-2-amine —— C20H19FN4O3S
5-(4-{2-[(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)oxy]pyridin-3-yl}-2-fluorophenyl)pyrimidin-2-amine
—— 5-[4-[2-(1,1-Dihydroxythian-4-yl)sulfonylphenyl]-2-fluorophenyl]pyrimidin-2-amine;hydrochloride —— C21H23ClFN3O4S2
5-[4-[2-(1,1-Dihydroxythian-4-yl)sulfonylphenyl]-2-fluorophenyl]pyrimidin-2-amine;hydrochloride
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]benzenesulfonamide;2,2,2-trifluoroacetic acid —— C26H19F7N4O4S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]benzenesulfonamide;2,2,2-trifluoroacetic acid
—— [[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-ethylamino] 2,2,2-trifluoroacetate —— C20H16F4N4O4S
[[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-ethylamino] 2,2,2-trifluoroacetate
—— 1-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-3,3-dimethylbutan-2-one —— C22H22FN3O3S
1-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-3,3-dimethylbutan-2-one
—— 5-[3-fluoro-2'-(2-methoxypyrimidin-5-yl)biphenyl-4-yl]pyrazin-2-amine —— C21H16FN5O
5-[3-fluoro-2'-(2-methoxypyrimidin-5-yl)biphenyl-4-yl]pyrazin-2-amine
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-ethylbenzenesulfonamide —— C18H17FN4O2S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-ethylbenzenesulfonamide
—— (R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-methylpiperazine-1-carboxylate —— C26H30FN5O4S
(R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-methylpiperazine-1-carboxylate
—— 5-[4-(2-Tert-butylsulfonylpyridin-3-yl)-2-fluorophenyl]pyrimidin-2-amine;formic acid —— C20H21FN4O4S
5-[4-(2-Tert-butylsulfonylpyridin-3-yl)-2-fluorophenyl]pyrimidin-2-amine;formic acid
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(2-hydroxy-1,1-dimethylethyl)biphenyl-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C20H21FN4O3S
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(2-hydroxy-1,1-dimethylethyl)biphenyl-2-sulfonamide trifluoroacetic acid salt
—— 5-{3-fluoro-2'-[(4-methylpiperazin-1-yl)sulfonyl]-4'-(trifluoromethyl)biphenyl-4-yl}pyrimidin-2-amine —— C22H21F4N5O2S
5-{3-fluoro-2'-[(4-methylpiperazin-1-yl)sulfonyl]-4'-(trifluoromethyl)biphenyl-4-yl}pyrimidin-2-amine
—— 5-(3-fluoro-2'-{[(2R)-2-methylpiperazin-1-yl]sulfonyl}biphenyl-4-yl)pyrimidin-2-amine —— C21H22FN5O2S
5-(3-fluoro-2'-{[(2R)-2-methylpiperazin-1-yl]sulfonyl}biphenyl-4-yl)pyrimidin-2-amine
—— Tert-butyl 4-[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-methylpiperazine-1-carboxylate —— C26H30FN5O4S
Tert-butyl 4-[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-methylpiperazine-1-carboxylate
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(3-hydroxy-2,2-dimethylpropyl)biphenyl-2-sulfonamide —— C21H23FN4O3S
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-(3-hydroxy-2,2-dimethylpropyl)biphenyl-2-sulfonamide
—— 4'-(2-aminopyrimidin-5-yl)-N-(tert-butyl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C20H21FN4O2S
4'-(2-aminopyrimidin-5-yl)-N-(tert-butyl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide trifluoroacetic acid salt
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]-N-tert-butyl-5-(trifluoromethyl)benzamide —— C22H20F4N4O
2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]-N-tert-butyl-5-(trifluoromethyl)benzamide
—— 5-[2-Fluoro-4-[2-(2-morpholin-4-ylethylsulfonyl)pyridin-3-yl]phenyl]pyrimidin-2-amine;formic acid —— C22H24FN5O5S
5-[2-Fluoro-4-[2-(2-morpholin-4-ylethylsulfonyl)pyridin-3-yl]phenyl]pyrimidin-2-amine;formic acid
—— 2-(((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)methyl)quinazolin-4(3H)-one —— C25H18FN5O3S
2-(((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)methyl)quinazolin-4(3H)-one
—— N-tert-butyl-5-(2-fluoro-3-phenylphenyl)-4-(trifluoromethyl)pyrimidin-2-amine —— C21H19F4N3
N-tert-butyl-5-(2-fluoro-3-phenylphenyl)-4-(trifluoromethyl)pyrimidin-2-amine
—— 5-[2'-(5-aminopyrazin-2-yl)-3-fluorobiphenyl-4-yl]pyrimidin-2-amine —— C20H15FN6
5-[2'-(5-aminopyrazin-2-yl)-3-fluorobiphenyl-4-yl]pyrimidin-2-amine
—— [(1S)-1-[3-chloro-6-[4-(methoxycarbonylamino)-2-(2-methylbut-3-enoylamino)phenyl]pyridazin-4-yl]but-3-enyl]carbamic acid —— C22H24ClN5O5
[(1S)-1-[3-chloro-6-[4-(methoxycarbonylamino)-2-(2-methylbut-3-enoylamino)phenyl]pyridazin-4-yl]but-3-enyl]carbamic acid
—— 2-[4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonylpiperazin-1-yl]ethyl 2,2,2-trifluoroacetate —— C24H23F4N5O4S
2-[4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonylpiperazin-1-yl]ethyl 2,2,2-trifluoroacetate
—— [2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]-5-(trifluoromethyl)phenyl]-(1,1-dioxo-1,4-thiazinan-4-yl)methanone —— C22H18F4N4O3S
[2-[4-(2-aminopyrimidin-5-yl)-3-fluoro-phenyl]-5-(trifluoromethyl)phenyl]-(1,1-dioxo-1,4-thiazinan-4-yl)methanone
—— N-[(1S)-1-[3-chloro-6-[2-(2-methylbut-3-enoylamino)-4-nitrophenyl]pyridazin-4-yl]but-3-enyl]carbamate —— C20H19ClN5O5-
N-[(1S)-1-[3-chloro-6-[2-(2-methylbut-3-enoylamino)-4-nitrophenyl]pyridazin-4-yl]but-3-enyl]carbamate