中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-[[(2R)-oxolan-2-yl]methyl]pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H36FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-(4-bromo-2-fluorophenyl)-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C21H25BrFN3O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2,3-difluoro-4-(2-oxo-1,3-dihydroindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H30F2N4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(4-fluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H29FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(3-methyl-3,8-diazabicyclo[3.2.1]octan-8-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H38FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(methylcarbamoyl)thiophen-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H31FN4O4S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(3-methylbutanoyl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H36FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(methylcarbamoyl)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H33FN4O4 |
|
—— |
thiophen-2-ylmethyl (2R)-2-(4-chlorophenoxy)propanoate |
—— |
C14H13ClO3S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-[4-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H33FN4O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(ethylcarbamoyl)furan-2-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H33FN4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[2-[4-(1-acetyl-5-methylpyrazol-3-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H32FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(1,1-dimethyl-3-oxo-2-benzofuran-5-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H34FN3O5 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-2-[4-(3-carbamoylphenyl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C29H31FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(4-azido-2-fluorophenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C21H27FN6O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-5-(6-oxo-1H-pyridin-2-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H29FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-oxo-1H-pyridin-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H29FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(2-oxo-3H-1-benzofuran-5-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H32FN3O6 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(5-carbamoylthiophen-3-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H29FN4O4S |
|
—— |
tert-butyl (1R,3S,4S)-3-[(1-cyano-2-dibenzofuran-2-ylethyl)carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H29N3O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(1-ethylpiperidin-4-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H39FN4O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(1-tert-butylpyrazol-4-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H36FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2-ethyl-1,3-thiazol-5-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H31FN4O3S |
|
—— |
Thiophen-2-ylmethyl 5-(1,3-benzothiazol-2-yl)thiophene-2-carboxylate |
—— |
C17H11NO2S3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3-cyclopropylsulfonylphenyl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H34FN3O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[1-(benzenesulfonyl)pyrazol-4-yl]-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H32FN5O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(2,4-difluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H28F2N4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2,3-difluoro-4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H32F2N4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(4-bromo-2-fluorophenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C21H27BrFN3O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[(Z)-1-amino-3-(2-methoxyacetyl)iminoprop-1-en-2-yl]-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H34FN5O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H39BFN3O6 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(2-cyano-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H29N5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1H-pyrazol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C24H28FN5O3 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(4-methylsulfinamoylphenyl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C29H33FN4O4S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(2-fluoro-4-pyrrolidin-3-ylphenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C25H35FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-pyrazolo[1,5-a]pyrimidin-3-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H29FN6O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-(1,3,4,6,7,9a-hexahydropyrido[2,1-c][1,4]oxazin-8-yl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H37FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(4-methylpiperazine-1-carbonyl)furan-2-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H38FN5O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)piperidin-3-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H43FN4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-3-(1-fluoro-6-morpholin-4-yl-5,6,7,8-tetrahydronaphthalen-2-yl)-1-methoxy-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H42FN3O6 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-[1-(oxolan-3-yl)-2,3,3a,4,6,6a-hexahydropyrrolo[3,4-b]pyrrol-5-yl]phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H44FN5O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(1-oxo-3H-2-benzofuran-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H30FN3O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-[1-[(2-methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]-2-oxo-3H-indol-5-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C39H48FN5O6 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(9-fluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H29FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(oxan-2-ylmethyl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H38FN5O4 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methylindazol-6-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C30H32FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(3-methylsulfonylphenyl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H32FN3O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(furan-2-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C25H28FN3O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-3-[4-(2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[2,3-c]pyrrol-5-yl)-2-fluorophenyl]-1-amino-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H38FN5O4 |
|
—— |
Tert-butyl 4-[3-(1-aminoethenylsulfanyl)propyl]piperazine-1-carboxylate |
—— |
C14H27N3O2S |
|