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—— methyl 2-[(2S)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C24H27N5O6S2
methyl 2-[(2S)-1-[3-[(Z)-[3-(3-methoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 2-[(2S)-1-[7-methyl-3-[(Z)-[3-(3-methylbutyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C25H29N5O5S2
methyl 2-[(2S)-1-[7-methyl-3-[(Z)-[3-(3-methylbutyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl (2Z)-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-7-methyl-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H32N2O5S
methyl (2Z)-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-7-methyl-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1R,9S,13E,16S)-13-[[4-(difluoromethoxy)phenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H18F2N2O5S
methyl (1R,9S,13E,16S)-13-[[4-(difluoromethoxy)phenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl 2-[(2R)-1-[7-methyl-3-[(Z)-[3-(3-methylbutyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C25H29N5O5S2
methyl 2-[(2R)-1-[7-methyl-3-[(Z)-[3-(3-methylbutyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 2-[(2R)-1-[7-methyl-4-oxo-3-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C25H29N5O5S2
methyl 2-[(2R)-1-[7-methyl-4-oxo-3-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 2-[(2S)-1-[7-methyl-4-oxo-3-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C25H29N5O5S2
methyl 2-[(2S)-1-[7-methyl-4-oxo-3-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— methyl 4-[(Z)-[3-(4-ethylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]benzoate —— C20H17NO3S2
methyl 4-[(Z)-[3-(4-ethylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]benzoate
—— methylsulfonyl (3S,4R,5R)-3-benzoyl-2,2-difluoro-3,4,5-trihydroxy-6-oxo-6-phenylhexanoate —— C20H18F2O9S
methylsulfonyl (3S,4R,5R)-3-benzoyl-2,2-difluoro-3,4,5-trihydroxy-6-oxo-6-phenylhexanoate
—— methyl (1R,9S,13E,16R)-13-[[4-(difluoromethoxy)phenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H18F2N2O5S
methyl (1R,9S,13E,16R)-13-[[4-(difluoromethoxy)phenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl 2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoate —— C12H11NO4S2
methyl 2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoate
—— methyl (1R,9S,13E,16R)-9-methyl-14-oxo-13-(thiophen-2-ylmethylidene)-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C20H16N2O4S2
methyl (1R,9S,13E,16R)-9-methyl-14-oxo-13-(thiophen-2-ylmethylidene)-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16S)-9-methyl-14-oxo-13-(thiophen-2-ylmethylidene)-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C20H16N2O4S2
methyl (1R,9S,13E,16S)-9-methyl-14-oxo-13-(thiophen-2-ylmethylidene)-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16R)-13-[(2-hydroxy-3-methoxyphenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H20N2O6S
methyl (1R,9S,13E,16R)-13-[(2-hydroxy-3-methoxyphenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16R)-9-methyl-14-oxo-13-[(4-propan-2-yloxyphenyl)methylidene]-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C25H24N2O5S
methyl (1R,9S,13E,16R)-9-methyl-14-oxo-13-[(4-propan-2-yloxyphenyl)methylidene]-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16S)-13-[(2-hydroxy-3-methoxyphenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H20N2O6S
methyl (1R,9S,13E,16S)-13-[(2-hydroxy-3-methoxyphenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,13S,17R)-13-methyl-15-sulfanylidene-12-oxa-14,16-diazatetracyclo[11.3.1.02,11.03,8]heptadeca-2(11),3,5,7,9-pentaene-17-carboxylate —— C17H16N2O3S
methyl (1R,13S,17R)-13-methyl-15-sulfanylidene-12-oxa-14,16-diazatetracyclo[11.3.1.02,11.03,8]heptadeca-2(11),3,5,7,9-pentaene-17-carboxylate
—— methyl (1R,9S,13E,16S)-9-methyl-14-oxo-13-[(4-propan-2-yloxyphenyl)methylidene]-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C25H24N2O5S
methyl (1R,9S,13E,16S)-9-methyl-14-oxo-13-[(4-propan-2-yloxyphenyl)methylidene]-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16R)-9-methyl-13-[(4-nitrophenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C22H17N3O6S
methyl (1R,9S,13E,16R)-9-methyl-13-[(4-nitrophenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16S)-9-methyl-13-[(4-nitrophenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C22H17N3O6S
methyl (1R,9S,13E,16S)-9-methyl-13-[(4-nitrophenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1S,9R,13R)-9-methyl-11-methylsulfanyl-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2,4,6,11-tetraene-13-carboxylate —— C14H16N2O3S
methyl (1S,9R,13R)-9-methyl-11-methylsulfanyl-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2,4,6,11-tetraene-13-carboxylate
—— methyl (1R,9S,13E,16R)-9-methyl-13-[(4-methylphenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H20N2O4S
methyl (1R,9S,13E,16R)-9-methyl-13-[(4-methylphenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16R)-13-[(2,4-dichlorophenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C22H16Cl2N2O4S
methyl (1R,9S,13E,16R)-13-[(2,4-dichlorophenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,9S,13E,16S)-9-methyl-13-[(4-methylphenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C23H20N2O4S
methyl (1R,9S,13E,16S)-9-methyl-13-[(4-methylphenyl)methylidene]-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1S,9R,13S)-9-methyl-11-methylsulfanyl-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2,4,6,11-tetraene-13-carboxylate —— C14H16N2O3S
methyl (1S,9R,13S)-9-methyl-11-methylsulfanyl-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2,4,6,11-tetraene-13-carboxylate
—— methyl (1R,9S,13E,16S)-13-[(2,4-dichlorophenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C22H16Cl2N2O4S
methyl (1R,9S,13E,16S)-13-[(2,4-dichlorophenyl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1R,13S,17S)-13-methyl-15-sulfanylidene-12-oxa-14,16-diazatetracyclo[11.3.1.02,11.03,8]heptadeca-2(11),3,5,7,9-pentaene-17-carboxylate —— C17H16N2O3S
methyl (1R,13S,17S)-13-methyl-15-sulfanylidene-12-oxa-14,16-diazatetracyclo[11.3.1.02,11.03,8]heptadeca-2(11),3,5,7,9-pentaene-17-carboxylate
—— methyl 2-[[(1R,4S)-4,7,7-trimethyl-2,3-dioxobicyclo[2.2.1]heptane-1-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H25NO5S
methyl 2-[[(1R,4S)-4,7,7-trimethyl-2,3-dioxobicyclo[2.2.1]heptane-1-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl N-[(Z)-[cyclohexyl(phenyl)methylidene]amino]carbamate —— C15H20N2O2
methyl N-[(Z)-[cyclohexyl(phenyl)methylidene]amino]carbamate
—— methyl 4-[[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaene-1-carbonyl]amino]benzoate —— C25H25N3O3
methyl 4-[[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaene-1-carbonyl]amino]benzoate
—— methyl (2Z)-2-[[4-[2-(2-bromo-4,5-dimethylanilino)-2-oxoethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H28BrN3O5S
methyl (2Z)-2-[[4-[2-(2-bromo-4,5-dimethylanilino)-2-oxoethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[[(1S,2S,4S)-2-bromo-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate —— C19H22BrNO4
methyl 2-[[(1S,2S,4S)-2-bromo-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate
—— methyl 2-[(1S,2R,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]benzoate —— C17H17NO4
methyl 2-[(1S,2R,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]benzoate
—— methyl (2Z)-2-(3-ethoxybenzylidene)-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22N2O4S
methyl (2Z)-2-(3-ethoxybenzylidene)-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaene-1-carbonyl]amino]benzoate —— C25H25N3O3
methyl 2-[[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaene-1-carbonyl]amino]benzoate
—— methyl 2-[(5Z)-5-[(5-chloro-2-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C15H14ClNO5S
methyl 2-[(5Z)-5-[(5-chloro-2-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— methyl 2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate —— C12H21NO2
methyl 2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate
—— methyl (2Z)-2-[[4-[2-(3,4-dimethylanilino)-2-oxoethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29N3O5S
methyl (2Z)-2-[[4-[2-(3,4-dimethylanilino)-2-oxoethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[[2-[(5S,7S)-3-(4-methylphenyl)-1-adamantyl]acetyl]amino]benzoate —— C27H31NO3
methyl 4-[[2-[(5S,7S)-3-(4-methylphenyl)-1-adamantyl]acetyl]amino]benzoate
—— methyl (2Z)-2-(4-ethoxy-3-methoxybenzylidene)-7-methyl-3-oxo-5-[4-(propan-2-yl)phenyl]-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H30N2O5S
methyl (2Z)-2-(4-ethoxy-3-methoxybenzylidene)-7-methyl-3-oxo-5-[4-(propan-2-yl)phenyl]-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z)-2-[(4-ethoxy-3-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24N2O5S
methyl (2Z)-2-[(4-ethoxy-3-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 5-(4-ethylphenyl)-1-[(5R,7R)-3-methyl-1-adamantyl]-4,6-dioxopyrrolo[3,4-c]pyrazole-3-carboxylate —— C26H29N3O4
methyl 5-(4-ethylphenyl)-1-[(5R,7R)-3-methyl-1-adamantyl]-4,6-dioxopyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl 3-[(3E)-3-(phenylhydrazinylidene)indol-2-yl]propanoate —— C18H17N3O2
methyl 3-[(3E)-3-(phenylhydrazinylidene)indol-2-yl]propanoate
—— methyl 2-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate —— C12H21NO2
methyl 2-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate
—— methyl 2-[[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate —— C12H21NO2
methyl 2-[[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]acetate
—— methyl 2-[(5Z)-5-{[1-(4-chlorobenzyl)-1H-indol-3-yl]methylidene}-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoate —— C27H19ClN2O3S2
methyl 2-[(5Z)-5-{[1-(4-chlorobenzyl)-1H-indol-3-yl]methylidene}-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoate
—— methyl N-[[(1E)-1-(6-oxocyclohexa-2,4-dien-1-ylidene)propyl]amino]carbamate —— C11H14N2O3
methyl N-[[(1E)-1-(6-oxocyclohexa-2,4-dien-1-ylidene)propyl]amino]carbamate
—— methyl 4-[[(E)-(5-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]benzoate —— C15H12N2O5
methyl 4-[[(E)-(5-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]benzoate
—— methyl 5-(4-ethylphenyl)-1-[(5S,7S)-3-methyl-1-adamantyl]-4,6-dioxopyrrolo[3,4-c]pyrazole-3-carboxylate —— C26H29N3O4
methyl 5-(4-ethylphenyl)-1-[(5S,7S)-3-methyl-1-adamantyl]-4,6-dioxopyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl 4-[[2-[(5R,7R)-3-(4-methylphenyl)-1-adamantyl]acetyl]amino]benzoate —— C27H31NO3
methyl 4-[[2-[(5R,7R)-3-(4-methylphenyl)-1-adamantyl]acetyl]amino]benzoate