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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 2-[5-[[2-(2-cyanopropan-2-yl)pyridine-4-carbonyl]amino]-2-methylphenyl]-4-morpholin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxylate —— C33H39N7O4
tert-butyl 2-[5-[[2-(2-cyanopropan-2-yl)pyridine-4-carbonyl]amino]-2-methylphenyl]-4-morpholin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxylate
—— Tert-butyl 2-cyano-2-(5-methylpyridazin-3-yl)acetate —— C12H15N3O2
Tert-butyl 2-cyano-2-(5-methylpyridazin-3-yl)acetate
—— Tert-butyl 3-((4-chloro-6-morpholinopyrimidin-2-yl)amino)azetidine-1-carboxylate —— C16H24ClN5O3
Tert-butyl 3-((4-chloro-6-morpholinopyrimidin-2-yl)amino)azetidine-1-carboxylate
—— Tert-butyl 4-(4-methyl-3-(1-methyl-5-morpholino-6-oxo-1,6-dihydropyridin-3-yl)benzamido)-2-(trifluoromethyl)benzylcarbamate —— C31H35F3N4O5
Tert-butyl 4-(4-methyl-3-(1-methyl-5-morpholino-6-oxo-1,6-dihydropyridin-3-yl)benzamido)-2-(trifluoromethyl)benzylcarbamate
—— tert-butyl 2-(2-methyl-5-((3-(trifluoromethyl)phenyl)carbamoyl)phenyl)-4-morpholino-5H-pyrrolo[3,4-d]pyrimidine-6(7H)-carboxylate —— C30H32F3N5O4
tert-butyl 2-(2-methyl-5-((3-(trifluoromethyl)phenyl)carbamoyl)phenyl)-4-morpholino-5H-pyrrolo[3,4-d]pyrimidine-6(7H)-carboxylate
—— Tert-butyl 3-((4-chloro-6-morpholinopyrimidin-2-yl)oxy)azetidine-1-carboxylate —— C16H23ClN4O4
Tert-butyl 3-((4-chloro-6-morpholinopyrimidin-2-yl)oxy)azetidine-1-carboxylate
—— tert-butyl 4-(1-acryloylazetidin-3-yl)-3-methylpiperazine-1-carboxylate —— C16H27N3O3
tert-butyl 4-(1-acryloylazetidin-3-yl)-3-methylpiperazine-1-carboxylate
—— Tert-butyl 4-[2-[7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate —— C24H32N4O3
Tert-butyl 4-[2-[7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate
—— tert-butyl (4S,5R)-4-(2,4-dipropoxyphenyl)-6-methylidene-2-sulfanylidene-1,3-diazinane-5-carboxylate —— C22H32N2O4S
tert-butyl (4S,5R)-4-(2,4-dipropoxyphenyl)-6-methylidene-2-sulfanylidene-1,3-diazinane-5-carboxylate
—— tert-butyl (4R,5S)-4-(2,4-dipropoxyphenyl)-6-methylidene-2-sulfanylidene-1,3-diazinane-5-carboxylate —— C22H32N2O4S
tert-butyl (4R,5S)-4-(2,4-dipropoxyphenyl)-6-methylidene-2-sulfanylidene-1,3-diazinane-5-carboxylate
—— tert-butyl 4-(((5-bromo-2-hydrazinylpyridin-4-yl)oxy)methyl)piperidine-1-carboxylate —— C16H25BrN4O3
tert-butyl 4-(((5-bromo-2-hydrazinylpyridin-4-yl)oxy)methyl)piperidine-1-carboxylate
—— Tert-butyl 4-[2-[7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate —— C23H30N4O3
Tert-butyl 4-[2-[7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate
—— tert-butyl 3-(4-(2-(4-chloro-5-isopropyl-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate —— C24H37ClN4O4
tert-butyl 3-(4-(2-(4-chloro-5-isopropyl-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate
—— Tert-butyl 4-[3-(3-fluoro-7-methoxy-5-methylpyrido[3,4-b]indol-9-yl)propyl]piperazine-1-carboxylate —— C25H33FN4O3
Tert-butyl 4-[3-(3-fluoro-7-methoxy-5-methylpyrido[3,4-b]indol-9-yl)propyl]piperazine-1-carboxylate
—— (Tert-butylcarbamoyl)methyl 5,6-dichloropyridine-3-carboxylate —— C12H14Cl2N2O3
(Tert-butylcarbamoyl)methyl 5,6-dichloropyridine-3-carboxylate
—— tert-butyl 2-[[(4S)-4-[[2-[2-(2-aminoethoxy)ethoxy]acetyl]amino]-5-[(2-methylpropan-2-yl)oxy]-5-oxopentanoyl]amino]-5-(ethylamino)-5-oxopentanoate —— C26H48N4O9
tert-butyl 2-[[(4S)-4-[[2-[2-(2-aminoethoxy)ethoxy]acetyl]amino]-5-[(2-methylpropan-2-yl)oxy]-5-oxopentanoyl]amino]-5-(ethylamino)-5-oxopentanoate
—— tert-butyl N-[4-[[(5S)-5-[[2-[2-(2-aminoethoxy)ethoxy]acetyl]amino]-6-oxoheptyl]carbamoyl]phenyl]carbamate —— C25H40N4O7
tert-butyl N-[4-[[(5S)-5-[[2-[2-(2-aminoethoxy)ethoxy]acetyl]amino]-6-oxoheptyl]carbamoyl]phenyl]carbamate
—— tert-butyl 2-amino-5-[[1-[(2-methylpropan-2-yl)oxy]-5-[2-[2-[2-[[(3S)-7-[[4-[(2-methylpropan-2-yl)oxycarbonylamino]benzoyl]amino]-2-oxoheptan-3-yl]amino]-2-oxoethoxy]ethoxy]ethylamino]-1,5-dioxopentan-2-yl]amino]-5-oxopentanoate —— C43H70N6O13
tert-butyl 2-amino-5-[[1-[(2-methylpropan-2-yl)oxy]-5-[2-[2-[2-[[(3S)-7-[[4-[(2-methylpropan-2-yl)oxycarbonylamino]benzoyl]amino]-2-oxoheptan-3-yl]amino]-2-oxoethoxy]ethoxy]ethylamino]-1,5-dioxopentan-2-yl]amino]-5-oxopentanoate
—— Tert-butyl 2-[[1-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]-2-oxoethyl]imidazol-2-yl]methyl-[2-[2-[(decylamino)methyl]imidazol-1-yl]acetyl]amino]acetate —— C40H67N7O8
Tert-butyl 2-[[1-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]-2-oxoethyl]imidazol-2-yl]methyl-[2-[2-[(decylamino)methyl]imidazol-1-yl]acetyl]amino]acetate
—— tert-butyl (3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[3-[2-[2-[2-[2-[2-[2-[5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-3-tritylsulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoyl]amino]propanoyl]amino]-3-(3-tritylimidazol-4-yl)propanoyl]amino]-4-oxo-4-(tritylamino)butanoyl]amino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]propanoyl]amino]-4-[[(2S)-1-[[(2S)-4-methyl-1-[[(2R)-3-methyl-1-oxo-1-[[(2S)-3-oxo-1-tritylsulfanylbutan-2-yl]amino]butan-2-yl]amino]-1-oxopentan-2-yl]amino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]-1-oxopropan-2-yl]amino]-4-oxobutanoate —— C180H216N18O26S3
tert-butyl (3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[3-[2-[2-[2-[2-[2-[2-[5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-3-tritylsulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoyl]amino]propanoyl]amino]-3-(3-tritylimidazol-4-yl)propanoyl]amino]-4-oxo-4-(tritylamino)butanoyl]amino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]propanoyl]amino]-4-[[(2S)-1-[[(2S)-4-methyl-1-[[(2R)-3-methyl-1-oxo-1-[[(2S)-3-oxo-1-tritylsulfanylbutan-2-yl]amino]butan-2-yl]amino]-1-oxopentan-2-yl]amino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]-1-oxopropan-2-yl]amino]-4-oxobutanoate
—— tert-butyl N-[2-[2-[2-(2-aminoethoxy)ethyl-(2-oxopropyl)amino]ethoxy]ethyl]carbamate —— C16H33N3O5
tert-butyl N-[2-[2-[2-(2-aminoethoxy)ethyl-(2-oxopropyl)amino]ethoxy]ethyl]carbamate
—— tert-butyl (4S)-5-(methylamino)-5-oxo-4-(2-oxopyrrolidin-1-yl)pentanoate —— C14H24N2O4
tert-butyl (4S)-5-(methylamino)-5-oxo-4-(2-oxopyrrolidin-1-yl)pentanoate
—— tert-butyl 5-[[(1S)-1-cyano-2-[4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]ethyl]carbamoyl]-2-oxa-6-azabicyclo[3.3.1]nonane-6-carboxylate —— C31H36N4O5
tert-butyl 5-[[(1S)-1-cyano-2-[4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]ethyl]carbamoyl]-2-oxa-6-azabicyclo[3.3.1]nonane-6-carboxylate
—— Tert-butyl 5-(benzenecarbonothioylsulfanyl)-2-methyl-4-phenylpentanoate —— C23H28O2S2
Tert-butyl 5-(benzenecarbonothioylsulfanyl)-2-methyl-4-phenylpentanoate
—— Tert-butyl 4-[4-[5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]benzoyl]-1,4-diazepane-1-carboxylate 1232418-06-2 C29H31N7O4
Tert-butyl 4-[4-[5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]benzoyl]-1,4-diazepane-1-carboxylate
—— tert-butyl 4-[4-[(3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate —— C28H32N4O3S
tert-butyl 4-[4-[(3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate
—— tert-butyl 4-[(Z)-4-[4-[(2-methylpropan-2-yl)oxycarbonyl]phenoxy]but-2-enoxy]benzoate —— C26H32O6
tert-butyl 4-[(Z)-4-[4-[(2-methylpropan-2-yl)oxycarbonyl]phenoxy]but-2-enoxy]benzoate
—— tert-butyl N-[(1S)-1-cyano-2-[4-(2-methyl-1,1-dioxo-3H-1,2-benzothiazol-5-yl)phenyl]ethyl]carbamate —— C22H25N3O4S
tert-butyl N-[(1S)-1-cyano-2-[4-(2-methyl-1,1-dioxo-3H-1,2-benzothiazol-5-yl)phenyl]ethyl]carbamate
—— tert-butyl 3-[4-[(3Z)-3-[[4-[2-(diethylamino)ethylcarbamoyl]-3,5-dimethyl-1H-pyrrol-2-yl]methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]pyrrolidine-1-carboxylate —— C34H44N6O4S
tert-butyl 3-[4-[(3Z)-3-[[4-[2-(diethylamino)ethylcarbamoyl]-3,5-dimethyl-1H-pyrrol-2-yl]methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl N-[4-(3-chlorophenyl)-5-fluoro-6-[(4-methylphenyl)methyl]-1,3-benzothiazol-2-yl]carbamate —— C26H24ClFN2O2S
tert-butyl N-[4-(3-chlorophenyl)-5-fluoro-6-[(4-methylphenyl)methyl]-1,3-benzothiazol-2-yl]carbamate
—— tert-butyl 4-[4-[(3Z)-3-[(4-methoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate —— C30H34N4O5S
tert-butyl 4-[4-[(3Z)-3-[(4-methoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate
—— tert-butyl (1R,5S)-5-[[(1S)-1-cyano-2-[4-(4-cyano-3-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-oxa-6-azabicyclo[3.2.1]octane-6-carboxylate —— C29H32N4O6S
tert-butyl (1R,5S)-5-[[(1S)-1-cyano-2-[4-(4-cyano-3-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-oxa-6-azabicyclo[3.2.1]octane-6-carboxylate
—— tert-butyl 3-(3-cyano-7-oxo-6-propan-2-yl-1H-pyrazolo[1,5-a]pyrimidin-5-yl)-2,5-dihydropyrrole-1-carboxylate —— C19H23N5O3
tert-butyl 3-(3-cyano-7-oxo-6-propan-2-yl-1H-pyrazolo[1,5-a]pyrimidin-5-yl)-2,5-dihydropyrrole-1-carboxylate
—— tert-butyl N-[3-(3-cyano-6-ethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl)phenyl]carbamate —— C20H21N5O3
tert-butyl N-[3-(3-cyano-6-ethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl)phenyl]carbamate
—— tert-butyl 1-[[(1S)-2-(4-bromo-2-fluorophenyl)-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate —— C22H27BrFN3O3
tert-butyl 1-[[(1S)-2-(4-bromo-2-fluorophenyl)-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl N-[4-[[5-[[2-(2-ethoxyethoxy)acetyl]amino]-6-(methylamino)-6-oxohexyl]carbamoyl]phenyl]carbamate —— C25H40N4O7
tert-butyl N-[4-[[5-[[2-(2-ethoxyethoxy)acetyl]amino]-6-(methylamino)-6-oxohexyl]carbamoyl]phenyl]carbamate
—— tert-butyl 4-[4-[(3Z)-2-oxo-3-(4,5,6,7-tetrahydro-1H-indol-2-ylmethylidene)-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate —— C30H34N4O3S
tert-butyl 4-[4-[(3Z)-2-oxo-3-(4,5,6,7-tetrahydro-1H-indol-2-ylmethylidene)-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate
—— Tert-butyl 3-[4-(2-oxo-1,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]pyrrolidine-1-carboxylate —— C20H23N3O3S
Tert-butyl 3-[4-(2-oxo-1,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]pyrrolidine-1-carboxylate
—— Trimethyl-[[5-[4-(4-methylphenyl)sulfonylphenyl]sulfonyl-2-[4-[4-(4-methylsulfonylphenyl)sulfonylphenyl]sulfonylbenzoyl]sulfonylphenyl]methyl]azanium —— C43H40NO13S6+
Trimethyl-[[5-[4-(4-methylphenyl)sulfonylphenyl]sulfonyl-2-[4-[4-(4-methylsulfonylphenyl)sulfonylphenyl]sulfonylbenzoyl]sulfonylphenyl]methyl]azanium
—— tert-butyl 4-[4-[(3Z)-3-(1H-indol-2-ylmethylidene)-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate —— C30H30N4O3S
tert-butyl 4-[4-[(3Z)-3-(1H-indol-2-ylmethylidene)-2-oxo-1H-indol-5-yl]-1,3-thiazol-2-yl]piperidine-1-carboxylate
—— Tert-butyl 4-[4-(4-fluoro-3-methylphenyl)-1-(2-hydroxyethyl)imidazol-2-yl]-4-[2-[hydroxy(dimethyl)silyl]-2-methylpropyl]piperidine-1-carboxylate —— C28H44FN3O4Si
Tert-butyl 4-[4-(4-fluoro-3-methylphenyl)-1-(2-hydroxyethyl)imidazol-2-yl]-4-[2-[hydroxy(dimethyl)silyl]-2-methylpropyl]piperidine-1-carboxylate
—— tert-butyl N-[2-[[2-chloro-5-(3-ethoxy-4-methoxybut-1-ynyl)pyrimidin-4-yl]amino]ethyl]carbamate —— C18H27ClN4O4
tert-butyl N-[2-[[2-chloro-5-(3-ethoxy-4-methoxybut-1-ynyl)pyrimidin-4-yl]amino]ethyl]carbamate
—— tert-butyl N-[(1S)-1-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]carbamate —— C16H18F3N3O4
tert-butyl N-[(1S)-1-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]carbamate
—— Tert-butyl 4-[4-(4-fluoro-3-methylphenyl)-1-[2-(oxan-2-yloxy)ethyl]imidazol-2-yl]-4-[2-[hydroxy(dimethyl)silyl]-2-methylpropyl]piperidine-1-carboxylate —— C33H52FN3O5Si
Tert-butyl 4-[4-(4-fluoro-3-methylphenyl)-1-[2-(oxan-2-yloxy)ethyl]imidazol-2-yl]-4-[2-[hydroxy(dimethyl)silyl]-2-methylpropyl]piperidine-1-carboxylate
—— tert-butyl N-[2-[(2-ethyl-5-methylpyrimidin-4-yl)amino]ethyl]carbamate —— C14H24N4O2
tert-butyl N-[2-[(2-ethyl-5-methylpyrimidin-4-yl)amino]ethyl]carbamate
—— tert-butyl N-[4-[[7-[(1S,5R)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl]quinoxalin-5-yl]amino]cyclohexyl]carbamate —— C25H35N5O3
tert-butyl N-[4-[[7-[(1S,5R)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl]quinoxalin-5-yl]amino]cyclohexyl]carbamate
—— tert-butyl N-[4-[(6-morpholin-4-yl-2,1,3-benzoxadiazol-4-yl)amino]cyclohexyl]carbamate —— C21H31N5O4
tert-butyl N-[4-[(6-morpholin-4-yl-2,1,3-benzoxadiazol-4-yl)amino]cyclohexyl]carbamate
—— tert-butyl N-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-[[(3R,4S)-1-cyclopropyl-3-fluoropiperidin-4-yl]amino]-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate —— C39H58ClFN6O5Si
tert-butyl N-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-[[(3R,4S)-1-cyclopropyl-3-fluoropiperidin-4-yl]amino]-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate
—— Tert-butyl 4-[2-[[4-(7-morpholin-4-ylquinoxalin-5-yl)oxycyclohexyl]amino]pyrimidin-5-yl]piperidine-1-carboxylate —— C32H43N7O4
Tert-butyl 4-[2-[[4-(7-morpholin-4-ylquinoxalin-5-yl)oxycyclohexyl]amino]pyrimidin-5-yl]piperidine-1-carboxylate
—— tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(5-chloro-4-(3,5-dimethyl-isoxazol-4-yl)-6-((tetrahydro-2H-pyran-4-yl)methylamino)pyrimidin-2-yl) phenoxy)propyl(methyl)carbamate —— C36H54ClN5O6Si
tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(5-chloro-4-(3,5-dimethyl-isoxazol-4-yl)-6-((tetrahydro-2H-pyran-4-yl)methylamino)pyrimidin-2-yl) phenoxy)propyl(methyl)carbamate