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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[4-(1-benzyl-3,6-dihydro-2H-pyridin-5-yl)-2-fluorophenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C33H41FN4O4
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[4-(1-benzyl-3,6-dihydro-2H-pyridin-5-yl)-2-fluorophenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(2-methoxyethyl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C27H34FN5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(2-methoxyethyl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-[1-(oxan-4-yl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H36FN5O4
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-[1-(oxan-4-yl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(7-azaspiro[3.5]non-2-en-2-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H37FN4O3
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(7-azaspiro[3.5]non-2-en-2-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C29H31FN4O5
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C30H42FN5O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl N-[(2S)-3-methyl-1-oxo-1-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[[(1S,2S,6R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]methylamino]propan-2-yl]amino]-3-phenylpropan-2-yl]amino]butan-2-yl]carbamate —— C33H51BN4O7
tert-butyl N-[(2S)-3-methyl-1-oxo-1-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[[(1S,2S,6R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]methylamino]propan-2-yl]amino]-3-phenylpropan-2-yl]amino]butan-2-yl]carbamate
—— tert-butyl (4S)-5-hydroxy-4-(3-oxo-3-phenylmethoxypropyl)-5-(trifluoromethyl)-1,3-oxazolidine-3-carboxylate —— C19H24F3NO6
tert-butyl (4S)-5-hydroxy-4-(3-oxo-3-phenylmethoxypropyl)-5-(trifluoromethyl)-1,3-oxazolidine-3-carboxylate
—— tert-butyl N-[3-[6-[2-[(4E,6E,8E)-2-methyl-3-methylidene-8-(1,3,3-trimethylindol-2-ylidene)octa-4,6-dien-2-yl]anilino]hexanoylamino]propyl]-N-[4-[(2-methylpropan-2-yl)oxycarbonyl-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]amino]butyl]carbamate —— C58H90N6O7
tert-butyl N-[3-[6-[2-[(4E,6E,8E)-2-methyl-3-methylidene-8-(1,3,3-trimethylindol-2-ylidene)octa-4,6-dien-2-yl]anilino]hexanoylamino]propyl]-N-[4-[(2-methylpropan-2-yl)oxycarbonyl-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]amino]butyl]carbamate
—— Thiophen-2-ylmethyl cyclopropanecarboxylate —— C9H10O2S
Thiophen-2-ylmethyl cyclopropanecarboxylate
—— Tert-butyl 2-[[2-[4-[5-[5-(fluoromethyl)-1-phenylpyrazol-4-yl]-1,2,4-oxadiazol-3-yl]phenyl]-2-hydroxyacetyl]amino]acetate —— C26H26FN5O5
Tert-butyl 2-[[2-[4-[5-[5-(fluoromethyl)-1-phenylpyrazol-4-yl]-1,2,4-oxadiazol-3-yl]phenyl]-2-hydroxyacetyl]amino]acetate
—— tert-butyl (3S)-3-(6-bromo-1H-benzimidazol-2-yl)-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C18H22BrN3O2
tert-butyl (3S)-3-(6-bromo-1H-benzimidazol-2-yl)-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (2S)-2-[5-(5-bromo-1-benzofuran-2-yl)-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate —— C24H28BrN3O3
tert-butyl (2S)-2-[5-(5-bromo-1-benzofuran-2-yl)-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate
—— Trimethoxy-[4-[methoxy(dimethyl)silyl]phenyl]silane —— C12H22O4Si2
Trimethoxy-[4-[methoxy(dimethyl)silyl]phenyl]silane
—— tert-butyl (3S)-3-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-benzimidazol-2-yl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C24H34BN3O4
tert-butyl (3S)-3-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-benzimidazol-2-yl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (3S)-3-[5-(6-bromopyridin-3-yl)-1H-imidazol-2-yl]-2-azabicyclo[2.2.1]heptane-2-carboxylate —— C19H23BrN4O2
tert-butyl (3S)-3-[5-(6-bromopyridin-3-yl)-1H-imidazol-2-yl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— tert-butyl (2S,3aS,7aS)-2-[5-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate —— C28H40BN3O4
tert-butyl (2S,3aS,7aS)-2-[5-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate
—— tert-butyl 4-(1-acetyl-4-amino-2,3-dimethyl-3,4-dihydro-2H-quinolin-6-yl)-2-methylpiperazine-1-carboxylate —— C23H36N4O3
tert-butyl 4-(1-acetyl-4-amino-2,3-dimethyl-3,4-dihydro-2H-quinolin-6-yl)-2-methylpiperazine-1-carboxylate
—— tert-butyl (2S)-2-[5-[4-[5-[2-[(3S)-2-[(2-methylpropan-2-yl)oxycarbonyl]-2-azabicyclo[2.2.1]heptan-3-yl]-1H-imidazol-5-yl]pyridin-2-yl]phenyl]-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate —— C41H51N7O4
tert-butyl (2S)-2-[5-[4-[5-[2-[(3S)-2-[(2-methylpropan-2-yl)oxycarbonyl]-2-azabicyclo[2.2.1]heptan-3-yl]-1H-imidazol-5-yl]pyridin-2-yl]phenyl]-1H-imidazol-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindole-1-carboxylate
—— Trimethoxysilylmethyl 3-cyano-2,3-dimethylbutanoate —— C11H21NO5Si
Trimethoxysilylmethyl 3-cyano-2,3-dimethylbutanoate
—— tert-butyl 4-(2-((5-methyl-4-(1-(2-methylbenzoyl)indolin-5-yl)thiazol-2-yl)amino)-2-oxoethyl)piperazine-1-carboxylate —— C31H37N5O4S
tert-butyl 4-(2-((5-methyl-4-(1-(2-methylbenzoyl)indolin-5-yl)thiazol-2-yl)amino)-2-oxoethyl)piperazine-1-carboxylate
—— tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[4-(methylcarbamoyl)anilino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C33H45N5O4
tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[4-(methylcarbamoyl)anilino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— tert-butyl N-[(E)-6-oxaspiro[4.5]decan-9-ylideneamino]carbamate —— C14H24N2O3
tert-butyl N-[(E)-6-oxaspiro[4.5]decan-9-ylideneamino]carbamate
—— tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-[4-(methylcarbamoyl)anilino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C33H45N5O4
tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-[4-(methylcarbamoyl)anilino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— trans-1-(cyclopropylcarbonyl)-2,6-dimethyl-4-(4-methylphenylamino)-1,2,3,4-tetrahydroquinoline —— C22H26N2O
trans-1-(cyclopropylcarbonyl)-2,6-dimethyl-4-(4-methylphenylamino)-1,2,3,4-tetrahydroquinoline
—— tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[(4-methylpyrimidin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C30H42N6O3
tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[(4-methylpyrimidin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[(5-methylpyrazin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C30H42N6O3
tert-butyl 4-[1-acetyl-2-cyclopropyl-3-methyl-4-[(5-methylpyrazin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— tert-butyl 4-((2S,3R,4R)-1-acetyl-4-((4-(methoxycarbonyl)phenyl)amino)-2,3-dimethyl-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylic acid —— C29H38N4O5
tert-butyl 4-((2S,3R,4R)-1-acetyl-4-((4-(methoxycarbonyl)phenyl)amino)-2,3-dimethyl-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylic acid
—— tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-[(5-methylpyrazin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C30H42N6O3
tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-[(5-methylpyrazin-2-yl)amino]-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-4-[(5-fluoropyridin-2-yl)amino]-3-methyl-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate —— C30H40FN5O3
tert-butyl 4-[(2S,3R,4R)-1-acetyl-2-cyclopropyl-4-[(5-fluoropyridin-2-yl)amino]-3-methyl-3,4-dihydro-2H-quinolin-6-yl]-2-methylpiperazine-1-carboxylate
—— tert-butyl 5-(1-acetyl-4-amino-2,3-dimethyl-3,4-dihydro-2H-quinolin-6-yl)-2,5-diazabicyclo[2.2.2]octane-2-carboxylate —— C24H36N4O3
tert-butyl 5-(1-acetyl-4-amino-2,3-dimethyl-3,4-dihydro-2H-quinolin-6-yl)-2,5-diazabicyclo[2.2.2]octane-2-carboxylate
—— tert-butyl 4-((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylate —— C27H38N6O3
tert-butyl 4-((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylate
—— Tert-butyl 2-[[5-(3-benzyl-4-oxophthalazin-1-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetate —— C23H22N4O4S
Tert-butyl 2-[[5-(3-benzyl-4-oxophthalazin-1-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetate
—— tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-(2,3-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate —— C38H54ClN7O5Si
tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-(2,3-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate
—— tert-butyl 5-(aminomethyl)-1H-imidazole-1-carboxylate —— C9H15N3O2
tert-butyl 5-(aminomethyl)-1H-imidazole-1-carboxylate
—— tert-butyl 3-(3-(4-(3,5-dimethyl-3H-1,2,3-triazol-4-yl)-5-methyl-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-2-yl)phenoxy)-2-hydroxy-propyl(methyl)carbamate —— C29H41N7O5
tert-butyl 3-(3-(4-(3,5-dimethyl-3H-1,2,3-triazol-4-yl)-5-methyl-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-2-yl)phenoxy)-2-hydroxy-propyl(methyl)carbamate
—— tert-butyl N-[4-(1,1-difluoroethylsulfanyl)phenyl]carbamate —— C13H17F2NO2S
tert-butyl N-[4-(1,1-difluoroethylsulfanyl)phenyl]carbamate
—— tert-butyl-[(2R)-1-[4-chloro-3-[4-chloro-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]butan-2-yl]oxy-dimethylsilane —— C26H35Cl2N3O3Si
tert-butyl-[(2R)-1-[4-chloro-3-[4-chloro-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]butan-2-yl]oxy-dimethylsilane
—— tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-(1,3-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate —— C38H54ClN7O5Si
tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-(1,3-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate
—— tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy)propylcarbamate —— C26H46BNO6Si
tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy)propylcarbamate
—— tert-butyl N-[tert-butyl(dimethyl)silyl]oxy-N-[3-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]propyl]carbamate —— C26H46BNO6Si
tert-butyl N-[tert-butyl(dimethyl)silyl]oxy-N-[3-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]propyl]carbamate
—— tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-chloro-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate —— C31H44Cl2N4O5Si
tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[4-chloro-3-[4-chloro-6-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate
—— tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[3-(4,6-dichloro-5-methylpyrimidin-2-yl)-4-fluorophenoxy]propyl]-N-methylcarbamate —— C26H38Cl2FN3O4Si
tert-butyl N-[2-[tert-butyl(dimethyl)silyl]oxy-3-[3-(4,6-dichloro-5-methylpyrimidin-2-yl)-4-fluorophenoxy]propyl]-N-methylcarbamate
—— tert-butyl-[1-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]azetidin-3-yl]carbamic acid —— C27H30N6O4
tert-butyl-[1-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]azetidin-3-yl]carbamic acid
—— tert-butyl N-[3-(3-bromophenoxy)-2-hydroxypropyl]-N-methylcarbamate —— C30H44Br2N2O8
tert-butyl N-[3-(3-bromophenoxy)-2-hydroxypropyl]-N-methylcarbamate
—— tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-chloro-5-(4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-2-yl) phenoxy)propyl(methyl)carbamate —— C36H54ClN5O6Si
tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-chloro-5-(4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-2-yl) phenoxy)propyl(methyl)carbamate
—— tert-butyl 3-(3-bromophenoxy)-2-hydroxypropyl(methyl)carbamate —— C15H22BrNO4
tert-butyl 3-(3-bromophenoxy)-2-hydroxypropyl(methyl)carbamate
—— tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(4-((4,6-di methyl-2-oxo-2,3-dihydropyridin-3-yl)methylcarbamoyl)-1-isopropyl-1H-pyrazolo[3,4-b]pyridin-6-yl)phenoxy)propyl(methyl)carbamate —— C39H56N6O6Si
tert-butyl 2-(tert-butyldimethylsilyloxy)-3-(3-(4-((4,6-di methyl-2-oxo-2,3-dihydropyridin-3-yl)methylcarbamoyl)-1-isopropyl-1H-pyrazolo[3,4-b]pyridin-6-yl)phenoxy)propyl(methyl)carbamate
—— Tert-butyl 5-cyclopropyl-2,7-diazaspiro[3.5]nonane-2-carboxylate —— C15H26N2O2
Tert-butyl 5-cyclopropyl-2,7-diazaspiro[3.5]nonane-2-carboxylate
—— tert-butyl N-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-3-[3-[4-(3,5-dimethyl-1,2-oxazol-4-yl)-6-[(1-methylpiperidin-4-yl)amino]pyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate —— C36H56N6O5Si
tert-butyl N-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-3-[3-[4-(3,5-dimethyl-1,2-oxazol-4-yl)-6-[(1-methylpiperidin-4-yl)amino]pyrimidin-2-yl]phenoxy]propyl]-N-methylcarbamate