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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-5-phenoxyindazol-3-yl]methyl]amino]ethyl]carbamate —— C28H38N4O4
tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-5-phenoxyindazol-3-yl]methyl]amino]ethyl]carbamate
—— tert-butyl 4-(cyanomethyl)-4-[3-[3-fluoro-4-(propan-2-ylsulfamoyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C27H34FN7O5S
tert-butyl 4-(cyanomethyl)-4-[3-[3-fluoro-4-(propan-2-ylsulfamoyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[4-(3,5-dimethylpyrazol-1-yl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C29H33N7O4
tert-butyl 5-(cyanomethyl)-5-[3-[4-(3,5-dimethylpyrazol-1-yl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-(2-oxa-5-azabicyclo[2.2.1]heptane-5-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C31H36N6O6
tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-(2-oxa-5-azabicyclo[2.2.1]heptane-5-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[4-[1-(dimethylamino)-2,2,2-trifluoroethyl]anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C28H33F3N6O4
tert-butyl 5-(cyanomethyl)-5-[3-[4-[1-(dimethylamino)-2,2,2-trifluoroethyl]anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-(quinolin-3-ylamino)-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C27H28N6O4
tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-(quinolin-3-ylamino)-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl N-[2-[[5-(4-aminophenoxy)-1-[(2R)-oxan-2-yl]indazol-3-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C28H39N5O4
tert-butyl N-[2-[[5-(4-aminophenoxy)-1-[(2R)-oxan-2-yl]indazol-3-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-[2-(trifluoromethyl)piperidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C30H35F3N6O4
tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-[2-(trifluoromethyl)piperidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(trifluoromethyl)pyrrolidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C29H34F3N7O3
tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(trifluoromethyl)pyrrolidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-(morpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C30H36N6O6
tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-(morpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)oxane-2-carboxylate —— C18H23N5O4
tert-butyl 5-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)oxane-2-carboxylate
—— tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(3-hydroxypiperidine-1-carbonyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C38H48F3N5O5
tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(3-hydroxypiperidine-1-carbonyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl N-[2-[2-[5-cyclohexyl-1-(oxan-2-yl)indazol-3-yl]ethylamino]ethyl]-N-methylcarbamate —— C28H44N4O3
tert-butyl N-[2-[2-[5-cyclohexyl-1-(oxan-2-yl)indazol-3-yl]ethylamino]ethyl]-N-methylcarbamate
—— tert-butyl 5-(cyanomethyl)-5-[3-[(2-morpholin-4-ylquinolin-6-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C31H35N7O5
tert-butyl 5-(cyanomethyl)-5-[3-[(2-morpholin-4-ylquinolin-6-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-(1-pyrrolidin-1-ylethyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C30H38N6O4
tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-(1-pyrrolidin-1-ylethyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[(2-fluoropyridin-4-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C23H25FN6O4
tert-butyl 5-(cyanomethyl)-5-[3-[(2-fluoropyridin-4-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— Thiophen-2-yl-[4-[3-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]methanone —— C16H15F3N2O3S2
Thiophen-2-yl-[4-[3-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]methanone
—— tert-butyl 5-(cyanomethyl)-5-[3-[4-(2,6-dimethylmorpholine-4-carbonyl)-3-methylanilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C32H40N6O6
tert-butyl 5-(cyanomethyl)-5-[3-[4-(2,6-dimethylmorpholine-4-carbonyl)-3-methylanilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-(quinolin-6-ylamino)-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C27H28N6O4
tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-(quinolin-6-ylamino)-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl (2S,5S)-5-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)oxane-2-carboxylate —— C18H23N5O4
tert-butyl (2S,5S)-5-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)oxane-2-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-(4-morpholin-4-ylsulfonylanilino)-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C28H34N6O7S
tert-butyl 5-(cyanomethyl)-5-[3-(4-morpholin-4-ylsulfonylanilino)-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(propan-2-ylamino)propan-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C30H41N7O3
tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(propan-2-ylamino)propan-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-Butyl 4-(2-acrylamidoethyl)piperidine-1-carboxylate —— C15H26N2O3
tert-Butyl 4-(2-acrylamidoethyl)piperidine-1-carboxylate
—— tert-butyl (2R)-2-[(2-fluorophenyl)methylcarbamoyl]pyrrolidine-1-carboxylate —— C17H23FN2O3
tert-butyl (2R)-2-[(2-fluorophenyl)methylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-(trifluoromethylsulfonyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C25H27F3N6O5S
tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-(trifluoromethylsulfonyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl (2S)-2-[(2-fluorophenyl)methylcarbamoyl]pyrrolidine-1-carboxylate —— C17H23FN2O3
tert-butyl (2S)-2-[(2-fluorophenyl)methylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl 4-{4-(benzyloxy)-3-[(4-fluorophenyl)amino]-1H-pyrazolo[4,3-c]pyridin-1-yl}-4-(cyanomethyl)piperidine-1-carboxylate —— C31H33FN6O3
tert-butyl 4-{4-(benzyloxy)-3-[(4-fluorophenyl)amino]-1H-pyrazolo[4,3-c]pyridin-1-yl}-4-(cyanomethyl)piperidine-1-carboxylate
—— tert-butyl 4-(4-(benzyloxy)-3-((3-(N,N-dimethylsulfamoyl) phenyl)amino)-1H-pyrazolo[4,3-c]pyridin-1-yl)-4-(cyanomethyl)piperidine-1-carboxylate —— C33H39N7O5S
tert-butyl 4-(4-(benzyloxy)-3-((3-(N,N-dimethylsulfamoyl) phenyl)amino)-1H-pyrazolo[4,3-c]pyridin-1-yl)-4-(cyanomethyl)piperidine-1-carboxylate
—— tert-butyl 5-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]-1-methylisoindole-2-carboxylate —— C27H30N6O3
tert-butyl 5-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]-1-methylisoindole-2-carboxylate
—— tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(3-hydroxyazetidine-1-carbonyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C36H44F3N5O5
tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(3-hydroxyazetidine-1-carbonyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl N-methyl-N-[2-[methyl-[[1-(oxan-2-yl)-5-(oxan-4-yl)indazol-3-yl]methyl]amino]ethyl]carbamate;N,5-dimethoxy-N-methyl-1H-indazole-3-carboxamide —— C38H55N7O7
tert-butyl N-methyl-N-[2-[methyl-[[1-(oxan-2-yl)-5-(oxan-4-yl)indazol-3-yl]methyl]amino]ethyl]carbamate;N,5-dimethoxy-N-methyl-1H-indazole-3-carboxamide
—— Tert-butyl 4-[2-[7-methoxy-1-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate —— C24H29F3N4O3
Tert-butyl 4-[2-[7-methoxy-1-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate
—— tert-butyl 5-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]-1-methyl-1,3-dihydroisoindole-2-carboxylate —— C27H32N6O3
tert-butyl 5-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]-1-methyl-1,3-dihydroisoindole-2-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[3-[3-methyl-4-(morpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C30H37N7O5
tert-butyl 4-(cyanomethyl)-4-[3-[3-methyl-4-(morpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 3-[4-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]phenyl]-8-azabicyclo[3.2.1]octane-8-carboxylate —— C31H38N6O3
tert-butyl 3-[4-[[1-(2-cyanocyclohexyl)-4-oxo-2H-pyrazolo[4,3-c]pyridin-3-yl]amino]phenyl]-8-azabicyclo[3.2.1]octane-8-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[3-[3-methyl-4-(3-oxa-8-azabicyclo[3.2.1]octane-8-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C32H39N7O5
tert-butyl 4-(cyanomethyl)-4-[3-[3-methyl-4-(3-oxa-8-azabicyclo[3.2.1]octane-8-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-(3-methyl-4-pyrazol-1-ylanilino)-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C28H31N7O4
tert-butyl 5-(cyanomethyl)-5-[3-(3-methyl-4-pyrazol-1-ylanilino)-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl N-[2-[[3-[(2R,5R)-5-[tert-butyl(dimethyl)silyl]oxyspiro[5.5]undecan-2-yl]-1-(oxan-2-yl)pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C35H64N4O4Si
tert-butyl N-[2-[[3-[(2R,5R)-5-[tert-butyl(dimethyl)silyl]oxyspiro[5.5]undecan-2-yl]-1-(oxan-2-yl)pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— thian-4-yl 4-(cyanomethyl)-4-[3-[4-(dimethylsulfamoyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C27H33N7O5S2
thian-4-yl 4-(cyanomethyl)-4-[3-[4-(dimethylsulfamoyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 3-(3-(acrylamido)azetidin-1-yl)azetidine-1-carboxylate —— C14H23N3O3
tert-butyl 3-(3-(acrylamido)azetidin-1-yl)azetidine-1-carboxylate
—— tert-butyl 5-[3-[(2-tert-butyl-1-oxo-3H-isoindol-5-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]-5-(cyanomethyl)oxane-2-carboxylate —— C30H36N6O5
tert-butyl 5-[3-[(2-tert-butyl-1-oxo-3H-isoindol-5-yl)amino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]-5-(cyanomethyl)oxane-2-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-(pentafluoro-λ6-sulfanyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C24H27F5N6O3S
tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-(pentafluoro-λ6-sulfanyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butylmethyl(2-(methyl((5-((tetrahydrofuran-3-yl)oxy)-1H-indazol-3-yl)methyl)amino)ethyl)carbamate —— C21H32N4O4
tert-butylmethyl(2-(methyl((5-((tetrahydrofuran-3-yl)oxy)-1H-indazol-3-yl)methyl)amino)ethyl)carbamate
—— Tert-butyl 3-[4-[2-(4-chloro-5-ethyl-2-methoxyanilino)acetyl]piperazin-1-yl]azetidine-1-carboxylate —— C23H35ClN4O4
Tert-butyl 3-[4-[2-(4-chloro-5-ethyl-2-methoxyanilino)acetyl]piperazin-1-yl]azetidine-1-carboxylate
—— tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(trifluoromethyl)piperidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C30H36F3N7O3
tert-butyl 4-(cyanomethyl)-4-[4-oxo-3-[4-[2-(trifluoromethyl)piperidin-2-yl]anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— Tert-butyl 5-[3-(4-chloroanilino)-4-phenylmethoxypyrazolo[4,3-c]pyridin-1-yl]-5-(cyanomethyl)oxane-2-carboxylate —— C31H32ClN5O4
Tert-butyl 5-[3-(4-chloroanilino)-4-phenylmethoxypyrazolo[4,3-c]pyridin-1-yl]-5-(cyanomethyl)oxane-2-carboxylate
—— Tert-butyl 4-[[2-[2-methoxy-3-[(2-methylpropan-2-yl)oxycarbonyl]phenyl]-1-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]carbamoyl]piperidine-1-carboxylate —— C35H53BN2O8
Tert-butyl 4-[[2-[2-methoxy-3-[(2-methylpropan-2-yl)oxycarbonyl]phenyl]-1-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]carbamoyl]piperidine-1-carboxylate
—— Tert-butyl 2-[3-benzamido-6-(trifluoromethyl)pyridin-2-yl]oxyacetate —— C19H19F3N2O4
Tert-butyl 2-[3-benzamido-6-(trifluoromethyl)pyridin-2-yl]oxyacetate
—— tert-butyl 5-(3-amino-4-(benzyloxy)-1H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)tetrahydro-2H-pyran-2-carboxylate —— C25H29N5O4
tert-butyl 5-(3-amino-4-(benzyloxy)-1H-pyrazolo[4,3-c]pyridin-1-yl)-5-(cyanomethyl)tetrahydro-2H-pyran-2-carboxylate
—— Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate —— C43H72BN3O9Si
Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate