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—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(trifluoromethyl)thiophen-2-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C26H27F4N3O3S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(trifluoromethyl)thiophen-2-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2,5-dimethylpyrazol-3-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C26H32FN5O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2,5-dimethylpyrazol-3-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(N-cyano-S-methylsulfonimidoyl)phenyl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H32FN5O4S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(N-cyano-S-methylsulfonimidoyl)phenyl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2-ethylpyrazol-3-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C26H32FN5O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2-ethylpyrazol-3-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1-propan-2-ylpiperidin-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H41FN4O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1-propan-2-ylpiperidin-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[1-[(1-acetylpiperidin-4-yl)methyl]pyrazol-4-yl]-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H41FN6O4
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[1-[(1-acetylpiperidin-4-yl)methyl]pyrazol-4-yl]-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(4-ethylpiperazin-1-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H38FN5O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(4-ethylpiperazin-1-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H40FN5O5S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-oxo-3H-2-benzofuran-5-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H32FN3O6
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-oxo-3H-2-benzofuran-5-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-piperidin-1-ylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H39FN4O5S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-piperidin-1-ylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C28H38FN5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C30H35FN4O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,3-dihydroisoindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-morpholin-4-ylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C31H37FN4O6S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-morpholin-4-ylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(4-sulfamoylphenyl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate —— C28H31FN4O5S
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(4-sulfamoylphenyl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2,3-difluoro-4-(4-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C28H31F2N3O5S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2,3-difluoro-4-(4-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-propan-2-yl-3,6-dihydro-2H-pyridin-4-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H41FN4O4
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-propan-2-yl-3,6-dihydro-2H-pyridin-4-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(1,3,4,6,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-8-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H37FN4O4
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(1,3,4,6,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-8-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(3-oxo-1H-2-benzofuran-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H30FN3O5
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(3-oxo-1H-2-benzofuran-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-propan-2-ylpiperidin-4-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H43FN4O4
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(1-propan-2-ylpiperidin-4-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(1-methylpiperidin-4-yl)-2-oxo-3H-indol-6-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C35H42FN5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(1-methylpiperidin-4-yl)-2-oxo-3H-indol-6-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(4-methylpiperazine-1-carbonyl)thiophen-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C31H38FN5O4S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(4-methylpiperazine-1-carbonyl)thiophen-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-imidazo[1,2-a]pyrazin-2-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H29FN6O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-imidazo[1,2-a]pyrazin-2-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— Tert-butyl 2-[2-(benzhydrylideneamino)-2-cyanoethyl]carbazole-9-carboxylate —— C33H29N3O2
Tert-butyl 2-[2-(benzhydrylideneamino)-2-cyanoethyl]carbazole-9-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-fluoro-3-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H39F2N5O5S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-fluoro-3-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(5-ethoxycarbonylthiophen-2-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C28H32FN3O5S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(5-ethoxycarbonylthiophen-2-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-cyano-4,9-difluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H27F2N5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-cyano-4,9-difluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-imidazo[1,2-b]pyridazin-2-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H29FN6O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-imidazo[1,2-b]pyridazin-2-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(1H-indazol-5-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C22H27N5O3
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(1H-indazol-5-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— Thiophen-2-ylmethyl 2-(4-chloro-2-methylphenoxy)acetate —— C14H13ClO3S
Thiophen-2-ylmethyl 2-(4-chloro-2-methylphenoxy)acetate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[5-(6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl)thiophen-3-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H35FN6O4S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[5-(6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl)thiophen-3-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(4-ethoxycarbonylpyrazol-1-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H32FN5O5
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(4-ethoxycarbonylpyrazol-1-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(2,3-difluoro-4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C21H27F2N3O5
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(2,3-difluoro-4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(dimethylcarbamoyl)pyrazol-1-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H33FN6O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(dimethylcarbamoyl)pyrazol-1-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2,3-difluoro-4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C30H34F2N4O5
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2,3-difluoro-4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[4-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-2-fluorophenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C26H37BFN3O6
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[4-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-2-fluorophenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(3,4,9-trifluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C28H27F3N4O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(3,4,9-trifluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(pyrrolidine-1-carbonyl)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H37FN4O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(pyrrolidine-1-carbonyl)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[2-(methylamino)-3H-benzimidazol-5-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H33FN6O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[2-(methylamino)-3H-benzimidazol-5-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,2R,4S,5S,7S)-7-[[1-cyano-2-[2-fluoro-4-(1-oxo-3,4-dihydro-2H-isoquinolin-6-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate —— C31H33FN4O4
tert-butyl (1R,2R,4S,5S,7S)-7-[[1-cyano-2-[2-fluoro-4-(1-oxo-3,4-dihydro-2H-isoquinolin-6-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(4-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C28H32FN3O5S
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(4-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(2-methoxyethyl)-3-methylpiperazin-1-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H42FN5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(2-methoxyethyl)-3-methylpiperazin-1-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)-3,6-dihydro-2H-pyridin-4-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C30H41FN4O5
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)-3,6-dihydro-2H-pyridin-4-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(5-methoxycarbonylfuran-2-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H30FN3O6
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(5-methoxycarbonylfuran-2-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-amino-3-(1H-indazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C22H29N5O4
tert-butyl (1R,3S,4S)-3-[[1-amino-3-(1H-indazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)piperidin-4-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C30H43FN4O5
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)piperidin-4-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1,3,3-trimethyl-2-oxoindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H37FN4O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1,3,3-trimethyl-2-oxoindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— Tert-butyl 2-(2-amino-2-cyanoethyl)carbazole-9-carboxylate —— C20H21N3O2
Tert-butyl 2-(2-amino-2-cyanoethyl)carbazole-9-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2-ethoxy-1,3-thiazol-4-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C26H31FN4O4S
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2-ethoxy-1,3-thiazol-4-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl 6-[4-[(2S)-2-cyano-2-[[(1R,3S,4S)-2-[1-[(2-methylpropan-2-yl)oxy]ethenyl]-2-azabicyclo[2.2.1]heptane-3-carbonyl]amino]ethyl]-3-fluorophenyl]-2,6-diazaspiro[3.3]heptane-2-carboxylate —— C32H44FN5O4
tert-butyl 6-[4-[(2S)-2-cyano-2-[[(1R,3S,4S)-2-[1-[(2-methylpropan-2-yl)oxy]ethenyl]-2-azabicyclo[2.2.1]heptane-3-carbonyl]amino]ethyl]-3-fluorophenyl]-2,6-diazaspiro[3.3]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[4-(cyclopropylcarbamoyl)-6-oxo-5H-phenanthridin-8-yl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C32H35N5O5
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[4-(cyclopropylcarbamoyl)-6-oxo-5H-phenanthridin-8-yl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate