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—— methyl 2-[6-oxo-2-[(2R)-1-oxo-1-[(2-propan-2-ylpyrazol-3-yl)amino]propan-2-yl]sulfanyl-1H-pyrimidin-4-yl]acetate —— C16H21N5O4S
methyl 2-[6-oxo-2-[(2R)-1-oxo-1-[(2-propan-2-ylpyrazol-3-yl)amino]propan-2-yl]sulfanyl-1H-pyrimidin-4-yl]acetate
—— methyl 2-[6-oxo-2-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1H-pyrimidin-4-yl]acetate —— C17H15N3O4S
methyl 2-[6-oxo-2-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1H-pyrimidin-4-yl]acetate
—— methyl 2-[6-oxo-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1H-pyrimidin-4-yl]acetate —— C16H14N4O4S
methyl 2-[6-oxo-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1H-pyrimidin-4-yl]acetate
—— methyl 4-[[(1S)-2-[4-(1-benzothiophene-2-carbonyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C31H32N2O5S
methyl 4-[[(1S)-2-[4-(1-benzothiophene-2-carbonyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl 4-methyl-3-[[(2S)-1-oxo-1-(2-oxoimidazolidin-1-yl)propan-2-yl]amino]benzoate —— C15H19N3O4
methyl 4-methyl-3-[[(2S)-1-oxo-1-(2-oxoimidazolidin-1-yl)propan-2-yl]amino]benzoate
—— methyl (1R,9S,13E,16S)-13-[(1-ethyl-3-methylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C22H22N4O4S
methyl (1R,9S,13E,16S)-13-[(1-ethyl-3-methylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl 2-[2-[2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H19N3O5S
methyl 2-[2-[2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— Methyl 3-[2-oxo-2-[[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]ethoxy]benzoate —— C18H15F3N2O5
Methyl 3-[2-oxo-2-[[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]ethoxy]benzoate
—— methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(2,6-dichlorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate —— C28H27Cl3N2O4
methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(2,6-dichlorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate
—— Methyl 3-[2-(ethoxycarbonylamino)-2-oxoethoxy]benzoate —— C13H15NO6
Methyl 3-[2-(ethoxycarbonylamino)-2-oxoethoxy]benzoate
—— methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(5-chlorothiophen-2-yl)sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate —— C25H26Cl2N2O5S2
methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(5-chlorothiophen-2-yl)sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 2-[2-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C15H21N3O5S
methyl 2-[2-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[(2R)-1-(1-adamantylamino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C20H27N3O4S
methyl 2-[2-[(2R)-1-(1-adamantylamino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-(4-acetamidophenyl)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H17N3O5S
methyl 2-[2-[2-(4-acetamidophenyl)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-(2,6-difluorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate —— C28H27ClF2N2O4
methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-(2,6-difluorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 4-[[(1S)-2-[4-(4-bromobenzoyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C29H31BrN2O5
methyl 4-[[(1S)-2-[4-(4-bromobenzoyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl (2Z)-2-[2-[(3S,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate —— C26H23N3O3S
methyl (2Z)-2-[2-[(3S,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate
—— methyl 4-[[(1S)-1-(4-chlorophenyl)-2-(4-thiophen-2-ylsulfonylpiperazin-1-yl)ethoxy]methyl]benzoate —— C25H27ClN2O5S2
methyl 4-[[(1S)-1-(4-chlorophenyl)-2-(4-thiophen-2-ylsulfonylpiperazin-1-yl)ethoxy]methyl]benzoate
—— methyl 4-[[(1R)-2-[4-(1-benzothiophene-2-carbonyl)piperazin-1-yl]-1-(4-chlorophenyl)ethoxy]methyl]benzoate —— C30H29ClN2O4S
methyl 4-[[(1R)-2-[4-(1-benzothiophene-2-carbonyl)piperazin-1-yl]-1-(4-chlorophenyl)ethoxy]methyl]benzoate
—— methyl (2E)-2-[2-[(3S,3aS,7Z)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate —— C26H23N3O3S
methyl (2E)-2-[2-[(3S,3aS,7Z)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate
—— methyl 4-[[(1R)-2-[4-(2,6-dichlorobenzoyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C29H30Cl2N2O5
methyl 4-[[(1R)-2-[4-(2,6-dichlorobenzoyl)piperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl 3-[(Z)-2-cyano-3-[(5-methyl-1,2-oxazol-3-yl)amino]-3-oxoprop-1-enyl]-1H-indole-4-carboxylate —— C18H14N4O4
methyl 3-[(Z)-2-cyano-3-[(5-methyl-1,2-oxazol-3-yl)amino]-3-oxoprop-1-enyl]-1H-indole-4-carboxylate
—— methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(2,6-difluorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate —— C28H27ClF2N2O4
methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-(2,6-difluorobenzoyl)piperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 4-[[(1S)-2-[4-(3,5-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C28H30F2N2O6S
methyl 4-[[(1S)-2-[4-(3,5-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl 3-[[(Z)-2-cyano-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)prop-2-enoyl]amino]thiophene-2-carboxylate —— C17H12N4O3S
methyl 3-[[(Z)-2-cyano-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)prop-2-enoyl]amino]thiophene-2-carboxylate
—— methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-(5-chlorothiophen-2-yl)sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate —— C25H26Cl2N2O5S2
methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-(5-chlorothiophen-2-yl)sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 3-methoxy-4-[[5-[(3R)-3-methylpiperidin-1-yl]sulfonyl-1-[[(2S)-oxolan-2-yl]methyl]benzimidazol-2-yl]sulfanylmethyl]benzoate —— C28H35N3O6S2
methyl 3-methoxy-4-[[5-[(3R)-3-methylpiperidin-1-yl]sulfonyl-1-[[(2S)-oxolan-2-yl]methyl]benzimidazol-2-yl]sulfanylmethyl]benzoate
—— methyl (2E)-2-[2-[(3S,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate —— C26H23N3O3S
methyl (2E)-2-[2-[(3S,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-4-oxo-1,3-thiazol-5-ylidene]acetate
—— methyl (2E)-2-[(5R)-9-(1,3-dithiolan-2-ylidene)-3-oxo-5-phenyl-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate —— C22H20N2O3S3
methyl (2E)-2-[(5R)-9-(1,3-dithiolan-2-ylidene)-3-oxo-5-phenyl-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate
—— methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-[2-(2,3-dimethoxyphenyl)ethylcarbamoyl]piperazin-1-yl]ethoxy]methyl]benzoate —— C32H38ClN3O6
methyl 4-[[(1S)-1-(4-chlorophenyl)-2-[4-[2-(2,3-dimethoxyphenyl)ethylcarbamoyl]piperazin-1-yl]ethoxy]methyl]benzoate
—— methyl (5E)-2-(3,4-dichloroanilino)-4-oxo-5-[[4-(2,2,2-trifluoroethyl)phenyl]methylidene]thiophene-3-carboxylate —— C21H14Cl2F3NO3S
methyl (5E)-2-(3,4-dichloroanilino)-4-oxo-5-[[4-(2,2,2-trifluoroethyl)phenyl]methylidene]thiophene-3-carboxylate
—— methyl 2-[2-[2-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C18H25N3O4S
methyl 2-[2-[2-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl (1S,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocycloheptane-1-carboxylate —— C16H17ClO3
methyl (1S,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocycloheptane-1-carboxylate
—— methyl (2E)-2-[(5S)-9-(1,3-dithiolan-2-ylidene)-5-(4-methoxyphenyl)-3-oxo-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate —— C23H22N2O4S3
methyl (2E)-2-[(5S)-9-(1,3-dithiolan-2-ylidene)-5-(4-methoxyphenyl)-3-oxo-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate
—— methyl (1R,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocycloheptane-1-carboxylate —— C16H17ClO3
methyl (1R,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocycloheptane-1-carboxylate
—— methyl 4-[(2,5-dichlorophenyl)carbamoyl]-2-[3-[(5E)-5-[(3-methylphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoylamino]benzoate —— C29H23Cl2N3O6S
methyl 4-[(2,5-dichlorophenyl)carbamoyl]-2-[3-[(5E)-5-[(3-methylphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoylamino]benzoate
—— methyl (1S,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocyclohexane-1-carboxylate —— C15H15ClO3
methyl (1S,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocyclohexane-1-carboxylate
—— methyl (2E)-2-[(5R)-9-(1,3-dithiolan-2-ylidene)-5-(4-methoxyphenyl)-3-oxo-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate —— C23H22N2O4S3
methyl (2E)-2-[(5R)-9-(1,3-dithiolan-2-ylidene)-5-(4-methoxyphenyl)-3-oxo-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate
—— methyl (2E)-2-[(5S)-9-(1,3-dithiolan-2-ylidene)-3-oxo-5-phenyl-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate —— C22H20N2O3S3
methyl (2E)-2-[(5S)-9-(1,3-dithiolan-2-ylidene)-3-oxo-5-phenyl-5,6,7,8-tetrahydro-[1,3]thiazolo[2,3-b]quinazolin-2-ylidene]acetate
—— methyl 2-[2-[2-[4-(difluoromethoxy)phenyl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C16H14F2N2O5S
methyl 2-[2-[2-[4-(difluoromethoxy)phenyl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H16N4O4S
methyl 2-[2-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-(2-methoxy-2-oxoethyl)sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C10H12N2O5S
methyl 2-[2-(2-methoxy-2-oxoethyl)sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-[2-(2,3-dimethoxyphenyl)ethylcarbamoyl]piperazin-1-yl]ethoxy]methyl]benzoate —— C32H38ClN3O6
methyl 4-[[(1R)-1-(4-chlorophenyl)-2-[4-[2-(2,3-dimethoxyphenyl)ethylcarbamoyl]piperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 2-[2-[2-[(2R)-2-carbamoylpiperidin-1-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C15H20N4O5S
methyl 2-[2-[2-[(2R)-2-carbamoylpiperidin-1-yl]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-[cyclopropyl-[(2-fluorophenyl)methyl]amino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C19H20FN3O4S
methyl 2-[2-[2-[cyclopropyl-[(2-fluorophenyl)methyl]amino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-methyl-5-[2-[2-(4-methylpiperidin-1-yl)-2-oxoethoxy]-2-oxoethyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C19H23N3O6S
methyl 2-methyl-5-[2-[2-(4-methylpiperidin-1-yl)-2-oxoethoxy]-2-oxoethyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— methyl (1R,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocyclohexane-1-carboxylate —— C15H15ClO3
methyl (1R,3Z)-3-[(4-chlorophenyl)methylidene]-2-oxocyclohexane-1-carboxylate
—— Methyl 4-[[[2-(4-acetamidophenyl)sulfanylacetyl]amino]methyl]benzoate —— C19H20N2O4S
Methyl 4-[[[2-(4-acetamidophenyl)sulfanylacetyl]amino]methyl]benzoate
—— methyl 5-[2-[2-[[(1R)-1-cyclopropylethyl]amino]-2-oxoethoxy]-2-oxoethyl]-2-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C18H21N3O6S
methyl 5-[2-[2-[[(1R)-1-cyclopropylethyl]amino]-2-oxoethoxy]-2-oxoethyl]-2-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— methyl 5-[2-(3,3-dimethyl-2-oxobutoxy)-2-oxoethyl]-2-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C17H20N2O6S
methyl 5-[2-(3,3-dimethyl-2-oxobutoxy)-2-oxoethyl]-2-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate