申请人:The Upjohn Company
公开号:US04357347A1
公开(公告)日:1982-11-02
Phenylcarbamoylbenzimidates of the formula ##STR1## wherein X.sub.1 is selected from the group consisting of methyl, trifluoromethyl, chlorine, fluorine and bromine; X.sub.2 is selected from the group consisting of hydrogen, methyl, trifluoromethyl, chlorine, fluorine and bromine; R is alkyl of from 1 to 5 carbon atoms; X.sub.3 and X.sub.4 can be the same or different and are selected from the group consisting of hydrogen, chlorine and bromine; X.sub.5 is selected from the group consisting of hydrogen, chlorine, bromine and trifluoromethyl; and X.sub.6 is selected from the group consisting of cyano and nitro; with the proviso that when X.sub.1 and X.sub.2 are chlorine or when X.sub.1 is fluorine and X.sub.2 is hydrogen then R, X.sub.3, X.sub.4, X.sub.5 and X.sub.6 are respectively not 1-methylethyl, chlorine, hydrogen, chlorine and nitro; with the further proviso that when X.sub.1 is fluorine and X.sub.2 is hydrogen then R, X.sub.3, X.sub.4, X.sub.5 and X.sub.6 are respectively not 1-methylethyl, chlorine, hydrogen, hydrogen and nitro; and with the further proviso that when X.sub. 1 is florine or methyl and X.sub.2 is hydrogen then R, X.sub.3, X.sub.4, X.sub.5 and X.sub.6 are respectively not ethyl, hydrogen, hydrogen, hydrogen and nitro; and with the proviso that when X.sub.1 and X.sub.2 are florine, then R, X.sub.3, X.sub.4, X.sub.5 and X.sub.6 are respectively not ethyl, chlorine, hydrogen, chlorine and nitro.
该文本描述了公式为 ##STR1## 的苯基
氨基甲酰
苯并咪唑,其中 X.sub.1 选自甲基、三
氟甲基、
氯、
氟和
溴的群组;X.sub.2 选自氢、甲基、三
氟甲基、
氯、
氟和
溴的群组;R 是1至5个碳原子的烷基;X.sub.3 和 X.sub.4 可以相同也可以不同,选自氢、
氯和
溴的群组;X.sub.5 选自氢、
氯、
溴和三
氟甲基的群组;X.sub.6 选自
氰基和硝基的群组;但是当 X.sub.1 和 X.sub.2 为
氯时,或者当 X.sub.1 为
氟且 X.sub.2 为氢时,那么 R、X.sub.3、X.sub.4、X.sub.5 和 X.sub.6 分别不是1-甲基乙基、
氯、氢、
氯和硝基;进一步地,当 X.sub.1 为
氟且 X.sub.2 为氢时,那么 R、X.sub.3、X.sub.4、X.sub.5 和 X.sub.6 分别不是1-甲基乙基、
氯、氢、氢和硝基;当 X.sub.1 为
氟或甲基且 X.sub.2 为氢时,那么 R、X.sub.3、X.sub.4、X.sub.5 和 X.sub.6 分别不是乙基、氢、氢、氢和硝基;而当 X.sub.1 和 X.sub.2 为
氟时,那么 R、X.sub.3、X.sub.4、X.sub.5 和 X.sub.6 分别不是乙基、
氯、氢、
氯和硝基。