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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylcarbamate —— C27H30F2N8O2
methyl N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylcarbamate
—— 3-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-propan-2-yloxyphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]oxypropanenitrile —— C29H32F2N8O2
3-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-propan-2-yloxyphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]oxypropanenitrile
—— 4-amino-1-[(2R,3R,4S,5S)-3-azido-5-ethyl-5-fluoro-3,4-dimethyloxolan-2-yl]pyrimidin-2-one —— C12H17FN6O2
4-amino-1-[(2R,3R,4S,5S)-3-azido-5-ethyl-5-fluoro-3,4-dimethyloxolan-2-yl]pyrimidin-2-one
—— N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-(2,6-difluoro-4-propan-2-yloxyphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]acetamide —— C29H33F2N7O2
N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-(2,6-difluoro-4-propan-2-yloxyphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]acetamide
—— methyl N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-[2,6-difluoro-4-(oxolan-3-yloxy)phenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]-N-methylcarbamate —— C31H35F2N7O4
methyl N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-[2,6-difluoro-4-(oxolan-3-yloxy)phenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]-N-methylcarbamate
—— 1-[(2R,3R,4R,5R)-3-chloro-5-ethyl-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione —— C12H17ClN2O3
1-[(2R,3R,4R,5R)-3-chloro-5-ethyl-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione
—— N-[4-[(1R,3S)-3-aminocyclohexyl]pyridin-3-yl]-2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-amine —— C24H24F2N6
N-[4-[(1R,3S)-3-aminocyclohexyl]pyridin-3-yl]-2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-amine
—— 4-amino-1-[(2R,3R,4S,5S)-5-ethyl-3,5-difluoro-3,4-dimethyloxolan-2-yl]pyrimidin-2-one —— C12H17F2N3O2
4-amino-1-[(2R,3R,4S,5S)-5-ethyl-3,5-difluoro-3,4-dimethyloxolan-2-yl]pyrimidin-2-one
—— 1-[(2R,3R,4S,5S)-5-ethyl-3,5-difluoro-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione —— C12H16F2N2O3
1-[(2R,3R,4S,5S)-5-ethyl-3,5-difluoro-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione
—— N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylsulfonylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylacetamide —— C27H30F2N8O3S
N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylsulfonylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylacetamide
—— N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]acetamide —— C26H28F2N8O
N-[(3R,4S,5S)-3-amino-1-[3-[[2-(2,6-difluoro-4-methylphenyl)imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]acetamide
—— N-[4-[(1R,3R,4S,5S)-3-amino-5-methyl-4-methylsulfonylcyclohexyl]pyridin-3-yl]-2-[2,6-difluoro-4-(oxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-amine —— C28H30F2N6O3S
N-[4-[(1R,3R,4S,5S)-3-amino-5-methyl-4-methylsulfonylcyclohexyl]pyridin-3-yl]-2-[2,6-difluoro-4-(oxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-amine
—— 1-[(2R,3R,4R,5R)-3-chloro-5-fluoro-5-(hydroxymethyl)-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione —— C11H14ClFN2O4
1-[(2R,3R,4R,5R)-3-chloro-5-fluoro-5-(hydroxymethyl)-3,4-dimethyloxolan-2-yl]pyrimidine-2,4-dione
—— N-[(3R,4S,5S)-3-amino-1-[3-[[2-[4-(4-cyanooxan-4-yl)-2,6-difluorophenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylacetamide —— C32H35F2N9O2
N-[(3R,4S,5S)-3-amino-1-[3-[[2-[4-(4-cyanooxan-4-yl)-2,6-difluorophenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-5-methylpiperidin-4-yl]-N-methylacetamide
—— N-[4-[(3R,4S,5S)-3-amino-5-methyl-4-methylsulfonylcyclohexyl]pyridin-3-yl]-2-[4-(ethoxymethyl)-2,6-difluorophenyl]imidazo[1,5-b]pyridazin-7-amine —— C28H32F2N6O3S
N-[4-[(3R,4S,5S)-3-amino-5-methyl-4-methylsulfonylcyclohexyl]pyridin-3-yl]-2-[4-(ethoxymethyl)-2,6-difluorophenyl]imidazo[1,5-b]pyridazin-7-amine
—— N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-[2,6-difluoro-4-(3-fluorooxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]acetamide —— C29H30F3N7O2
N-[(1S,2R,4R,6S)-2-amino-4-[3-[[2-[2,6-difluoro-4-(3-fluorooxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-yl]amino]pyridin-4-yl]-6-methylcyclohexyl]acetamide
—— N-[4-[(1R,3S,5S)-3-amino-5-methylcyclohexyl]pyridin-3-yl]-2-[2,6-difluoro-4-(oxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-amine —— C27H28F2N6O
N-[4-[(1R,3S,5S)-3-amino-5-methylcyclohexyl]pyridin-3-yl]-2-[2,6-difluoro-4-(oxetan-3-yl)phenyl]imidazo[1,5-b]pyridazin-7-amine
—— N'-[(E)-(4-ethoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-4,6-diphenylpyrimidine-2-carbohydrazide —— C26H22N4O3
N'-[(E)-(4-ethoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-4,6-diphenylpyrimidine-2-carbohydrazide
—— N'-methyl-N-pyrimidin-4-ylmethanimidamide —— C6H8N4
N'-methyl-N-pyrimidin-4-ylmethanimidamide
—— N-[4-[(6-methylpyrimidin-4-yl)amino]cyclohexyl]acetamide —— C13H20N4O
N-[4-[(6-methylpyrimidin-4-yl)amino]cyclohexyl]acetamide
—— 6-(2-hydroxyethylamino)-2-[2-methoxyethyl(methyl)amino]-N-[3-(methylamino)propyl]pyrimidine-4-carboxamide —— C15H28N6O3
6-(2-hydroxyethylamino)-2-[2-methoxyethyl(methyl)amino]-N-[3-(methylamino)propyl]pyrimidine-4-carboxamide
—— N-(azetidin-3-yl)-2-tert-butyl-6-propan-2-ylpyrimidin-4-amine —— C14H24N4
N-(azetidin-3-yl)-2-tert-butyl-6-propan-2-ylpyrimidin-4-amine
—— 3-(4,6-Dimethylpyrimidin-2-yl)-1-[4-[4-(4-methylphenyl)phthalazin-1-yl]piperazin-1-yl]propan-1-one —— C28H30N6O
3-(4,6-Dimethylpyrimidin-2-yl)-1-[4-[4-(4-methylphenyl)phthalazin-1-yl]piperazin-1-yl]propan-1-one
—— 4-(3-Methyl-5-phenylphenyl)-2,6-diphenylpyrimidine —— C29H22N2
4-(3-Methyl-5-phenylphenyl)-2,6-diphenylpyrimidine
—— 1-N-(6-ethylpyrimidin-4-yl)-4-N,4-N-dimethylcyclohexane-1,4-diamine —— C14H24N4
1-N-(6-ethylpyrimidin-4-yl)-4-N,4-N-dimethylcyclohexane-1,4-diamine
—— methyl 4-[3-[4-[[7-[(1E,3E)-2,4-bis(trifluoromethyl)hexa-1,3,5-trienyl]-5-oxo-6-oxa-4-azaspiro[2.4]heptan-4-yl]methyl]-2-methylsulfanylpyrimidin-5-yl]-4-methoxyphenyl]-3-methylbenzoate —— C35H31F6N3O5S
methyl 4-[3-[4-[[7-[(1E,3E)-2,4-bis(trifluoromethyl)hexa-1,3,5-trienyl]-5-oxo-6-oxa-4-azaspiro[2.4]heptan-4-yl]methyl]-2-methylsulfanylpyrimidin-5-yl]-4-methoxyphenyl]-3-methylbenzoate
—— N-[(3S)-oxolan-3-yl]-6-propan-2-ylpyrimidin-4-amine —— C11H17N3O
N-[(3S)-oxolan-3-yl]-6-propan-2-ylpyrimidin-4-amine
—— N-(azetidin-3-yl)-2-tert-butyl-6-methylpyrimidin-4-amine —— C12H20N4
N-(azetidin-3-yl)-2-tert-butyl-6-methylpyrimidin-4-amine
—— 6-ethyl-2-methoxy-N-(oxetan-3-yl)pyrimidin-4-amine —— C10H15N3O2
6-ethyl-2-methoxy-N-(oxetan-3-yl)pyrimidin-4-amine
—— 6-ethyl-5-methyl-N-(oxetan-3-yl)pyrimidin-4-amine —— C10H15N3O
6-ethyl-5-methyl-N-(oxetan-3-yl)pyrimidin-4-amine
—— 8-[3,5-bis(trifluoromethyl)phenyl]-5-({5-[4-fluoro-2-methoxy-5-(propan-2-yl)phenyl]-2-(methylsulfanyl)pyrimidin-4-yl} methyl)-7-oxa-5-azaspiro[3.4]octan-6-one 1616347-74-0 C30H28F7N3O3S
8-[3,5-bis(trifluoromethyl)phenyl]-5-({5-[4-fluoro-2-methoxy-5-(propan-2-yl)phenyl]-2-(methylsulfanyl)pyrimidin-4-yl} methyl)-7-oxa-5-azaspiro[3.4]octan-6-one
—— 1-[3-[(2,6-Dimethylpyrimidin-4-yl)amino]azetidin-1-yl]ethanone —— C11H16N4O
1-[3-[(2,6-Dimethylpyrimidin-4-yl)amino]azetidin-1-yl]ethanone
—— 1-[(1R,2R,3S,4S)-4-fluoro-1,2,3,5-tetrahydroxy-2-methylpentyl]pyrimidine-2,4-dione —— C10H15FN2O6
1-[(1R,2R,3S,4S)-4-fluoro-1,2,3,5-tetrahydroxy-2-methylpentyl]pyrimidine-2,4-dione
—— N'-[(E)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-4,6-dimethylpyrimidine-2-carbohydrazide —— C15H16N4O3
N'-[(E)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-4,6-dimethylpyrimidine-2-carbohydrazide
—— [[(2S,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-2,4-difluoro-3-hydroxy-4-prop-1-en-2-yloxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate —— C12H17F2N2O14P3
[[(2S,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-2,4-difluoro-3-hydroxy-4-prop-1-en-2-yloxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
—— 4-amino-1-[(2R,3R,5R)-3-azido-5-fluoro-5-(hydroxymethyl)-3-methyloxolan-2-yl]pyrimidin-2-one —— C10H13FN6O3
4-amino-1-[(2R,3R,5R)-3-azido-5-fluoro-5-(hydroxymethyl)-3-methyloxolan-2-yl]pyrimidin-2-one
—— 4-[(2-Butoxy-4,6-dimethylpyridin-3-yl)methyl]-6-methyl-9-[2-(methylamino)pyrimidin-5-yl]-7-propan-2-yloxy-2,3-dihydro-1,4-benzoxazepin-5-one —— C30H39N5O4
4-[(2-Butoxy-4,6-dimethylpyridin-3-yl)methyl]-6-methyl-9-[2-(methylamino)pyrimidin-5-yl]-7-propan-2-yloxy-2,3-dihydro-1,4-benzoxazepin-5-one
—— 1-methyl-2-[4-(methylamino)-6,7,8,9-tetrahydro-5H-cyclohepta[d]pyrimidin-2-yl]cyclohexane-1-carboxylic acid —— C18H27N3O2
1-methyl-2-[4-(methylamino)-6,7,8,9-tetrahydro-5H-cyclohepta[d]pyrimidin-2-yl]cyclohexane-1-carboxylic acid
—— 6-methyl-N-[1-(2-methylsulfonylethyl)azetidin-3-yl]pyrimidin-4-amine —— C11H18N4O2S
6-methyl-N-[1-(2-methylsulfonylethyl)azetidin-3-yl]pyrimidin-4-amine
—— N-methyl-N-[4-[(6-methylpyrimidin-4-yl)amino]cyclohexyl]acetamide —— C14H22N4O
N-methyl-N-[4-[(6-methylpyrimidin-4-yl)amino]cyclohexyl]acetamide
—— 3-Ethyl-[1,2]thiazolo[4,5-c]pyridazine —— C7H7N3S
3-Ethyl-[1,2]thiazolo[4,5-c]pyridazine
—— 2-[butyl(methyl)amino]-6-(2-methoxyethylamino)-N-methylpyrimidine-4-carboxamide —— C14H25N5O2
2-[butyl(methyl)amino]-6-(2-methoxyethylamino)-N-methylpyrimidine-4-carboxamide
—— 6-(2-Methoxyethylamino)pyrimidine-4-carbaldehyde —— C8H11N3O2
6-(2-Methoxyethylamino)pyrimidine-4-carbaldehyde
—— N-(azetidin-3-yl)-6-ethyl-2-methoxypyrimidin-4-amine —— C10H16N4O
N-(azetidin-3-yl)-6-ethyl-2-methoxypyrimidin-4-amine
—— [1,2]Thiazolo[5,4-c]pyridazine —— C5H3N3S
[1,2]Thiazolo[5,4-c]pyridazine
—— 1-[3-[(6-Methylpyrimidin-4-yl)amino]azetidin-1-yl]propan-1-one —— C11H16N4O
1-[3-[(6-Methylpyrimidin-4-yl)amino]azetidin-1-yl]propan-1-one
—— Cyclobutyl-[3-[(6-propan-2-ylpyrimidin-4-yl)amino]azetidin-1-yl]methanone —— C15H22N4O
Cyclobutyl-[3-[(6-propan-2-ylpyrimidin-4-yl)amino]azetidin-1-yl]methanone
—— N-[3-(2-methoxyethoxy)cyclobutyl]-6-propan-2-ylpyrimidin-4-amine —— C14H23N3O2
N-[3-(2-methoxyethoxy)cyclobutyl]-6-propan-2-ylpyrimidin-4-amine
—— (5E)-1-[(4-fluorophenyl)methyl]-5-[(3-hydroxypropylamino)methylidene]-1,3-diazinane-2,4,6-trione —— C15H16FN3O4
(5E)-1-[(4-fluorophenyl)methyl]-5-[(3-hydroxypropylamino)methylidene]-1,3-diazinane-2,4,6-trione
—— 5-methyl-N-(oxan-4-yl)pyridazin-3-amine —— C10H15N3O
5-methyl-N-(oxan-4-yl)pyridazin-3-amine