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—— methyl 4-[[(1S,4S,6R)-6-bromo-4,5,5-trimethylbicyclo[2.1.1]hexane-1-carbonyl]amino]benzoate —— C18H22BrNO3
methyl 4-[[(1S,4S,6R)-6-bromo-4,5,5-trimethylbicyclo[2.1.1]hexane-1-carbonyl]amino]benzoate
—— methyl (2S)-2-[[(5R,7R)-3-(4-nitrophenyl)adamantane-1-carbonyl]amino]propanoate —— C21H26N2O5
methyl (2S)-2-[[(5R,7R)-3-(4-nitrophenyl)adamantane-1-carbonyl]amino]propanoate
—— methyl (3R)-4-(4-methoxyphenyl)-5-[N-(4-methylphenyl)-C-phenylcarbonimidoyl]imino-3-(trichloromethyl)-1,2,4-thiadiazolidine-2-carboxylate —— C26H23Cl3N4O3S
methyl (3R)-4-(4-methoxyphenyl)-5-[N-(4-methylphenyl)-C-phenylcarbonimidoyl]imino-3-(trichloromethyl)-1,2,4-thiadiazolidine-2-carboxylate
—— methyl (3S,5S)-3,5-dimethyladamantane-1-carboxylate —— C14H22O2
methyl (3S,5S)-3,5-dimethyladamantane-1-carboxylate
—— methyl 3-[[(5S,7S)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]benzoate —— C26H29NO3
methyl 3-[[(5S,7S)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]benzoate
—— methyl (3R,5R)-3,5-dimethyladamantane-1-carboxylate —— C14H22O2
methyl (3R,5R)-3,5-dimethyladamantane-1-carboxylate
—— methyl (2R)-2-[[(5R,7R)-3-(4-nitrophenyl)adamantane-1-carbonyl]amino]propanoate —— C21H26N2O5
methyl (2R)-2-[[(5R,7R)-3-(4-nitrophenyl)adamantane-1-carbonyl]amino]propanoate
—— methyl 2-[(2S)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C23H25N5O6S2
methyl 2-[(2S)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl (2E,5S)-2-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H21ClN2O6S
methyl (2E,5S)-2-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl [(5Z)-5-(3-bromo-5-chloro-2-methoxybenzylidene)-4-oxo-3-phenyl-2-thioxoimidazolidin-1-yl]acetate —— C20H16BrClN2O4S
methyl [(5Z)-5-(3-bromo-5-chloro-2-methoxybenzylidene)-4-oxo-3-phenyl-2-thioxoimidazolidin-1-yl]acetate
—— methyl (2E,5R)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H21ClN2O6S
methyl (2E,5R)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 3-[[(5R,7R)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]benzoate —— C26H29NO3
methyl 3-[[(5R,7R)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]benzoate
—— methyl (2S)-3-methyl-2-[[(5S,7S)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]butanoate —— C24H33NO3
methyl (2S)-3-methyl-2-[[(5S,7S)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]butanoate
—— methyl 2-[(2R)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C23H25N5O6S2
methyl 2-[(2R)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 2-[(5Z)-5-[[1-(3-nitrophenyl)pyrrol-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C18H15N3O6S
methyl 2-[(5Z)-5-[[1-(3-nitrophenyl)pyrrol-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— methyl 2-[[(5R,7R)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]acetate —— C21H27NO3
methyl 2-[[(5R,7R)-3-(4-methylphenyl)adamantane-1-carbonyl]amino]acetate
—— methyl (2E,5S)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H21ClN2O6S
methyl (2E,5S)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-5-(4-methoxycarbonylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5S)-2-[[5-(2,5-dichlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H20Cl2N2O4S2
methyl (2E,5S)-2-[[5-(2,5-dichlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5R)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H21ClN2O4S2
methyl (2E,5R)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5S)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H21ClN2O4S2
methyl (2E,5S)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-7-methyl-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[(2S)-1-[3-[(Z)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C24H21N5O6S2
methyl 2-[(2S)-1-[3-[(Z)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl (5R,7R)-3-(4-nitrophenyl)adamantane-1-carboxylate —— C18H21NO4
methyl (5R,7R)-3-(4-nitrophenyl)adamantane-1-carboxylate
—— methyl N-[4-[(3R)-3-[[4-(pyrimidin-2-ylsulfamoyl)phenyl]carbamoyl]piperidin-1-yl]sulfonylphenyl]carbamate —— C24H26N6O7S2
methyl N-[4-[(3R)-3-[[4-(pyrimidin-2-ylsulfamoyl)phenyl]carbamoyl]piperidin-1-yl]sulfonylphenyl]carbamate
—— methyl 3-[(1R,2R,6S,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate —— C19H17NO4
methyl 3-[(1R,2R,6S,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate
—— methyl (2E,5R)-5-(4-tert-butylphenyl)-7-methyl-2-[[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H34N4O3S
methyl (2E,5R)-5-(4-tert-butylphenyl)-7-methyl-2-[[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate —— C17H15NO4
methyl 3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate
—— methyl 3-[(1R,2S,6S,7R)-3,5-dioxo-10-propan-2-ylidene-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate —— C20H19NO4
methyl 3-[(1R,2S,6S,7R)-3,5-dioxo-10-propan-2-ylidene-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate
—— methyl 4-(5-{(E)-[1-(2,3-dimethylphenyl)-4,6-dioxo-2-thioxotetrahydropyrimidin-5(2H)-ylidene]methyl}furan-2-yl)benzoate —— C25H20N2O5S
methyl 4-(5-{(E)-[1-(2,3-dimethylphenyl)-4,6-dioxo-2-thioxotetrahydropyrimidin-5(2H)-ylidene]methyl}furan-2-yl)benzoate
—— methyl 3-[(1R,2R,6R,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate —— C19H17NO4
methyl 3-[(1R,2R,6R,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate
—— methyl 3-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1-benzothiophene-2-carboxylate —— C27H30N2O5S2
methyl 3-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1-benzothiophene-2-carboxylate
—— methyl 3-[(1R,2S,6S,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate —— C19H17NO4
methyl 3-[(1R,2S,6S,7R)-3,5-dioxospiro[4-azatricyclo[5.2.1.02,6]dec-8-ene-10,1'-cyclopropane]-4-yl]benzoate
—— methyl 2-[[[5-bromo-2-[[(Z)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]-phenylmethyl]amino]acetate —— C23H21BrN2O3
methyl 2-[[[5-bromo-2-[[(Z)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]-phenylmethyl]amino]acetate
—— methyl 4-[2-[[4-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1,3-thiazol-4-yl]benzoate —— C28H31N3O5S2
methyl 4-[2-[[4-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1,3-thiazol-4-yl]benzoate
—— methyl N-[4-[(3S)-3-[[4-(pyrimidin-2-ylsulfamoyl)phenyl]carbamoyl]piperidin-1-yl]sulfonylphenyl]carbamate —— C24H26N6O7S2
methyl N-[4-[(3S)-3-[[4-(pyrimidin-2-ylsulfamoyl)phenyl]carbamoyl]piperidin-1-yl]sulfonylphenyl]carbamate
—— methyl 4-[2-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1,3-thiazol-4-yl]benzoate —— C28H31N3O5S2
methyl 4-[2-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1,3-thiazol-4-yl]benzoate
—— methyl (2E,5S)-5-(4-tert-butylphenyl)-7-methyl-2-[[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H34N4O3S
methyl (2E,5S)-5-(4-tert-butylphenyl)-7-methyl-2-[[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[(5Z)-5-[(3-bromo-5-chloro-4-hydroxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C14H11BrClNO5S
methyl 2-[(5Z)-5-[(3-bromo-5-chloro-4-hydroxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— methyl 5-phenyl-3-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]thiophene-2-carboxylate —— C29H32N2O5S2
methyl 5-phenyl-3-[[4-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]thiophene-2-carboxylate
—— methyl 4-[[(Z)-(3-chloro-5-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-(4-chlorophenyl)methyl]amino]pentanoate —— C20H21Cl2NO3
methyl 4-[[(Z)-(3-chloro-5-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-(4-chlorophenyl)methyl]amino]pentanoate
—— methyl 2-[(2R)-1-[3-[(Z)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C24H21N5O6S2
methyl 2-[(2R)-1-[3-[(Z)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 4-{(Z)-[3-(1-ethoxy-1-oxopropan-2-yl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}benzoate —— C17H17NO6S
methyl 4-{(Z)-[3-(1-ethoxy-1-oxopropan-2-yl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}benzoate
—— methyl N-[4-[(3S)-3-(4-benzhydrylpiperazine-1-carbonyl)piperidin-1-yl]sulfonylphenyl]carbamate —— C31H36N4O5S
methyl N-[4-[(3S)-3-(4-benzhydrylpiperazine-1-carbonyl)piperidin-1-yl]sulfonylphenyl]carbamate
—— methyl N-[4-[(3R)-3-(4-benzhydrylpiperazine-1-carbonyl)piperidin-1-yl]sulfonylphenyl]carbamate —— C31H36N4O5S
methyl N-[4-[(3R)-3-(4-benzhydrylpiperazine-1-carbonyl)piperidin-1-yl]sulfonylphenyl]carbamate
—— methyl 3-[[4-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1-benzothiophene-2-carboxylate —— C27H30N2O5S2
methyl 3-[[4-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]amino]-1-benzothiophene-2-carboxylate
—— methyl (2E,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[(4-phenylmethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H26N2O5S
methyl (2E,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[(4-phenylmethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5R)-2-[(3-methoxy-4-pentoxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N2O6S
methyl (2E,5R)-2-[(3-methoxy-4-pentoxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5R)-2-[[3-methoxy-4-(3-methylbutoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N2O6S
methyl (2E,5R)-2-[[3-methoxy-4-(3-methylbutoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-methyl-2-[(2Z)-2-[6-methyl-2-(4-methylphenyl)chromen-4-ylidene]hydrazinyl]-1,3-thiazole-5-carboxylate —— C23H21N3O3S
methyl 4-methyl-2-[(2Z)-2-[6-methyl-2-(4-methylphenyl)chromen-4-ylidene]hydrazinyl]-1,3-thiazole-5-carboxylate
—— methyl (2E,5R)-5-(4-methoxyphenyl)-2-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28N2O6S
methyl (2E,5R)-5-(4-methoxyphenyl)-2-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[2-[(2Z)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6,8-dimethylchromen-4-yl]hydrazinyl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H23N3O5S
methyl 2-[2-[(2Z)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6,8-dimethylchromen-4-yl]hydrazinyl]-4-methyl-1,3-thiazole-5-carboxylate