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中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl 2-[(1S,11R,12S,16R)-11-(4-methoxybenzoyl)-13,15-dioxo-9,10,14-triazatetracyclo[8.6.0.02,7.012,16]hexadeca-2,4,6,8-tetraen-14-yl]benzoate —— C29H23N3O6
methyl 2-[(1S,11R,12S,16R)-11-(4-methoxybenzoyl)-13,15-dioxo-9,10,14-triazatetracyclo[8.6.0.02,7.012,16]hexadeca-2,4,6,8-tetraen-14-yl]benzoate
—— methyl 2-[(1R,11R,12S,16R)-11-(4-methoxybenzoyl)-13,15-dioxo-9,10,14-triazatetracyclo[8.6.0.02,7.012,16]hexadeca-2,4,6,8-tetraen-14-yl]benzoate —— C29H23N3O6
methyl 2-[(1R,11R,12S,16R)-11-(4-methoxybenzoyl)-13,15-dioxo-9,10,14-triazatetracyclo[8.6.0.02,7.012,16]hexadeca-2,4,6,8-tetraen-14-yl]benzoate
—— methyl (1R,2S,3R,4R)-3-[(4-methylphenyl)carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylate —— C17H19NO3
methyl (1R,2S,3R,4R)-3-[(4-methylphenyl)carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylate
—— methyl 4-[(3R,3aS,6aS)-5-(4-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]benzoate —— C25H19N3O7
methyl 4-[(3R,3aS,6aS)-5-(4-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]benzoate
—— methyl 2-(4-ethoxycarbonylphenyl)imino-3-(3-morpholin-4-ylpropyl)-4-oxo-1,3-thiazine-6-carboxylate;hydrochloride —— C22H28ClN3O6S
methyl 2-(4-ethoxycarbonylphenyl)imino-3-(3-morpholin-4-ylpropyl)-4-oxo-1,3-thiazine-6-carboxylate;hydrochloride
—— methyl 4-[(3S,3aS,6aS)-5-(4-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]benzoate —— C25H19N3O7
methyl 4-[(3S,3aS,6aS)-5-(4-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-3-yl]benzoate
—— methyl (1S,3S,6S,9S)-8-benzyl-6-methyl-4-oxo-9-phenyl-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate —— C23H23NO5
methyl (1S,3S,6S,9S)-8-benzyl-6-methyl-4-oxo-9-phenyl-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate
—— methyl (1S,3S,6R,9S)-8-benzyl-6-methyl-4-oxo-9-phenyl-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate —— C23H23NO5
methyl (1S,3S,6R,9S)-8-benzyl-6-methyl-4-oxo-9-phenyl-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate
—— morpholin-4-yl-[(5S,7S)-3-(1,2,4-triazol-1-yl)-1-adamantyl]methanone —— C17H24N4O2
morpholin-4-yl-[(5S,7S)-3-(1,2,4-triazol-1-yl)-1-adamantyl]methanone
—— methyl 4-[(3R,3aR,6aS)-3-(3-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate —— C25H19N3O7
methyl 4-[(3R,3aR,6aS)-3-(3-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate
—— methyl 4-[(3S,3aR,6aS)-3-(3-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate —— C25H19N3O7
methyl 4-[(3S,3aR,6aS)-3-(3-nitrophenyl)-4,6-dioxo-2-phenyl-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate
—— methyl (1R,2S,3S,4R)-3-[(4-methylphenyl)carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylate —— C17H19NO3
methyl (1R,2S,3S,4R)-3-[(4-methylphenyl)carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylate
—— morpholin-4-yl-[(5R,7R)-3-(1,2,4-triazol-1-yl)-1-adamantyl]methanone —— C17H24N4O2
morpholin-4-yl-[(5R,7R)-3-(1,2,4-triazol-1-yl)-1-adamantyl]methanone
—— methyl (2E)-2-[(1S,4R,7R)-7-(bromomethyl)-4,7-dimethyl-3-oxo-2-bicyclo[2.2.1]heptanylidene]-2-hydroxyacetate —— C13H17BrO4
methyl (2E)-2-[(1S,4R,7R)-7-(bromomethyl)-4,7-dimethyl-3-oxo-2-bicyclo[2.2.1]heptanylidene]-2-hydroxyacetate
—— methyl (5R,6R,7R)-5-hydroxy-7-(4-methoxyphenyl)-5-methyl-3-(trifluoromethyl)-7,8-dihydro-6H-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C16H17F3N4O4
methyl (5R,6R,7R)-5-hydroxy-7-(4-methoxyphenyl)-5-methyl-3-(trifluoromethyl)-7,8-dihydro-6H-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (1S,3S,6R,9S)-9-(2,4-dimethylphenyl)-6,8-dimethyl-4-oxo-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate —— C19H23NO5
methyl (1S,3S,6R,9S)-9-(2,4-dimethylphenyl)-6,8-dimethyl-4-oxo-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate
—— methyl (1S,3S,6R,9R)-9-(2,4-dimethylphenyl)-6,8-dimethyl-4-oxo-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate —— C19H23NO5
methyl (1S,3S,6R,9R)-9-(2,4-dimethylphenyl)-6,8-dimethyl-4-oxo-2,5-dioxa-8-azatricyclo[4.4.0.01,3]decane-3-carboxylate
—— methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5S)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[(Z)-[4-(2,4-dichlorophenyl)-2-[[(2R)-oxolan-2-yl]methylimino]-1,3-thiazol-3-yl]iminomethyl]benzoate —— C23H21Cl2N3O3S
methyl 4-[(Z)-[4-(2,4-dichlorophenyl)-2-[[(2R)-oxolan-2-yl]methylimino]-1,3-thiazol-3-yl]iminomethyl]benzoate
—— methyl (5R)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5R)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5S)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5R)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
methyl (5S)-7-ethyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26FN3O4S
methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-7-ethyl-5-(4-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5S)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5S)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5R)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2S)-3-(2-chlorophenyl)-2-cyano-3-oxopropanoate —— C11H8ClNO3
methyl (2S)-3-(2-chlorophenyl)-2-cyano-3-oxopropanoate
—— methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 3-[[(3R)-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]carbamoylamino]benzoate —— C33H28N4O5
methyl 3-[[(3R)-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]carbamoylamino]benzoate
—— methyl (5R)-5-(3-chlorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22ClN3O4S
methyl (5R)-5-(3-chlorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-7-ethyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
methyl (5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-7-ethyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27N3O4S
methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2,5-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5R)-5-(2,5-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H29N3O4S
methyl (5R)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H25N3O4S
methyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate