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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (3S)-3-[[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-methylpyrrolidine-1-carboxylate —— C21H28BrN5O4
tert-butyl (3S)-3-[[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-methylpyrrolidine-1-carboxylate
—— Tert-butyl 3-[[1-methyl-2-oxo-3-(2-trimethylsilylethoxymethyl)-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-propan-2-ylazetidine-1-carboxylate —— C28H45N5O5Si
Tert-butyl 3-[[1-methyl-2-oxo-3-(2-trimethylsilylethoxymethyl)-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-propan-2-ylazetidine-1-carboxylate
—— (trans)-2-(2,2-difluoro-benzo[1,3]dioxol-5-yl)-cyclopropanecarboxylic acid ethyl ester —— C13H12F2O4
(trans)-2-(2,2-difluoro-benzo[1,3]dioxol-5-yl)-cyclopropanecarboxylic acid ethyl ester
—— Tert-butyl 2-methyl-3-[(1-methyl-2-oxo-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl)amino]azetidine-1-carboxylate —— C20H29N5O4
Tert-butyl 2-methyl-3-[(1-methyl-2-oxo-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl)amino]azetidine-1-carboxylate
—— tert-butyl 3-[(8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl)-methylamino]-3-methylazetidine-1-carboxylate —— C21H28BrN5O4
tert-butyl 3-[(8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl)-methylamino]-3-methylazetidine-1-carboxylate
—— Tricyclo[5.3.1.03,8]undeca-1(11),5,7,9-tetraen-4-ol —— C11H10O
Tricyclo[5.3.1.03,8]undeca-1(11),5,7,9-tetraen-4-ol
—— tert-butyl (2S,4S)-4-[9H-fluoren-9-yl(methoxycarbonyl)amino]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidine-1-carboxylate —— C35H39N3O5
tert-butyl (2S,4S)-4-[9H-fluoren-9-yl(methoxycarbonyl)amino]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl 3-[[8-[(Z)-2-ethoxyethenyl]-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-methylazetidine-1-carboxylate —— C24H33N5O5
tert-butyl 3-[[8-[(Z)-2-ethoxyethenyl]-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]-3-methylazetidine-1-carboxylate
—— tert-butyl 4-[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]piperidine-1-carboxylate —— C21H27BrN4O4
tert-butyl 4-[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]piperidine-1-carboxylate
—— Tert-butyl 3-((8-bromo-1-methyl-2-oxo-1,2,3,5-tetrahydrobenzo[5,6][1,4]oxazino[3,4-c][1,2,4]triazin-9-yl)amino)-3-methylazetidine-1-carboxylate —— C20H26BrN5O4
Tert-butyl 3-((8-bromo-1-methyl-2-oxo-1,2,3,5-tetrahydrobenzo[5,6][1,4]oxazino[3,4-c][1,2,4]triazin-9-yl)amino)-3-methylazetidine-1-carboxylate
—— tert-butyl 3-methyl-3-[2-[(1S)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]ethyl]azetidine-1-carboxylate —— C22H30N4O4
tert-butyl 3-methyl-3-[2-[(1S)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]ethyl]azetidine-1-carboxylate
—— tert-butyl 4-[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]piperidine-1-carboxylate —— C21H28N4O4
tert-butyl 4-[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]piperidine-1-carboxylate
—— Tetradecan-3-yl 2-bromopropanoate —— C17H33BrO2
Tetradecan-3-yl 2-bromopropanoate
—— Tert-butyl 2-methyl-3-[(1-methyl-2-oxo-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-3-yl)amino]azetidine-1-carboxylate —— C20H27N5O4
Tert-butyl 2-methyl-3-[(1-methyl-2-oxo-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-3-yl)amino]azetidine-1-carboxylate
—— tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]carbamate —— C26H28BrN3O4
tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]carbamate
—— tert-butyl N-[5-[(2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]carbamate —— C26H29N3O4
tert-butyl N-[5-[(2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]carbamate
—— (trans)-2-(5-formyl-furan-2-yl)-cyclopropanecarboxylic acid ethyl ester —— C11H12O4
(trans)-2-(5-formyl-furan-2-yl)-cyclopropanecarboxylic acid ethyl ester
—— tert-butyl N-[1-[[(3S)-5-[(S)-(2-cyanophenyl)-(2H-indazol-3-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate —— C33H35N7O4
tert-butyl N-[1-[[(3S)-5-[(S)-(2-cyanophenyl)-(2H-indazol-3-yl)methyl]-4-oxo-2,3-dihydro-1H-1,5-benzodiazepin-3-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl 4-[[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]methyl]piperidine-1-carboxylate —— C22H29BrN4O4
tert-butyl 4-[[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]methyl]piperidine-1-carboxylate
—— tert-butyl (2S)-2-[[[(4S)-9-sulfooxy-7-oxa-5,9-diazatricyclo[3.2.1.11,6]nonane-4-carbonyl]amino]oxymethyl]piperidine-1-carboxylate —— C18H30N4O9S
tert-butyl (2S)-2-[[[(4S)-9-sulfooxy-7-oxa-5,9-diazatricyclo[3.2.1.11,6]nonane-4-carbonyl]amino]oxymethyl]piperidine-1-carboxylate
—— (trans)-2-(2-fluoropyridin-4-yl)-cyclopropanecarboxylic acid ethyl ester —— C11H12FNO2
(trans)-2-(2-fluoropyridin-4-yl)-cyclopropanecarboxylic acid ethyl ester
—— tert-butyl 2-[[(1S)-8-fluoro-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]azetidine-1-carboxylate —— C19H24FN5O4
tert-butyl 2-[[(1S)-8-fluoro-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]azetidine-1-carboxylate
—— tert-butyl N-[1-cyclohexyl-2-[(2S,4S)-4-(9H-fluoren-9-ylmethoxycarbonylamino)-2-(1,2,3,4-tetrahydronaphthalen-1-ylcarbamoyl)pyrrolidin-1-yl]-2-oxoethyl]carbamate —— C43H52N4O6
tert-butyl N-[1-cyclohexyl-2-[(2S,4S)-4-(9H-fluoren-9-ylmethoxycarbonylamino)-2-(1,2,3,4-tetrahydronaphthalen-1-ylcarbamoyl)pyrrolidin-1-yl]-2-oxoethyl]carbamate
—— Tert-butyl-[4-(2-ethylphenoxy)butyl]azanium —— C16H28NO+
Tert-butyl-[4-(2-ethylphenoxy)butyl]azanium
—— tert-butyl 3-[(1,8-dimethyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl)methylamino]azetidine-1-carboxylate —— C21H29N5O4
tert-butyl 3-[(1,8-dimethyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl)methylamino]azetidine-1-carboxylate
—— tert-butyl (3S)-3-[[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]pyrrolidine-1-carboxylate —— C20H27N5O4
tert-butyl (3S)-3-[[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]pyrrolidine-1-carboxylate
—— tert-butyl N-[3-[5-bromo-2-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propoxy]-3-propoxyphenoxy]propyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate —— C30H49BrN2O9
tert-butyl N-[3-[5-bromo-2-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propoxy]-3-propoxyphenoxy]propyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— tert-butyl N-[2-[3-(4-amino-2-but-2-ynylphenoxy)-5-(trifluoromethyl)anilino]ethyl]carbamate —— C24H28F3N3O3
tert-butyl N-[2-[3-(4-amino-2-but-2-ynylphenoxy)-5-(trifluoromethyl)anilino]ethyl]carbamate
—— tert-butyl 4-[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]-3-methylpiperidine-1-carboxylate —— C22H29BrN4O4
tert-butyl 4-[(1R)-8-bromo-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]-3-methylpiperidine-1-carboxylate
—— tert-butyl (3R)-3-[[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]pyrrolidine-1-carboxylate —— C20H27N5O4
tert-butyl (3R)-3-[[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]amino]pyrrolidine-1-carboxylate
—— tert-butyl N-[2-(2-aminopropylamino)propyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate —— C16H33N3O4
tert-butyl N-[2-(2-aminopropylamino)propyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— tert-butyl 3-methyl-3-[2-[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]ethyl]azetidine-1-carboxylate —— C22H30N4O4
tert-butyl 3-methyl-3-[2-[(1R)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-9-yl]ethyl]azetidine-1-carboxylate
—— tert-butyl N-[3-[[2-[2-[(2S,4S)-4-amino-2-(propan-2-ylcarbamoyl)pyrrolidin-1-yl]cyclohexyl]-2-oxoethyl]amino]-3-oxopropyl]-N-methylcarbamate —— C25H45N5O5
tert-butyl N-[3-[[2-[2-[(2S,4S)-4-amino-2-(propan-2-ylcarbamoyl)pyrrolidin-1-yl]cyclohexyl]-2-oxoethyl]amino]-3-oxopropyl]-N-methylcarbamate
—— tert-butyl N-[2-[2-[4-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-6-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-4-(trifluoromethyl)phenyl]sulfanylethyl]carbamate —— C44H56F6N8O9S
tert-butyl N-[2-[2-[4-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-6-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-4-(trifluoromethyl)phenyl]sulfanylethyl]carbamate
—— tert-butyl 4-[3-fluoro-2-[(1S)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-8-yl]phenyl]piperazine-1-carboxylate —— C26H30FN5O4
tert-butyl 4-[3-fluoro-2-[(1S)-1-methyl-2-oxo-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-8-yl]phenyl]piperazine-1-carboxylate
—— ((trans)-2-thiophen-3-yl-cyclopropylmethyl)-carbamic acid benzyl ester —— C16H17NO2S
((trans)-2-thiophen-3-yl-cyclopropylmethyl)-carbamic acid benzyl ester
—— tert-butyl (3R)-3-[2-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-6-[[4-[3-[hydroxy(oxido)amino]-5-(trifluoromethyl)phenoxy]phenyl]carbamoylamino]-4-(trifluoromethyl)phenoxy]pyrrolidine-3-carboxylate —— C46H57F6N8O12-
tert-butyl (3R)-3-[2-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-6-[[4-[3-[hydroxy(oxido)amino]-5-(trifluoromethyl)phenoxy]phenyl]carbamoylamino]-4-(trifluoromethyl)phenoxy]pyrrolidine-3-carboxylate
—— tert-butyl N-[N'-[5-[3-[3-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-2-[(3R)-pyrrolidin-3-yl]oxy-5-(trifluoromethyl)anilino]-5-oxopentyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamimidoyl]carbamate —— C41H50F6N8O8
tert-butyl N-[N'-[5-[3-[3-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-2-[(3R)-pyrrolidin-3-yl]oxy-5-(trifluoromethyl)anilino]-5-oxopentyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamimidoyl]carbamate
—— (trans)-2-(4-methylpyridin-2-yl)-cyclopropanecarboxylic acid ethyl ester —— C12H15NO2
(trans)-2-(4-methylpyridin-2-yl)-cyclopropanecarboxylic acid ethyl ester
—— Trifluoro-(2-phenylmethoxycyclopropyl)boranuide —— C10H11BF3O-
Trifluoro-(2-phenylmethoxycyclopropyl)boranuide
—— [trans-2-Tert-butoxycarbonylcyclopropyl]-trifluoro-boranuide —— C8H13BF3O2-
[trans-2-Tert-butoxycarbonylcyclopropyl]-trifluoro-boranuide
—— tert-butyl N-[2-[2-[3-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-6-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-4-(trifluoromethyl)phenyl]sulfanylethyl]carbamate —— C44H56F6N8O9S
tert-butyl N-[2-[2-[3-[3-amino-5-(trifluoromethyl)phenoxy]-N-carbamoylanilino]-6-[5-[bis[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]pentanoylamino]-4-(trifluoromethyl)phenyl]sulfanylethyl]carbamate
—— tert-butyl N-[1-(5-bromo-4-cyano-1,3-thiazol-2-yl)piperidin-3-yl]carbamate —— C14H19BrN4O2S
tert-butyl N-[1-(5-bromo-4-cyano-1,3-thiazol-2-yl)piperidin-3-yl]carbamate
—— (trans)-2-(5-cyano-pyridin-2-yl)-cyclopropanecarboxylic acid ethyl ester —— C12H12N2O2
(trans)-2-(5-cyano-pyridin-2-yl)-cyclopropanecarboxylic acid ethyl ester
—— (trans)-2-(6-trifluoromethyl-pyridin-3-yl)-cyclopropanecarboxylic acid ethyl ester —— C12H12F3NO2
(trans)-2-(6-trifluoromethyl-pyridin-3-yl)-cyclopropanecarboxylic acid ethyl ester
—— tert-butyl 2-[[(2S)-1-[[(1S)-2-[(3S,5S)-5-(benzylcarbamoyl)-3-(9H-fluoren-9-ylmethoxycarbonylamino)pyrrolidin-3-yl]-1-cyclohexyl-2-oxoethyl]amino]-1-oxopropan-2-yl]amino]acetate —— C44H55N5O7
tert-butyl 2-[[(2S)-1-[[(1S)-2-[(3S,5S)-5-(benzylcarbamoyl)-3-(9H-fluoren-9-ylmethoxycarbonylamino)pyrrolidin-3-yl]-1-cyclohexyl-2-oxoethyl]amino]-1-oxopropan-2-yl]amino]acetate
—— tert-butyl N-[3-[[2-[2-[(2S,4S)-4-amino-2-(benzylcarbamoyl)pyrrolidin-1-yl]cyclohexyl]-2-oxoethyl]amino]-3-oxopropyl]-N-methylcarbamate —— C29H45N5O5
tert-butyl N-[3-[[2-[2-[(2S,4S)-4-amino-2-(benzylcarbamoyl)pyrrolidin-1-yl]cyclohexyl]-2-oxoethyl]amino]-3-oxopropyl]-N-methylcarbamate
—— (trans)-2-(3-Trifluoromethyl-phenyl)-cyclopropanecarboxylic acid ethyl ester —— C13H13F3O2
(trans)-2-(3-Trifluoromethyl-phenyl)-cyclopropanecarboxylic acid ethyl ester
—— [trans-2-Carboxycyclopropyl]-trifluoro-boranuide —— C4H5BF3O2-
[trans-2-Carboxycyclopropyl]-trifluoro-boranuide
—— tert-butyl 3-[(2E)-2-hydrazinylideneethyl]-3-methylazetidine-1-carboxylate —— C11H21N3O2
tert-butyl 3-[(2E)-2-hydrazinylideneethyl]-3-methylazetidine-1-carboxylate