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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl N-[3-[[(Z)-3-[2-(4-cyanoanilino)-4-(propylamino)pyrimidin-5-yl]prop-2-enyl]amino]-3-oxopropyl]carbamate —— C25H33N7O3
tert-butyl N-[3-[[(Z)-3-[2-(4-cyanoanilino)-4-(propylamino)pyrimidin-5-yl]prop-2-enyl]amino]-3-oxopropyl]carbamate
—— tert-butyl (4-(((benzyloxycarbonyl)amino)methyl)tetrahydro-2H-pyran-4-yl)carbamate —— C19H28N2O5
tert-butyl (4-(((benzyloxycarbonyl)amino)methyl)tetrahydro-2H-pyran-4-yl)carbamate
—— tert-butyl N-[(2S)-1-[5-[2-(ethylamino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C23H38N6O3
tert-butyl N-[(2S)-1-[5-[2-(ethylamino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[2-oxo-2-[4-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]piperidin-1-yl]ethyl]carbamate —— C27H40N8O4
tert-butyl N-[2-oxo-2-[4-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]piperidin-1-yl]ethyl]carbamate
—— tert-butyl N-methyl-N-[(2S)-1-[5-[2-[4-(methylcarbamoyl)anilino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]carbamate —— C30H43N7O4
tert-butyl N-methyl-N-[(2S)-1-[5-[2-[4-(methylcarbamoyl)anilino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]carbamate
—— tert-butyl (2S)-2-[5-[2-(1H-indazol-5-ylamino)-4-(3-methoxypropylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate —— C30H40N8O4
tert-butyl (2S)-2-[5-[2-(1H-indazol-5-ylamino)-4-(3-methoxypropylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl (2S)-2-[5-[2-(1H-indazol-5-ylamino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate —— C27H34N8O3
tert-butyl (2S)-2-[5-[2-(1H-indazol-5-ylamino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl N-[3-[2-[2-(3-cyanoanilino)-4-(propylamino)pyrimidin-5-yl]ethynyl]cyclobutyl]carbamate —— C25H30N6O2
tert-butyl N-[3-[2-[2-(3-cyanoanilino)-4-(propylamino)pyrimidin-5-yl]ethynyl]cyclobutyl]carbamate
—— tert-butyl N-[(2S)-1-[5-[2-(2,2-dimethylpropylamino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C26H44N6O3
tert-butyl N-[(2S)-1-[5-[2-(2,2-dimethylpropylamino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-morpholin-4-ylpyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C27H36FN7O4
tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-morpholin-4-ylpyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[3-[[2-(cinnolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H39N9O4
tert-butyl N-[(2S)-1-[3-[[2-(cinnolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C27H38FN7O3
tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H41N7O5
tert-butyl N-[(2S)-1-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[3-[2-[2-chloro-4-[methyl(propyl)amino]pyrimidin-5-yl]ethynyl]anilino]-1-oxopropan-2-yl]-N-methylcarbamate —— C25H32ClN5O3
tert-butyl N-[(2S)-1-[3-[2-[2-chloro-4-[methyl(propyl)amino]pyrimidin-5-yl]ethynyl]anilino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[[5-[2-(4-cyanoanilino)-4-(cyclopropylamino)pyrimidin-5-yl]-3,3-dimethylpent-4-ynyl]amino]-1-oxopropan-2-yl]-N-methylcarbamate —— C30H39N7O3
tert-butyl N-[(2S)-1-[[5-[2-(4-cyanoanilino)-4-(cyclopropylamino)pyrimidin-5-yl]-3,3-dimethylpent-4-ynyl]amino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-pyrrolidin-1-ylpyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C27H36FN7O3
tert-butyl N-[(2S)-1-[5-[2-[(2-fluoropyridin-4-yl)amino]-4-pyrrolidin-1-ylpyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[2-(4-cyano-3-fluoroanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H36FN7O3
tert-butyl N-[(2S)-1-[5-[2-(4-cyano-3-fluoroanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl (2-(4-(propylamino)-2-((2-(pyridin-4-yl)ethyl)amino)pyrimidine-5-carboxamido)ethyl)carbamate —— C22H33N7O3
tert-butyl (2-(4-(propylamino)-2-((2-(pyridin-4-yl)ethyl)amino)pyrimidine-5-carboxamido)ethyl)carbamate
—— tert-butyl N-[(2S)-1-[5-[2-[3-(difluoromethoxy)anilino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H38F2N6O4
tert-butyl N-[(2S)-1-[5-[2-[3-(difluoromethoxy)anilino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-methyl-N-[(2S)-1-[3-[2-[4-[methyl(propyl)amino]-2-(2-pyridin-4-ylethylamino)pyrimidin-5-yl]ethynyl]anilino]-1-oxopropan-2-yl]carbamate —— C32H41N7O3
tert-butyl N-methyl-N-[(2S)-1-[3-[2-[4-[methyl(propyl)amino]-2-(2-pyridin-4-ylethylamino)pyrimidin-5-yl]ethynyl]anilino]-1-oxopropan-2-yl]carbamate
—— tert-butyl ((1S*,3R*)-3-(methoxy(methyl)carbamoyl)cyclohexyl)carbamate —— C14H26N2O4
tert-butyl ((1S*,3R*)-3-(methoxy(methyl)carbamoyl)cyclohexyl)carbamate
—— tert-butyl (2S,4S)-4-hydroxy-2-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate —— C29H41N7O6
tert-butyl (2S,4S)-4-hydroxy-2-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl N-[(2S)-1-[5-[2-(4-carbamoylanilino)-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C29H41N7O4
tert-butyl N-[(2S)-1-[5-[2-(4-carbamoylanilino)-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[(2S)-1-[5-[4-(cyclopropylamino)-2-[(6-methoxypyridin-2-yl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C27H37N7O4
tert-butyl N-[(2S)-1-[5-[4-(cyclopropylamino)-2-[(6-methoxypyridin-2-yl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl methyl(2-oxo-2-((3-(2-((phthalazin-6-yl)amino)-4-(propylamino)pyrimidine-5-carboxamido)propyl)amino)ethyl)carbamate —— C27H37N9O4
tert-butyl methyl(2-oxo-2-((3-(2-((phthalazin-6-yl)amino)-4-(propylamino)pyrimidine-5-carboxamido)propyl)amino)ethyl)carbamate
—— tert-butyl N-[(2S)-1-[5-[2-[4-(cyclopropylcarbamoyl)anilino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C32H45N7O4
tert-butyl N-[(2S)-1-[5-[2-[4-(cyclopropylcarbamoyl)anilino]-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[3-oxo-3-[2-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]ethylamino]propyl]carbamate —— C25H38N8O4
tert-butyl N-[3-oxo-3-[2-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]ethylamino]propyl]carbamate
—— tert-butyl N-[(2S)-1-[5-[2-(3-fluoroanilino)-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H39FN6O3
tert-butyl N-[(2S)-1-[5-[2-(3-fluoroanilino)-4-[methyl(propyl)amino]pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— Tert-butyl ((1S,3R)-3-ethynylcyclopentyl)carbamate —— C12H19NO2
Tert-butyl ((1S,3R)-3-ethynylcyclopentyl)carbamate
—— tert-butyl N-[2-oxo-2-[2-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]ethylamino]ethyl]carbamate —— C24H36N8O4
tert-butyl N-[2-oxo-2-[2-[[4-(propylamino)-2-(2-pyridin-4-ylethylamino)pyrimidine-5-carbonyl]amino]ethylamino]ethyl]carbamate
—— tert-butyl N-[2-[5-[2-(4-carbamoylanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-2-oxoethyl]carbamate —— C26H35N7O4
tert-butyl N-[2-[5-[2-(4-carbamoylanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-2-oxoethyl]carbamate
—— tert-butyl N-[(1S,3R)-3-[2-[2-(4-cyanoanilino)-4-(cyclopropylamino)pyrimidin-5-yl]ethynyl]cyclohexyl]carbamate —— C27H32N6O2
tert-butyl N-[(1S,3R)-3-[2-[2-(4-cyanoanilino)-4-(cyclopropylamino)pyrimidin-5-yl]ethynyl]cyclohexyl]carbamate
—— tert-butyl N-methyl-N-[(2S)-1-[5-[2-[(3-methyl-1,2-thiazol-5-yl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]carbamate —— C25H37N7O3S
tert-butyl N-methyl-N-[(2S)-1-[5-[2-[(3-methyl-1,2-thiazol-5-yl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]carbamate
—— tert-butyl N-[(2S)-1-[5-[2-(4-fluoro-3-methoxyanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate —— C28H39FN6O4
tert-butyl N-[(2S)-1-[5-[2-(4-fluoro-3-methoxyanilino)-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-methyl-N-[2-oxo-2-[3-[[2-(phthalazin-6-ylamino)-6-(propylamino)-1,2-dihydropyrimidine-5-carbonyl]amino]propylamino]ethyl]carbamate —— C27H39N9O4
tert-butyl N-methyl-N-[2-oxo-2-[3-[[2-(phthalazin-6-ylamino)-6-(propylamino)-1,2-dihydropyrimidine-5-carbonyl]amino]propylamino]ethyl]carbamate
—— tert-butyl (2S)-2-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate —— C29H41N7O5
tert-butyl (2S)-2-[5-[4-(3-methoxypropylamino)-2-[(2-methoxypyridin-4-yl)amino]pyrimidin-5-yl]pent-4-ynylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl (3-cyano-1,5-dimethoxypentan-3-yl)carbamate —— C13H24N2O4
tert-butyl (3-cyano-1,5-dimethoxypentan-3-yl)carbamate
—— tert-butyl N-[(2S)-1-[[2-[2-(3-fluoroanilino)-4-(propylamino)pyrimidin-5-yl]-1,3-benzoxazol-6-yl]amino]-1-oxopropan-2-yl]carbamate —— C28H32FN7O4
tert-butyl N-[(2S)-1-[[2-[2-(3-fluoroanilino)-4-(propylamino)pyrimidin-5-yl]-1,3-benzoxazol-6-yl]amino]-1-oxopropan-2-yl]carbamate
—— tert-butyl N-[3-[[2-(cinnolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propyl]carbamate —— C24H32N8O3
tert-butyl N-[3-[[2-(cinnolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propyl]carbamate
—— tert-butyl N-[(2S)-1-[[(1S,3R)-3-[2-[2-(3-fluoroanilino)-4-(2-methoxyethylamino)pyrimidin-5-yl]ethynyl]cyclohexyl]amino]-1-oxopropan-2-yl]-N-methylcarbamate —— C30H41FN6O4
tert-butyl N-[(2S)-1-[[(1S,3R)-3-[2-[2-(3-fluoroanilino)-4-(2-methoxyethylamino)pyrimidin-5-yl]ethynyl]cyclohexyl]amino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl N-[5-[2-(4-cyanoanilino)-4-(1,5-dihydropyrazol-2-yl)pyrimidin-5-yl]pent-4-ynyl]carbamate —— C24H27N7O2
tert-butyl N-[5-[2-(4-cyanoanilino)-4-(1,5-dihydropyrazol-2-yl)pyrimidin-5-yl]pent-4-ynyl]carbamate
—— tert-butyl N-[(2S)-1-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]anilino]-1-oxopropan-2-yl]-N-methylcarbamate —— C32H38N8O4
tert-butyl N-[(2S)-1-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]anilino]-1-oxopropan-2-yl]-N-methylcarbamate
—— tert-butyl (2S)-4,4-difluoro-2-[5-[2-(4-fluoroanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-2-methylpyrrolidine-1-carboxylate —— C27H33F3N6O3
tert-butyl (2S)-4,4-difluoro-2-[5-[2-(4-fluoroanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-2-methylpyrrolidine-1-carboxylate
—— tert-butyl N-[2-[[3-[[2-(4-carbamoylanilino)-4-(propylamino)pyrimidine-5-carbonyl]amino]cyclohexyl]amino]-2-oxoethyl]-N-methylcarbamate —— C29H42N8O5
tert-butyl N-[2-[[3-[[2-(4-carbamoylanilino)-4-(propylamino)pyrimidine-5-carbonyl]amino]cyclohexyl]amino]-2-oxoethyl]-N-methylcarbamate
—— tert-butyl (2S,4S)-2-[5-[2-(4-cyanoanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-4-fluoro-2-methylpyrrolidine-1-carboxylate —— C28H34FN7O3
tert-butyl (2S,4S)-2-[5-[2-(4-cyanoanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-4-fluoro-2-methylpyrrolidine-1-carboxylate
—— tert-butyl N-[2-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-2-oxoethyl]carbamate —— C27H36N8O4
tert-butyl N-[2-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-2-oxoethyl]carbamate
—— tert-butyl (2S,4S)-2-[5-[2-(4-fluoroanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-2,4-dimethylpyrrolidine-1-carboxylate —— C28H37FN6O3
tert-butyl (2S,4S)-2-[5-[2-(4-fluoroanilino)-4-(methylamino)pyrimidin-5-yl]pent-4-ynylcarbamoyl]-2,4-dimethylpyrrolidine-1-carboxylate
—— tert-butyl N-[1-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-2-methyl-1-oxopropan-2-yl]carbamate —— C29H40N8O4
tert-butyl N-[1-[3-[[2-(isoquinolin-6-ylamino)-4-(propylamino)pyrimidine-5-carbonyl]amino]propylamino]-2-methyl-1-oxopropan-2-yl]carbamate
—— tert-butyl N-[2-[[3-[[2-(4-carbamoylanilino)-4-(propylamino)pyrimidine-5-carbonyl]amino]cyclohexyl]amino]-2-oxoethyl]carbamate —— C28H40N8O5
tert-butyl N-[2-[[3-[[2-(4-carbamoylanilino)-4-(propylamino)pyrimidine-5-carbonyl]amino]cyclohexyl]amino]-2-oxoethyl]carbamate
—— tert-butyl 3-((3-aminophenyl)amino)piperidine-1-carboxylate —— C16H25N3O2
tert-butyl 3-((3-aminophenyl)amino)piperidine-1-carboxylate