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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,5-dimethyl-3-propan-2-yl-7,8-dihydro-6H-imidazo[1,2-b]pyridazine —— C11H19N3
2,5-dimethyl-3-propan-2-yl-7,8-dihydro-6H-imidazo[1,2-b]pyridazine
—— 2,3,5-trimethyl-7,8-dihydro-6H-imidazo[1,2-b]pyridazine —— C9H15N3
2,3,5-trimethyl-7,8-dihydro-6H-imidazo[1,2-b]pyridazine
—— N-[(4-chloro-2-fluorophenyl)methyl]-4-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-2-amine —— C17H11ClF4N4
N-[(4-chloro-2-fluorophenyl)methyl]-4-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-2-amine
—— 3-[2-(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)hydrazinyl]benzoate —— C11H7N4O4S-
3-[2-(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)hydrazinyl]benzoate
—— N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine —— C18H14F4N4
N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine
—— N-[(2,4-difluorophenyl)methyl]-2-(2-fluoropyridin-3-yl)pyrimidin-4-amine —— C16H11F3N4
N-[(2,4-difluorophenyl)methyl]-2-(2-fluoropyridin-3-yl)pyrimidin-4-amine
—— 6-(2,4-difluoro-N-methylanilino)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C23H19F5N6O3
6-(2,4-difluoro-N-methylanilino)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— 6-(2,4-difluoro-N-methylanilino)-N-(4-oxocyclohexyl)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C24H20F5N5O2
6-(2,4-difluoro-N-methylanilino)-N-(4-oxocyclohexyl)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— 2-[4-(2-aminopyrimidin-5-yl)-2,3-difluorophenyl]-N-methylbenzenesulfonamide;2,2,2-trifluoroacetic acid —— C19H15F5N4O4S
2-[4-(2-aminopyrimidin-5-yl)-2,3-difluorophenyl]-N-methylbenzenesulfonamide;2,2,2-trifluoroacetic acid
—— 4-[[[2-[5-(Trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one —— C19H14F3N5O
4-[[[2-[5-(Trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one
—— 5-[3-fluoro-2'-(morpholin-4-ylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine trifluoroacetic acid salt —— (x)C2HF3O2*C20H19FN4O3S
5-[3-fluoro-2'-(morpholin-4-ylsulfonyl)biphenyl-4-yl]pyrimidin-2-amine trifluoroacetic acid salt
—— 2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2R)-1-hydroxypropan-2-yl]benzenesulfonamide;2,2,2-trifluoroacetic acid —— C21H20F4N4O5S
2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]-N-[(2R)-1-hydroxypropan-2-yl]benzenesulfonamide;2,2,2-trifluoroacetic acid
—— 6-(2,4-difluoro-N-methylanilino)-N-[(1-pyridin-3-ylcyclopentyl)methyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C29H25F5N6O
6-(2,4-difluoro-N-methylanilino)-N-[(1-pyridin-3-ylcyclopentyl)methyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— 5-[4-[2-(5-Aminopyrimidin-2-yl)sulfonylphenyl]-2-fluorophenyl]pyrimidin-2-amine —— C20H15FN6O2S
5-[4-[2-(5-Aminopyrimidin-2-yl)sulfonylphenyl]-2-fluorophenyl]pyrimidin-2-amine
—— N-methyl-2-phenyl-2-[[2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]acetamide —— C19H16F3N5O
N-methyl-2-phenyl-2-[[2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]acetamide
—— N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine —— C17H20F3N5
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine
—— N-[(2-fluorophenyl)methyl]-2-(2-fluoropyridin-3-yl)pyrimidin-4-amine —— C16H12F2N4
N-[(2-fluorophenyl)methyl]-2-(2-fluoropyridin-3-yl)pyrimidin-4-amine
—— 4-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}piperazin-2-one trifluoroacetic acid salt —— (x)C2HF3O2*C20H18FN5O3S
4-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}piperazin-2-one trifluoroacetic acid salt
—— 6-[(2,4-difluorophenyl)methylamino]-N-[(1-pyridin-3-ylcyclopentyl)methyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C29H25F5N6O
6-[(2,4-difluorophenyl)methylamino]-N-[(1-pyridin-3-ylcyclopentyl)methyl]-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— N-(2,1,3-benzothiadiazol-4-yl)-6-(2,4-difluoro-N-methylanilino)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C24H14F5N7OS
N-(2,1,3-benzothiadiazol-4-yl)-6-(2,4-difluoro-N-methylanilino)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— 4'-(2-aminopyrimidin-5-yl)-N-cyclopropyl-3'-fluorobiphenyl-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C19H17FN4O2S
4'-(2-aminopyrimidin-5-yl)-N-cyclopropyl-3'-fluorobiphenyl-2-sulfonamide trifluoroacetic acid salt
—— [4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-2-oxopiperazin-1-yl] 2,2,2-trifluoroacetate —— C22H17F4N5O5S
[4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-2-oxopiperazin-1-yl] 2,2,2-trifluoroacetate
—— N-[(2-fluorophenyl)methyl]-2-(6-fluoropyridin-3-yl)pyrimidin-4-amine —— C16H12F2N4
N-[(2-fluorophenyl)methyl]-2-(6-fluoropyridin-3-yl)pyrimidin-4-amine
—— (3S)-1-[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonylpyrrolidine-3-carboxamide —— C21H20FN5O3S
(3S)-1-[2-[4-(2-aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonylpyrrolidine-3-carboxamide
—— 2-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-2-methylpropanamide —— C20H19FN4O3S
2-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-2-methylpropanamide
—— 6-(2,4-difluoro-N-methylanilino)-N-imidazo[1,2-a]pyridin-5-yl-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide —— C25H16F5N7O
6-(2,4-difluoro-N-methylanilino)-N-imidazo[1,2-a]pyridin-5-yl-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carboxamide
—— {[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]oxy}acetic acid —— C18H14FN3O3
{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]oxy}acetic acid
—— (3R)-1-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]carbonyl}pyrrolidin-3-ol —— C21H19FN4O2
(3R)-1-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]carbonyl}pyrrolidin-3-ol
—— 5-[3-fluoro-2'-(pyrimidin-2-yloxy)-4'-(trifluoromethyl)biphenyl-4-yl]pyrimidin-2-amine —— C21H13F4N5O
5-[3-fluoro-2'-(pyrimidin-2-yloxy)-4'-(trifluoromethyl)biphenyl-4-yl]pyrimidin-2-amine
—— [[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-cyclopropylamino] 2,2,2-trifluoroacetate —— C21H16F4N4O4S
[[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-cyclopropylamino] 2,2,2-trifluoroacetate
—— 5-[3-fluoro-2'-(morpholin-4-ylcarbonyl)biphenyl-4-yl]pyrimidin-2-amine —— C21H19FN4O2
5-[3-fluoro-2'-(morpholin-4-ylcarbonyl)biphenyl-4-yl]pyrimidin-2-amine
—— N-(2-phenylethyl)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine —— C18H15F3N4
N-(2-phenylethyl)-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine
—— N-[(2,4-difluorophenyl)methyl]-6-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine —— C17H11F5N4
N-[(2,4-difluorophenyl)methyl]-6-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine
—— 5-[4-[2-(1,1-Dihydroxy-1,2-thiazolidin-2-yl)phenyl]-2-fluorophenyl]pyrimidin-2-amine —— C19H19FN4O2S
5-[4-[2-(1,1-Dihydroxy-1,2-thiazolidin-2-yl)phenyl]-2-fluorophenyl]pyrimidin-2-amine
—— 4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-(hydroxymethyl)piperazine-1-carboxylic acid —— C22H22FN5O5S
4-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfonyl-3-(hydroxymethyl)piperazine-1-carboxylic acid
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(1R)-2,2,2-trifluoro-1-methylethyl]biphenyl-2-carboxamide —— C20H16F4N4O
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(1R)-2,2,2-trifluoro-1-methylethyl]biphenyl-2-carboxamide
—— N-methyl-N-pyridin-3-yl-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine —— C16H12F3N5
N-methyl-N-pyridin-3-yl-2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-amine
—— 5-[2'-(1,1-dioxidoisothiazolidin-2-yl)-3-fluorobiphenyl-4-yl]pyrimidin-2-amine —— C19H17FN4O2S
5-[2'-(1,1-dioxidoisothiazolidin-2-yl)-3-fluorobiphenyl-4-yl]pyrimidin-2-amine
—— N-methyl-1-[[[2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]methyl]cyclopropane-1-carboxamide —— C16H16F3N5O
N-methyl-1-[[[2-[5-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]methyl]cyclopropane-1-carboxamide
—— 5-{2'-[(4-aminopyrimidin-2-yl)oxy]-3-fluoro-4'-(trifluoromethyl)biphenyl-4-yl}pyrimidin-2-amine —— C21H14F4N6O
5-{2'-[(4-aminopyrimidin-2-yl)oxy]-3-fluoro-4'-(trifluoromethyl)biphenyl-4-yl}pyrimidin-2-amine
—— 5-(4-chloro-2-fluoro-3-methylphenyl)pyrazin-2-amine —— C11H9ClFN3
5-(4-chloro-2-fluoro-3-methylphenyl)pyrazin-2-amine
—— 5-{3-fluoro-2'-[(3R)-piperidin-3-yloxy]biphenyl-4-yl}pyrimidin-2-amine —— C21H21FN4O
5-{3-fluoro-2'-[(3R)-piperidin-3-yloxy]biphenyl-4-yl}pyrimidin-2-amine
—— 6-[(Z)-(4-chlorophenyl)methylideneamino]-5-methyl-3-phenyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C19H13ClN4OS2
6-[(Z)-(4-chlorophenyl)methylideneamino]-5-methyl-3-phenyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— (1,1-Dioxo-1,4-thiazinan-4-yl)-[2-(3-fluoro-4-pyrimidin-5-ylphenyl)phenyl]methanone —— C21H18FN3O3S
(1,1-Dioxo-1,4-thiazinan-4-yl)-[2-(3-fluoro-4-pyrimidin-5-ylphenyl)phenyl]methanone
—— [[2-[4-(2-Aminopyrimidin-5-yl)-2,3-difluorophenyl]phenyl]sulfonyl-tert-butylamino] 2,2,2-trifluoroacetate —— C22H19F5N4O4S
[[2-[4-(2-Aminopyrimidin-5-yl)-2,3-difluorophenyl]phenyl]sulfonyl-tert-butylamino] 2,2,2-trifluoroacetate
—— 5-[3-fluoro-2'-(pyrazin-2-ylsulfanyl)biphenyl-4-yl]pyrimidin-2-amine hydrochloride —— C20H14FN5S*(x)ClH
5-[3-fluoro-2'-(pyrazin-2-ylsulfanyl)biphenyl-4-yl]pyrimidin-2-amine hydrochloride
—— 5-{2'-[(5-aminopyrimidin-4-yl)sulfonyl]-3-fluorobiphenyl-4-yl}pyrimidin-2-amine hydrochloride —— C20H15FN6O2S*(x)ClH
5-{2'-[(5-aminopyrimidin-4-yl)sulfonyl]-3-fluorobiphenyl-4-yl}pyrimidin-2-amine hydrochloride
—— N-benzyl-2-(5-methoxypyridin-3-yl)pyrimidin-4-amine —— C17H16N4O
N-benzyl-2-(5-methoxypyridin-3-yl)pyrimidin-4-amine
—— 6-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfanylpyrimidin-4-amine;formic acid —— C21H17FN6O2S
6-[2-[4-(2-Aminopyrimidin-5-yl)-3-fluorophenyl]phenyl]sulfanylpyrimidin-4-amine;formic acid
—— 4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(1R)-2,2,2-trifluoro-1-methylethyl]biphenyl-2-sulfonamide trifluoroacetic acid salt —— (x)C2HF3O2*C19H16F4N4O2S
4'-(2-aminopyrimidin-5-yl)-3'-fluoro-N-[(1R)-2,2,2-trifluoro-1-methylethyl]biphenyl-2-sulfonamide trifluoroacetic acid salt