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—— Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate —— C43H72BN3O9Si
Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate
—— Tert-butyl 2-methoxy-3-[2-[[2-[3-[(2-methylpropan-2-yl)oxycarbonylamino]pyrrolidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate —— C35H54BN3O8
Tert-butyl 2-methoxy-3-[2-[[2-[3-[(2-methylpropan-2-yl)oxycarbonylamino]pyrrolidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate
—— Tert-butyl 2-methoxy-3-[2-[[2-[4-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]piperazin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate —— C36H56BN3O8
Tert-butyl 2-methoxy-3-[2-[[2-[4-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]piperazin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate
—— tert-butyl N-[2-[[3-[3-(3-methoxypropylcarbamoyl)-4,4-dimethylcyclohexyl]-1-(oxan-2-yl)pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C31H55N5O5
tert-butyl N-[2-[[3-[3-(3-methoxypropylcarbamoyl)-4,4-dimethylcyclohexyl]-1-(oxan-2-yl)pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— Tert-butyl 3-[2-[[2-[4-hydroxy-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate —— C36H56BN3O9
Tert-butyl 3-[2-[[2-[4-hydroxy-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate
—— tert-butyl 3-(hydroxymethyl)-4-(1-isopropyl-1H-pyrazol-5-yl)-2,5-dihydro-1H-pyrrole-1-carboxylate —— C16H25N3O3
tert-butyl 3-(hydroxymethyl)-4-(1-isopropyl-1H-pyrazol-5-yl)-2,5-dihydro-1H-pyrrole-1-carboxylate
—— tert-butyl N-[2-[[3-[(5S)-1,1-dimethyl-2-oxaspiro[4.5]dec-7-en-8-yl]-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C29H48N4O4
tert-butyl N-[2-[[3-[(5S)-1,1-dimethyl-2-oxaspiro[4.5]dec-7-en-8-yl]-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— tert-butyl N-[[4-[2-(dimethylamino)-2-oxoethoxy]-3-ethoxyphenyl]methylideneamino]carbamate —— C18H27N3O5
tert-butyl N-[[4-[2-(dimethylamino)-2-oxoethoxy]-3-ethoxyphenyl]methylideneamino]carbamate
—— Tert-butyl-dimethyl-[7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[4.5]dec-6-en-10-yl]oxysilane —— C22H41BO3Si
Tert-butyl-dimethyl-[7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[4.5]dec-6-en-10-yl]oxysilane
—— tert-butyl 4-[2-[7-oxo-5-(trifluoromethyl)-2H-pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate —— C23H27F3N4O3
tert-butyl 4-[2-[7-oxo-5-(trifluoromethyl)-2H-pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate
—— tert-butyl N-[2-[[4-(3,3-dimethyl-1-oxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-3-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C29H50N4O4
tert-butyl N-[2-[[4-(3,3-dimethyl-1-oxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-3-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— Tert-butyl 2-[[5-(1,3-benzothiazol-2-ylsulfanylmethyl)-4-benzyl-1,2,4-triazol-3-yl]sulfanyl]acetate —— C23H24N4O2S3
Tert-butyl 2-[[5-(1,3-benzothiazol-2-ylsulfanylmethyl)-4-benzyl-1,2,4-triazol-3-yl]sulfanyl]acetate
—— tert-butyl N-(2-{ [(3-{5-[(tert-butyldimethylsilyl)oxy]spiro[5.5]undec-2-en-2-yl}-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl] (methyl)amino}ethyl)-N-methylcarbamate —— C35H62N4O4Si
tert-butyl N-(2-{ [(3-{5-[(tert-butyldimethylsilyl)oxy]spiro[5.5]undec-2-en-2-yl}-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl] (methyl)amino}ethyl)-N-methylcarbamate
—— tert-butyl N-[2-[[3-(1,1-dimethyl-2-oxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C29H50N4O4
tert-butyl N-[2-[[3-(1,1-dimethyl-2-oxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— Tert-butyl 4-[3-[3-fluoro-7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate —— C24H31FN4O3
Tert-butyl 4-[3-[3-fluoro-7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate
—— tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-3-(4-oxocyclohexyl)pyrazol-4-yl]methyl]amino]ethyl]carbamate —— C24H40N4O4
tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-3-(4-oxocyclohexyl)pyrazol-4-yl]methyl]amino]ethyl]carbamate
—— tert-butyl 5-[4-[[methyl-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]methyl]-1-[(2R)-oxan-2-yl]pyrazol-3-yl]indazole-1-carboxylate —— C29H42N6O5
tert-butyl 5-[4-[[methyl-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]methyl]-1-[(2R)-oxan-2-yl]pyrazol-3-yl]indazole-1-carboxylate
—— tert-butyl 3-(4-(2-((5-bromo-2-carbamoyl-4-chlorophenyl)amino)acetyl)piperazin-1-yl)azetidine-1-carboxylate —— C21H29BrClN5O4
tert-butyl 3-(4-(2-((5-bromo-2-carbamoyl-4-chlorophenyl)amino)acetyl)piperazin-1-yl)azetidine-1-carboxylate
—— tert-butyl 3-(4-(4,5-dichloro-2-methoxybenzylcarbamoyl)piperidin-1-yl)azetidine-1-carboxylate —— C22H31Cl2N3O4
tert-butyl 3-(4-(4,5-dichloro-2-methoxybenzylcarbamoyl)piperidin-1-yl)azetidine-1-carboxylate
—— tert-butyl 3-(4-acryloylpiperazin-1-yl)azetidine-1-carboxylate —— C15H25N3O3
tert-butyl 3-(4-acryloylpiperazin-1-yl)azetidine-1-carboxylate
—— tert-butyl 4-[3-(3-fluoro-5-methyl-7-oxo-2H-pyrido[3,4-b]indol-9-yl)propyl]piperazine-1-carboxylate —— C24H31FN4O3
tert-butyl 4-[3-(3-fluoro-5-methyl-7-oxo-2H-pyrido[3,4-b]indol-9-yl)propyl]piperazine-1-carboxylate
—— tert-butyl methyl(2-(methyl((5-((tetrahydro-2H-pyran-4-yl)oxy)-1H-indazol-3-yl)methyl)amino)ethyl)carbamate —— C22H34N4O4
tert-butyl methyl(2-(methyl((5-((tetrahydro-2H-pyran-4-yl)oxy)-1H-indazol-3-yl)methyl)amino)ethyl)carbamate
—— tert-butyl N-[2-[[5-[3-[10-[tert-butyl(dimethyl)silyl]oxyspiro[4.5]dec-7-en-7-yl]oxan-2-yl]-1H-pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C34H60N4O4Si
tert-butyl N-[2-[[5-[3-[10-[tert-butyl(dimethyl)silyl]oxyspiro[4.5]dec-7-en-7-yl]oxan-2-yl]-1H-pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— tert-butyl N-[2-[[3-(1,4-dioxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C26H44N4O5
tert-butyl N-[2-[[3-(1,4-dioxaspiro[4.5]decan-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— Tert-butyl 4-[3-[7-methoxy-5-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate —— C25H31F3N4O3
Tert-butyl 4-[3-[7-methoxy-5-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate
—— Tert-butyl 4-[2-[7-methoxy-5-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate —— C24H29F3N4O3
Tert-butyl 4-[2-[7-methoxy-5-(trifluoromethyl)pyrido[3,4-b]indol-9-yl]ethyl]piperazine-1-carboxylate
—— tert-butyl 4-[2-(3-fluoro-1-methyl-7-oxo-2H-pyrido[3,4-b]indol-9-yl)ethyl]piperazine-1-carboxylate —— C23H29FN4O3
tert-butyl 4-[2-(3-fluoro-1-methyl-7-oxo-2H-pyrido[3,4-b]indol-9-yl)ethyl]piperazine-1-carboxylate
—— tert-butyl 6-bromo-[1,2,4]triazolo[4,3-a]pyridine-7-carboxylate —— C11H12BrN3O2
tert-butyl 6-bromo-[1,2,4]triazolo[4,3-a]pyridine-7-carboxylate
—— tert-butyl N-(2-[[(3-[1,4-dioxaspiro[4.5]decan-8-yl]-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl](methyl)amino]ethyl)-N-methylcarbamate —— C26H44N4O5
tert-butyl N-(2-[[(3-[1,4-dioxaspiro[4.5]decan-8-yl]-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl](methyl)amino]ethyl)-N-methylcarbamate
—— Tert-butyl 4-[3-[7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate —— C25H34N4O3
Tert-butyl 4-[3-[7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate
—— tert-butyl N-methyl-N-[2-[methyl-[[5-(4-nitrophenoxy)-1-[(2R)-oxan-2-yl]indazol-3-yl]methyl]amino]ethyl]carbamate —— C28H37N5O6
tert-butyl N-methyl-N-[2-[methyl-[[5-(4-nitrophenoxy)-1-[(2R)-oxan-2-yl]indazol-3-yl]methyl]amino]ethyl]carbamate
—— tert-butyl 3-(4-(2-(5-chloro-4-ethyl-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate —— C23H35ClN4O4
tert-butyl 3-(4-(2-(5-chloro-4-ethyl-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate
—— tert-butyl N-(2-{[(3-{10-[(tert-butyldimethylsilyl)oxy]spiro[4.5]decan-7-yl}-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl] (methyl)amino}ethyl)-N-methylcarbamate —— C34H62N4O4Si
tert-butyl N-(2-{[(3-{10-[(tert-butyldimethylsilyl)oxy]spiro[4.5]decan-7-yl}-1-(oxan-2-yl)-1H-pyrazol-4-yl)methyl] (methyl)amino}ethyl)-N-methylcarbamate
—— tert-butyl 5-oxotetrahydro-2H-pyran-2-carboxylate —— C10H16O4
tert-butyl 5-oxotetrahydro-2H-pyran-2-carboxylate
—— Tert-butyl 3-[4-[2-(5-bromo-4-chloro-2-methoxyanilino)propanoyl]piperazin-1-yl]azetidine-1-carboxylate —— C22H32BrClN4O4
Tert-butyl 3-[4-[2-(5-bromo-4-chloro-2-methoxyanilino)propanoyl]piperazin-1-yl]azetidine-1-carboxylate
—— trimethyl-[[2-(2-pyrrolidin-1-ylphenyl)-2,3-dihydro-1H-indol-7-yl]oxy]silane —— C21H28N2OSi
trimethyl-[[2-(2-pyrrolidin-1-ylphenyl)-2,3-dihydro-1H-indol-7-yl]oxy]silane
—— tert-butyl 3-(5-bromo-3,7-dihydroxy-3H-1,2-benzothiazol-2-yl)-3-methylbutanoate —— C16H22BrNO4S
tert-butyl 3-(5-bromo-3,7-dihydroxy-3H-1,2-benzothiazol-2-yl)-3-methylbutanoate
—— tert-butyl 3-(4-(2-(4-bromo-5-chloro-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate —— C21H30BrClN4O4
tert-butyl 3-(4-(2-(4-bromo-5-chloro-2-methoxyphenylamino)acetyl)piperazin-1-yl)azetidine-1-carboxylate
—— tert-butyl N-[[2,4-bis(difluoromethoxy)phenyl]methylideneamino]carbamate —— C14H16F4N2O4
tert-butyl N-[[2,4-bis(difluoromethoxy)phenyl]methylideneamino]carbamate
—— tert-butyl N-(2-bromo-3-formyl-6-phenylmethoxyphenoxy)-N-ethylcarbamate —— C21H24BrNO5
tert-butyl N-(2-bromo-3-formyl-6-phenylmethoxyphenoxy)-N-ethylcarbamate
—— tert-butyl (3R,4R)-3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-3-[2-[2-(2,5-dioxopyrrol-1-yl)ethoxy]ethylamino]-2,2-dimethyl-3-oxopropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C42H51F3N6O8
tert-butyl (3R,4R)-3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-3-[2-[2-(2,5-dioxopyrrol-1-yl)ethoxy]ethylamino]-2,2-dimethyl-3-oxopropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-4-[6-(2,5-dioxopyrrol-1-yl)hexanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C47H57F3N6O8
tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-4-[6-(2,5-dioxopyrrol-1-yl)hexanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-3-[2-[2-(2,5-dioxopyrrol-1-yl)ethoxy]ethylamino]-2,2-dimethyl-3-oxopropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C42H51F3N6O8
tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-3-[2-[2-(2,5-dioxopyrrol-1-yl)ethoxy]ethylamino]-2,2-dimethyl-3-oxopropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.2.2]nona-1(7),5,8-trien-7-yl]oxy]silane —— C21H28N2OSi
Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.2.2]nona-1(7),5,8-trien-7-yl]oxy]silane
—— tert-butyl N-[1-[4-(cycloheptylcarbamoyl)-3-fluorophenyl]ethyl]carbamate —— C21H31FN2O3
tert-butyl N-[1-[4-(cycloheptylcarbamoyl)-3-fluorophenyl]ethyl]carbamate
—— tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethylpropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-hydroxypyrrolidine-1-carboxylate —— C34H44F2N4O5
tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethylpropyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-hydroxypyrrolidine-1-carboxylate
—— tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-(methylamino)-4-oxobutyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C36H46F3N5O5
tert-butyl 3-[[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-(methylamino)-4-oxobutyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]pyrrolidine-1-carboxylate —— C35H44F2N4O5
tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]pyrrolidine-1-carboxylate
—— tert-Butyl 4-oxopiperidine-3-carboxylate —— C10H17NO3
tert-Butyl 4-oxopiperidine-3-carboxylate
—— tert-butyl (5Z)-5-(cyanomethylidene)oxane-2-carboxylate —— C12H17NO3
tert-butyl (5Z)-5-(cyanomethylidene)oxane-2-carboxylate