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中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl 2-[2-[(2R)-1-(4-chloroanilino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C16H16ClN3O4S
methyl 2-[2-[(2R)-1-(4-chloroanilino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[(2R)-1-(4-acetylanilino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C18H19N3O5S
methyl 2-[2-[(2R)-1-(4-acetylanilino)-1-oxopropan-2-yl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[6-oxo-2-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]sulfanyl-1H-pyrimidin-4-yl]acetate —— C17H19N3O4S
methyl 2-[6-oxo-2-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]sulfanyl-1H-pyrimidin-4-yl]acetate
—— Methyl 3-[[2-(1,3-dioxo-2-azaspiro[4.5]decan-2-yl)acetyl]amino]-4-methylbenzoate —— C20H24N2O5
Methyl 3-[[2-(1,3-dioxo-2-azaspiro[4.5]decan-2-yl)acetyl]amino]-4-methylbenzoate
—— methyl 2-[2-[2-[[(1R)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H18ClN3O4S
methyl 2-[2-[2-[[(1R)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-(2-methoxy-5-methylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H19N3O5S
methyl 2-[2-[2-(2-methoxy-5-methylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-(3-chloro-2-methylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C16H16ClN3O4S
methyl 2-[2-[2-(3-chloro-2-methylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-(6-oxo-2-propylsulfanyl-1H-pyrimidin-4-yl)acetate —— C10H14N2O3S
methyl 2-(6-oxo-2-propylsulfanyl-1H-pyrimidin-4-yl)acetate
—— Methyl 4-[(1,3-dioxo-2-azaspiro[4.5]decan-2-yl)methyl]benzoate —— C18H21NO4
Methyl 4-[(1,3-dioxo-2-azaspiro[4.5]decan-2-yl)methyl]benzoate
—— methyl 2-[2-[2-(2,6-difluoroanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C15H13F2N3O4S
methyl 2-[2-[2-(2,6-difluoroanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-(1-adamantylamino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C19H25N3O4S
methyl 2-[2-[2-(1-adamantylamino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 4-[[(1R)-1-(3-methoxyphenyl)-2-[4-[2-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate —— C29H31F3N2O6S
methyl 4-[[(1R)-1-(3-methoxyphenyl)-2-[4-[2-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 2-[2-[(4-bromophenyl)methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate —— C14H13BrN2O3S
methyl 2-[2-[(4-bromophenyl)methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2-[2-[2-(2-methylsulfanylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C16H17N3O4S2
methyl 2-[2-[2-(2-methylsulfanylanilino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl (3S)-2-[2-(5-phenyltetrazol-2-yl)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C20H19N5O3
methyl (3S)-2-[2-(5-phenyltetrazol-2-yl)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— methyl 4-[[(1S)-1-(3-methoxyphenyl)-2-[4-[2-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate —— C29H31F3N2O6S
methyl 4-[[(1S)-1-(3-methoxyphenyl)-2-[4-[2-(trifluoromethyl)phenyl]sulfonylpiperazin-1-yl]ethoxy]methyl]benzoate
—— methyl 2-[2-[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C15H14N4O4S2
methyl 2-[2-[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 4-[(S)-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]methyl]benzoate —— C32H35N5O6S
methyl 4-[(S)-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]methyl]benzoate
—— methyl (3S)-2-[2-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)oxyacetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C18H19N3O6
methyl (3S)-2-[2-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)oxyacetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— methyl (3R)-2-[2-(2-carbamoylphenoxy)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C20H20N2O5
methyl (3R)-2-[2-(2-carbamoylphenoxy)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— methyl 3-[(Z)-2-cyano-3-oxo-3-(2-phenylethylamino)prop-1-enyl]-1H-indole-4-carboxylate —— C22H19N3O3
methyl 3-[(Z)-2-cyano-3-oxo-3-(2-phenylethylamino)prop-1-enyl]-1H-indole-4-carboxylate
—— methyl (3S)-2-[2-(4-acetamidophenoxy)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C21H22N2O5
methyl (3S)-2-[2-(4-acetamidophenoxy)acetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— methyl 2-[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H17N3O6S
methyl 2-[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl-6-oxo-1H-pyrimidin-4-yl]acetate
—— methyl 2,4-dimethyl-5-[(2S)-2-(naphthalen-1-ylamino)propanoyl]-1H-pyrrole-3-carboxylate —— C21H22N2O3
methyl 2,4-dimethyl-5-[(2S)-2-(naphthalen-1-ylamino)propanoyl]-1H-pyrrole-3-carboxylate
—— methyl 5-[(2S)-2-(3-chloro-2-methylanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H21ClN2O3
methyl 5-[(2S)-2-(3-chloro-2-methylanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl 5-[[(E)-3-(1-benzyltriazol-4-yl)prop-2-enoyl]oxymethyl]-2-methylfuran-3-carboxylate —— C20H19N3O5
methyl 5-[[(E)-3-(1-benzyltriazol-4-yl)prop-2-enoyl]oxymethyl]-2-methylfuran-3-carboxylate
—— methyl (3R)-2-[2-(2-hydroxy-4-methylbenzoyl)oxyacetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C21H21NO6
methyl (3R)-2-[2-(2-hydroxy-4-methylbenzoyl)oxyacetyl]-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— methyl 4-[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C28H26N4O4S2
methyl 4-[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— methyl 4-[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C28H26N4O4S2
methyl 4-[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— methyl 4-[(R)-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]methyl]benzoate —— C32H35N5O6S
methyl 4-[(R)-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]methyl]benzoate
—— methyl 3-[[(Z)-3-quinolin-2-ylprop-2-enoyl]oxymethyl]benzoate —— C21H17NO4
methyl 3-[[(Z)-3-quinolin-2-ylprop-2-enoyl]oxymethyl]benzoate
—— methyl 5-[(2S)-2-(cycloheptylamino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H28N2O3
methyl 5-[(2S)-2-(cycloheptylamino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl 1-[2-[(E)-3-(1-benzyltriazol-4-yl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate —— C21H24N4O5
methyl 1-[2-[(E)-3-(1-benzyltriazol-4-yl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate
—— methyl 2-[[3-[4-[(2S)-butan-2-yl]phenyl]-7-chloro-4-oxoquinazolin-2-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C28H25ClN4O4S2
methyl 2-[[3-[4-[(2S)-butan-2-yl]phenyl]-7-chloro-4-oxoquinazolin-2-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— methyl 5-[(2S)-2-(2-methoxyanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H22N2O4
methyl 5-[(2S)-2-(2-methoxyanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl 5-[(2S)-2-(2,5-dimethylanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C19H24N2O3
methyl 5-[(2S)-2-(2,5-dimethylanilino)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl (5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
methyl (5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
methyl (5R)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H34N4O4S
methyl (5R)-7-ethyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[[2-[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C22H29N3O3S
methyl 2-[[2-[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— methyl (5R)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
methyl (5R)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[[3-[4-[(2R)-butan-2-yl]phenyl]-7-chloro-4-oxoquinazolin-2-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C28H25ClN4O4S2
methyl 2-[[3-[4-[(2R)-butan-2-yl]phenyl]-7-chloro-4-oxoquinazolin-2-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H34N4O4S
methyl (5S)-7-ethyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
methyl (5R)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[[(1S)-2-[4-(2,4-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C28H30F2N2O6S
methyl 4-[[(1S)-2-[4-(2,4-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl (5S)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
methyl (5S)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[[(1R)-2-[4-(2,4-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate —— C28H30F2N2O6S
methyl 4-[[(1R)-2-[4-(2,4-difluorophenyl)sulfonylpiperazin-1-yl]-1-(3-methoxyphenyl)ethoxy]methyl]benzoate
—— methyl (5S)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
methyl (5S)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O4S
methyl (5R)-7-ethyl-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(3-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O4S
methyl (5S)-7-ethyl-5-(3-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate