Process for converting a carboxamide to a thiocarboxamide includes reacting (a) a substrate that comprises a heteroatom-containing moiety and a carboxamide moiety with (b) a dialkyl dithiophosphate and/or a salt thereof. The heteroatom-containing moiety includes a heteroatom selected from the group consisting of N, O, and S. Processes for preparing piperidine-4-thiocarboxamide are described.
将羧酰胺转化为
硫代羧酰胺的过程包括将(a)包含杂原子基团和羧酰胺基团的底物与(b)二烷基
二硫代磷酸盐和/或其盐反应。杂原子基团包括从N、O和S组成的杂原子。描述了制备
吡啶-4-
硫代羧酰胺的过程。