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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl N-[2-[[3-(2,6-dichloro-3,5-dimethoxyphenyl)-2-oxo-1-[[3-(propanoylamino)phenyl]methyl]-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]carbamate —— C35H37Cl2N7O6
tert-butyl N-[2-[[3-(2,6-dichloro-3,5-dimethoxyphenyl)-2-oxo-1-[[3-(propanoylamino)phenyl]methyl]-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]carbamate
—— tert-butyl N-[(3R,4S)-4-[[6-(3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate —— C25H31N5O6
tert-butyl N-[(3R,4S)-4-[[6-(3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate
—— tert-butyl N-[2-[[3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-[(3-nitrophenyl)methyl]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]carbamate —— C32H31Cl2N7O7
tert-butyl N-[2-[[3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-[(3-nitrophenyl)methyl]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]carbamate
—— tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[1-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)cyclohexa-2,4-dien-1-yl]oxypropyl]-N-methylcarbamate —— C28H52BNO6Si
tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[1-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)cyclohexa-2,4-dien-1-yl]oxypropyl]-N-methylcarbamate
—— tert-butyl (3R,4S)-4-azidotetrahydrofuran-3-yl carbamate —— C9H16N4O3
tert-butyl (3R,4S)-4-azidotetrahydrofuran-3-yl carbamate
—— tert-butyl N-[2-[[6-(3,5-dimethoxyphenyl)-7-methoxyquinazolin-2-yl]amino]cyclohexyl]carbamate —— C28H36N4O5
tert-butyl N-[2-[[6-(3,5-dimethoxyphenyl)-7-methoxyquinazolin-2-yl]amino]cyclohexyl]carbamate
—— tert-butyl N-[4-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]thiolan-3-yl]carbamate —— C25H29Cl2N5O5S
tert-butyl N-[4-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]thiolan-3-yl]carbamate
—— tert-butyl N-[5-[(4-ethylpiperazin-1-yl)methyl]-2-nitrophenyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate —— C23H36N4O6
tert-butyl N-[5-[(4-ethylpiperazin-1-yl)methyl]-2-nitrophenyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— tert-butyl N-[2-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]-4-oxocyclopentyl]carbamate —— C26H29Cl2N5O6
tert-butyl N-[2-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]-4-oxocyclopentyl]carbamate
—— tert-butyl (3S)-3-[[6-(3,5-dimethoxyphenyl)-2-methylsulfanyl-7-oxopyrido[2,3-d]pyrimidin-8-yl]methyl]pyrrolidine-1-carboxylate —— C26H32N4O5S
tert-butyl (3S)-3-[[6-(3,5-dimethoxyphenyl)-2-methylsulfanyl-7-oxopyrido[2,3-d]pyrimidin-8-yl]methyl]pyrrolidine-1-carboxylate
—— tert-butyl N-[(3R,4S)-4-[[8-[[(3R)-1-acetylpyrrolidin-3-yl]methyl]-6-(2,6-dichloro-3,5-dimethoxyphenyl)-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate —— C31H38Cl2N6O7
tert-butyl N-[(3R,4S)-4-[[8-[[(3R)-1-acetylpyrrolidin-3-yl]methyl]-6-(2,6-dichloro-3,5-dimethoxyphenyl)-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate
—— tert-butyl N-[2-[[3-(3,5-dimethoxyphenyl)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]-5-(4-ethylpiperazin-1-yl)phenyl]carbamate —— C32H42N8O5
tert-butyl N-[2-[[3-(3,5-dimethoxyphenyl)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]-5-(4-ethylpiperazin-1-yl)phenyl]carbamate
—— tert-butyl 3-[3-(3,5-dimethoxyphenyl)-2-oxo-7-[[2-(prop-2-enoylamino)cyclohexyl]amino]-4H-pyrimido[4,5-d]pyrimidin-1-yl]piperidine-1-carboxylate —— C33H45N7O6
tert-butyl 3-[3-(3,5-dimethoxyphenyl)-2-oxo-7-[[2-(prop-2-enoylamino)cyclohexyl]amino]-4H-pyrimido[4,5-d]pyrimidin-1-yl]piperidine-1-carboxylate
—— tert-butyl N-[(3R,4S)-4-[[6-(2-fluoro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate —— C25H30FN5O6
tert-butyl N-[(3R,4S)-4-[[6-(2-fluoro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate
—— Tert-butyl (2-nitro-5-(piperidin-1-yl)phenyl)carbamate —— C16H23N3O4
Tert-butyl (2-nitro-5-(piperidin-1-yl)phenyl)carbamate
—— tert-butyl N-[(3R,4S)-4-[[6-(3,5-dimethoxy-2,6-dimethylphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate —— C27H35N5O6
tert-butyl N-[(3R,4S)-4-[[6-(3,5-dimethoxy-2,6-dimethylphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate
—— tert-butyl (2-amino-4-(1-methyl-1H-pyrazol-4-yl)phenyl)carbamate —— C15H20N4O2
tert-butyl (2-amino-4-(1-methyl-1H-pyrazol-4-yl)phenyl)carbamate
—— Tert-butyl 3-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]-4-(prop-2-enoylamino)pyrrolidine-1-carboxylate —— C28H32Cl2N6O6
Tert-butyl 3-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]-4-(prop-2-enoylamino)pyrrolidine-1-carboxylate
—— tert-butyl N-[(3R,4S)-4-[[6-[5-[(3-tert-butylphenyl)carbamoyl]-2-chlorophenyl]-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate —— C34H39ClN6O5
tert-butyl N-[(3R,4S)-4-[[6-[5-[(3-tert-butylphenyl)carbamoyl]-2-chlorophenyl]-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]carbamate
—— Tert-butyl 3-amino-4-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]pyrrolidine-1-carboxylate —— C25H30Cl2N6O5
Tert-butyl 3-amino-4-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]pyrrolidine-1-carboxylate
—— tert-butyl (4-(1-methyl-1H-pyrazol-4-yl)-2-nitrophenyl)carbamate —— C15H18N4O4
tert-butyl (4-(1-methyl-1H-pyrazol-4-yl)-2-nitrophenyl)carbamate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C31H36N4O4
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-oxo-1,3-dihydroindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H34N4O4
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-oxo-1,3-dihydroindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[4-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C29H36N4O5S
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[4-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-oxo-3,4-dihydro-2H-isoquinolin-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C31H36N4O4
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-oxo-3,4-dihydro-2H-isoquinolin-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-2-[4-(4-carbamoylphenyl)phenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C29H34N4O4
tert-butyl (3S)-3-[[(1S)-2-[4-(4-carbamoylphenyl)phenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-cyanopyridin-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C28H31N5O3
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-cyanopyridin-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C28H30F3N3O3
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[3-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C29H36N4O5S
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[3-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(4-ethylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H37N3O5S
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(4-ethylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl 7-[(3E)-hexa-1,3,5-trien-3-yl]-1,1-dioxo-1,2,7-thiadiazepane-2-carboxylate —— C15H24N2O4S
tert-butyl 7-[(3E)-hexa-1,3,5-trien-3-yl]-1,1-dioxo-1,2,7-thiadiazepane-2-carboxylate
—— tert-butyl 3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,1-dioxo-3H-1,2-benzothiazol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H35FN4O5S
tert-butyl 3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,1-dioxo-3H-1,2-benzothiazol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(2S)-1-amino-3-(4-bromophenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C22H30BrN3O4
tert-butyl (3S)-3-[[(2S)-1-amino-3-(4-bromophenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3-cyano-4-methylsulfonylphenyl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H33FN4O5S
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3-cyano-4-methylsulfonylphenyl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(4-cyano-3-fluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C29H31FN4O3
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(4-cyano-3-fluorophenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C29H35N3O5S
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(3-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-oxo-2,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H34N4O4
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(1-oxo-2,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[1-(2-methoxyethyl)-2-oxo-3H-indol-6-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C33H40N4O5
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-[1-(2-methoxyethyl)-2-oxo-3H-indol-6-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl N-[[4-(3-aminoazetidin-1-yl)pyrimidin-2-yl]-butylamino]-N-[1-(2-chloropyrimidin-4-yl)azetidin-3-yl]carbamate —— C23H34ClN9O2
tert-butyl N-[[4-(3-aminoazetidin-1-yl)pyrimidin-2-yl]-butylamino]-N-[1-(2-chloropyrimidin-4-yl)azetidin-3-yl]carbamate
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C31H37FN4O3
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— Trimethyl-[2-[4-(oxetan-3-yloxymethyl)phenyl]ethynyl]silane —— C15H20O2Si
Trimethyl-[2-[4-(oxetan-3-yloxymethyl)phenyl]ethynyl]silane
—— tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-oxo-1,3-dihydroindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C30H34N4O4
tert-butyl (3S)-3-[[(1S)-1-cyano-2-[4-(2-oxo-1,3-dihydroindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl N-[1-[4-(3-aminoazetidin-1-yl)pyrimidin-2-yl]butylamino]-N-[1-(2-chloropyrimidin-4-yl)azetidin-3-yl]carbamate —— C23H34ClN9O2
tert-butyl N-[1-[4-(3-aminoazetidin-1-yl)pyrimidin-2-yl]butylamino]-N-[1-(2-chloropyrimidin-4-yl)azetidin-3-yl]carbamate
—— Trimethyl-[2-[4-[[2-methyl-2-(oxan-2-yloxy)propoxy]methyl]phenyl]ethynyl]silane —— C21H32O3Si
Trimethyl-[2-[4-[[2-methyl-2-(oxan-2-yloxy)propoxy]methyl]phenyl]ethynyl]silane
—— tert-butyl (4S)-4-(1-benzoyloxyhexadecyl)-2,2-dimethyl-1,3-oxazolidine-3-carboxylate —— C33H55NO5
tert-butyl (4S)-4-(1-benzoyloxyhexadecyl)-2,2-dimethyl-1,3-oxazolidine-3-carboxylate
—— tert-butyl N-[6'-[(2-methylpropan-2-yl)oxycarbonylamino]-3-oxospiro[2-benzofuran-1,9'-xanthene]-3'-yl]carbamate —— C30H30N2O7
tert-butyl N-[6'-[(2-methylpropan-2-yl)oxycarbonylamino]-3-oxospiro[2-benzofuran-1,9'-xanthene]-3'-yl]carbamate
—— tert-butyl (4S)-4-[(E)-1-benzoyloxyhexadec-2-enyl]-2,2-dimethyl-1,3-oxazolidine-3-carboxylate —— C33H53NO5
tert-butyl (4S)-4-[(E)-1-benzoyloxyhexadec-2-enyl]-2,2-dimethyl-1,3-oxazolidine-3-carboxylate
—— tert-butyl N-[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-pyridin-2-ylpyrrolidin-3-yl]carbamate —— C18H25N5O4S
tert-butyl N-[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-pyridin-2-ylpyrrolidin-3-yl]carbamate
—— tert-butyl N-[(3R,4R)-1-(1-methylimidazol-4-yl)sulfonyl-4-piperidin-2-ylpyrrolidin-3-yl]carbamate —— C18H31N5O4S
tert-butyl N-[(3R,4R)-1-(1-methylimidazol-4-yl)sulfonyl-4-piperidin-2-ylpyrrolidin-3-yl]carbamate
—— tert-butyl (6S,6aS)-3-[[3-[[(6S,6aS)-2-methoxy-5-[(2-methylpropan-2-yl)oxycarbonyl]-6-(oxan-2-yloxy)-11-oxo-6a,7,8,9-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxymethyl]-5-methylphenyl]methoxy]-2-methoxy-6-(oxan-2-yloxy)-11-oxo-6a,7,8,9-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzodiazepine-5-carboxylate —— C55H72N4O14
tert-butyl (6S,6aS)-3-[[3-[[(6S,6aS)-2-methoxy-5-[(2-methylpropan-2-yl)oxycarbonyl]-6-(oxan-2-yloxy)-11-oxo-6a,7,8,9-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxymethyl]-5-methylphenyl]methoxy]-2-methoxy-6-(oxan-2-yloxy)-11-oxo-6a,7,8,9-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzodiazepine-5-carboxylate